| Compound ID |
Compound Name |
Compound Formula |
|
CP0499901
|
1-[1-(2-Isobutylamino-ethyl)-1H-indazol-5-yl]-3-(4-phenoxy-phenyl)-urea
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|
C26H29N5O2
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0486548
|
1-[1-(2-Cyclopentylamino-ethyl)-1H-indazol-5-yl]-3-(4-phenoxy-phenyl)-urea
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|
C27H29N5O2
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0483655
|
1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-1,3-dihydro-imidazol-2-one
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|
C28H27N5O2
|
1
|
| 1 |
IC50 = 5.9 nM
|
|
|
|
CP0378101
|
1-[1-(3-Cyclopentylamino-propyl)-1H-indazol-5-yl]-3-(4-phenoxy-phenyl)-urea
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|
C28H31N5O2
|
1
|
| 1 |
IC50 = 8.5 nM
|
|
|
|
CP0408146
|
1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea
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|
C26H27N5O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0511996
|
1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-imidazolidin-2-one
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|
C28H29N5O2
|
1
|
| 1 |
IC50 = 19.8 nM
|
|
|
|
CP0382283
|
1-[2-(4-Phenoxy-phenyl)-ethyl]-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea
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|
C28H31N5O2
|
1
|
| 1 |
IC50 = 34.3 nM
|
|
|
|
CP0401319
|
1-{1-[2-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-ethyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea
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|
C28H31N5O3
|
1
|
| 1 |
IC50 = 38.7 nM
|
|
|
|
CP0378102
|
1-(3-{5-[3-(4-Phenoxy-phenyl)-ureido]-indazol-1-yl}-propyl)-piperidine-4-carboxylic acid amide
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|
C29H32N6O3
|
1
|
| 1 |
IC50 = 40.6 nM
|
|
|
|
CP0515945
|
1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea
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|
C27H29N5O2
|
1
|
| 1 |
IC50 = 41.3 nM
|
|
|
|
CP0483661
|
1-(4-Phenoxy-benzyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea
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|
C27H29N5O2
|
1
|
| 1 |
IC50 = 78.5 nM
|
|
|
|
CP0486549
|
1-{1-[3-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-propyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea
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|
C29H33N5O3
|
1
|
| 1 |
IC50 = 82.9 nM
|
|
|
|
CP0394804
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-3,5-dimethoxy-4-methylbenzamide
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|
C23H28N2O5
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0562127
|
1-{1-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea
Show/Hide
|
C28H31N5O3
|
1
|
| 1 |
IC50 = 91.5 nM
|
|
|
|
CP0382281
|
1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea
Show/Hide
|
C27H29N5O2
|
1
|
| 1 |
IC50 = 113 nM
|
|
|
|
CP0541586
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-3,5-dimethoxybenzamide
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|
C22H26N2O5
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0495031
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-3-methoxybenzamide
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|
C21H24N2O4
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0499902
|
1-(2-{5-[3-(4-Phenoxy-phenyl)-ureido]-indazol-1-yl}-ethyl)-piperidine-4-carboxylic acid amide
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|
C28H30N6O3
|
1
|
| 1 |
IC50 = 134 nM
|
|
|
|
CP0486484
|
1-{1-[2-(3,3-Difluoro-pyrrolidin-1-yl)-ethyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea
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|
C26H25F2N5O2
|
1
|
| 1 |
IC50 = 305 nM
|
|
|
|
CP0445642
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-[4-(3-cyanophenyl)phenyl]acetamide
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|
C28H27N3O3
|
1
|
| 1 |
IC50 = 380 nM
|
|
|
|
CP0448050
|
1-(4-Phenoxy-benzyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea
Show/Hide
|
C27H29N5O2
|
1
|
| 1 |
IC50 = 508 nM
|
|
|
|
CP0518139
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-[4-(2-methoxyphenyl)phenyl]acetamide
Show/Hide
|
C28H30N2O4
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0541587
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-3,5-dichlorobenzamide
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|
C20H20Cl2N2O3
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0445478
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-3-(trifluoromethoxy)benzamide
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|
C21H21F3N2O4
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0562126
|
1-[2-(4-Phenoxy-phenyl)-ethyl]-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea
Show/Hide
|
C28H31N5O2
|
1
|
| 1 |
IC50 = 545 nM
|
|
|
|
CP0515567
|
3-Methoxy-N-[1-((E)-3-phenyl-allyl)-piperidin-4-yl]-benzamide
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|
C22H26N2O2
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0391664
|
1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea
Show/Hide
|
C26H27N5O2
|
1
|
| 1 |
IC50 = 581 nM
|
|
|
|
CP0431234
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-(4-phenylphenyl)acetamide
Show/Hide
|
C27H28N2O3
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0449084
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-[4-(4-methoxyphenyl)phenyl]acetamide
Show/Hide
|
C28H30N2O4
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0522509
|
N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-2-[4-(3-methoxyphenyl)phenyl]acetamide
Show/Hide
|
C28H30N2O4
|
1
|
| 1 |
IC50 = 890 nM
|
|
|
|
CP0499909
|
1-(1-Benzyl-piperidin-4-yl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-5-yl]-urea
Show/Hide
|
C26H34N6O
|
1
|
| 1 |
IC50 = 971 nM
|
|
|
|
CP0486506
|
1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-4-yl]-urea
Show/Hide
|
C27H29N5O2
|
1
|
| 1 |
IC50 = 1053 nM
|
|
|
|
CP0431048
|
1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-4-yl]-urea
Show/Hide
|
C26H27N5O2
|
1
|
| 1 |
IC50 = 1851 nM
|
|
|
|
CP0401307
|
1-(1-Benzyl-piperidin-4-yl)-3-[1-(2-pyrrolidin-1-yl-ethyl)-1H-indazol-6-yl]-urea
Show/Hide
|
C26H34N6O
|
1
|
| 1 |
IC50 = 4509 nM
|
|
|
|
CP0514279
|
1-{1-[2-(4-Hydroxy-piperidin-1-yl)-ethyl]-1H-indazol-5-yl}-3-(4-phenoxy-phenyl)-urea
Show/Hide
|
C27H29N5O3
|
1
|
| 1 |
IC50 = 6130 nM
|
|
|
