Brief Information of the Cell Line and Protein
Cell Line ID: CL000423 , IGROV-1
Synonyms
Igrov-1
IGROV 1
IGR-OV1
IGROV1
Igrov1
IGR.OV1
IGROV
OV1/P
OV1/p
OV1-P
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_1304
Protein ID: PT01873 , Trifunctional purine biosynthetic protein adenosine-3
Gene Name GART
Organism Homo sapiens, Human
Protein Classification Enzyme
Uniprot ID P22102
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000423  Protein ID: PT01873
 
Compound ID Compound Name Compound Formula
CP0387048
(2S)-2-[[4-[4-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)butyl]thiophene-2-carbonyl]amino]pentanedioic acid
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C20H23N5O6S
 1
1
IC50 = 1.79 nM
   TI
   LI
   LO
   TS
CP0260881
(2S)-2-[[5-[4-(2-amino-4-oxo-3,7-dihydropyrrolo[2,3-d]pyrimidin-6-yl)butyl]thiophene-3-carbonyl]amino]pentanedioic acid
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C20H23N5O6S
 1
1
IC50 = 2.03 nM
   TI
   LI
   LO
   TS
CP0330758
(S)-2-({5-[4-(2-Amino-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]-pyrimidin-6-yl)-butyl]-thiophene-2-carbonyl}-amino)-pentanedioicAcid
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C20H23N5O6S
 1
1
IC50 = 3.46 nM
   TI
   LI
   LO
   TS
CP0046082
(2S)-2-[(4-{2-[(6R)-2-amino-4-oxo-1H,4H,5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-6-yl]ethyl}phenyl)formamido]pentanedioic acid
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C21H25N5O6
 1
1
IC50 = 5.77 nM
   TI
   LI
   LO
   TS