Brief Information of the Compound and Protein
Compound Name
1-(2-{5-[3-(4-Phenoxy-phenyl)-ureido]-indazol-1-yl}-ethyl)-piperidine-4-carboxylic acid amide
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PubChem ID
CID: 11386451
SID: 16480503
Canonical SMILES
NC(=O)C1CCN(CCn2ncc3cc(NC(=O)Nc4ccc(Oc5ccccc5)cc4)ccc23)CC1
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Compound Formula C28H30N6O3
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q8JZL2
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  1
1
IC50 = 134 nM
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