| Compound ID |
Compound Name |
Compound Formula |
|
CP0406634
|
5-[[2-fluoro-4-(1-methylpyrazol-4-yl)phenyl]methyl]-2H-pyrazolo[4,3-c]quinolin-3-one
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|
C21H16FN5O
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0000324
|
2-acetoxyethyl(trimethyl)ammonium;bromide
Show/Hide
|
C7H16NO2+
|
2
|
| 1 |
EC50 = 1.1 nM
|
|
|
| 2 |
EC50 = 27000 nM
|
|
|
|
CP0433184
|
5-[(4-pyrazol-1-ylphenyl)methyl]-2H-pyrazolo[4,3-c]quinolin-3-one
Show/Hide
|
C20H15N5O
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0371787
|
5-(4-Hexyloxy-[1,2,5]thiadiazol-3-yl)-1-methyl-1,2,3,6-tetrahydro-pyridine; oxalic acid
Show/Hide
|
C14H23N3OS
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0305211
|
1-(1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-benzo[d]imidazol-2(3H)-one
Show/Hide
|
C25H32N4O
|
1
|
| 1 |
EC50 = 6.5 nM
|
|
|
|
CP0398671
|
N-[1-[3-(6-fluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]propanamide
Show/Hide
|
C20H28FN3O2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0381256
|
N-[1-[3-(6,7-difluoro-3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]propanamide
Show/Hide
|
C19H25F2N3O3
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0082269
|
1-benzyl-2,3-dihydro-1H-indole-2,3-dione
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|
C15H11NO2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0515358
|
1-[(4-pyrazol-1-ylphenyl)methyl]indole-2,3-dione
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|
C18H13N3O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0420948
|
1-[3-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-3,4-dihydro-1,5-naphthyridin-2-one
Show/Hide
|
C23H27N5O2
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0377069
|
N-[1-[3-(6,7-difluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-(3,4-dimethoxyphenyl)acetamide
Show/Hide
|
C27H33F2N3O4
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0506103
|
N-[1-[3-(6,7-difluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C25H29F2N3O2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0128076
|
8-Chloro-11-piperazin-1-yl-5H-dibenzo[b,e][1,4]diazepine
Show/Hide
|
C17H17ClN4
|
2
|
| 1 |
EC50 = 18 nM
|
|
|
| 2 |
EC50 = 140 nM
|
|
|
|
CP0427852
|
N-[1-[3-(5-fluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]propanamide
Show/Hide
|
C20H28FN3O2
|
1
|
| 1 |
EC50 = 19 nM
|
|
|
|
CP0398672
|
N-[1-[3-(7-fluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]propanamide
Show/Hide
|
C20H28FN3O2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0402343
|
N-[1-[3-(6,7-difluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]propanamide
Show/Hide
|
C20H27F2N3O2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0482046
|
1-[3-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-3,4-dihydro-1,8-naphthyridin-2-one
Show/Hide
|
C23H27N5O2
|
1
|
| 1 |
EC50 = 20 nM
|
|
|
|
CP0507197
|
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]propanamide
Show/Hide
|
C19H27N3O3
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
|
CP0507697
|
4-[3-[4-(6-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-1,4-benzoxazin-3-one
Show/Hide
|
C23H25FN4O3
|
1
|
| 1 |
EC50 = 44 nM
|
|
|
|
CP0504765
|
2-methyl-N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]propanamide
Show/Hide
|
C20H29N3O3
|
1
|
| 1 |
EC50 = 46 nM
|
|
|
|
CP0387736
|
N-[1-[3-(2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C25H31N3O2
|
1
|
| 1 |
EC50 = 48 nM
|
|
|
|
CP0374396
|
N-[1-[3-(6-fluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C25H30FN3O2
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0398633
|
N-[1-[3-(7-fluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C25H30FN3O2
|
1
|
| 1 |
EC50 = 51 nM
|
|
|
|
CP0026924
|
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C24H29N3O3
|
2
|
| 1 |
EC50 = 61 nM
|
|
|
| 2 |
EC50 = 97 nM
|
|
|
|
CP0482070
|
4-[3-[4-(5-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-1,4-benzoxazin-3-one
Show/Hide
|
C23H25FN4O3
|
1
|
| 1 |
EC50 = 66 nM
|
|
|
|
CP0455528
|
5-fluoro-1-[3-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C24H27FN4O2
|
1
|
| 1 |
EC50 = 68 nM
|
|
|
|
CP0439897
|
4-[3-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-1,4-benzoxazin-3-one
Show/Hide
|
C23H26N4O3
|
1
|
| 1 |
EC50 = 73 nM
|
|
|
|
CP0427853
|
N-[1-[3-(6,7-difluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]acetamide
Show/Hide
|
C19H25F2N3O2
|
1
|
| 1 |
EC50 = 86 nM
|
|
|
|
CP0400349
|
N-[1-[3-(3-oxo-1,4-benzothiazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0375830
|
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]cyclopropanecarboxamide
Show/Hide
|
C20H27N3O3
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0425952
|
1-[3-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C24H28N4O2
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0425956
|
4-[3-[4-(4-fluoro-2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-1,4-benzoxazin-3-one
Show/Hide
|
C23H25FN4O3
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0499476
|
N-[1-[3-(7-methoxy-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C26H33N3O3
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0377068
|
2-(3-Methoxy-phenyl)-N-{1-[3-(3-oxo-2,3-dihydro-benzo[1,4]oxazin-4-yl)-(propyl]-piperidin-4-yl}-acetamide
Show/Hide
|
C25H31N3O4
|
1
|
| 1 |
EC50 = 130 nM
|
|
|
|
CP0029624
|
4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one
Show/Hide
|
C20H31NO
|
2
|
| 1 |
EC50 = 150 nM
|
|
|
| 2 |
EC50 = 500 nM
|
|
|
|
CP0400355
|
N-[1-[3-(5-fluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C25H30FN3O2
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0381254
|
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]cyclobutanecarboxamide
Show/Hide
|
C21H29N3O3
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0425957
|
1-[3-[4-(1H-indol-5-yl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C25H29N3O
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0477314
|
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]acetamide
Show/Hide
|
C18H25N3O3
|
1
|
| 1 |
EC50 = 180 nM
|
|
|
|
CP0427848
|
N-[1-[3-(8-fluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C25H30FN3O2
|
1
|
| 1 |
EC50 = 290 nM
|
|
|
|
CP0439898
|
8-fluoro-1-[3-[4-(2-oxo-3H-benzimidazol-1-yl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
Show/Hide
|
C24H27FN4O2
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0400352
|
N-[1-[3-(8-fluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]propanamide
Show/Hide
|
C20H28FN3O2
|
1
|
| 1 |
EC50 = 310 nM
|
|
|
|
CP0377067
|
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]cyclopentanecarboxamide
Show/Hide
|
C22H31N3O3
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0462008
|
OXIPEROMIDE
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|
C20H23N3O2
|
1
|
| 1 |
EC50 = 400 nM
|
|
|
|
CP0521938
|
5-benzyl-2-[(2,5-dimethylphenyl)methyl]pyrazolo[4,3-c]quinolin-3-one
Show/Hide
|
C26H23N3O
|
1
|
| 1 |
EC50 = 473 nM
|
|
|
|
CP0427851
|
N-[1-[3-(6-methoxy-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C26H33N3O3
|
1
|
| 1 |
EC50 = 560 nM
|
|
|
|
CP0055373
|
1-(2-fluoro-4-(1-methyl-1H-pyrazol-4-yl)benzyl)indoline-2,3-dione
Show/Hide
|
C19H14FN3O2
|
1
|
| 1 |
EC50 = 830 nM
|
|
|
|
CP0379273
|
2-[4,6-difluoro-1-[[6-(1-methylpyrazol-4-yl)pyridin-3-yl]methyl]indol-3-yl]sulfonyl-N-(5-methyl-1,2-oxazol-3-yl)acetamide
Show/Hide
|
C24H20F2N6O4S
|
1
|
| 1 |
EC50 = 845 nM
|
|
|
|
CP0499477
|
N-methyl-N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C25H31N3O3
|
1
|
| 1 |
EC50 = 910 nM
|
|
|
|
CP0400350
|
N-[1-[3-(3-oxo-1,4-benzoxazin-4-yl)propyl]piperidin-4-yl]-3-phenylpropanamide
Show/Hide
|
C25H31N3O3
|
1
|
| 1 |
EC50 = 970 nM
|
|
|
|
CP0120956
|
3-amino-5-chloro-N-cyclopropyl-4,6-dimethylthieno[2,3-b]pyridine-2-carboxamide
Show/Hide
|
C13H14ClN3OS
|
1
|
| 1 |
EC50 = 970 nM
|
|
|
|
CP0377066
|
N-[1-[3-(2-oxo-1,3-benzoxazol-3-yl)propyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C23H27N3O3
|
1
|
| 1 |
EC50 = 1100 nM
|
|
|
|
CP0455529
|
4-[3-[4-(2-oxo-1H-imidazo[4,5-c]pyridin-3-yl)piperidin-1-yl]propyl]-1,4-benzoxazin-3-one
Show/Hide
|
C22H25N5O3
|
1
|
| 1 |
EC50 = 1200 nM
|
|
|
|
CP0443620
|
4-[3-[4-(2-oxo-1H-imidazo[4,5-b]pyridin-3-yl)piperidin-1-yl]propyl]-1,4-benzoxazin-3-one
Show/Hide
|
C22H25N5O3
|
1
|
| 1 |
EC50 = 1700 nM
|
|
|
|
CP0379740
|
2-methyl-5-[(4-pyrazol-1-ylphenyl)methyl]pyrazolo[4,3-c]quinolin-3-one
Show/Hide
|
C21H17N5O
|
1
|
| 1 |
EC50 = 2430 nM
|
|
|
|
CP0379206
|
5-benzyl-2-(pyridin-2-ylmethyl)pyrazolo[4,3-c]quinolin-3-one
Show/Hide
|
C23H18N4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0379737
|
5-benzyl-2-methylpyrazolo[4,3-c]quinolin-3-one
Show/Hide
|
C18H15N3O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0379738
|
5-benzyl-2-(pyridin-4-ylmethyl)pyrazolo[4,3-c]quinolin-3-one
Show/Hide
|
C23H18N4O
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0120957
|
3-amino-5-chloro-4,6-dimethyl-N-(pyridin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxamide
Show/Hide
|
C16H15ClN4OS
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0397064
|
2-[(2,5-dimethylphenyl)methyl]-1H-pyrazolo[4,3-c]quinolin-3-one
Show/Hide
|
C19H17N3O
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0379739
|
2-benzyl-5-[(4-pyrazol-1-ylphenyl)methyl]pyrazolo[4,3-c]quinolin-3-one
Show/Hide
|
C27H21N5O
|
1
|
| 1 |
EC50 > 10 nM
|
|
|
|
CP0041613
|
Anapriline
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|
C16H21NO2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0066236
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-8-yl)oxy]propan-2-ol
Show/Hide
|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0366351
|
1-(dimethylamino)-3-[(2-methyl-1H-1,2-benzazaborinin-5-yl)oxy]propan-2-ol
Show/Hide
|
C14H21BN2O2
|
2
|
| 1 |
EC50 > 5011.87 nM
|
|
|
| 2 |
IC50 > 5011.87 nM
|
|
|
|
CP0666404
|
Tiotropium bromide
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|
C19H24BrNO5S2
|
3
|
| 1 |
IC50 = 0.03162 nM
|
|
|
| 2 |
IC50 = 0.1 nM
|
|
|
| 3 |
IC50 = 0.22 nM
|
|
|
|
CP0696953
|
Aclidinium bromide
Show/Hide
|
C26H30BrNO4S2
|
2
|
| 1 |
IC50 = 0.1 nM
|
|
|
| 2 |
IC50 = 0.14 nM
|
|
|
|
CP0860527
|
GLYCOPYRROLATE
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|
C19H28BrNO3
|
1
|
| 1 |
IC50 = 0.1259 nM
|
|
|
|
CP0666488
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C25H28BrNO3S2
|
1
|
| 1 |
IC50 = 0.14 nM
|
|
|
|
CP0705209
|
(3R)-3-{[(2S)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl)acetyl]-oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H36BrNO4S
|
1
|
| 1 |
IC50 = 0.15 nM
|
|
|
|
CP0852883
|
(3R)-3-{[(2S)-2-Hydroxy-2-phenyl-2-(2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H32BrNO4S
|
1
|
| 1 |
IC50 = 0.16 nM
|
|
|
|
CP0418147
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2S)-cyclopentyl(hydroxy)2-thienylacetate
Show/Hide
|
C18H25NO3S
|
1
|
| 1 |
IC50 = 0.19 nM
|
|
|
|
CP0086732
|
(3R)-1-Azabicyclo[2.2.2]oct-3-ylhydroxy(di-2-thienyl)acetate
Show/Hide
|
C17H19NO3S2
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0431075
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2S)-hydroxy(phenyl)2-thienylacetate
Show/Hide
|
C19H21NO3S
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0397014
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2R)-hydroxy(phenyl)2-thienylacetate
Show/Hide
|
C19H21NO3S
|
1
|
| 1 |
IC50 = 0.23 nM
|
|
|
|
CP0896422
|
(3R)-3-{[(9-Hydroxy-9H-xanthen-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32BrNO5
|
1
|
| 1 |
IC50 = 0.23 nM
|
|
|
|
CP0918897
|
(3R)-3-{[Hydroxy(di-3-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H30BrNO4S2
|
1
|
| 1 |
IC50 = 0.23 nM
|
|
|
|
CP0439371
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl(2R)-cyclopentyl(hydroxy)2-thienylacetate
Show/Hide
|
C18H25NO3S
|
1
|
| 1 |
IC50 = 0.24 nM
|
|
|
|
CP0462648
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl9-hydroxy-9H-fluorene-9-carboxylate
Show/Hide
|
C21H21NO3
|
1
|
| 1 |
IC50 = 0.26 nM
|
|
|
|
CP0851960
|
(3R)-3-{[(9-Methyl-9H-xanthen-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34BrNO4
|
1
|
| 1 |
IC50 = 0.28 nM
|
|
|
|
CP0868133
|
(3R)-3-{[(9-Hydroxy-9H-xanthen-9-yl)carbonyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30BrNO4
|
1
|
| 1 |
IC50 = 0.29 nM
|
|
|
|
CP0874933
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(4-phenylbutyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H32BrNO3S2
|
1
|
| 1 |
IC50 = 0.29 nM
|
|
|
|
CP0369702
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl9H-xanthene-9-carboxylate
Show/Hide
|
C21H21NO3
|
1
|
| 1 |
IC50 = 0.31 nM
|
|
|
|
CP0918903
|
(3R)-3-{[Hydroxy(diphenyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H34BrNO4
|
1
|
| 1 |
IC50 = 0.31 nM
|
|
|
|
CP0868135
|
(3R)-3-[(Di-2-thienylacetyl)oxy]-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H30BrNO3S2
|
1
|
| 1 |
IC50 = 0.34 nM
|
|
|
|
CP0217648
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] 2-hydroxy-2,2-diphenylacetate
Show/Hide
|
C21H23NO3
|
1
|
| 1 |
IC50 = 0.36 nM
|
|
|
|
CP0893211
|
(3R)-3-{[(2R)-2-Hydroxy-2-phenyl-2-(2-thienyl)acetyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H32BrNO4S
|
1
|
| 1 |
IC50 = 0.38 nM
|
|
|
|
CP0456355
|
(R)-quinuclidin-3-yl phenyl(thiophen-3-ylmethyl)carbamate
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0456356
|
(R)-quinuclidin-3-yl phenyl(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C19H22N2O2S
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0501199
|
(R)-quinuclidin-3-yl benzyl(phenyl)carbamate
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0846167
|
(R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H31BrN2O3S
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0911595
|
(R)-1-(2-phenoxyethyl)-3-(phenyl(thiophen-3-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H31BrN2O3S
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0441678
|
(2S)-N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-cyclopentyl-2-hydroxy-2-thiophen-2-ylacetamide
Show/Hide
|
C18H26N2O2S
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0499035
|
(3R)-1-Heptyl-3-{[hydroxy(di-2-thienyl)acetyl]oxy}-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C24H34BrNO3S2
|
1
|
| 1 |
IC50 = 0.41 nM
|
|
|
|
CP0462649
|
(3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-methyl-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C18H22BrNO3S2
|
1
|
| 1 |
IC50 = 0.43 nM
|
|
|
|
CP0891026
|
(3R)-1-(2-Phenylethyl)-3-[(9H-xanthen-9-ylcarbonyl)oxy]-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30BrNO3
|
1
|
| 1 |
IC50 = 0.44 nM
|
|
|
|
CP0851961
|
(3R)-3-[(2,2-Di-2-thienylpropanoyl)oxy]-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H32BrNO3S2
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0874051
|
(3R)-3-{[(9-Hydroxy-9H-fluoren-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32BrNO4
|
1
|
| 1 |
IC50 = 0.63 nM
|
|
|
|
CP0459211
|
(R)-quinuclidin-3-yl butyl(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C17H26N2O2S
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0502914
|
(R)-quinuclidin-3-yl pentyl(phenyl)carbamate
Show/Hide
|
C19H28N2O2
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0868134
|
(3R)-3-{[(2R)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl)acetyl]-oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H36BrNO4S
|
1
|
| 1 |
IC50 = 0.81 nM
|
|
|
|
CP0390751
|
(R)-quinuclidin-3-yl 3-fluorophenyl(3,4,5-trifluorobenzyl)carbamate
Show/Hide
|
C21H20F4N2O2
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0387223
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-hydroxy-2,2-dithiophen-2-ylacetamide
Show/Hide
|
C17H20N2O2S2
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0478198
|
(R)-quinuclidin-3-yl m-tolyl(2,4,5-trifluorobenzyl)carbamate
Show/Hide
|
C22H23F3N2O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0482224
|
(R)-quinuclidin-3-yl phenethyl(phenyl)carbamate
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0851406
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0859004
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C24H29BrN2O2S3
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0502913
|
(R)-quinuclidin-3-yl butyl(phenyl)carbamate
Show/Hide
|
C18H26N2O2
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0906344
|
(R)-3-((3-fluorophenyl)(3,4,5-trifluorobenzyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H29BrF4N2O3
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0891027
|
(3R)-3-{[(9-Hydroxy-9H-fluoren-9-yl)carbonyl]oxy}-1-(2-phenylethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H30BrNO3
|
1
|
| 1 |
IC50 = 1.12 nM
|
|
|
|
CP0920325
|
(3R)-3-{[(9-Methyl-9H-fluoren-9-yl)carbonyl]oxy}-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34BrNO3
|
1
|
| 1 |
IC50 = 1.26 nM
|
|
|
|
CP0916859
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H33BrN2O2S
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0917225
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H35BrN2O3
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0488363
|
(R)-quinuclidin-3-yl 3-fluorobenzyl(3-fluorophenyl)carbamate
Show/Hide
|
C21H22F2N2O2
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0909075
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H35BrN2O2
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0891718
|
(R)-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0846146
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H33BrN2O3
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0891721
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C25H35BrN2O2S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0895086
|
(R)-3-(phenyl(thiophen-3-ylmethyl)carbamoyloxy)-1-(3-(thiophen-2-yl)propyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0864661
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(2-phenoxyethyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C25H29BrN2O3S2
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0501201
|
(R)-quinuclidin-3-yl bis(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C18H22N2O2S2
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0912372
|
(R)-1-(2-phenoxyethyl)-3-(m-tolyl(2,4,5-trifluorobenzyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H32BrF3N2O3
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0847622
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-(3-phenylpropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C27H37BrN2O2
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0070586
|
Ipratropium Bromide
Show/Hide
|
C20H30BrNO3
|
2
|
| 1 |
IC50 = 2.65 nM
|
|
|
| 2 |
IC50 = 2.9 nM
|
|
|
|
CP0802380
|
quinuclidin-4-yl biphenyl-2-ylcarbamate hydrochloride
Show/Hide
|
C20H23ClN2O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0912371
|
(R)-1-(3-phenylpropyl)-3-(m-tolyl(2,4,5-trifluorobenzyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C31H34BrF3N2O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0505031
|
(3R)-1-Heptyl-3-{[(9-hydroxy-9H-fluoren-9-yl)carbonyl]-oxy}-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C28H36BrNO3
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0864662
|
(R)-3-(2-hydroxy-2,2-di(thiophen-2-yl)acetamido)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O3S2
|
1
|
| 1 |
IC50 = 4.4 nM
|
|
|
|
CP0673968
|
SID50106181
Show/Hide
|
C21H26INO2
|
2
|
| 1 |
IC50 = 4.5 nM
|
|
|
| 2 |
Ki = 1.1 nM
|
|
|
|
CP0847983
|
(R)-1-(3-phenoxypropyl)-3-(9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C30H33BrN2O3
|
1
|
| 1 |
IC50 = 4.9 nM
|
|
|
|
CP0026865
|
2-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine
Show/Hide
|
C18H19ClN4
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0398693
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2-hydroxy-2,2-diphenylacetamide
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 = 6.1 nM
|
|
|
|
CP0477682
|
1-[(2R)-4-(5-fluoro-3-methylpyridin-2-yl)-2-methylpiperazin-1-yl]-4-quinolin-5-ylbutan-1-one
Show/Hide
|
C24H27FN4O
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0390680
|
(R)-quinuclidin-3-yl benzyl(4-fluorophenyl)carbamate
Show/Hide
|
C21H23FN2O2
|
1
|
| 1 |
IC50 = 8.3 nM
|
|
|
|
CP0375586
|
(R)-quinuclidin-3-yl benzyl(thiophen-2-ylmethyl)carbamate
Show/Hide
|
C20H24N2O2S
|
1
|
| 1 |
IC50 = 8.8 nM
|
|
|
|
CP0459214
|
(R)-1-methyl-3-(phenyl(thiophen-2-ylmethyl)carbamoyloxy)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C20H25BrN2O2S
|
1
|
| 1 |
IC50 = 9.2 nM
|
|
|
|
CP0025667
|
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
|
C18H19ClN4
|
1
|
| 1 |
IC50 = 9.4 nM
|
|
|
|
CP0379242
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-9-hydroxyfluorene-9-carboxamide
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
IC50 = 9.8 nM
|
|
|
|
CP0490579
|
6-[(2R,6R)-4-[3-(1,3-benzothiazol-7-ylsulfonyl)propanoyl]-2,6-dimethylpiperazin-1-yl]pyridine-3-carbonitrile
Show/Hide
|
C22H23N5O3S2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0411467
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-9H-xanthene-9-carboxamide
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
IC50 = 13.4 nM
|
|
|
|
CP0505885
|
(3R)-1-Azabicyclo[2.2.2]oct-3-yl 10,11-dihydro-5H-dibenzo-[a,d][7]annulene-5-carboxylate
Show/Hide
|
C23H25NO2
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0845813
|
(R)-3-(benzyl(phenyl)carbamoyloxy)-1-phenethyl-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H33BrN2O2
|
1
|
| 1 |
IC50 = 15.1 nM
|
|
|
|
CP0213707
|
8-Methoxy-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine
Show/Hide
|
C19H22N4O
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0469097
|
1-(4-pyridin-4-ylpiperazin-1-yl)-4-quinolin-5-ylbutan-1-one
Show/Hide
|
C22H24N4O
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0459212
|
(R)-quinuclidin-3-yl phenyl(propyl)carbamate
Show/Hide
|
C17H24N2O2
|
1
|
| 1 |
IC50 = 26.7 nM
|
|
|
|
CP0048902
|
11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepin-8-ol
Show/Hide
|
C18H20N4O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0469803
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-N-methyl-9H-xanthene-9-carboxamide
Show/Hide
|
C22H24N2O2
|
1
|
| 1 |
IC50 = 30.1 nM
|
|
|
|
CP0903846
|
(R)-3-(butyl(phenyl)carbamoyloxy)-1-phenethyl-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H35BrN2O2
|
1
|
| 1 |
IC50 = 33.3 nM
|
|
|
|
CP0398694
|
N-[(3R)-1-azabicyclo[2.2.2]octan-3-yl]-2,2-dithiophen-2-ylacetamide
Show/Hide
|
C17H20N2OS2
|
1
|
| 1 |
IC50 = 34.8 nM
|
|
|
|
CP0135432
|
[6-(4-methylpiperazin-1-yl)-11H-benzo[b][1,4]benzodiazepin-3-yl] trifluoromethanesulfonate
Show/Hide
|
C19H19F3N4O3S
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0184885
|
11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepin-2-ol
Show/Hide
|
C18H20N4O
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0196783
|
[6-(4-methylpiperazin-1-yl)-11H-benzo[b][1,4]benzodiazepin-3-yl] methanesulfonate
Show/Hide
|
C19H22N4O3S
|
1
|
| 1 |
IC50 = 38 nM
|
|
|
|
CP0100094
|
2-Methoxy-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]diazepine
Show/Hide
|
C19H22N4O
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0478197
|
(R)-quinuclidin-3-yl benzyl(p-tolyl)carbamate
Show/Hide
|
C22H26N2O2
|
1
|
| 1 |
IC50 = 39.7 nM
|
|
|
|
CP0882813
|
(R)-3-(2,2-di(thiophen-2-yl)acetamido)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C26H31BrN2O2S2
|
1
|
| 1 |
IC50 = 53.8 nM
|
|
|
|
CP0218798
|
[3-chloro-6-(4-methylpiperazin-1-yl)-11H-benzo[b][1,4]benzodiazepin-8-yl] trifluoromethanesulfonate
Show/Hide
|
C19H18ClF3N4O3S
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0846145
|
SOLIFENACIN SUCCINATE
Show/Hide
|
C27H32N2O6
|
1
|
| 1 |
IC50 = 63.5 nM
|
|
|
|
CP0935343
|
(R)-1-(3-(1H-pyrrol-1-yl)propyl)-3-(N-methyl-9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C29H34BrN3O2
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0896423
|
(3R)-1-Benzyl-3-{[hydroxy(di-2-thienyl)acetyl]oxy}-1-azoniabicyclo[2.2.2]octane bromide
Show/Hide
|
C24H26BrNO3S2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0393505
|
N-[3-oxo-3-(4-pyridin-4-ylpiperazin-1-yl)propyl]quinoline-5-sulfonamide
Show/Hide
|
C21H23N5O3S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0868278
|
(R)-1-(3-(biphenyl-4-yloxy)propyl)-3-(N-methyl-9H-xanthene-9-carboxamido)-1-azoniabicyclo[2.2.2]octane chloride
Show/Hide
|
C37H39ClN2O3
|
1
|
| 1 |
IC50 = 281.4 nM
|
|
|
|
CP0864660
|
(R)-3-(9-hydroxy-9H-fluorene-9-carboxamido)-1-(3-(methyl(phenyl)amino)propyl)-1-azoniabicyclo[2.2.2]octane chloride
Show/Hide
|
C31H36ClN3O2
|
1
|
| 1 |
IC50 = 290.8 nM
|
|
|
|
CP0390678
|
(R)-quinuclidin-3-yl diphenylcarbamate
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
IC50 = 319.4 nM
|
|
|
|
CP0469061
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-2,3,4,5,6-pentafluorobenzamide
Show/Hide
|
C19H17ClF5N3O
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0390681
|
(R)-quinuclidin-3-yl isopropyl(phenyl)carbamate
Show/Hide
|
C17H24N2O2
|
1
|
| 1 |
IC50 = 428 nM
|
|
|
|
CP0133741
|
[6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzothiazepin-8-yl] trifluoromethanesulfonate
Show/Hide
|
C19H18F3N3O3S2
|
1
|
| 1 |
IC50 = 460 nM
|
|
|
|
CP0196982
|
[6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzoxazepin-8-yl] trifluoromethanesulfonate
Show/Hide
|
C19H18F3N3O4S
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0401466
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-2,5-bis(trifluoromethyl)benzamide
Show/Hide
|
C21H20ClF6N3O
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0577417
|
1-[4-(3-fluoropyridin-4-yl)piperazin-1-yl]-4-quinolin-5-ylbutan-1-one
Show/Hide
|
C22H23FN4O
|
1
|
| 1 |
IC50 = 490 nM
|
|
|
|
CP0372956
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-2-methoxybenzamide
Show/Hide
|
C20H24ClN3O2
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0373153
|
2-chloro-N-(3-chloro-4-(4-ethylpiperazin-1-yl)phenyl)benzamide
Show/Hide
|
C19H21Cl2N3O
|
1
|
| 1 |
IC50 = 960 nM
|
|
|
|
CP0207272
|
[6-(4-methylpiperazin-1-yl)-11H-benzo[b][1,4]benzodiazepin-8-yl] methanesulfonate
Show/Hide
|
C19H22N4O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0209256
|
[6-(4-methylpiperazin-1-yl)-11H-benzo[b][1,4]benzodiazepin-8-yl] trifluoromethanesulfonate
Show/Hide
|
C19H19F3N4O3S
|
2
|
| 1 |
IC50 = 1200 nM
|
|
|
| 2 |
IC50 > 1000 nM
|
|
|
|
CP0506234
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3-methylbenzamide
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0493960
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3,5-bis(trifluoromethyl)benzamide
Show/Hide
|
C21H20ClF6N3O
|
1
|
| 1 |
IC50 = 2600 nM
|
|
|
|
CP0507717
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-4-methylbenzamide
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0514007
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C20H21ClF3N3O
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0372793
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]benzamide
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
|
CP0372958
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-4-methoxybenzamide
Show/Hide
|
C20H24ClN3O2
|
1
|
| 1 |
IC50 = 3200 nM
|
|
|
|
CP0469062
|
N-[3-chloro-4-(4-ethylpiperazin-1-yl)phenyl]-3,4-difluorobenzamide
Show/Hide
|
C19H20ClF2N3O
|
1
|
| 1 |
IC50 = 4700 nM
|
|
|
|
CP0008601
|
4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl)
Show/Hide
|
C21H23ClFNO2
|
1
|
| 1 |
IC50 = 5500 nM
|
|
|
|
CP0076121
|
13-chloro-10-(4-methylpiperazin-1-yl)-2-oxa-9-azatricyclo[9.4.0.0^{3,8}]pentadeca-1(11),3,5,7,9,12,14-heptaene
Show/Hide
|
C18H18ClN3O
|
1
|
| 1 |
IC50 = 5500 nM
|
|
|
|
CP0448294
|
(R)-2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-1-methyl-piperidine
Show/Hide
|
C22H25N
|
1
|
| 1 |
Kd = 1.53 nM
|
|
|
|
CP0897105
|
2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-1-methyl-piperidine
Show/Hide
|
C22H25N
|
1
|
| 1 |
Kd = 1.75 nM
|
|
|
|
CP0948456
|
2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl-piperidine
Show/Hide
|
C22H25N
|
1
|
| 1 |
Kd = 2.7 nM
|
|
|
|
CP0496337
|
2-[(E)-2-(9,9a-Dihydro-4aH-xanthen-9-yl)-vinyl]-1-methyl-piperidine
Show/Hide
|
C21H25NO
|
1
|
| 1 |
Kd = 3.35 nM
|
|
|
|
CP0448319
|
(S)-2-[(E)-2-(9,10-Dihydro-anthracen-9-yl)-vinyl]-1-methyl-piperidine
Show/Hide
|
C22H25N
|
1
|
| 1 |
Kd = 4.92 nM
|
|
|
|
CP0410597
|
2-[3-(10H-Anthracen-9-ylidene)-propyl]-1-methyl-piperidine
Show/Hide
|
C23H27N
|
1
|
| 1 |
Kd = 4.99 nM
|
|
|
|
CP0440269
|
2-[(E)-3-(9,10-Dihydro-anthracen-9-yl)-allyl]-1-methyl-piperidine
Show/Hide
|
C23H27N
|
1
|
| 1 |
Kd = 5.23 nM
|
|
|
|
CP0470231
|
(R)-2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl-piperidine
Show/Hide
|
C22H25N
|
1
|
| 1 |
Kd = 11.6 nM
|
|
|
|
CP0461109
|
(S)-2-[2-(10H-Anthracen-9-ylidene)-ethyl]-1-methyl-piperidine
Show/Hide
|
C22H25N
|
1
|
| 1 |
Kd = 24.2 nM
|
|
|
|
CP0054849
|
(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methyl-6-(S)-methyl-piperidin-2-yl)-vinyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C22H35NO2
|
3
|
| 1 |
Kd = 148 nM
|
|
|
| 2 |
Kd = 168 nM
|
|
|
| 3 |
Ki = 4.5 nM
|
|
|
|
CP0430934
|
(2S,6R)-1,2-Dimethyl-6-[(E)-2-((3S,3aR,4R,4aS,8aR,9aS)-3-methyl-dodecahydro-naphtho[2,3-c]furan-4-yl)-vinyl]-piperidine
Show/Hide
|
C22H37NO
|
1
|
| 1 |
Kd = 167 nM
|
|
|
|
CP0472252
|
(1S,3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-vinyl]-3-methyl-dodecahydro-naphtho[2,3-c]furan-1-ol
Show/Hide
|
C22H37NO2
|
1
|
| 1 |
Kd = 423 nM
|
|
|
|
CP0440092
|
(S)-1-{(1R,2R,3S,4aR,8aS)-1-[(E)-2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-vinyl]-3-hydroxymethyl-decahydro-naphthalen-2-yl}-ethanol
Show/Hide
|
C22H39NO2
|
1
|
| 1 |
Kd = 494 nM
|
|
|
|
CP0465184
|
Acetic acid (S)-1-{(1R,2R,3S,4aR,8aS)-3-acetoxymethyl-1-[(E)-2-((2R,6S)-1,6-dimethyl-piperidin-2-yl)-vinyl]-decahydro-naphthalen-2-yl}-ethyl ester
Show/Hide
|
C26H43NO4
|
1
|
| 1 |
Kd = 604.7 nM
|
|
|
|
CP0501173
|
2-((E)-2-Anthracen-9-yl-vinyl)-1-methyl-piperidine
Show/Hide
|
C22H23N
|
1
|
| 1 |
Kd = 679 nM
|
|
|
|
CP0431696
|
Acetic acid (1R,3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-((2R,6S)-1,6-dimethyl-piperidin-2-yl)-vinyl]-3-methyl-dodecahydro-naphtho[2,3-c]furan-1-yl ester
Show/Hide
|
C24H39NO3
|
1
|
| 1 |
Kd = 866 nM
|
|
|
|
CP0406349
|
2,2-Dimethyl-propionic acid (1R,3S,3aR,4R,4aS,8aR,9aS)-4-[(E)-2-((2R,6S)-1,6-dimethyl-piperidin-2-yl)-vinyl]-3-methyl-dodecahydro-naphtho[2,3-c]furan-1-yl ester
Show/Hide
|
C27H45NO3
|
1
|
| 1 |
Kd = 2520 nM
|
|
|
|
CP0207650
|
(4R,5S)-5-Methyl-4-[(E)-3-((R)-1-methyl-piperidin-2-yl)-allyl]-dihydro-furan-2-one
Show/Hide
|
C14H23NO2
|
1
|
| 1 |
Kd = 9700 nM
|
|
|
|
CP0477680
|
6-[3-[3-(1,3-benzothiazol-7-ylsulfonyl)propanoyl]-3,8-diazabicyclo[3.2.1]octan-8-yl]pyridine-3-carbonitrile
Show/Hide
|
C22H21N5O3S2
|
2
|
| 1 |
Ki = 0.14 nM
|
|
|
| 2 |
Ki = 19 nM
|
|
|
|
CP0487381
|
[(2S,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H32INO2
|
1
|
| 1 |
Ki = 0.302 nM
|
|
|
|
CP0472767
|
(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)methyl-trimethylazanium;iodide
Show/Hide
|
C20H32INO2
|
1
|
| 1 |
Ki = 0.5248 nM
|
|
|
|
CP0491606
|
7-(3-bromo-5-methoxyphenyl)-1,3-dimethyl-7,8-dihydropyrazolo[3,4-d][1,3]thiazepin-4-one
Show/Hide
|
C15H16BrN3O2S
|
1
|
| 1 |
Ki = 0.594 nM
|
|
|
|
CP0516427
|
1-[(2S,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H29NO2
|
1
|
| 1 |
Ki = 0.7943 nM
|
|
|
|
CP0101233
|
2-(4-Hydroxy-phenyl)-2-phenyl-propionic acid 2-diethylamino-ethyl ester
Show/Hide
|
C21H27NO3
|
1
|
| 1 |
Ki = 0.881 nM
|
|
|
|
CP0109931
|
ATROPEN
Show/Hide
|
C17H23NO3
|
1
|
| 1 |
Ki = 0.922 nM
|
|
|
|
CP0390370
|
1-[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H23NO2
|
1
|
| 1 |
Ki = 1.259 nM
|
|
|
|
CP0468712
|
S-[2-(diethylamino)ethyl] 2-hydroxy-2,2-diphenylethanethioate
Show/Hide
|
C20H25NO2S
|
1
|
| 1 |
Ki = 1.29 nM
|
|
|
|
CP0491603
|
2-(diethylamino)ethyl 2-cyclohexyl-2-hydroxy-2-thiophen-2-ylacetate
Show/Hide
|
C18H29NO3S
|
1
|
| 1 |
Ki = 1.32 nM
|
|
|
|
CP0421081
|
1-(6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl)-N,N-dimethylmethanamine
Show/Hide
|
C19H29NO2
|
1
|
| 1 |
Ki = 1.38 nM
|
|
|
|
CP0540935
|
2-[2-[6-[8-[6-[bis[2-oxo-2-(6-oxo-5H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)ethyl]amino]hexyl-methylamino]octyl-methylamino]hexylamino]acetyl]-2,4,9,15-tetrazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-10-one
Show/Hide
|
C63H76N14O6
|
1
|
| 1 |
Ki = 1.585 nM
|
|
|
|
CP0850774
|
METHYLBENACTYZIUM BROMIDE
Show/Hide
|
C21H28BrNO3
|
1
|
| 1 |
Ki = 1.59 nM
|
|
|
|
CP0436551
|
1-(bicyclo[2.2.1]hept-5-en-2-yl)-1-phenyl-3-(piperidin-1-yl)propan-1-ol
Show/Hide
|
C21H29NO
|
1
|
| 1 |
Ki = 2.36 nM
|
|
|
|
CP0080609
|
1-Cyclohexyl-4-{1-[4-(4-methoxy-benzenesulfonyl)-phenyl]-vinyl}-piperidine
Show/Hide
|
C26H33NO3S
|
1
|
| 1 |
Ki = 2.8 nM
|
|
|
|
CP0056034
|
11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
|
C19H21N5O2
|
1
|
| 1 |
Ki = 2.818 nM
|
|
|
|
CP0516424
|
Flotros
Show/Hide
|
C25H30ClNO3
|
1
|
| 1 |
Ki = 3.467 nM
|
|
|
|
CP0058613
|
CAS_132947
Show/Hide
|
C64H77N13O6
|
1
|
| 1 |
Ki = 3.548 nM
|
|
|
|
CP0296594
|
(3S,3aR,4R,4aS,8aR,9aS)-4-[2-((2R,6S)-1,6-Dimethyl-piperidin-2-yl)-ethyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C22H37NO2
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0465680
|
(3S)-3-[[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 4.571 nM
|
|
|
|
CP0521081
|
[(2R,6R)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium
Show/Hide
|
C20H32NO2+
|
1
|
| 1 |
Ki = 5.012 nM
|
|
|
|
CP0673820
|
2-(2,2-diphenylacetoxy)-N,N,N-triethylethanaminiumiodide
Show/Hide
|
C22H30INO2
|
1
|
| 1 |
Ki = 5.75 nM
|
|
|
|
CP0822547
|
2-(2,2-diphenylacetoxy)-N,N-diethyl-Nmethylethanaminiumbromide
Show/Hide
|
C21H28BrNO2
|
1
|
| 1 |
Ki = 5.78 nM
|
|
|
|
CP0849067
|
11-{2-[[(1S,2R)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
Show/Hide
|
C28H34N4O10
|
1
|
| 1 |
Ki = 6.31 nM
|
|
|
|
CP0167280
|
4-{1-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-vinyl}-[1,4']bipiperidinyl-1'-carboxylic acid ethyl ester
Show/Hide
|
C28H36N2O5S
|
1
|
| 1 |
Ki = 6.5 nM
|
|
|
|
CP0175835
|
Isoptpo Hyoscine
Show/Hide
|
C17H21NO4
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0420726
|
2-(diethylamino)ethyl 2-(1-hydroxycyclohexyl)-2-phenylacetate
Show/Hide
|
C20H31NO3
|
1
|
| 1 |
Ki = 7.75 nM
|
|
|
|
CP0471590
|
(3R)-3-[[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 8.913 nM
|
|
|
|
CP0203329
|
4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)-1-(piperidin-4-yl)piperidine
Show/Hide
|
C25H32N2O3S
|
1
|
| 1 |
Ki = 9.1 nM
|
|
|
|
CP0564271
|
[(2R,6S)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H32INO2
|
1
|
| 1 |
Ki = 9.333 nM
|
|
|
|
CP0414398
|
[(2R,5R)-5-cyclohexyl-5-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H32INO2
|
1
|
| 1 |
Ki = 9.772 nM
|
|
|
|
CP0433352
|
3-(diethylamino)propyl (3S)-3-methyl-2-phenylpentanoate
Show/Hide
|
C19H31NO2
|
1
|
| 1 |
Ki = 10.7 nM
|
|
|
|
CP0849144
|
11-{2-[[(1R,2S)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
Show/Hide
|
C28H34N4O10
|
1
|
| 1 |
Ki = 12.59 nM
|
|
|
|
CP0164673
|
2,2-Diphenyl-propionic acid 2-diethylamino-ethyl ester
Show/Hide
|
C21H27NO2
|
1
|
| 1 |
Ki = 15.1 nM
|
|
|
|
CP0473020
|
[(2R,5S)-5-cyclohexyl-5-phenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H32INO2
|
1
|
| 1 |
Ki = 15.49 nM
|
|
|
|
CP0449731
|
2-(4-methoxyphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C22H25NO3
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0473019
|
1-[(2R,6R)-6-cyclohexyl-6-phenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
|
C19H29NO2
|
1
|
| 1 |
Ki = 20.89 nM
|
|
|
|
CP0858320
|
11-{2-[[(1R,2R)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
Show/Hide
|
C28H34N4O10
|
1
|
| 1 |
Ki = 22.39 nM
|
|
|
|
CP0209448
|
4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)-1-(propylsulfonyl)piperidine
Show/Hide
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C28H38N2O5S2
|
1
|
| 1 |
Ki = 25.7 nM
|
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CP0225899
|
AQ-RA 741
Show/Hide
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C27H37N5O2
|
1
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| 1 |
Ki = 28.84 nM
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CP0217520
|
AF-DX 384
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C27H38N6O2
|
1
|
| 1 |
Ki = 30.9 nM
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CP0406396
|
N,N-dimethyl-1-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]methanamine
Show/Hide
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C19H22N2
|
1
|
| 1 |
Ki = 34.67 nM
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CP0475081
|
1-[(2R)-6,6-diphenyl-1,4-dioxan-2-yl]-N,N-dimethylmethanamine
Show/Hide
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C19H23NO2
|
1
|
| 1 |
Ki = 35.48 nM
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CP0516425
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[(2R)-5,5-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO2
|
1
|
| 1 |
Ki = 36.31 nM
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CP0401540
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(octahydro-quinolin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C25H41NO2
|
1
|
| 1 |
Ki = 38 nM
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|
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CP0386733
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C24H27NO4
|
1
|
| 1 |
Ki = 41.69 nM
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|
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CP0220544
|
1-(4-(4-(1-(4-(4-methoxyphenylsulfonyl)phenyl)vinyl)piperidin-1-yl)piperidin-1-yl)butan-1-one
Show/Hide
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C29H38N2O4S
|
1
|
| 1 |
Ki = 42 nM
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CP0397949
|
N,N-dimethyl-2-[3-[phenyl(pyridin-2-yl)methyl]-1H-inden-2-yl]ethanamine
Show/Hide
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C25H26N2
|
1
|
| 1 |
Ki = 43.65 nM
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|
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CP0849141
|
11-{2-[[(1S,2S)-2-(Dimethylamino)cyclohexyl](methyl)amino]acetyl}-6,11-dihydro-5H-benzo[e]pyrido[3,2-b][1,4]diazepin-6-one Dioxalate
Show/Hide
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C28H34N4O10
|
1
|
| 1 |
Ki = 45.71 nM
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CP0002227
|
SOLIFENACIN
Show/Hide
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C23H26N2O2
|
1
|
| 1 |
Ki = 51.29 nM
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CP0375774
|
N,N-dimethyl-2-[3-(2-pyridin-2-ylpropan-2-yl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H26N2
|
1
|
| 1 |
Ki = 52.48 nM
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CP0489025
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(3S)-3-[[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 54.95 nM
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CP0490256
|
1,3-benzodioxol-5-ylmethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C22H23NO4
|
1
|
| 1 |
Ki = 60 nM
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|
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CP0517270
|
[(2R,5S,6R)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
|
C20H26INO2
|
1
|
| 1 |
Ki = 64.57 nM
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CP0462407
|
4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]piperidine-1-carboxamide
Show/Hide
|
C25H33F3N6OS
|
1
|
| 1 |
Ki = 66.07 nM
|
|
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CP0386735
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 67.61 nM
|
|
|
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CP0842192
|
2-(2,2-diphenylacetoxy)-N,N,Ntrimethylethanaminiumbromide
Show/Hide
|
C19H24BrNO2
|
1
|
| 1 |
Ki = 85.7 nM
|
|
|
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CP0489900
|
2-(4-fluorophenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C22H24FNO2
|
1
|
| 1 |
Ki = 100 nM
|
|
|
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CP0368307
|
5-[5-[3-[1-[2-fluoro-4-(trifluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
Show/Hide
|
C23H26F4N6OS
|
1
|
| 1 |
Ki = 109.65 nM
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|
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CP0390368
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 120.23 nM
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|
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CP0381106
|
(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(Adamantan-1-ylamino)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C26H41NO2
|
1
|
| 1 |
Ki = 136 nM
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|
|
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CP0380642
|
5-[5-[3-[(2S,3R)-2-[2-fluoro-4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
Show/Hide
|
C23H25F4N5OS
|
1
|
| 1 |
Ki = 138.04 nM
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|
|
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CP0425615
|
2-thiophen-3-ylethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C20H23NO2S
|
1
|
| 1 |
Ki = 140 nM
|
|
|
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CP0403962
|
2-[6-chloro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C20H23ClN2
|
1
|
| 1 |
Ki = 151.36 nM
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|
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CP0449403
|
N,N-dimethyl-2-[3-(1-phenylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H25N
|
1
|
| 1 |
Ki = 158.49 nM
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|
|
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CP0410687
|
(3R)-3-[[(2S)-6,6-diphenyl-1,4-dioxan-2-yl]methoxy]-1-azabicyclo[2.2.2]octane
Show/Hide
|
C24H29NO3
|
1
|
| 1 |
Ki = 162.18 nM
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|
|
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CP0385601
|
2-(diethylamino)ethyl 2,2-diphenylbutanoate
Show/Hide
|
C22H29NO2
|
1
|
| 1 |
Ki = 166 nM
|
|
|
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CP0398325
|
4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]thiadiazole
Show/Hide
|
C21H23F3N6S2
|
1
|
| 1 |
Ki = 169.82 nM
|
|
|
|
CP0425606
|
1-Ethyl-4-phenyl-1,2,5,6-tetrahydro-pyridine-3-carboxylic acid 2-(4-methoxy-phenyl)-ethyl ester; oxalic acid
Show/Hide
|
C23H27NO3
|
1
|
| 1 |
Ki = 170 nM
|
|
|
|
CP0398323
|
N-[4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]cyclohexyl]acetamide
Show/Hide
|
C27H36F3N5OS
|
1
|
| 1 |
Ki = 173.78 nM
|
|
|
|
CP0432187
|
2-(diethylamino)ethyl 2-(2,6-dimethylphenyl)-2-hydroxy-2-phenylacetate
Show/Hide
|
C22H29NO3
|
1
|
| 1 |
Ki = 176 nM
|
|
|
|
CP0502977
|
(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-(3-thiomorpholin-4-yl-propyl)-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C20H33NO2S
|
1
|
| 1 |
Ki = 179 nM
|
|
|
|
CP0271112
|
N,N-dimethyl-2-[3-[(1S)-1-pyridin-2-ylethyl]-1H-inden-2-yl]ethanamine
Show/Hide
|
C20H24N2
|
1
|
| 1 |
Ki = 190.55 nM
|
|
|
|
CP0415329
|
[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C24H27NO4
|
1
|
| 1 |
Ki = 190.55 nM
|
|
|
|
CP0410686
|
[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2R)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C25H29NO4
|
1
|
| 1 |
Ki = 194.98 nM
|
|
|
|
CP0875549
|
1-(4-Hydroxy-4,4-diphenyl-butyl)-1-methyl-piperidinium iodide
Show/Hide
|
C22H30INO
|
1
|
| 1 |
Ki = 199.53 nM
|
|
|
|
CP0440870
|
2-(2-methylphenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H27NO2
|
1
|
| 1 |
Ki = 200 nM
|
|
|
|
CP0465375
|
2-(1,3-benzodioxol-5-yl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H25NO4
|
1
|
| 1 |
Ki = 200 nM
|
|
|
|
CP0418487
|
2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-methyl-5-phenyl-3,6-dihydro-2H-pyridine-4-carboxylate
Show/Hide
|
C23H25NO3
|
1
|
| 1 |
Ki = 210 nM
|
|
|
|
CP0453174
|
(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-(3-morpholin-4-yl-propyl)-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C20H33NO3
|
1
|
| 1 |
Ki = 222 nM
|
|
|
|
CP0416602
|
2-[6-chloro-3-(1-pyridin-2-ylpropyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H25ClN2
|
1
|
| 1 |
Ki = 223.87 nM
|
|
|
|
CP0214556
|
5-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]pyridine-2-carboxamide
Show/Hide
|
C25H27F3N6OS
|
1
|
| 1 |
Ki = 223.87 nM
|
|
|
|
CP0403951
|
N-methyl-N-[[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]methyl]propan-2-amine
Show/Hide
|
C21H26N2
|
1
|
| 1 |
Ki = 229.09 nM
|
|
|
|
CP0436921
|
N,N-dimethyl-2-[3-(1-pyridin-2-ylpropyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C21H26N2
|
1
|
| 1 |
Ki = 239.88 nM
|
|
|
|
CP0414198
|
2-(4-bromophenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C22H24BrNO2
|
1
|
| 1 |
Ki = 240 nM
|
|
|
|
CP0392151
|
N,N-dimethyl-2-[3-(1-pyridin-2-ylbutyl)-1H-inden-2-yl]ethanamine
Show/Hide
|
C22H28N2
|
1
|
| 1 |
Ki = 245.47 nM
|
|
|
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CP0380480
|
(2R,3S)-5-[3-[[4-methyl-5-(oxan-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptane
Show/Hide
|
C24H31F3N4OS
|
1
|
| 1 |
Ki = 251.19 nM
|
|
|
|
CP0300572
|
3-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]benzamide
Show/Hide
|
C26H28F3N5OS
|
1
|
| 1 |
Ki = 263.03 nM
|
|
|
|
CP0220610
|
Bietamiverine
Show/Hide
|
C19H30N2O2
|
1
|
| 1 |
Ki = 271 nM
|
|
|
|
CP0418483
|
2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H25NO3
|
1
|
| 1 |
Ki = 290 nM
|
|
|
|
CP0398327
|
1-methyl-4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]pyridin-2-one
Show/Hide
|
C25H28F3N5OS
|
1
|
| 1 |
Ki = 302 nM
|
|
|
|
CP0481591
|
(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(3,4-Dihydro-1H-isoquinolin-2-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C25H35NO2
|
1
|
| 1 |
Ki = 304 nM
|
|
|
|
CP0380644
|
4-methyl-5-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-oxazole
Show/Hide
|
C23H26F3N5OS
|
1
|
| 1 |
Ki = 309.03 nM
|
|
|
|
CP0467583
|
(3S,3aR,4R,4aS,8aR,9aS)-4-(3-[1,4']Bipiperidinyl-1'-yl-propyl)-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C26H44N2O2
|
1
|
| 1 |
Ki = 312 nM
|
|
|
|
CP0398324
|
5-[5-[3-[(2R,3R)-2-[2-fluoro-4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
Show/Hide
|
C23H25F4N5OS
|
1
|
| 1 |
Ki = 323.59 nM
|
|
|
|
CP0425885
|
2-(3-fluorophenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C21H22FNO2
|
1
|
| 1 |
Ki = 330 nM
|
|
|
|
CP0397929
|
2-[5-fluoro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C20H23FN2
|
1
|
| 1 |
Ki = 331.13 nM
|
|
|
|
CP0507911
|
2-(4-methylsulfanylphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C22H25NO2S
|
1
|
| 1 |
Ki = 340 nM
|
|
|
|
CP0399359
|
(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(2-Ethyl-piperidin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C23H39NO2
|
1
|
| 1 |
Ki = 341 nM
|
|
|
|
CP0403738
|
2-[5-chloro-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C20H23ClN2
|
1
|
| 1 |
Ki = 346.74 nM
|
|
|
|
CP0381564
|
(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(2,5-Dimethyl-piperazin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C22H38N2O2
|
1
|
| 1 |
Ki = 353 nM
|
|
|
|
CP0425827
|
2-pyridin-4-ylethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
Ki = 370 nM
|
|
|
|
CP0398322
|
4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-3H-pyridin-2-one
Show/Hide
|
C24H26F3N5OS
|
1
|
| 1 |
Ki = 371.54 nM
|
|
|
|
CP0378379
|
(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(3-methyl-piperidin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C22H37NO2
|
1
|
| 1 |
Ki = 376 nM
|
|
|
|
CP0122473
|
1-methyl-5-[4-methyl-5-[3-[1-[4-(trifluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]pyridin-2-one
Show/Hide
|
C25H29F3N6OS
|
1
|
| 1 |
Ki = 380.19 nM
|
|
|
|
CP0386736
|
[(3R)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
|
C24H27NO4
|
1
|
| 1 |
Ki = 380.19 nM
|
|
|
|
CP0398329
|
5-[5-[3-[(2S,3R)-2-[4-fluoro-2-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
Show/Hide
|
C23H25F4N5OS
|
1
|
| 1 |
Ki = 389.05 nM
|
|
|
|
CP0441004
|
(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(2-methyl-piperidin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C22H37NO2
|
1
|
| 1 |
Ki = 399 nM
|
|
|
|
CP0418484
|
2-pyridin-2-ylethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
Ki = 410 nM
|
|
|
|
CP0466978
|
(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(3,3-Dimethyl-piperidin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C23H39NO2
|
1
|
| 1 |
Ki = 416 nM
|
|
|
|
CP0851168
|
DIPHENIDOL HYDROCHLORIDE
Show/Hide
|
C21H28ClNO
|
1
|
| 1 |
Ki = 426.58 nM
|
|
|
|
CP0428746
|
(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-(3-piperidin-1-yl-propyl)-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C21H35NO2
|
1
|
| 1 |
Ki = 427 nM
|
|
|
|
CP0524558
|
4-[3-((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-1-oxo-dodecahydro-naphtho[2,3-c]furan-4-yl)-propyl]-piperazine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C25H42N2O4
|
1
|
| 1 |
Ki = 445 nM
|
|
|
|
CP0372479
|
N,N-diethyl-2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
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C22H28N2
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1
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| 1 |
Ki = 446.68 nM
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CP0398326
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4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]benzamide
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C26H28F3N5OS
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1
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| 1 |
Ki = 457.09 nM
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CP0437729
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(4-Cyclohexyl-piperazin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C26H44N2O2
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1
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| 1 |
Ki = 464 nM
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CP0488918
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2-(3-methoxyphenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C23H27NO3
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1
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| 1 |
Ki = 470 nM
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CP0458157
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4-methyl-5-[4-methyl-5-[3-[(2S,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-oxazole
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C23H26F3N5OS
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1
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| 1 |
Ki = 478.63 nM
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CP0134104
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5-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-3H-pyridin-2-one
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C24H26F3N5OS
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1
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| 1 |
Ki = 489.78 nM
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CP0516426
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[(2R,5R,6R)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C20H26INO2
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1
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| 1 |
Ki = 501.19 nM
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CP0507905
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2-(4-methylsulfonylphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C22H25NO4S
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1
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| 1 |
Ki = 510 nM
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CP0420595
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6-methyl-5-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]pyridine-2-carboxamide
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C26H29F3N6OS
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1
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| 1 |
Ki = 512.86 nM
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CP0156301
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2-(diethylamino)ethyl 2-(4-chlorophenyl)sulfanylbenzoate
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C19H22ClNO2S
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1
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| 1 |
Ki = 519 nM
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CP0487384
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[(2R,5R)-5-benzhydryl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C21H28INO2
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1
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| 1 |
Ki = 524.81 nM
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CP0487380
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trimethyl-[[(2R,5S)-5,6,6-triphenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
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C26H30INO2
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1
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| 1 |
Ki = 549.54 nM
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CP0437730
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(4-methyl-piperidin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H37NO2
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1
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| 1 |
Ki = 554 nM
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CP0481480
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2-(4-chlorophenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C22H24ClNO2
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1
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| 1 |
Ki = 560 nM
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CP0441146
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N,N-dimethyl-2-[6-methyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C21H26N2
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1
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| 1 |
Ki = 562.34 nM
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CP0445692
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5-[5-[3-[(2S,3S)-2-[4-fluoro-2-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-4-methyl-1,2,4-triazol-3-yl]-4-methyl-1,3-oxazole
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C23H25F4N5OS
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1
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| 1 |
Ki = 562.34 nM
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CP0432842
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-(4-methyl-piperazin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
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C21H36N2O2
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1
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| 1 |
Ki = 579 nM
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CP0392927
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-((S)-3-methyl-piperazin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C21H36N2O2
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1
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| 1 |
Ki = 581 nM
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CP0493835
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(2,6-Dimethyl-morpholin-4-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H37NO3
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1
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| 1 |
Ki = 601 nM
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CP0436507
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N-(2-fluoroethyl)-N-methyl-2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
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C21H25FN2
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1
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| 1 |
Ki = 602.56 nM
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CP0851172
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4-(4-hydroxy-4,4-diphenylbutyl)piperazine-1,4-diium dichloride
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C20H28Cl2N2O
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1
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| 1 |
Ki = 602.56 nM
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CP0851174
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1-(4-hydroxy-4,4-diphenylbutyl)-4-[1-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperidin-1-ium-4-yl]-1-methylpiperidin-1-ium diiodide
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C44H58I2N2O2
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1
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| 1 |
Ki = 602.56 nM
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CP0317889
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5-[3-[(4-methyl-5-pyridin-3-yl-1,2,4-triazol-3-yl)sulfanyl]propyl]-1-[2-(trifluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrole
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C24H27F3N6S
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1
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| 1 |
Ki = 630.96 nM
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CP0386734
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[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-2-methyl-6,6-diphenyl-1,4-dioxane-2-carboxylate
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C25H29NO4
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1
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| 1 |
Ki = 660.69 nM
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CP0179022
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2-[4-[4-methyl-5-[3-[(2R,3S)-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]phenyl]-1,3-oxazole
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C28H28F3N5OS
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1
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| 1 |
Ki = 676.08 nM
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CP0479714
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trimethyl-[[(2R,5R)-5,6,6-triphenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
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C26H30INO2
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1
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| 1 |
Ki = 676.08 nM
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CP0237860
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4-methyl-5-[4-methyl-5-[3-[(2S,3R)-2-phenyl-5-azaspiro[2.4]heptan-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-oxazole
Show/Hide
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C22H27N5OS
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1
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| 1 |
Ki = 741.31 nM
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CP0851169
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1-(4-hydroxy-4,4-diphenylbutyl)-4-[1-(4-hydroxy-4,4-diphenylbutyl)piperidin-1-ium-4-yl]piperidin-1-ium dichloride
Show/Hide
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C42H54Cl2N2O2
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1
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| 1 |
Ki = 794.33 nM
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CP0425890
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2-(4-nitrophenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C22H24N2O4
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1
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| 1 |
Ki = 810 nM
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CP0473022
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[(2R,5S)-5-benzhydryl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
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C21H28INO2
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1
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| 1 |
Ki = 831.76 nM
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CP0441685
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[3-((R)-3-methyl-piperazin-1-yl)-propyl]-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C21H36N2O2
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1
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| 1 |
Ki = 857 nM
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CP0406408
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N,N-dimethyl-2-[5-methylsulfanyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C21H26N2S
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1
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| 1 |
Ki = 870.96 nM
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CP0449839
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N-methyl-N-[2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethyl]propan-2-amine
Show/Hide
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C22H28N2
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1
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| 1 |
Ki = 870.96 nM
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CP0425886
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2-(3-methylphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C22H25NO2
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1
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| 1 |
Ki = 880 nM
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CP0372485
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N,N-dimethyl-3-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]propan-1-amine
Show/Hide
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C21H26N2
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1
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| 1 |
Ki = 891.25 nM
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CP0464098
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3-(2,3-dihydro-1-benzofuran-5-yl)propyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C24H27NO3
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1
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| 1 |
Ki = 920 nM
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CP0468678
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2-[di(propan-2-yl)amino]ethyl 2-hydroxy-2,2-diphenylacetate
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C22H29NO3
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1
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| 1 |
Ki = 971 nM
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CP0066235
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4-methyl-5-[4-methyl-5-[3-(1-phenyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl)propylsulfanyl]-1,2,4-triazol-3-yl]-1,3-oxazole
Show/Hide
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C22H28N6OS
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1
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| 1 |
Ki = 1000 nM
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CP0364090
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5-[3-[[4-methyl-5-(oxan-4-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-1-phenyl-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrole
Show/Hide
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C23H33N5OS
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1
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| 1 |
Ki = 1023.29 nM
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CP0466831
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3-methylbut-2-enyl 2-[2-(diethylamino)ethylsulfanyl]-2-phenylacetate
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C19H29NO2S
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1
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| 1 |
Ki = 1040 nM
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CP0372523
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2-[1-[2-(2-pyrrolidin-1-ylethyl)-3H-inden-1-yl]ethyl]pyridine
Show/Hide
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C22H26N2
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1
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| 1 |
Ki = 1047.13 nM
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CP0479764
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N-[3-[1-[2-(8-chloro-6-oxo-5H-pyrido[2,3-b][1,4]benzodiazepin-11-yl)-2-oxoethyl]piperidin-4-yl]propyl]-N-ethyl-2,2-dimethylpentanamide
Show/Hide
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C31H42ClN5O3
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1
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| 1 |
Ki = 1071.52 nM
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CP0862110
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N1,N3-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N3-dimethylpropane-1,3-diaminium chloride
Show/Hide
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C37H48Cl2N2O2
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1
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| 1 |
Ki = 1348.96 nM
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CP0490487
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(3,5-Dimethyl-piperazin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C22H38N2O2
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1
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| 1 |
Ki = 1361 nM
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CP0484746
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C24H27NO3
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1
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| 1 |
Ki = 1390 nM
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CP0437455
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[(2R,5S,6S)-5,6-diphenyl-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki = 1412.54 nM
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CP0381409
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11-[2-[(4aS,8aR)-4-methyl-2,3,4a,5,6,7,8,8a-octahydroquinoxalin-1-yl]acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
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C23H27N5O2
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1
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| 1 |
Ki = 1445.44 nM
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CP0455460
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(3-Hydroxy-piperidin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C21H35NO3
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1
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| 1 |
Ki = 1533 nM
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CP0372477
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2-[6-methoxy-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
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C21H26N2O
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1
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| 1 |
Ki = 1548.82 nM
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CP0397931
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N,N-dimethyl-2-[3-(pyridin-2-ylmethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C19H22N2
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1
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| 1 |
Ki = 1584.89 nM
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CP0492466
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N,N-dimethyl-2-[5-methyl-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C21H26N2
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1
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| 1 |
Ki = 1621.81 nM
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CP0420656
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(2R,3S)-5-[3-[[4-methyl-5-(2-methylpyridin-3-yl)-1,2,4-triazol-3-yl]sulfanyl]propyl]-2-[4-(trifluoromethyl)phenyl]-5-azaspiro[2.4]heptane
Show/Hide
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C25H28F3N5S
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1
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| 1 |
Ki = 1659.59 nM
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CP0386732
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[(3S)-1-azabicyclo[2.2.2]octan-3-yl] (2S)-6,6-diphenyl-1,4-dioxane-2-carboxylate
Show/Hide
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C24H27NO4
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1
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| 1 |
Ki = 1698.24 nM
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CP0489883
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2-(2-methoxyphenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H27NO3
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1
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| 1 |
Ki = 1730 nM
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CP0404647
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4-[4-methyl-5-[3-[1-[4-(trifluoromethyl)phenyl]-2,3,3a,4,6,6a-hexahydropyrrolo[2,3-c]pyrrol-5-yl]propylsulfanyl]-1,2,4-triazol-3-yl]-1H-pyridin-2-one
Show/Hide
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C24H27F3N6OS
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1
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| 1 |
Ki = 1737.8 nM
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CP0139209
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N,N-dimethyl-2-[3-[(1R)-1-pyridin-2-ylethyl]-1H-inden-2-yl]ethanamine
Show/Hide
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C20H24N2
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1
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| 1 |
Ki = 1862.09 nM
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CP0372527
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2-[1-[2-(2-piperidin-1-ylethyl)-3H-inden-1-yl]ethyl]pyridine
Show/Hide
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C23H28N2
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1
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| 1 |
Ki = 1905.46 nM
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CP0139207
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9-Methoxy-2-methyl-11,12-dihydro-3H,6aH,13H-6-oxa-3,12a-diaza-benzo[a]cyclopenta[h]anthracene-1-carboxylic acid ethyl ester
Show/Hide
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C23H24N2O4
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1
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| 1 |
Ki = 2290.87 nM
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CP0381581
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11-[2-[(4aR,8aR)-4-methyl-2,3,4a,5,6,7,8,8a-octahydroquinoxalin-1-yl]acetyl]-5H-pyrido[2,3-b][1,4]benzodiazepin-6-one
Show/Hide
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C23H27N5O2
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1
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| 1 |
Ki = 2290.87 nM
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CP0479717
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trimethyl-[[(2R,5R)-5-phenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C14H22INO2
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1
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| 1 |
Ki = 2344.23 nM
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CP0425828
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 4-(3-methoxyphenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C24H27NO4
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1
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| 1 |
Ki = 2430 nM
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CP0473017
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trimethyl-[[(2R,5S)-5-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2S
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1
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| 1 |
Ki = 2691.53 nM
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CP0476763
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2-(4-methoxy-3-methylphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H27NO3
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1
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| 1 |
Ki = 2700 nM
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CP0875550
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4-(4-Hydroxy-4,4-diphenyl-butyl)-1,1-dimethyl-piperazin-1-ium iodide
Show/Hide
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C22H31IN2O
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1
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| 1 |
Ki = 2951.21 nM
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CP0470619
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(4-methoxyphenyl)methyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C22H25NO3
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1
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| 1 |
Ki = 3060 nM
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CP0472770
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trimethyl-[[(2R,6R)-6-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2S
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1
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| 1 |
Ki = 3090.3 nM
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CP0472769
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trimethyl-[[(2R,6S)-6-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2S
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1
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| 1 |
Ki = 3162.28 nM
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CP0425883
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3-(4-methoxyphenyl)propyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C24H29NO3
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1
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| 1 |
Ki = 3290 nM
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CP0424269
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2-(dimethylamino)ethyl 3-(pyridin-3-ylmethyl)-1H-indene-2-carboxylate
Show/Hide
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C20H22N2O2
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1
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| 1 |
Ki = 3548.13 nM
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CP0399353
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N,N-dimethyl-2-[3-(pyridin-3-ylmethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C19H22N2
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1
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| 1 |
Ki = 3715.35 nM
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CP0403766
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2-[5-methoxy-3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]-N,N-dimethylethanamine
Show/Hide
|
C21H26N2O
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1
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| 1 |
Ki = 3715.35 nM
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CP0472768
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trimethyl-[[(2R,5R)-5-(4-phenylsulfanylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
|
C20H26INO2S
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1
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| 1 |
Ki = 3715.35 nM
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CP0505786
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N,N-dimethyl-2-[3-(pyridin-4-ylmethyl)-1H-inden-2-yl]ethanamine
Show/Hide
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C19H22N2
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1
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| 1 |
Ki = 4265.8 nM
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CP0404155
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4-[2-[3-(1-pyridin-2-ylethyl)-1H-inden-2-yl]ethyl]morpholine
Show/Hide
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C22H26N2O
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1
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| 1 |
Ki = 4365.16 nM
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CP0479720
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[(2R,6R)-6-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO4S
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1
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| 1 |
Ki = 5128.61 nM
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CP0425882
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 4-(2-fluorophenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H24FNO3
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1
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| 1 |
Ki = 5270 nM
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CP0404384
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2-(dimethylamino)ethyl 3-(pyridin-2-ylmethyl)-1H-indene-2-carboxylate
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C20H22N2O2
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1
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| 1 |
Ki = 5370.32 nM
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CP0471232
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4-(4-methoxyphenyl)butyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
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C24H29NO3
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1
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| 1 |
Ki = 5400 nM
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CP0862120
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1-(4-hydroxy-4,4-diphenylbutyl)-4-(1-methylpiperidin-1-ium-4-yl)piperidin-1-ium dichloride
Show/Hide
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C27H40Cl2N2O
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1
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| 1 |
Ki = 5754.4 nM
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CP0425891
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2-(3,4-dimethoxyphenyl)ethyl 1-methyl-5-phenyl-3,6-dihydro-2H-pyridine-4-carboxylate
Show/Hide
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C23H27NO4
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1
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| 1 |
Ki = 6160 nM
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CP0425826
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2-(4-methoxyphenoxy)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C22H25NO4
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1
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| 1 |
Ki = 6190 nM
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CP0479629
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[(2R,5S)-5-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO3S
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1
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| 1 |
Ki = 6760.83 nM
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CP0479715
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[(2R,6R)-6-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO3S
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1
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| 1 |
Ki = 6760.83 nM
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CP0862114
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1,4-Bis-(4-hydroxy-4,4-diphenyl-butyl)-1-methyl-piperazin-1-ium iodide
Show/Hide
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C37H45IN2O2
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1
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| 1 |
Ki = 7079.46 nM
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CP0862121
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N1,N3-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N1,N3,N3-tetramethylpropane-1,3-diaminium iodide
Show/Hide
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C39H52I2N2O2
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1
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| 1 |
Ki = 7244.36 nM
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CP0851171
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4-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperazine-1,4-diium dichloride
Show/Hide
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C21H30Cl2N2O
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1
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| 1 |
Ki = 7762.47 nM
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CP0464077
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-ethyl-4-(4-fluorophenyl)-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C24H26FNO3
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1
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| 1 |
Ki = 7900 nM
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CP0851569
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1-(3,5-dichlorophenyl)piperazine
Show/Hide
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C10H12Cl2N2
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1
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| 1 |
Ki = 7943.28 nM
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CP0913741
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4-(1,1-dimethylpiperidin-1-ium-4-yl)-1-(4-hydroxy-4,4-diphenylbutyl)-1-methylpiperidin-1-ium diiodide
Show/Hide
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C29H44I2N2O
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1
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| 1 |
Ki = 8317.64 nM
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CP0479708
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[(2R,6S)-6-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO4S
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1
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| 1 |
Ki = 8317.64 nM
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CP0464076
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 4-(2-methoxyphenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C24H27NO4
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1
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| 1 |
Ki = 8350 nM
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CP0387007
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[(2R,5S)-5-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO4S
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1
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| 1 |
Ki > 10000 nM
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CP0421082
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trimethyl-[[(2R,5S)-5-phenyl-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C14H22INO2
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1
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| 1 |
Ki > 10000 nM
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CP0473016
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[(2R,5S)-5-(4-benzylphenyl)-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C21H28INO2
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1
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| 1 |
Ki > 10000 nM
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CP0473018
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[(2R,5R)-5-[4-(benzenesulfonyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO4S
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1
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| 1 |
Ki > 10000 nM
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CP0479627
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trimethyl-[[(2R,5S)-5-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0479628
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trimethyl-[[(2R,5R)-5-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0479654
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trimethyl-[[(2R,6R)-6-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0479711
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trimethyl-[[(2R,6S)-6-(4-phenylphenyl)-1,4-dioxan-2-yl]methyl]azanium;iodide
Show/Hide
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C20H26INO2
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1
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| 1 |
Ki > 10000 nM
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CP0487382
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[(2R,5R)-5-(4-benzylphenyl)-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C21H28INO2
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1
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| 1 |
Ki > 10000 nM
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CP0491695
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[(2R,6S)-6-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO3S
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1
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| 1 |
Ki > 10000 nM
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CP0516423
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[(2R,5R)-5-[4-(benzenesulfinyl)phenyl]-1,4-dioxan-2-yl]methyl-trimethylazanium;iodide
Show/Hide
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C20H26INO3S
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1
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| 1 |
Ki > 10000 nM
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CP0464101
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2-(3-fluoro-4-methoxyphenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H26FNO3
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1
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| 1 |
Ki = 11700 nM
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CP0404254
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N-[2-(dimethylamino)ethyl]-3-(pyridin-2-ylmethyl)-1H-indene-2-carboxamide
Show/Hide
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C20H23N3O
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1
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| 1 |
Ki = 16218.1 nM
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CP0851173
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1-(4-Hydroxy-4,4-diphenyl-butyl)-1-methyl-4-phenyl-piperazin-1-ium iodide
Show/Hide
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C27H33IN2O
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1
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| 1 |
Ki = 17378.01 nM
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CP0069240
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4-(piperazin-1-yl)-1H-indole
Show/Hide
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C12H15N3
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1
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| 1 |
Ki > 19952.62 nM
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CP0184743
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4-methyl-2-piperazin-1-ylquinoline
Show/Hide
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C14H17N3
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1
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| 1 |
Ki > 19952.62 nM
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CP0364794
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1-(2,3-dichlorophenyl)piperazine
Show/Hide
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C10H12Cl2N2
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1
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| 1 |
Ki > 19952.62 nM
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CP0418482
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2-naphthalen-1-ylethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C25H25NO2
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1
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| 1 |
Ki = 24400 nM
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CP0425884
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2-(3,4-dimethoxyphenyl)ethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H27NO4
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1
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| 1 |
Ki = 25300 nM
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CP0862112
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N1,N2-bis(4-hydroxy-4,4-diphenylbutyl)-N1,N1,N2,N2-tetramethylethane-1,2-diaminium iodide
Show/Hide
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C38H50I2N2O2
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1
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| 1 |
Ki = 26302.68 nM
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CP0471231
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2-(3,4-dimethoxyphenyl)ethyl 4-(3-fluorophenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H26FNO4
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1
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| 1 |
Ki = 27000 nM
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CP0416829
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N-[2-(dimethylamino)ethyl]-3-(pyridin-3-ylmethyl)-1H-indene-2-carboxamide
Show/Hide
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C20H23N3O
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1
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| 1 |
Ki = 48977.88 nM
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CP0375776
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N-[2-(dimethylamino)ethyl]-3-(pyridin-4-ylmethyl)-1H-indene-2-carboxamide
Show/Hide
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C20H23N3O
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1
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| 1 |
Ki = 53703.18 nM
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CP0425887
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ethyl 1-[1-(2,6-dichlorobenzoyl)piperidin-4-yl]-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C26H28Cl2N2O3
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1
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| 1 |
Ki > 100000 nM
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CP0425888
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ethyl 1-[2-(1,3-benzodioxol-5-yl)ethyl]-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H25NO4
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1
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| 1 |
Ki > 100000 nM
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CP0425889
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 4-(3-fluorophenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H24FNO3
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1
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| 1 |
Ki > 100000 nM
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CP0434325
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ethyl 1-[1-(2,6-dimethylbenzoyl)piperidin-4-yl]-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C28H34N2O3
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1
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| 1 |
Ki > 100000 nM
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CP0449730
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2,3-dihydro-1-benzofuran-5-ylmethyl 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C22H23NO3
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1
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| 1 |
Ki > 100000 nM
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CP0464075
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ethyl 1-[2-(4-methoxyphenyl)ethyl]-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C23H27NO3
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1
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| 1 |
Ki > 100000 nM
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CP0471233
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 2-(1-methyl-3,6-dihydro-2H-pyridin-4-yl)benzoate
Show/Hide
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C23H25NO3
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1
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| 1 |
Ki > 100000 nM
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CP0471234
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ethyl 1-[2-(2,3-dihydro-1-benzofuran-5-yl)ethyl]-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C24H27NO3
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1
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| 1 |
Ki > 100000 nM
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CP0476764
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[(2S)-1-(4-methoxyphenyl)propan-2-yl] 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C24H29NO3
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1
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| 1 |
Ki > 100000 nM
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CP0476765
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2-(3,4-dimethoxyphenyl)ethyl 4-(2-fluorophenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H26FNO4
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1
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| 1 |
Ki > 100000 nM
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CP0476766
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 1-butyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C26H31NO3
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1
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| 1 |
Ki > 100000 nM
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CP0476767
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2-(4-methoxyphenyl)ethyl 1-[(4-methoxyphenyl)methyl]-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C29H31NO4
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1
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| 1 |
Ki > 100000 nM
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CP0484745
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2-(3,4,5-trimethoxyphenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C25H31NO5
|
1
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| 1 |
Ki > 100000 nM
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CP0488904
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ethyl 1-[1-(4-methylphenyl)sulfonylpiperidin-4-yl]-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
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C26H32N2O4S
|
1
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| 1 |
Ki > 100000 nM
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CP0488906
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ethyl 4-phenyl-1-(2-phenylethyl)-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C22H25NO2
|
1
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| 1 |
Ki > 100000 nM
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CP0488907
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2-(3,4-dimethoxyphenyl)ethyl 4-(2-methoxyphenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C24H29NO5
|
1
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| 1 |
Ki > 100000 nM
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CP0488908
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2-(4-methoxyphenyl)ethyl 1-butyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C25H31NO3
|
1
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| 1 |
Ki > 100000 nM
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CP0488929
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2-(4-methoxyphenyl)ethyl 4-phenyl-1-propyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C24H29NO3
|
1
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| 1 |
Ki > 100000 nM
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CP0507910
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2-(2,4,6-trimethylphenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C25H31NO2
|
1
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| 1 |
Ki > 100000 nM
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CP0511553
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2-(4-methylsulfonylphenyl)ethyl 1-ethyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C23H27NO4S
|
1
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| 1 |
Ki > 100000 nM
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CP0515836
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2-(2,3-dihydro-1-benzofuran-5-yl)ethyl 4-phenyl-1-propyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C25H29NO3
|
1
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| 1 |
Ki > 100000 nM
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CP0521680
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2-(3,4-dimethoxyphenyl)ethyl 4-(3-methoxyphenyl)-1-methyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C24H29NO5
|
1
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| 1 |
Ki > 100000 nM
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CP0521681
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(2-methoxy-2-phenylethyl) 1-methyl-4-phenyl-3,6-dihydro-2H-pyridine-5-carboxylate
Show/Hide
|
C22H25NO3
|
1
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| 1 |
Ki > 100000 nM
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CP0406685
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(3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-(3-piperazin-1-yl-propyl)-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
|
C20H34N2O2
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1
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| 1 |
Ki > 420 nM
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CP0392943
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(3S,3aR,4R,4aS,8aR,9aS)-4-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-3-methyl-decahydro-naphtho[2,3-c]furan-1-one
Show/Hide
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C21H35NO3
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1
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| 1 |
Ki > 900 nM
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