| Compound ID |
Compound Name |
Compound Formula |
|
CP0055947
|
(15S)-prostaglandin E2
Show/Hide
|
C20H32O5
|
1
|
| 1 |
IC50 < 3 nM
|
|
|
|
CP0168917
|
Omidenepag
Show/Hide
|
C23H22N6O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0440482
|
De-117
Show/Hide
|
C26H28N6O4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0058712
|
N-[5-(2,6-dichlorophenyl)-1,3,4-thiadiazol-2-yl]-4-ethyl-2,3-dihydro-1,4-benzoxazine-6-carboxamide
Show/Hide
|
C19H16Cl2N4O2S
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0493926
|
1-ethyl-4-fluoro-N-[5-[1-(2-hydroxy-2-methylpropanoyl)-4-methylpiperidin-4-yl]-1,3,4-thiadiazol-2-yl]indazole-6-carboxamide
Show/Hide
|
C22H27FN6O3S
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0535739
|
N-[5-(1-acetyl-4-methylpiperidin-4-yl)-1,3,4-thiadiazol-2-yl]-1-ethyl-4-fluoroindazole-6-carboxamide
Show/Hide
|
C20H23FN6O2S
|
1
|
| 1 |
Ki = 11.7 nM
|
|
|
|
CP0483468
|
4-chloro-N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-ethylindazole-6-carboxamide
Show/Hide
|
C15H14ClN5OS
|
1
|
| 1 |
Ki = 14.1 nM
|
|
|
|
CP0380091
|
1-ethyl-4-fluoro-N-[5-[1-(2-hydroxyacetyl)-4-methylpiperidin-4-yl]-1,3,4-thiadiazol-2-yl]indazole-6-carboxamide
Show/Hide
|
C20H23FN6O3S
|
1
|
| 1 |
Ki = 14.5 nM
|
|
|
|
CP0534613
|
1-ethyl-4-fluoro-N-[5-[1-(2-hydroxypropanoyl)-4-methylpiperidin-4-yl]-1,3,4-thiadiazol-2-yl]indazole-6-carboxamide
Show/Hide
|
C21H25FN6O3S
|
1
|
| 1 |
Ki = 16.5 nM
|
|
|
|
CP0397467
|
(E)-3-[2-[(E)-3-[4-[2-(1-cyanoisoindol-2-yl)ethoxy]-3-methoxyphenyl]prop-1-enyl]phenyl]prop-2-enoic acid
Show/Hide
|
C30H26N2O4
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0087631
|
(E)-3-[2-[(E)-3-[4-[2-(2,4-dinitroanilino)ethoxy]-3-methoxyphenyl]prop-1-enyl]phenyl]prop-2-enoic acid
Show/Hide
|
C27H25N3O8
|
1
|
| 1 |
Ki = 23.4 nM
|
|
|
|
CP0314860
|
(E)-3-[2-[(E)-3-[4-[2-(1-cyanoisoindol-2-yl)ethoxy]-3-methoxyphenyl]prop-1-enyl]phenyl]-N-thiophen-2-ylsulfonylprop-2-enamide
Show/Hide
|
C34H29N3O5S2
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0401842
|
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-ethyl-4-fluoroindazole-6-carboxamide
Show/Hide
|
C15H14FN5OS
|
1
|
| 1 |
Ki = 38.3 nM
|
|
|
|
CP0499805
|
N-[5-(1-acetyl-3-methylpyrrolidin-3-yl)-1,3,4-thiadiazol-2-yl]-1-ethyl-4-fluoroindazole-6-carboxamide
Show/Hide
|
C19H21FN6O2S
|
1
|
| 1 |
Ki = 53.1 nM
|
|
|
|
CP0499804
|
N-[5-(1-acetyl-3-methylazetidin-3-yl)-1,3,4-thiadiazol-2-yl]-1-ethyl-4-fluoroindazole-6-carboxamide
Show/Hide
|
C18H19FN6O2S
|
1
|
| 1 |
Ki = 64.5 nM
|
|
|
|
CP0380092
|
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-4-ethyl-2,3-dihydro-1,4-benzoxazine-6-carboxamide
Show/Hide
|
C16H18N4O2S
|
1
|
| 1 |
Ki = 77 nM
|
|
|
|
CP0857864
|
1-(2-(4-((E)-3-(2-((E)-2-Carboxyvinyl)phenyl)allyl)-2-methoxyphenoxy)ethyl)-4-((1E,3E)-4-(4-(dimethylamino)phenyl)buta-1,3-dienyl)-2,6-dimethylpyridinium boron tetrafluoride
Show/Hide
|
C40H43BF4N2O4
|
1
|
| 1 |
Ki = 135 nM
|
|
|
|
CP0924841
|
1-(2-(4-((E)-3-(2-((E)-2-Carboxyvinyl)phenyl)allyl)-2-methoxyphenoxy)ethyl)-4-(4-(dimethylamino)styryl)-2,6-dimethylpyridinium borontetrafluoride
Show/Hide
|
C38H41BF4N2O4
|
1
|
| 1 |
Ki = 218.5 nM
|
|
|
|
CP0508755
|
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-ethylindazole-6-carboxamide
Show/Hide
|
C15H15N5OS
|
1
|
| 1 |
Ki = 310 nM
|
|
|
|
CP0390337
|
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-propan-2-ylindazole-6-carboxamide
Show/Hide
|
C16H17N5OS
|
1
|
| 1 |
Ki = 584 nM
|
|
|
|
CP0917448
|
5-(3-(2-(4-((E)-3-(2-((E)-2-Carboxyvinyl)phenyl)allyl)-2-methoxyphenoxy)ethyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid
Show/Hide
|
C42H34N2O9S
|
1
|
| 1 |
Ki = 678.4 nM
|
|
|
|
CP0401841
|
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-methylindazole-6-carboxamide
Show/Hide
|
C14H13N5OS
|
1
|
| 1 |
Ki = 1066 nM
|
|
|
|
CP0924952
|
4-(3-(2-(4-((E)-3-(2-((E)-2-Carboxyvinyl)phenyl)allyl)-2-methoxyphenoxy)ethyl)thioureido)-2-(6-hydroxy-3-oxo-3H-xanthen-9-yl)benzoic acid
Show/Hide
|
C42H34N2O9S
|
1
|
| 1 |
Ki = 1264.6 nM
|
|
|
|
CP0524936
|
(E)-3-[2-[(E)-3-[4-(2-aminoethoxy)-3-methoxyphenyl]prop-1-enyl]phenyl]prop-2-enoic acid
Show/Hide
|
C21H23NO4
|
1
|
| 1 |
Ki = 1496.8 nM
|
|
|
|
CP0380090
|
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-methylindazole-5-carboxamide
Show/Hide
|
C14H13N5OS
|
1
|
| 1 |
Ki = 5890 nM
|
|
|
|
CP0469649
|
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-1-methylpyrazolo[4,3-b]pyridine-6-carboxamide
Show/Hide
|
C13H12N6OS
|
1
|
| 1 |
Ki > 9650 nM
|
|
|
