US10717746, Example 51

N,N-dimethyl-2-[4-[4-(2-methyl-3-propan-2-ylbenzimidazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

(1S,3R)-3-acetamido-N-[5-chloro-4-(5,5-dimethyl-4,6-dihydropyrrolo[1,2-b]pyrazol-3-yl)pyridin-2-yl]cyclohexane-1-carboxamide

N,N-dimethyl-2-[4-[4-(6-oxo-1-propan-2-ylpyridazin-3-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

1-propan-2-yl-5-[2-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-2-one

US10717746, Example 25

N,N-dimethyl-2-[4-[4-(6-oxo-1-propan-2-ylpyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

2-[4-[4-(4-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]-N,N-dimethylacetamide

US9073922, 18

US10717746, Example 22

US10717746, Example 48

US10717746, Example 47

US10717746, Example 27

2-[4-[4-(4-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]ethanol

US10717746, Example 44

N,N-dimethyl-2-[4-[4-[1-(2-methylsulfanylethyl)-6-oxopyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

5-[2-[1-(2-oxo-2-piperidin-1-ylethyl)piperidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-propan-2-ylpyridin-2-one

US9073922, 29

5-[2-[1-(2-oxo-2-pyrrolidin-1-ylethyl)piperidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-propan-2-ylpyridin-2-one

US10717746, Example 66

N-methyl-2-[4-[4-(6-oxo-1-propan-2-ylpyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

US10717746, Example 63

US10717746, Example 2

5-[2-[1-(2,2-difluoroethyl)piperidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-propan-2-ylpyridin-2-one

5-(2-piperidin-4-yl-1H-pyrrolo[2,3-b]pyridin-4-yl)-1-propan-2-ylpyridin-2-one

US9067888, 33

[4-[2-[1-(2-hydroxyethyl)piperidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-4-yl]-3-methoxyphenyl]-pyrrolidin-1-ylmethanone

(1S,3R)-3-acetamido-N-(5-chloro-4-pyrazolo[1,5-a]pyridin-3-ylpyridin-2-yl)cyclohexane-1-carboxamide

4-[[4-[4-(4-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]phenyl]methyl]morpholine

US10717746, Example 39

US10717746, Example 16

US10717746, Example 82

[3-methoxy-4-(2-piperidin-4-yl-1H-pyrrolo[2,3-b]pyridin-4-yl)phenyl]-pyrrolidin-1-ylmethanone

US10717746, Example 43

1-[4-[4-(4-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]ethanone

US10717746, Example 8

5-[2-(1-acetylpiperidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1-propan-2-ylpyridin-2-one

2-[4-[4-(1-cyclobutyl-6-oxopyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]-N,N-dimethylacetamide

1-[4-[4-[2-methoxy-4-(pyrrolidine-1-carbonyl)phenyl]-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]ethanone

(1S,3R)-3-acetamido-N-[5-chloro-4-(1,5-dimethylpyrazol-4-yl)pyridin-2-yl]cyclohexane-1-carboxamide

US10717746, Example 3

US10717746, Example 10

N-[4-[4-(4-fluoro-2-methoxyphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]cyclohexyl]acetamide

N,N-dimethyl-2-[4-[4-[1-(2-methylpropyl)-6-oxopyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

N,N-dimethyl-2-[4-[4-(2-oxo-1-propan-2-ylpyrimidin-5-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

[3-methoxy-4-[2-(oxan-4-yl)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenyl]-pyrrolidin-1-ylmethanone

US10717746, Example 78

US10717746, Example 12

US10717746, Example 13

US10717746, Example 15

(1S,3R)-3-acetamido-N-[4-(2-methyl-3-propan-2-ylimidazol-4-yl)pyridin-2-yl]cyclohexane-1-carboxamide

2-[4-[4-(1-ethyl-6-oxopyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]-N,N-dimethylacetamide

2-[4-[4-[1-(2-methoxyethyl)-6-oxopyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]-N,N-dimethylacetamide

4-(4-fluoro-2-methoxyphenyl)-2-(oxan-4-yl)-1H-pyrrolo[2,3-b]pyridine

US10717746, Example 7

[3-methoxy-4-[2-[4-(morpholin-4-ylmethyl)phenyl]-1H-imidazo[4,5-b]pyridin-7-yl]phenyl]-pyrrolidin-1-ylmethanone

(1S,3R)-3-acetamido-N-(5-chloro-4-imidazo[1,2-a]pyridin-3-ylpyridin-2-yl)cyclohexane-1-carboxamide

US10717746, Example 11

(1S,3R)-3-acetamido-N-(5-chloro-4-(5-(4-hydroxybutyl)-1H-pyrazol-4-yl)pyridin-2-yl)cyclohexanecarboxamide

(1S,3R)-3-acetamido-N-(5-chloro-4-(5-(3-hydroxy-2,2-dimethylpropyl)-1H-pyrazol-4-yl)pyridin-2-yl)cyclohexanecarboxamide

(1S,3R)-3-acetamido-N-[5-chloro-4-(triazolo[1,5-a]pyridin-3-yl)pyridin-2-yl]cyclohexane-1-carboxamide

(1S,3R)-3-acetamido-N-[5-chloro-4-(2,3-dimethylimidazol-4-yl)pyridin-2-yl]cyclohexane-1-carboxamide

N,N-dimethyl-2-[4-[4-[1-(oxan-4-ylmethyl)-6-oxopyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

N,N-dimethyl-2-[4-[4-(1-methyl-6-oxopyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

N,N-dimethyl-2-[4-[4-[1-[2-(oxan-4-yl)ethyl]-6-oxopyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

N,N-dimethyl-2-[4-[4-[1-(oxan-4-yl)-6-oxopyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]acetamide

2-[4-[4-(4-methoxy-1-methyl-6-oxopyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-2-yl]piperidin-1-yl]-N,N-dimethylacetamide