Brief Information of the Cell Line and Protein
Cell Line ID: CL000013 , Sf9
Synonyms
SF9
sf9
SF-9
Sf-9
sf-9
Sf 9
Spodoptera frugiperda clone 9
Sf clone 9
IPLB-Sf-9AE
IPLB-SF-9AE
IPLB-SF-9
IPLB-Sf-9
IPLB-Sf9
Category Spontaneously immortalized cell line
Organism
Spodoptera frugiperda (Fall armyworm)
Cellosaurus ID
CVCL_0549
Protein ID: PT01366 , D(3) dopamine receptor
Gene Name DRD3
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P19020
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000013  Protein ID: PT01366
 
Compound ID Compound Name Compound Formula
CP0523741
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]pyridine-3-sulfonamide
   Show/Hide
C23H30Cl2N4O2S
 1
1
IC50 = 0.2 nM
   TI
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CP0459270
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]propanamide
   Show/Hide
C21H31Cl2N3O
 1
1
IC50 = 0.26 nM
   TI
   LI
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   TS
CP0450524
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]acetamide
   Show/Hide
C20H29Cl2N3O
 1
1
IC50 = 0.29 nM
   TI
   LI
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   TS
CP0467830
N-[4-[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]pyridine-3-sulfonamide
   Show/Hide
C24H31F3N4O2S
 1
1
IC50 = 0.3 nM
   TI
   LI
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   TS
CP0459271
[4-[2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]urea
   Show/Hide
C19H28Cl2N4O
 1
1
IC50 = 0.32 nM
   TI
   LI
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   TS
CP0432559
1-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-3-ethylurea
   Show/Hide
C21H32Cl2N4O
 1
1
IC50 = 0.34 nM
   TI
   LI
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   TS
CP0464137
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]pyridine-3-sulfonamide
   Show/Hide
C25H30F3N5O2S
 1
1
IC50 = 0.4 nM
   TI
   LI
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   TS
CP0432558
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-2,2,2-trifluoroacetamide
   Show/Hide
C20H26Cl2F3N3O
 1
1
IC50 = 0.41 nM
   TI
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   TS
CP0459269
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]methanesulfonamide
   Show/Hide
C19H29Cl2N3O2S
 1
1
IC50 = 0.48 nM
   TI
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   TS
CP0523742
4-pyrazol-1-yl-N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]cyclohexyl]benzenesulfonamide
   Show/Hide
C30H37F3N4O2S
 1
1
IC50 = 0.5 nM
   TI
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CP0533088
N-[4-[2-[4-(4-bromo-2-methoxyphenyl)piperazin-1-yl]ethyl]cyclohexyl]-4-methoxybenzenesulfonamide
   Show/Hide
C26H36BrN3O4S
 1
1
IC50 = 0.5 nM
   TI
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   TS
CP0432560
3-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-diethylurea
   Show/Hide
C23H36Cl2N4O
 1
1
IC50 = 0.62 nM
   TI
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   TS
CP0501623
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]-2-oxo-3,4-dihydro-1H-quinoline-6-sulfonamide
   Show/Hide
C29H34F3N5O3S
 1
1
IC50 = 0.7 nM
   TI
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   TS
CP0505453
N-[4-[2-[4-(3-cyanophenyl)piperazin-1-yl]ethyl]cyclohexyl]-3,4-dimethoxybenzenesulfonamide
   Show/Hide
C27H36N4O4S
 1
1
IC50 = 0.7 nM
   TI
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   TS
CP0371880
N-[4-[[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]sulfamoyl]phenyl]acetamide
   Show/Hide
C28H34F3N5O3S
 1
1
IC50 = 0.9 nM
   TI
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CP0513445
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]methanesulfonamide
   Show/Hide
C21H29F3N4O2S
 1
1
IC50 = 0.9 nM
   TI
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CP0533087
3-oxo-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)phenoxy)piperidin-1-yl)ethyl)cyclohexyl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-6-sulfonamide
   Show/Hide
C28H34F3N3O5S
 1
1
IC50 = 1 nM
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CP0667862
cariprazine hydrochloride
   Show/Hide
C21H33Cl3N4O
 1
1
IC50 = 1.6 nM
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CP0428657
N-[4-[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]acetamide
   Show/Hide
C21H30F3N3O
 1
1
IC50 = 1.9 nM
   TI
   LI
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   TS
CP0430627
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]acetamide
   Show/Hide
C22H29F3N4O
 1
1
IC50 = 1.9 nM
   TI
   LI
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   TS
CP0523740
N-[4-[2-[4-(2,5-dichloroanilino)piperidin-1-yl]ethyl]cyclohexyl]-4-fluorobenzenesulfonamide
   Show/Hide
C25H32Cl2FN3O2S
 1
1
IC50 = 2 nM
   TI
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   TS
CP0371879
N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]cyclohexyl]-1-benzothiophene-2-sulfonamide
   Show/Hide
C29H35F3N2O2S2
 1
1
IC50 = 2.6 nM
   TI
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CP0485806
N-[4-[2-[4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl]ethyl]cyclohexyl]pyridine-3-sulfonamide
   Show/Hide
C25H32F3N3O3S
 1
1
IC50 = 2.8 nM
   TI
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CP0505454
4-chloro-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)phenylamino)piperidin-1-yl)ethyl)cyclohexyl)benzenesulfonamide
   Show/Hide
C26H33ClF3N3O2S
 1
1
IC50 = 3 nM
   TI
   LI
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   TS
CP0510648
4-bromo-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)cyclohexyl)benzenesulfonamide
   Show/Hide
C26H30BrF3N4O2S
 1
1
IC50 = 3.3 nM
   TI
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CP0490420
N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]cyclohexyl]acetamide
   Show/Hide
C23H33F3N2O
 1
1
IC50 = 3.3 nM
   TI
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CP0847951
(R)-(-)-2-(4-Hydroxyphenyl)-apomorphine hydrochloride
   Show/Hide
C23H22ClNO3
 2
1
IC50 = 3.7 nM
   TI
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2
Ki = 1.78 nM
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CP0462568
4-chloro-N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]cyclohexyl]benzenesulfonamide
   Show/Hide
C27H34ClF3N2O2S
 1
1
IC50 = 3.8 nM
   TI
   LI
   LO
   TS
CP0525031
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]-6-methylpyridine-3-sulfonamide
   Show/Hide
C26H32F3N5O2S
 1
1
IC50 = 4.2 nM
   TI
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CP0528867
N-[4-[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]methanesulfonamide
   Show/Hide
C20H30F3N3O2S
 1
1
IC50 = 4.8 nM
   TI
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CP0566164
ethyl N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]ethyl]cyclohexyl]carbamate
   Show/Hide
C23H34F3N3O2
 1
1
IC50 = 5.1 nM
   TI
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CP0450523
N-[4-[2-[4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl]ethyl]cyclohexyl]acetamide
   Show/Hide
C22H31F3N2O2
 1
1
IC50 = 5.3 nM
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CP0467831
3-cyano-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)cyclohexyl)benzenesulfonamide
   Show/Hide
C27H30F3N5O2S
 1
1
IC50 = 5.8 nM
   TI
   LI
   LO
   TS
CP0489100
N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]ethyl]cyclohexyl]methanesulfonamide
   Show/Hide
C21H32F3N3O2S
 1
1
IC50 = 11 nM
   TI
   LI
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CP0852096
(R)-(-)-2-Phenyl-apomorphine hydrochloride
   Show/Hide
C23H22ClNO2
 2
1
IC50 = 14.7 nM
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2
Ki = 7.7 nM
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CP0893248
(R)-(-)-2-(4-dibenzo-furanyl)-apomorphine hydrochloride
   Show/Hide
C29H24ClNO3
 2
1
IC50 = 49.4 nM
   TI
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2
Ki = 22.3 nM
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CP0850567
Apomorphine hydrochloride
   Show/Hide
C17H18ClNO2
 2
1
IC50 = 69.5 nM
   TI
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2
Ki = 36.4 nM
   TI
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CP0933722
(R)-(-)-2-Methyl-apomorphine hydrochloride
   Show/Hide
C18H20ClNO2
 2
1
IC50 = 82.6 nM
   TI
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2
Ki = 40.1 nM
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CP0945489
(R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine dihydrochloride
   Show/Hide
C25H28Cl2N2O2
 2
1
IC50 = 178 nM
   TI
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2
Ki = 78.4 nM
   TI
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CP0529799
N-(9-benzyl-9-azabicyclo[3.3.1]nonan-3-yl)-5-iodo-2,3-dimethoxybenzamide
   Show/Hide
C24H29IN2O3
 1
1
Ki = 0.04 nM
   TI
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CP0565856
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (9-benzyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide
   Show/Hide
C27H29BrN2O2
 1
1
Ki = 0.04 nM
   TI
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   TS
CP0403054
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-pyrrolidin-3-yl)-amide
   Show/Hide
C23H29BrN2O2
 1
1
Ki = 0.2 nM
   TI
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   TS
CP0524584
7-Bromo-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C17H18BrN3S
 1
1
Ki = 0.25 nM
   TI
   LI
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   TS
CP0438611
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-3-yl)-amide
   Show/Hide
C26H31BrN2O2
 1
1
Ki = 0.4 nM
   TI
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CP0112004
1-((S)-8-Chloro-10,11-dihydro-dibenzo[b,f]thiepin-10-yl)-4-methyl-piperazine
   Show/Hide
C19H21ClN2S
 1
1
Ki = 0.4 nM
   TI
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CP0497003
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-3-yl)-amide
   Show/Hide
C26H31BrN2O2
 1
1
Ki = 0.4 nM
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CP0389732
CHEMBL2024677
   Show/Hide
C21H32Cl2N4O
 1
1
Ki = 0.44 nM
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CP0043442
Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C23H25Cl2N3OS
 1
1
Ki = 0.5 nM
   TI
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CP0049308
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-4-pyridin-2-ylbenzamide
   Show/Hide
C26H28Cl2N4O
 1
1
Ki = 0.6 nM
   TI
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CP0475720
3-[4-[2-[4-(2,5-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
   Show/Hide
C21H32Cl2N4O
 1
1
Ki = 0.66 nM
   TI
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CP0463525
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclohexyl-pyrrolidin-3-yl)-amide
   Show/Hide
C22H27BrN2O2
 1
1
Ki = 0.8 nM
   TI
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CP0110281
Biphenyl-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C27H29Cl2N3O
 1
1
Ki = 0.9 nM
   TI
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CP0035955
(R,S) 7-[(3-Iodo-allyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalen-2-ol
   Show/Hide
C16H22INO
 1
1
Ki = 0.99 nM
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CP0458768
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide
   Show/Hide
C23H23BrN2O2
 1
1
Ki = 1 nM
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CP0520569
US8802672, 1
   Show/Hide
C19H30Cl2N6O
 1
1
Ki < 1 nM
   TI
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CP0551366
US8802672, 10
   Show/Hide
C20H33Cl2N7O
 1
1
Ki < 1 nM
   TI
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CP0551367
US8802672, 11
   Show/Hide
C20H32Cl2N6O
 1
1
Ki < 1 nM
   TI
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CP0463704
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-benzyl-piperidin-4-yl)-amide
   Show/Hide
C24H25BrN2O2
 1
1
Ki = 1.1 nM
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CP0079495
9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C28H29Cl2N3O
 2
1
Ki = 1.1 nM
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2
Ki = 1.4 nM
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CP0162854
(+/-)-7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-2-ol
   Show/Hide
C16H25NO
 1
1
Ki = 1.18 nM
   TI
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CP0348511
N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]benzamide
   Show/Hide
C21H23Cl2N3O
 1
1
Ki = 1.3 nM
   TI
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CP0466022
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-benzyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C24H25BrN2O2
 1
1
Ki = 1.4 nM
   TI
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CP0302789
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-4-iodobenzamide
   Show/Hide
C21H24Cl2IN3O
 1
1
Ki = 1.4 nM
   TI
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CP0183672
9-Oxo-9H-fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C28H27Cl2N3O2
 2
1
Ki = 1.4 nM
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2
Ki = 1.6 nM
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CP0401591
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid ((R)-1-benzyl-pyrrolidin-3-yl)-amide
   Show/Hide
C23H23BrN2O2
 1
1
Ki = 1.6 nM
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CP0528868
3-[4-[2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
   Show/Hide
C21H33ClN4O
 1
1
Ki = 1.6 nM
   TI
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CP0534389
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclobutyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C21H25BrN2O2
 1
1
Ki = 1.9 nM
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CP0276368
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]quinoxaline-2-carboxamide
   Show/Hide
C23H25Cl2N5O
 1
1
Ki = 1.9 nM
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CP0193103
9-Oxo-9H-fluorene-4-carboxylic acid {5-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-pentyl}-amide
   Show/Hide
C29H29Cl2N3O2
 1
1
Ki = 2 nM
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CP0283831
7-Chloro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C17H18ClN3S
 1
1
Ki = 2 nM
   TI
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CP0520570
US8802672, 6
   Show/Hide
C20H32Cl2N6O
 1
1
Ki = 2 nM
   TI
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CP0539117
US8802672, 7
   Show/Hide
C22H35Cl2N7O2
 1
1
Ki = 2 nM
   TI
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CP0550501
US8802672, 2
   Show/Hide
C18H29Cl2N7O
 1
1
Ki = 2 nM
   TI
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CP0550520
US8802672, 8
   Show/Hide
C20H33Cl2N7O
 1
1
Ki = 2 nM
   TI
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CP0116811
5-Bromo-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-2,3-dimethoxy-benzamide
   Show/Hide
C23H28BrCl2N3O3
 1
1
Ki = 2.1 nM
   TI
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CP0462674
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C24H31BrN2O2
 1
1
Ki = 2.4 nM
   TI
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CP0527508
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-pyrrolidin-3-yl)-amide
   Show/Hide
C21H25BrN2O2
 1
1
Ki = 2.5 nM
   TI
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   TS
CP0457307
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C27H33BrN2O2
 1
1
Ki = 2.6 nM
   TI
   LI
   LO
   TS
CP0109326
5-Fluoro-1H-indole-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C23H25Cl2FN4O
 1
1
Ki = 2.6 nM
   TI
   LI
   LO
   TS
CP0498137
7-Fluoro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C17H18FN3S
 1
1
Ki = 2.7 nM
   TI
   LI
   LO
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CP0403673
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-pyrrolidin-3-yl)-amide
   Show/Hide
C23H29BrN2O2
 1
1
Ki = 2.9 nM
   TI
   LI
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CP0394485
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid ((R)-1-cyclohexyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C23H29BrN2O2
 1
1
Ki = 3.2 nM
   TI
   LI
   LO
   TS
CP0459272
3-[4-[2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
   Show/Hide
C21H32Cl2N4O
 1
1
Ki = 3.3 nM
   TI
   LI
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CP0501155
6-Amino-9H-fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C28H30Cl2N4O
 1
1
Ki = 3.5 nM
   TI
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CP0453332
2-[5-(5-Bromo-2,3-dimethoxy-phenyl)-1H-pyrrol-2-ylmethyl]-1,2,3,4-tetrahydro-isoquinoline
   Show/Hide
C22H23BrN2O2
 1
1
Ki = 3.8 nM
   TI
   LI
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   TS
CP0442046
2-[5-(5-Bromo-2,3-dimethoxy-phenyl)-1H-pyrrol-2-ylmethyl]-6,7-dimethoxy-1,2,3,4-tetrahydro-isoquinoline
   Show/Hide
C24H27BrN2O4
 1
1
Ki = 3.9 nM
   TI
   LI
   LO
   TS
CP0163132
(+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,14-octahydro-1H-benzo[4,5]cyclohepta[de]pyrido[2,1-a]isoquinolin-3-ol
   Show/Hide
C25H31NO
 1
1
Ki = 3.91 nM
   TI
   LI
   LO
   TS
CP0502805
7-Chloro-9-(4-methyl-[1,4]diazepan-1-yl)-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C18H20ClN3S
 1
1
Ki = 4.3 nM
   TI
   LI
   LO
   TS
CP0480711
9H-Fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C28H29Cl2N3O
 1
1
Ki = 4.5 nM
   TI
   LI
   LO
   TS
CP0100862
2-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-isoindole-1,3-dione
   Show/Hide
C22H23Cl2N3O2
 1
1
Ki = 4.8 nM
   TI
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CP0378868
N-[(Z)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]benzamide
   Show/Hide
C21H23Cl2N3O
 1
1
Ki = 4.9 nM
   TI
   LI
   LO
   TS
CP0446956
3-[4-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
   Show/Hide
C21H33ClN4O
 1
1
Ki = 4.95 nM
   TI
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CP0536697
CHEMBL2024525
   Show/Hide
C21H32Cl2N4O
 1
1
Ki = 5.4 nM
   TI
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CP0228520
2-{5-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-pentyl}-isoindole-1,3-dione
   Show/Hide
C23H25Cl2N3O2
 1
1
Ki = 5.6 nM
   TI
   LI
   LO
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CP0006107
CAS_85760-74-3
   Show/Hide
C13H21N3
 1
1
Ki = 5.65 nM
   TI
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CP0520943
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclohexyl-pyrrolidin-3-yl)-amide
   Show/Hide
C22H27BrN2O2
 1
1
Ki = 5.7 nM
   TI
   LI
   LO
   TS
CP0065124
9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
   Show/Hide
C28H27Cl2N3O
 1
1
Ki = 5.9 nM
   TI
   LI
   LO
   TS
CP0430205
9H-Fluorene-2-carboxylic acid {(Z)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
   Show/Hide
C28H27Cl2N3O
 1
1
Ki = 6 nM
   TI
   LI
   LO
   TS
CP0378073
9H-Fluorene-4-carboxylic acid {(Z)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
   Show/Hide
C28H27Cl2N3O
 1
1
Ki = 6.5 nM
   TI
   LI
   LO
   TS
CP0470402
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-bicyclo[3.3.1]non-9-yl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C26H33BrN2O2
 1
1
Ki = 7.5 nM
   TI
   LI
   LO
   TS
CP0052483
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-ethyl}-amide
   Show/Hide
C24H24BrCl2N3O2
 1
1
Ki = 8 nM
   TI
   LI
   LO
   TS
CP0077352
9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C17H19N3S
 1
1
Ki = 8.3 nM
   TI
   LI
   LO
   TS
CP0036333
(S)-3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-6-methoxy-benzamide
   Show/Hide
C15H20Cl2N2O3
 1
1
Ki = 9.25 nM
   TI
   LI
   LO
   TS
CP0048757
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C26H28BrCl2N3O2
 1
1
Ki = 10.2 nM
   TI
   LI
   LO
   TS
CP0048138
9H-Fluorene-9-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
   Show/Hide
C28H29Cl2N3O
 1
1
Ki = 11.1 nM
   TI
   LI
   LO
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CP0532372
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-bicyclo[3.3.1]non-9-yl-pyrrolidin-3-yl)-amide
   Show/Hide
C25H31BrN2O2
 1
1
Ki = 12 nM
   TI
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CP0374354
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-3-yl)-amide
   Show/Hide
C26H31BrN2O2
 1
1
Ki = 13 nM
   TI
   LI
   LO
   TS
CP0039958
(risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
   Show/Hide
C23H27FN4O2
 1
1
Ki = 13 nM
   TI
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   LO
   TS
CP0490421
3-[4-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
   Show/Hide
C21H33ClN4O
 1
1
Ki = 13.1 nM
   TI
   LI
   LO
   TS
CP0377962
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-bicyclo[3.3.1]non-9-yl-pyrrolidin-3-yl)-amide
   Show/Hide
C25H31BrN2O2
 1
1
Ki = 13.2 nM
   TI
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   TS
CP0008601
4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl)
   Show/Hide
C21H23ClFNO2
 3
1
Ki = 14.3 nM
   TI
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2
Ki = 18 nM
   TI
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3
Ki = 47 nM
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CP0406478
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-benzyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C24H25BrN2O2
 1
1
Ki = 14.6 nM
   TI
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CP0536696
1,1-dimethyl-3-[4-[2-(4-phenylpiperazin-1-yl)ethyl]cyclohexyl]urea
   Show/Hide
C21H34N4O
 1
1
Ki = 15.9 nM
   TI
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   TS
CP0432443
5-Bromo-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-2,3-dimethoxy-benzamide
   Show/Hide
C20H23BrN2O3
 1
1
Ki = 17.8 nM
   TI
   LI
   LO
   TS
CP0510381
1-Methyl-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C18H21N3S
 1
1
Ki = 18 nM
   TI
   LI
   LO
   TS
CP0372639
9H-Fluorene-4-carboxylic acid {(E)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
   Show/Hide
C28H27Cl2N3O
 1
1
Ki = 19 nM
   TI
   LI
   LO
   TS
CP0147752
1-(8-Chloro-10,11-dihydro-dibenzo[b,f]thiepin-10-yl)-4-methyl-piperazine
   Show/Hide
C19H21ClN2S
 1
1
Ki = 21 nM
   TI
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   LO
   TS
CP0048789
5-Bromo-N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-2,3-dimethoxy-benzamide
   Show/Hide
C22H27BrN2O5
 1
1
Ki = 21.4 nM
   TI
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   TS
CP0439629
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C22H27BrN2O2
 1
1
Ki = 30 nM
   TI
   LI
   LO
   TS
CP0189754
9H-Fluorene-9-carboxylic acid {3-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-propyl}-amide
   Show/Hide
C27H27Cl2N3O
 1
1
Ki = 34 nM
   TI
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   TS
CP0045063
2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3-b][1,5]benzodiazepine
   Show/Hide
C17H20N4S
 2
1
Ki = 39 nM
   TI
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2
Ki = 76 nM
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CP0438546
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (9-cycloheptyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide
   Show/Hide
C27H35BrN2O2
 1
1
Ki = 41 nM
   TI
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   LO
   TS
CP0185638
9-Oxo-9H-fluorene-4-carboxylic acid {3-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-propyl}-amide
   Show/Hide
C27H25Cl2N3O2
 1
1
Ki = 43 nM
   TI
   LI
   LO
   TS
CP0470382
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (9-cyclohexyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide
   Show/Hide
C26H33BrN2O2
 1
1
Ki = 48 nM
   TI
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   TS
CP0036921
3-HYDROXYTYRAMINE HYDROCHLORIDE
   Show/Hide
C8H11NO2
 1
1
Ki = 49.3 nM
   TI
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CP0461448
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C24H31BrN2O2
 1
1
Ki = 50 nM
   TI
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CP0466517
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C22H27BrN2O2
 1
1
Ki = 52 nM
   TI
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CP0438418
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-piperidin-4-yl)-amide
   Show/Hide
C24H31BrN2O2
 1
1
Ki = 58 nM
   TI
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   TS
CP0509389
1-{2-[4-(7-Chloro-9,10-dihydro-4-thia-10a-aza-benzo[f]azulen-9-yl)-piperazin-1-yl]-ethyl}-imidazolidin-2-one
   Show/Hide
C21H26ClN5OS
 1
1
Ki = 66 nM
   TI
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CP0438551
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C27H33BrN2O2
 1
1
Ki = 68 nM
   TI
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CP0463646
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-pyrrolidin-3-yl)-amide
   Show/Hide
C21H25BrN2O2
 1
1
Ki = 75 nM
   TI
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   TS
CP0442085
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2-(3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-amide
   Show/Hide
C23H23BrN2O2
 1
1
Ki = 81.6 nM
   TI
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CP0208243
9H-Fluorene-9-carboxylic acid [3-(4-phenyl-piperazin-1-yl)-propyl]-amide
   Show/Hide
C27H29N3O
 1
1
Ki = 84.5 nM
   TI
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CP0538897
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclobutyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C21H25BrN2O2
 1
1
Ki = 90 nM
   TI
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   TS
CP0460690
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-piperidin-4-yl)-amide
   Show/Hide
C27H33BrN2O2
 1
1
Ki = 92 nM
   TI
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CP0484590
9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene-1-carbaldehyde
   Show/Hide
C18H19N3OS
 1
1
Ki = 102 nM
   TI
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   LO
   TS
CP0394255
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl]-amide
   Show/Hide
C27H31BrN2O4
 1
1
Ki = 106.5 nM
   TI
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CP0082953
2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dimethoxyphenoxy)ethyl]amine;hydrochloride
   Show/Hide
C19H23NO5
 1
1
Ki = 107 nM
   TI
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CP0522332
(S)-7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C17H20ClN3S
 1
1
Ki = 110 nM
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CP0509454
[6-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepin-3-yl]methanol
   Show/Hide
C18H21N3OS
 1
1
Ki = 113 nM
   TI
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CP0456817
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-amide
   Show/Hide
C25H27BrN2O4
 1
1
Ki = 126.5 nM
   TI
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   TS
CP0431518
9H-Fluorene-4-carboxylic acid {3-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-propyl}-amide
   Show/Hide
C27H27Cl2N3O
 1
1
Ki = 139 nM
   TI
   LI
   LO
   TS
CP0241553
9H-Fluorene-2-carboxylic acid {3-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-propyl}-amide
   Show/Hide
C27H27Cl2N3O
 1
1
Ki = 199 nM
   TI
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   TS
CP0383914
9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-ynyl}-amide
   Show/Hide
C28H25Cl2N3O
 1
1
Ki = 214 nM
   TI
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   TS
CP0037227
7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-ol
   Show/Hide
C16H25NO
 1
1
Ki = 248 nM
   TI
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CP0535727
1-Isopropoxymethyl-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C21H27N3OS
 1
1
Ki = 278 nM
   TI
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   TS
CP0339117
5-Bromo-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-2-methoxy-benzamide
   Show/Hide
C19H21BrN2O2
 1
1
Ki = 310.7 nM
   TI
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CP0178464
N-[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]-2-methoxy-5-methylbenzamide
   Show/Hide
C24H32N2O4
 1
1
Ki = 313 nM
   TI
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CP0529519
7-Chloro-1-methoxymethyl-9-(4-methyl-piperazin-1-yl)-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene
   Show/Hide
C19H24ClN3OS
 1
1
Ki = 316 nM
   TI
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CP0025667
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
   Show/Hide
C18H19ClN4
 1
1
Ki = 319 nM
   TI
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CP0463526
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclohexyl-pyrrolidin-2-ylmethyl)-amide
   Show/Hide
C23H29BrN2O2
 1
1
Ki = 334 nM
   TI
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   TS
CP0382018
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-ynyl]benzamide
   Show/Hide
C21H21Cl2N3O
 1
1
Ki = 394 nM
   TI
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   TS
CP0465990
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclohexyl-piperidin-4-yl)-amide
   Show/Hide
C23H29BrN2O2
 1
1
Ki = 430 nM
   TI
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   TS
CP0080663
5-Bromo-N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-2-methoxy-benzamide
   Show/Hide
C21H25BrN2O4
 1
1
Ki = 488 nM
   TI
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CP0116813
5-Bromo-N-[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl]-2,3-dimethoxy-benzamide
   Show/Hide
C24H31BrN2O5
 1
1
Ki = 627 nM
   TI
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   TS
CP0046341
8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ol(SCH 23390)
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C17H18ClNO
 1
1
Ki = 768 nM
   TI
   LI
   LO
   TS
CP0465347
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-piperidin-4-yl)-amide
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C22H27BrN2O2
 1
1
Ki = 899 nM
   TI
   LI
   LO
   TS
CP0463091
9H-Fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-ynyl}-amide
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C28H25Cl2N3O
 1
1
Ki = 1080 nM
   TI
   LI
   LO
   TS
CP0538820
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-bicyclo[3.3.1]non-9-yl-piperidin-4-yl)-amide
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C26H33BrN2O2
 1
1
Ki = 1431 nM
   TI
   LI
   LO
   TS
CP0026495
CHEBI:51137
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C18H20N2
 1
1
Ki = 1524 nM
   TI
   LI
   LO
   TS
CP0001238
14C-5-hydroxy tryptamine creatinine disulfate
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C10H12N2O
 1
1
Ki = 2338 nM
   TI
   LI
   LO
   TS
CP0069692
(+)-yohimbine
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C21H26N2O3
 1
1
Ki = 2430 nM
   TI
   LI
   LO
   TS
CP0055980
N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-2-methoxy-5-methylbenzamide
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C22H28N2O4
 1
1
Ki = 3760 nM
   TI
   LI
   LO
   TS
CP0875029
9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene-1-carbaldehyde oxime
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C18H20N4OS
 1
1
Ki = 4255 nM
   TI
   LI
   LO
   TS
CP0038839
(4R,4aS,7aR,12bS)-3-allyl-4a,9-dihydroxy-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-7-one;hydrochloride
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C19H21NO4
 1
1
Ki > 20000 nM
   TI
   LI
   LO
   TS
CP0507024
9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene-1,10-dicarbaldehyde
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C19H19N3O2S
 1
1
Ki > 1000 nM
   TI
   LI
   LO
   TS
CP0041613
Anapriline
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C16H21NO2
 1
1
Ki > 5000 nM
   TI
   LI
   LO
   TS