N-benzyl-2-[benzyl-[3-(3,4-dimethoxyphenoxy)propyl]amino]acetamide

N-[(2-chlorophenyl)methyl]-2-[(3,4-difluorophenyl)methyl-[2-(3,4-dimethoxyphenoxy)ethyl]amino]acetamide

N-benzyl-2-[(3,4-difluorophenyl)methyl-[3-(3,4-dimethoxyphenoxy)propyl]amino]acetamide

[(3aR,6aS)-2-(6-fluoroquinazolin-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

N-benzyl-2-[2-(3,4-dimethoxyphenoxy)ethyl-(thiophen-2-ylmethyl)amino]acetamide

[(3aR,6aS)-2-(5-fluoro-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

N-benzyl-2-[3-(3,4-dimethoxyphenoxy)propyl-(thiophen-2-ylmethyl)amino]acetamide

[(7R)-4-(5-chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

N-[(2-chlorophenyl)methyl]-2-[2-(3,4-dimethoxyphenoxy)ethyl-[(4-fluorophenyl)methyl]amino]acetamide

2-[benzyl-[2-(3,4-dimethoxyphenoxy)ethyl]amino]-N-[(2-chlorophenyl)methyl]acetamide

[(3aR,6aS)-2-(1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

N-[(2-chlorophenyl)methyl]-2-[2-(3,4-dimethoxyphenoxy)ethyl-(thiophen-2-ylmethyl)amino]acetamide

[(3aR,6aS)-2-(5-chloro-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-(5-methyl-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

2-[(3,4-difluorophenyl)methyl-[2-(3,4-dimethoxyphenoxy)ethyl]amino]-N-(2-methylpropyl)acetamide

[(3aR,6aS)-2-(5-chloro-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[2-(triazol-2-yl)phenyl]methanone

2-[benzyl-[2-(3,4-dimethoxyphenoxy)ethyl]amino]-N-(2-methylpropyl)acetamide

[(3aR,6aS)-2-(5-methoxy-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

2-[2-(3,4-dimethoxyphenoxy)ethyl-(thiophen-2-ylmethyl)amino]-N-(2-methylpropyl)acetamide

[5-(5-chloro-1,3-benzoxazol-2-yl)-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-1-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-(5-chloro-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methoxy-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-[5-(trifluoromethyl)-1,3-benzoxazol-2-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

2-[2-(3,4-dimethoxyphenoxy)ethyl-[(4-fluorophenyl)methyl]amino]-N-(2-methylpropyl)acetamide

[(3aR,6aS)-2-(1,3-benzoxazol-2-yl)-3a,6a-difluoro-1,3,4,6-tetrahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aS,6aR)-2-(5-chloro-1,3-benzoxazol-2-yl)-3a,6a-difluoro-1,3,4,6-tetrahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-(1-methylbenzimidazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-(5-chloro-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-fluoro-2-(triazol-2-yl)phenyl]methanone

[(3aS,6aR)-2-(5-chloro-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[2-(triazol-2-yl)-5-(trifluoromethyl)phenyl]methanone

[2-(5-chloro-1,3-benzoxazol-2-yl)-3a-methyl-3,4,6,6a-tetrahydro-1H-pyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aS,6aR)-2-(5-chloro-1,3-benzothiazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-(5-chloro-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-chloro-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-(5-chloro-1,3-benzoxazol-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[2-(triazol-2-yl)-5-(trifluoromethoxy)phenyl]methanone

[(3aR,6aS)-2-quinazolin-4-yl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-[(5-chloro-1,3-benzoxazol-2-yl)methyl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-[4-(3-chlorophenyl)-1,3-oxazol-2-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aS,6aR)-2-[5-(trifluoromethoxy)-1,3-benzoxazol-2-yl]-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aS,6aR)-2-(4,5,6-trimethylpyrimidin-2-yl)-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[(3aR,6aS)-2-(5-chloro-1,3-benzoxazol-2-yl)-3a,6a-dimethyl-1,3,4,6-tetrahydropyrrolo[3,4-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[1-(5-chloro-1,3-benzoxazol-2-yl)-3,4,4a,5,7,7a-hexahydro-2H-pyrrolo[3,4-b]pyridin-6-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[6-(5-chloro-1,3-benzoxazol-2-yl)-3,4,4a,5,7,7a-hexahydro-2H-pyrrolo[3,4-b]pyridin-1-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

[1-(5-chloro-1,3-benzoxazol-2-yl)-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl]-[5-methyl-2-(triazol-2-yl)phenyl]methanone

4-(2-Chloro-6-fluoro-4-methoxybenzyl)-2-(3,4-dimethoxyphenyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

9-(4,6-dimethylpyrimidin-2-yl)-2-[(5-methoxy-1H-indol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-1-one

4-(2,6-Difluoro-4-methoxybenzyl)-2-(5,6-dimethoxypyridin-2-yl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

4-(2,6-Difluoro-4-methoxybenzyl)-2-(2,6-dimethoxypyridin-4-yl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

4-(2,6-Difluoro-4-methoxybenzyl)-2-(5,6-dimethoxypyridin-3-yl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

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2-(3,4-Dimethoxyphenyl)-4-(2,6-difluoro-4-methoxybenzyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

4-(2,6-difluoro-4-methoxybenzyl)-2-[6-methoxy-5-(methylamino)pyridin-3-yl]-2H-pyrido[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxide

4-(2-Chloro-6-fluorobenzyl)-2-(3,4-dimethoxyphenyl)-1,1-dioxo-1,4-dihydro-2H-1lambda'6'-benzo[1,2,4]thiadiazin-3-one

4-(2-Chloro-6-fluoro-4-methylbenzyl)-2-(3,4-dimethoxyphenyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

9-(4,6-dimethylpyrimidin-2-yl)-1-(1H-indol-4-ylmethyl)-1,9-diazaspiro[5.5]undecan-2-one

4-(2-chloro-4,6-difluorobenzyl)-2-(3,4-dimethoxyphenyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

9-(4,6-dimethylpyrimidin-2-yl)-2-[(5-phenyl-2H-triazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-1-one

2-(2,6-Dimethoxypyridin-4-yl)-4-(2,4,6-trifluorobenzyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

4-(2-Chloro-4,6-difluorobenzyl)-2-(5,6-dimethoxypyridin-3-yl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

2-(5,6-Dimethoxypyridin-2-yl)-4-(2,4,6-trifluorobenzyl)-2H-pyrido[2,3-e][1,2,4]thiadiazin-3(4H)-one 1,1-dioxide

2-(3,4-Dimethoxyphenyl)-4-(2,4,6-trifluorobenzyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

2-(5,6-dimethoxypyridin-3-yl)-1,1-dioxo-4-[(2,4,6-trifluorophenyl)methyl]pyrido[2,3-e][1,2,4]thiadiazin-3-one

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9-(4,6-dimethylpyrimidin-2-yl)-2-[(4-phenyl-1H-pyrazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-1-one

9-(4,6-dimethylpyrimidin-2-yl)-2-[(2-methyl-5-phenyltriazol-4-yl)methyl]-2,9-diazaspiro[5.5]undecan-1-one

2-(5,6-Dimethoxypyridin-3-yl)-4-(2,4,6-trifluorobenzyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

4-(2,4-Difluoro-6-methoxybenzyl)-2-(3,4-dimethoxyphenyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

2-(3,4-dimethoxyphenyl)-4-(2-fluorobenzyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

9-(4,6-dimethylpyrimidin-2-yl)-2-(2H-indazol-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-1-one

9-(4,6-dimethylpyrimidin-2-yl)-2-(1H-indol-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-1-one

4-(4-Chloro-2-fluorobenzyl)-2-(3,4-dimethoxyphenyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

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2-(1H-indol-3-ylmethyl)-9-(4-methoxypyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-1-one

9-(4,6-dimethylpyrimidin-2-yl)-2-(1H-pyrrolo[2,3-b]pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-1-one

9-(4,6-dimethylpyrimidin-2-yl)-2-[(1-methyl-4-phenylpyrazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-1-one

9-(4,6-dimethylpyrimidin-2-yl)-2-[(1-methylindol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-1-one

4-(2-Chloro-4-fluorobenzyl)-2-(3,4-dimethoxyphenyl)-1,1-dioxo-1,4-dihydro-2H-1lambda'6'-benzo[1,2,4]thiadiazin-3-one

2-(1H-indol-3-ylmethyl)-9-(4-methylpyrimidin-2-yl)-2,9-diazaspiro[5.5]undecan-1-one

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2-(2-Methoxypyridin-4-yl)-4-(2,4,6-trifluorobenzyl)-2H-1,2,4-benzothiadiazin-3(4H)-one 1,1-dioxide

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2-(1H-indol-4-ylmethyl)-9-quinoxalin-2-yl-2,9-diazaspiro[5.5]undecan-1-one

4-Benzyl-2-(3,4-dimethoxyphenyl)-1,1-dioxo-1,4-dihydro-2H-1lambda'6'-benzo[1,2,4]thiadiazin-3-one

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2-phenyl-1-(8-quinoxalin-2-yl-1,8-diazaspiro[4.5]decan-1-yl)ethanone

4-Benzo[1,3]dioxol-5-ylmethyl-2-(3,4-dimethoxyphenyl)-1,1-dioxo-1,4-dihydro-2H-1lambda'6'-benzo[1,2,4]thiadiazin-3-one

2-(1H-indol-3-ylmethyl)-9-pyrazin-2-yl-2,9-diazaspiro[5.5]undecan-1-one

2-(1H-indol-3-ylmethyl)-9-pyrimidin-2-yl-2,9-diazaspiro[5.5]undecan-1-one

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N-[2-[3-[[5-[3-(dimethylcarbamoyl)phenyl]-2-methoxyphenyl]sulfonylamino]anilino]ethyl]-3-methylbenzamide

1-(2-chlorobenzyl)-3-(3,4-dimethoxyphenyl)quinazoline-2,4(1H,3H)-dione