Compound ID |
Compound Name |
Compound Formula |
CP0523741
|
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]pyridine-3-sulfonamide
Show/Hide
|
C23H30Cl2N4O2S
|
1
|
1 |
IC50 = 0.2 nM
|
|
|
CP0459270
|
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]propanamide
Show/Hide
|
C21H31Cl2N3O
|
1
|
1 |
IC50 = 0.26 nM
|
|
|
CP0450524
|
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]acetamide
Show/Hide
|
C20H29Cl2N3O
|
1
|
1 |
IC50 = 0.29 nM
|
|
|
CP0467830
|
N-[4-[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]pyridine-3-sulfonamide
Show/Hide
|
C24H31F3N4O2S
|
1
|
1 |
IC50 = 0.3 nM
|
|
|
CP0459271
|
[4-[2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]urea
Show/Hide
|
C19H28Cl2N4O
|
1
|
1 |
IC50 = 0.32 nM
|
|
|
CP0432559
|
1-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-3-ethylurea
Show/Hide
|
C21H32Cl2N4O
|
1
|
1 |
IC50 = 0.34 nM
|
|
|
CP0464137
|
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]pyridine-3-sulfonamide
Show/Hide
|
C25H30F3N5O2S
|
1
|
1 |
IC50 = 0.4 nM
|
|
|
CP0432558
|
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-2,2,2-trifluoroacetamide
Show/Hide
|
C20H26Cl2F3N3O
|
1
|
1 |
IC50 = 0.41 nM
|
|
|
CP0459269
|
N-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]methanesulfonamide
Show/Hide
|
C19H29Cl2N3O2S
|
1
|
1 |
IC50 = 0.48 nM
|
|
|
CP0523742
|
4-pyrazol-1-yl-N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]cyclohexyl]benzenesulfonamide
Show/Hide
|
C30H37F3N4O2S
|
1
|
1 |
IC50 = 0.5 nM
|
|
|
CP0533088
|
N-[4-[2-[4-(4-bromo-2-methoxyphenyl)piperazin-1-yl]ethyl]cyclohexyl]-4-methoxybenzenesulfonamide
Show/Hide
|
C26H36BrN3O4S
|
1
|
1 |
IC50 = 0.5 nM
|
|
|
CP0432560
|
3-[4-[2-[4-(2,3-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-diethylurea
Show/Hide
|
C23H36Cl2N4O
|
1
|
1 |
IC50 = 0.62 nM
|
|
|
CP0501623
|
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]-2-oxo-3,4-dihydro-1H-quinoline-6-sulfonamide
Show/Hide
|
C29H34F3N5O3S
|
1
|
1 |
IC50 = 0.7 nM
|
|
|
CP0505453
|
N-[4-[2-[4-(3-cyanophenyl)piperazin-1-yl]ethyl]cyclohexyl]-3,4-dimethoxybenzenesulfonamide
Show/Hide
|
C27H36N4O4S
|
1
|
1 |
IC50 = 0.7 nM
|
|
|
CP0371880
|
N-[4-[[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]sulfamoyl]phenyl]acetamide
Show/Hide
|
C28H34F3N5O3S
|
1
|
1 |
IC50 = 0.9 nM
|
|
|
CP0513445
|
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]methanesulfonamide
Show/Hide
|
C21H29F3N4O2S
|
1
|
1 |
IC50 = 0.9 nM
|
|
|
CP0533087
|
3-oxo-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)phenoxy)piperidin-1-yl)ethyl)cyclohexyl)-3,4-dihydro-2H-benzo[b][1,4]oxazine-6-sulfonamide
Show/Hide
|
C28H34F3N3O5S
|
1
|
1 |
IC50 = 1 nM
|
|
|
CP0667862
|
cariprazine hydrochloride
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|
C21H33Cl3N4O
|
1
|
1 |
IC50 = 1.6 nM
|
|
|
CP0428657
|
N-[4-[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]acetamide
Show/Hide
|
C21H30F3N3O
|
1
|
1 |
IC50 = 1.9 nM
|
|
|
CP0430627
|
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]acetamide
Show/Hide
|
C22H29F3N4O
|
1
|
1 |
IC50 = 1.9 nM
|
|
|
CP0523740
|
N-[4-[2-[4-(2,5-dichloroanilino)piperidin-1-yl]ethyl]cyclohexyl]-4-fluorobenzenesulfonamide
Show/Hide
|
C25H32Cl2FN3O2S
|
1
|
1 |
IC50 = 2 nM
|
|
|
CP0371879
|
N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]cyclohexyl]-1-benzothiophene-2-sulfonamide
Show/Hide
|
C29H35F3N2O2S2
|
1
|
1 |
IC50 = 2.6 nM
|
|
|
CP0485806
|
N-[4-[2-[4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl]ethyl]cyclohexyl]pyridine-3-sulfonamide
Show/Hide
|
C25H32F3N3O3S
|
1
|
1 |
IC50 = 2.8 nM
|
|
|
CP0505454
|
4-chloro-N-((1r,4r)-4-(2-(4-(3-(trifluoromethyl)phenylamino)piperidin-1-yl)ethyl)cyclohexyl)benzenesulfonamide
Show/Hide
|
C26H33ClF3N3O2S
|
1
|
1 |
IC50 = 3 nM
|
|
|
CP0510648
|
4-bromo-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)cyclohexyl)benzenesulfonamide
Show/Hide
|
C26H30BrF3N4O2S
|
1
|
1 |
IC50 = 3.3 nM
|
|
|
CP0490420
|
N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]cyclohexyl]acetamide
Show/Hide
|
C23H33F3N2O
|
1
|
1 |
IC50 = 3.3 nM
|
|
|
CP0847951
|
(R)-(-)-2-(4-Hydroxyphenyl)-apomorphine hydrochloride
Show/Hide
|
C23H22ClNO3
|
2
|
1 |
IC50 = 3.7 nM
|
|
|
2 |
Ki = 1.78 nM
|
|
|
CP0462568
|
4-chloro-N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperidin-1-yl]ethyl]cyclohexyl]benzenesulfonamide
Show/Hide
|
C27H34ClF3N2O2S
|
1
|
1 |
IC50 = 3.8 nM
|
|
|
CP0525031
|
N-[4-[2-[4-[3-cyano-5-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]-6-methylpyridine-3-sulfonamide
Show/Hide
|
C26H32F3N5O2S
|
1
|
1 |
IC50 = 4.2 nM
|
|
|
CP0528867
|
N-[4-[2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethyl]cyclohexyl]methanesulfonamide
Show/Hide
|
C20H30F3N3O2S
|
1
|
1 |
IC50 = 4.8 nM
|
|
|
CP0566164
|
ethyl N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]ethyl]cyclohexyl]carbamate
Show/Hide
|
C23H34F3N3O2
|
1
|
1 |
IC50 = 5.1 nM
|
|
|
CP0450523
|
N-[4-[2-[4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl]ethyl]cyclohexyl]acetamide
Show/Hide
|
C22H31F3N2O2
|
1
|
1 |
IC50 = 5.3 nM
|
|
|
CP0467831
|
3-cyano-N-((1r,4r)-4-(2-(4-(3-cyano-5-(trifluoromethyl)phenyl)piperazin-1-yl)ethyl)cyclohexyl)benzenesulfonamide
Show/Hide
|
C27H30F3N5O2S
|
1
|
1 |
IC50 = 5.8 nM
|
|
|
CP0489100
|
N-[4-[2-[4-[[3-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]ethyl]cyclohexyl]methanesulfonamide
Show/Hide
|
C21H32F3N3O2S
|
1
|
1 |
IC50 = 11 nM
|
|
|
CP0852096
|
(R)-(-)-2-Phenyl-apomorphine hydrochloride
Show/Hide
|
C23H22ClNO2
|
2
|
1 |
IC50 = 14.7 nM
|
|
|
2 |
Ki = 7.7 nM
|
|
|
CP0893248
|
(R)-(-)-2-(4-dibenzo-furanyl)-apomorphine hydrochloride
Show/Hide
|
C29H24ClNO3
|
2
|
1 |
IC50 = 49.4 nM
|
|
|
2 |
Ki = 22.3 nM
|
|
|
CP0850567
|
Apomorphine hydrochloride
Show/Hide
|
C17H18ClNO2
|
2
|
1 |
IC50 = 69.5 nM
|
|
|
2 |
Ki = 36.4 nM
|
|
|
CP0933722
|
(R)-(-)-2-Methyl-apomorphine hydrochloride
Show/Hide
|
C18H20ClNO2
|
2
|
1 |
IC50 = 82.6 nM
|
|
|
2 |
Ki = 40.1 nM
|
|
|
CP0945489
|
(R)-(-)-2-(4-N,N-Dimethylaminophenyl)-apomorphine dihydrochloride
Show/Hide
|
C25H28Cl2N2O2
|
2
|
1 |
IC50 = 178 nM
|
|
|
2 |
Ki = 78.4 nM
|
|
|
CP0529799
|
N-(9-benzyl-9-azabicyclo[3.3.1]nonan-3-yl)-5-iodo-2,3-dimethoxybenzamide
Show/Hide
|
C24H29IN2O3
|
1
|
1 |
Ki = 0.04 nM
|
|
|
CP0565856
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (9-benzyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide
Show/Hide
|
C27H29BrN2O2
|
1
|
1 |
Ki = 0.04 nM
|
|
|
CP0403054
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-pyrrolidin-3-yl)-amide
Show/Hide
|
C23H29BrN2O2
|
1
|
1 |
Ki = 0.2 nM
|
|
|
CP0524584
|
7-Bromo-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C17H18BrN3S
|
1
|
1 |
Ki = 0.25 nM
|
|
|
CP0438611
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-3-yl)-amide
Show/Hide
|
C26H31BrN2O2
|
1
|
1 |
Ki = 0.4 nM
|
|
|
CP0112004
|
1-((S)-8-Chloro-10,11-dihydro-dibenzo[b,f]thiepin-10-yl)-4-methyl-piperazine
Show/Hide
|
C19H21ClN2S
|
1
|
1 |
Ki = 0.4 nM
|
|
|
CP0497003
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-3-yl)-amide
Show/Hide
|
C26H31BrN2O2
|
1
|
1 |
Ki = 0.4 nM
|
|
|
CP0389732
|
CHEMBL2024677
Show/Hide
|
C21H32Cl2N4O
|
1
|
1 |
Ki = 0.44 nM
|
|
|
CP0043442
|
Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C23H25Cl2N3OS
|
1
|
1 |
Ki = 0.5 nM
|
|
|
CP0049308
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-4-pyridin-2-ylbenzamide
Show/Hide
|
C26H28Cl2N4O
|
1
|
1 |
Ki = 0.6 nM
|
|
|
CP0475720
|
3-[4-[2-[4-(2,5-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
Show/Hide
|
C21H32Cl2N4O
|
1
|
1 |
Ki = 0.66 nM
|
|
|
CP0463525
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclohexyl-pyrrolidin-3-yl)-amide
Show/Hide
|
C22H27BrN2O2
|
1
|
1 |
Ki = 0.8 nM
|
|
|
CP0110281
|
Biphenyl-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C27H29Cl2N3O
|
1
|
1 |
Ki = 0.9 nM
|
|
|
CP0035955
|
(R,S) 7-[(3-Iodo-allyl)-propyl-amino]-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C16H22INO
|
1
|
1 |
Ki = 0.99 nM
|
|
|
CP0458768
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-benzyl-pyrrolidin-3-yl)-amide
Show/Hide
|
C23H23BrN2O2
|
1
|
1 |
Ki = 1 nM
|
|
|
CP0520569
|
US8802672, 1
Show/Hide
|
C19H30Cl2N6O
|
1
|
1 |
Ki < 1 nM
|
|
|
CP0551366
|
US8802672, 10
Show/Hide
|
C20H33Cl2N7O
|
1
|
1 |
Ki < 1 nM
|
|
|
CP0551367
|
US8802672, 11
Show/Hide
|
C20H32Cl2N6O
|
1
|
1 |
Ki < 1 nM
|
|
|
CP0463704
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-benzyl-piperidin-4-yl)-amide
Show/Hide
|
C24H25BrN2O2
|
1
|
1 |
Ki = 1.1 nM
|
|
|
CP0079495
|
9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C28H29Cl2N3O
|
2
|
1 |
Ki = 1.1 nM
|
|
|
2 |
Ki = 1.4 nM
|
|
|
CP0162854
|
(+/-)-7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-2-ol
Show/Hide
|
C16H25NO
|
1
|
1 |
Ki = 1.18 nM
|
|
|
CP0348511
|
N-[(E)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]benzamide
Show/Hide
|
C21H23Cl2N3O
|
1
|
1 |
Ki = 1.3 nM
|
|
|
CP0466022
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-benzyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C24H25BrN2O2
|
1
|
1 |
Ki = 1.4 nM
|
|
|
CP0302789
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]-4-iodobenzamide
Show/Hide
|
C21H24Cl2IN3O
|
1
|
1 |
Ki = 1.4 nM
|
|
|
CP0183672
|
9-Oxo-9H-fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C28H27Cl2N3O2
|
2
|
1 |
Ki = 1.4 nM
|
|
|
2 |
Ki = 1.6 nM
|
|
|
CP0401591
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid ((R)-1-benzyl-pyrrolidin-3-yl)-amide
Show/Hide
|
C23H23BrN2O2
|
1
|
1 |
Ki = 1.6 nM
|
|
|
CP0528868
|
3-[4-[2-[4-(2-chlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
Show/Hide
|
C21H33ClN4O
|
1
|
1 |
Ki = 1.6 nM
|
|
|
CP0534389
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclobutyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C21H25BrN2O2
|
1
|
1 |
Ki = 1.9 nM
|
|
|
CP0276368
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butyl]quinoxaline-2-carboxamide
Show/Hide
|
C23H25Cl2N5O
|
1
|
1 |
Ki = 1.9 nM
|
|
|
CP0193103
|
9-Oxo-9H-fluorene-4-carboxylic acid {5-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-pentyl}-amide
Show/Hide
|
C29H29Cl2N3O2
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0283831
|
7-Chloro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C17H18ClN3S
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0520570
|
US8802672, 6
Show/Hide
|
C20H32Cl2N6O
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0539117
|
US8802672, 7
Show/Hide
|
C22H35Cl2N7O2
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0550501
|
US8802672, 2
Show/Hide
|
C18H29Cl2N7O
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0550520
|
US8802672, 8
Show/Hide
|
C20H33Cl2N7O
|
1
|
1 |
Ki = 2 nM
|
|
|
CP0116811
|
5-Bromo-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-2,3-dimethoxy-benzamide
Show/Hide
|
C23H28BrCl2N3O3
|
1
|
1 |
Ki = 2.1 nM
|
|
|
CP0462674
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C24H31BrN2O2
|
1
|
1 |
Ki = 2.4 nM
|
|
|
CP0527508
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-pyrrolidin-3-yl)-amide
Show/Hide
|
C21H25BrN2O2
|
1
|
1 |
Ki = 2.5 nM
|
|
|
CP0457307
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C27H33BrN2O2
|
1
|
1 |
Ki = 2.6 nM
|
|
|
CP0109326
|
5-Fluoro-1H-indole-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C23H25Cl2FN4O
|
1
|
1 |
Ki = 2.6 nM
|
|
|
CP0498137
|
7-Fluoro-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C17H18FN3S
|
1
|
1 |
Ki = 2.7 nM
|
|
|
CP0403673
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-pyrrolidin-3-yl)-amide
Show/Hide
|
C23H29BrN2O2
|
1
|
1 |
Ki = 2.9 nM
|
|
|
CP0394485
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid ((R)-1-cyclohexyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C23H29BrN2O2
|
1
|
1 |
Ki = 3.2 nM
|
|
|
CP0459272
|
3-[4-[2-[4-(3,4-dichlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
Show/Hide
|
C21H32Cl2N4O
|
1
|
1 |
Ki = 3.3 nM
|
|
|
CP0501155
|
6-Amino-9H-fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C28H30Cl2N4O
|
1
|
1 |
Ki = 3.5 nM
|
|
|
CP0453332
|
2-[5-(5-Bromo-2,3-dimethoxy-phenyl)-1H-pyrrol-2-ylmethyl]-1,2,3,4-tetrahydro-isoquinoline
Show/Hide
|
C22H23BrN2O2
|
1
|
1 |
Ki = 3.8 nM
|
|
|
CP0442046
|
2-[5-(5-Bromo-2,3-dimethoxy-phenyl)-1H-pyrrol-2-ylmethyl]-6,7-dimethoxy-1,2,3,4-tetrahydro-isoquinoline
Show/Hide
|
C24H27BrN2O4
|
1
|
1 |
Ki = 3.9 nM
|
|
|
CP0163132
|
(+)-3-(tert-butyl)-(3S,4aS,13bS)-2,3,4,4a,8,9,13b,14-octahydro-1H-benzo[4,5]cyclohepta[de]pyrido[2,1-a]isoquinolin-3-ol
Show/Hide
|
C25H31NO
|
1
|
1 |
Ki = 3.91 nM
|
|
|
CP0502805
|
7-Chloro-9-(4-methyl-[1,4]diazepan-1-yl)-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C18H20ClN3S
|
1
|
1 |
Ki = 4.3 nM
|
|
|
CP0480711
|
9H-Fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C28H29Cl2N3O
|
1
|
1 |
Ki = 4.5 nM
|
|
|
CP0100862
|
2-{4-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-butyl}-isoindole-1,3-dione
Show/Hide
|
C22H23Cl2N3O2
|
1
|
1 |
Ki = 4.8 nM
|
|
|
CP0378868
|
N-[(Z)-4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-enyl]benzamide
Show/Hide
|
C21H23Cl2N3O
|
1
|
1 |
Ki = 4.9 nM
|
|
|
CP0446956
|
3-[4-[2-[4-(3-chlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
Show/Hide
|
C21H33ClN4O
|
1
|
1 |
Ki = 4.95 nM
|
|
|
CP0536697
|
CHEMBL2024525
Show/Hide
|
C21H32Cl2N4O
|
1
|
1 |
Ki = 5.4 nM
|
|
|
CP0228520
|
2-{5-[4-(2,3-Dichloro-phenyl)-piperazin-1-yl]-pentyl}-isoindole-1,3-dione
Show/Hide
|
C23H25Cl2N3O2
|
1
|
1 |
Ki = 5.6 nM
|
|
|
CP0006107
|
CAS_85760-74-3
Show/Hide
|
C13H21N3
|
1
|
1 |
Ki = 5.65 nM
|
|
|
CP0520943
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclohexyl-pyrrolidin-3-yl)-amide
Show/Hide
|
C22H27BrN2O2
|
1
|
1 |
Ki = 5.7 nM
|
|
|
CP0065124
|
9H-Fluorene-2-carboxylic acid {(E)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
Show/Hide
|
C28H27Cl2N3O
|
1
|
1 |
Ki = 5.9 nM
|
|
|
CP0430205
|
9H-Fluorene-2-carboxylic acid {(Z)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
Show/Hide
|
C28H27Cl2N3O
|
1
|
1 |
Ki = 6 nM
|
|
|
CP0378073
|
9H-Fluorene-4-carboxylic acid {(Z)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
Show/Hide
|
C28H27Cl2N3O
|
1
|
1 |
Ki = 6.5 nM
|
|
|
CP0470402
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-bicyclo[3.3.1]non-9-yl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C26H33BrN2O2
|
1
|
1 |
Ki = 7.5 nM
|
|
|
CP0052483
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {2-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-ethyl}-amide
Show/Hide
|
C24H24BrCl2N3O2
|
1
|
1 |
Ki = 8 nM
|
|
|
CP0077352
|
9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C17H19N3S
|
1
|
1 |
Ki = 8.3 nM
|
|
|
CP0036333
|
(S)-3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)-2-hydroxy-6-methoxy-benzamide
Show/Hide
|
C15H20Cl2N2O3
|
1
|
1 |
Ki = 9.25 nM
|
|
|
CP0048757
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C26H28BrCl2N3O2
|
1
|
1 |
Ki = 10.2 nM
|
|
|
CP0048138
|
9H-Fluorene-9-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-butyl}-amide
Show/Hide
|
C28H29Cl2N3O
|
1
|
1 |
Ki = 11.1 nM
|
|
|
CP0532372
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-bicyclo[3.3.1]non-9-yl-pyrrolidin-3-yl)-amide
Show/Hide
|
C25H31BrN2O2
|
1
|
1 |
Ki = 12 nM
|
|
|
CP0374354
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-3-yl)-amide
Show/Hide
|
C26H31BrN2O2
|
1
|
1 |
Ki = 13 nM
|
|
|
CP0039958
|
(risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
Show/Hide
|
C23H27FN4O2
|
1
|
1 |
Ki = 13 nM
|
|
|
CP0490421
|
3-[4-[2-[4-(4-chlorophenyl)piperazin-1-yl]ethyl]cyclohexyl]-1,1-dimethylurea
Show/Hide
|
C21H33ClN4O
|
1
|
1 |
Ki = 13.1 nM
|
|
|
CP0377962
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-bicyclo[3.3.1]non-9-yl-pyrrolidin-3-yl)-amide
Show/Hide
|
C25H31BrN2O2
|
1
|
1 |
Ki = 13.2 nM
|
|
|
CP0008601
|
4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl)
Show/Hide
|
C21H23ClFNO2
|
3
|
1 |
Ki = 14.3 nM
|
|
|
2 |
Ki = 18 nM
|
|
|
3 |
Ki = 47 nM
|
|
|
CP0406478
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-benzyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C24H25BrN2O2
|
1
|
1 |
Ki = 14.6 nM
|
|
|
CP0536696
|
1,1-dimethyl-3-[4-[2-(4-phenylpiperazin-1-yl)ethyl]cyclohexyl]urea
Show/Hide
|
C21H34N4O
|
1
|
1 |
Ki = 15.9 nM
|
|
|
CP0432443
|
5-Bromo-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-2,3-dimethoxy-benzamide
Show/Hide
|
C20H23BrN2O3
|
1
|
1 |
Ki = 17.8 nM
|
|
|
CP0510381
|
1-Methyl-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C18H21N3S
|
1
|
1 |
Ki = 18 nM
|
|
|
CP0372639
|
9H-Fluorene-4-carboxylic acid {(E)-4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-enyl}-amide
Show/Hide
|
C28H27Cl2N3O
|
1
|
1 |
Ki = 19 nM
|
|
|
CP0147752
|
1-(8-Chloro-10,11-dihydro-dibenzo[b,f]thiepin-10-yl)-4-methyl-piperazine
Show/Hide
|
C19H21ClN2S
|
1
|
1 |
Ki = 21 nM
|
|
|
CP0048789
|
5-Bromo-N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-2,3-dimethoxy-benzamide
Show/Hide
|
C22H27BrN2O5
|
1
|
1 |
Ki = 21.4 nM
|
|
|
CP0439629
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C22H27BrN2O2
|
1
|
1 |
Ki = 30 nM
|
|
|
CP0189754
|
9H-Fluorene-9-carboxylic acid {3-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-propyl}-amide
Show/Hide
|
C27H27Cl2N3O
|
1
|
1 |
Ki = 34 nM
|
|
|
CP0045063
|
2-methyl-4-(4-methylpiperazin-1-yl)-10H-thieno[2,3-b][1,5]benzodiazepine
Show/Hide
|
C17H20N4S
|
2
|
1 |
Ki = 39 nM
|
|
|
2 |
Ki = 76 nM
|
|
|
CP0438546
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (9-cycloheptyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide
Show/Hide
|
C27H35BrN2O2
|
1
|
1 |
Ki = 41 nM
|
|
|
CP0185638
|
9-Oxo-9H-fluorene-4-carboxylic acid {3-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-propyl}-amide
Show/Hide
|
C27H25Cl2N3O2
|
1
|
1 |
Ki = 43 nM
|
|
|
CP0470382
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (9-cyclohexyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide
Show/Hide
|
C26H33BrN2O2
|
1
|
1 |
Ki = 48 nM
|
|
|
CP0036921
|
3-HYDROXYTYRAMINE HYDROCHLORIDE
Show/Hide
|
C8H11NO2
|
1
|
1 |
Ki = 49.3 nM
|
|
|
CP0461448
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C24H31BrN2O2
|
1
|
1 |
Ki = 50 nM
|
|
|
CP0466517
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C22H27BrN2O2
|
1
|
1 |
Ki = 52 nM
|
|
|
CP0438418
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cycloheptyl-piperidin-4-yl)-amide
Show/Hide
|
C24H31BrN2O2
|
1
|
1 |
Ki = 58 nM
|
|
|
CP0509389
|
1-{2-[4-(7-Chloro-9,10-dihydro-4-thia-10a-aza-benzo[f]azulen-9-yl)-piperazin-1-yl]-ethyl}-imidazolidin-2-one
Show/Hide
|
C21H26ClN5OS
|
1
|
1 |
Ki = 66 nM
|
|
|
CP0438551
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C27H33BrN2O2
|
1
|
1 |
Ki = 68 nM
|
|
|
CP0463646
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-pyrrolidin-3-yl)-amide
Show/Hide
|
C21H25BrN2O2
|
1
|
1 |
Ki = 75 nM
|
|
|
CP0442085
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2-(3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-amide
Show/Hide
|
C23H23BrN2O2
|
1
|
1 |
Ki = 81.6 nM
|
|
|
CP0208243
|
9H-Fluorene-9-carboxylic acid [3-(4-phenyl-piperazin-1-yl)-propyl]-amide
Show/Hide
|
C27H29N3O
|
1
|
1 |
Ki = 84.5 nM
|
|
|
CP0538897
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclobutyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C21H25BrN2O2
|
1
|
1 |
Ki = 90 nM
|
|
|
CP0460690
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-adamantan-2-yl-piperidin-4-yl)-amide
Show/Hide
|
C27H33BrN2O2
|
1
|
1 |
Ki = 92 nM
|
|
|
CP0484590
|
9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene-1-carbaldehyde
Show/Hide
|
C18H19N3OS
|
1
|
1 |
Ki = 102 nM
|
|
|
CP0394255
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl]-amide
Show/Hide
|
C27H31BrN2O4
|
1
|
1 |
Ki = 106.5 nM
|
|
|
CP0082953
|
2,3-dihydro-1,4-benzodioxin-3-ylmethyl-[2-(2,6-dimethoxyphenoxy)ethyl]amine;hydrochloride
Show/Hide
|
C19H23NO5
|
1
|
1 |
Ki = 107 nM
|
|
|
CP0522332
|
(S)-7-Chloro-9-(4-methyl-piperazin-1-yl)-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C17H20ClN3S
|
1
|
1 |
Ki = 110 nM
|
|
|
CP0509454
|
[6-(4-methylpiperazin-1-yl)pyrrolo[2,1-b][1,3]benzothiazepin-3-yl]methanol
Show/Hide
|
C18H21N3OS
|
1
|
1 |
Ki = 113 nM
|
|
|
CP0456817
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-amide
Show/Hide
|
C25H27BrN2O4
|
1
|
1 |
Ki = 126.5 nM
|
|
|
CP0431518
|
9H-Fluorene-4-carboxylic acid {3-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-propyl}-amide
Show/Hide
|
C27H27Cl2N3O
|
1
|
1 |
Ki = 139 nM
|
|
|
CP0241553
|
9H-Fluorene-2-carboxylic acid {3-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-propyl}-amide
Show/Hide
|
C27H27Cl2N3O
|
1
|
1 |
Ki = 199 nM
|
|
|
CP0383914
|
9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-ynyl}-amide
Show/Hide
|
C28H25Cl2N3O
|
1
|
1 |
Ki = 214 nM
|
|
|
CP0037227
|
7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-ol
Show/Hide
|
C16H25NO
|
1
|
1 |
Ki = 248 nM
|
|
|
CP0535727
|
1-Isopropoxymethyl-9-(4-methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C21H27N3OS
|
1
|
1 |
Ki = 278 nM
|
|
|
CP0339117
|
5-Bromo-N-[2-(3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-2-methoxy-benzamide
Show/Hide
|
C19H21BrN2O2
|
1
|
1 |
Ki = 310.7 nM
|
|
|
CP0178464
|
N-[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)butyl]-2-methoxy-5-methylbenzamide
Show/Hide
|
C24H32N2O4
|
1
|
1 |
Ki = 313 nM
|
|
|
CP0529519
|
7-Chloro-1-methoxymethyl-9-(4-methyl-piperazin-1-yl)-9,10-dihydro-4-thia-10a-aza-benzo[f]azulene
Show/Hide
|
C19H24ClN3OS
|
1
|
1 |
Ki = 316 nM
|
|
|
CP0025667
|
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
|
C18H19ClN4
|
1
|
1 |
Ki = 319 nM
|
|
|
CP0463526
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclohexyl-pyrrolidin-2-ylmethyl)-amide
Show/Hide
|
C23H29BrN2O2
|
1
|
1 |
Ki = 334 nM
|
|
|
CP0382018
|
N-[4-[4-(2,3-dichlorophenyl)piperazin-1-yl]but-2-ynyl]benzamide
Show/Hide
|
C21H21Cl2N3O
|
1
|
1 |
Ki = 394 nM
|
|
|
CP0465990
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclohexyl-piperidin-4-yl)-amide
Show/Hide
|
C23H29BrN2O2
|
1
|
1 |
Ki = 430 nM
|
|
|
CP0080663
|
5-Bromo-N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-2-methoxy-benzamide
Show/Hide
|
C21H25BrN2O4
|
1
|
1 |
Ki = 488 nM
|
|
|
CP0116813
|
5-Bromo-N-[4-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-butyl]-2,3-dimethoxy-benzamide
Show/Hide
|
C24H31BrN2O5
|
1
|
1 |
Ki = 627 nM
|
|
|
CP0046341
|
8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ol(SCH 23390)
Show/Hide
|
C17H18ClNO
|
1
|
1 |
Ki = 768 nM
|
|
|
CP0465347
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-cyclopentyl-piperidin-4-yl)-amide
Show/Hide
|
C22H27BrN2O2
|
1
|
1 |
Ki = 899 nM
|
|
|
CP0463091
|
9H-Fluorene-4-carboxylic acid {4-[4-(2,3-dichloro-phenyl)-piperazin-1-yl]-but-2-ynyl}-amide
Show/Hide
|
C28H25Cl2N3O
|
1
|
1 |
Ki = 1080 nM
|
|
|
CP0538820
|
4-Bromo-1-methoxy-naphthalene-2-carboxylic acid (1-bicyclo[3.3.1]non-9-yl-piperidin-4-yl)-amide
Show/Hide
|
C26H33BrN2O2
|
1
|
1 |
Ki = 1431 nM
|
|
|
CP0026495
|
CHEBI:51137
Show/Hide
|
C18H20N2
|
1
|
1 |
Ki = 1524 nM
|
|
|
CP0001238
|
14C-5-hydroxy tryptamine creatinine disulfate
Show/Hide
|
C10H12N2O
|
1
|
1 |
Ki = 2338 nM
|
|
|
CP0069692
|
(+)-yohimbine
Show/Hide
|
C21H26N2O3
|
1
|
1 |
Ki = 2430 nM
|
|
|
CP0055980
|
N-[2-(6,7-dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)ethyl]-2-methoxy-5-methylbenzamide
Show/Hide
|
C22H28N2O4
|
1
|
1 |
Ki = 3760 nM
|
|
|
CP0875029
|
9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene-1-carbaldehyde oxime
Show/Hide
|
C18H20N4OS
|
1
|
1 |
Ki = 4255 nM
|
|
|
CP0038839
|
(4R,4aS,7aR,12bS)-3-allyl-4a,9-dihydroxy-2,4,5,6,7a,13-hexahydro-1H-4,12-methanobenzofuro[3,2-e]isoquinoline-7-one;hydrochloride
Show/Hide
|
C19H21NO4
|
1
|
1 |
Ki > 20000 nM
|
|
|
CP0507024
|
9-(4-Methyl-piperazin-1-yl)-4-thia-10a-aza-benzo[f]azulene-1,10-dicarbaldehyde
Show/Hide
|
C19H19N3O2S
|
1
|
1 |
Ki > 1000 nM
|
|
|
CP0041613
|
Anapriline
Show/Hide
|
C16H21NO2
|
1
|
1 |
Ki > 5000 nM
|
|
|