Compound ID |
Compound Name |
Compound Formula |
CP0073076
|
(2R)-2-[5-[6-amino-5-[(1R)-1-[5-fluoro-2-(triazol-2-yl)phenyl]ethoxy]pyridin-3-yl]-4-methyl-1,3-thiazol-2-yl]propane-1,2-diol
Show/Hide
|
C22H23FN6O3S
|
3
|
1 |
IC50 = 1.3 nM
|
|
|
2 |
IC50 = 21 nM
|
|
|
3 |
IC50 = 24 nM
|
|
|
CP0054448
|
6,6-dimethyl-8-[1-(oxan-4-ylmethyl)piperidin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile
Show/Hide
|
C30H33N3O2
|
1
|
1 |
IC50 = 17.9 nM
|
|
|
CP0066933
|
1256580-46-7
Show/Hide
|
C30H34N4O2
|
1
|
1 |
IC50 = 19 nM
|
|
|
CP0199533
|
9-ethyl-6,6-dimethyl-8-[1-(oxan-4-ylmethyl)-3,6-dihydro-2H-pyridin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile
Show/Hide
|
C32H35N3O2
|
1
|
1 |
IC50 = 49 nM
|
|
|
CP0059911
|
2-[[5-chloro-2-[[(6S)-6-[4-(2-hydroxyethyl)piperazin-1-yl]-1-methoxy-6,7,8,9-tetrahydro-5H-benzo[7]annulen-2-yl]amino]pyrimidin-4-yl]amino]-N-methylbenzamide
Show/Hide
|
C30H38ClN7O3
|
1
|
1 |
IC50 = 85 nM
|
|
|
CP0031719
|
(R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1-(piperidin-4-yl)-1H-pyrazol-4-yl)pyridin-2-amine
Show/Hide
|
C21H22Cl2FN5O
|
4
|
1 |
IC50 = 108 nM
|
|
|
2 |
IC50 = 261 nM
|
|
|
3 |
IC50 = 623 nM
|
|
|
4 |
IC50 = 838 nM
|
|
|
CP0095494
|
9-ethyl-6,6-dimethyl-8-[1-(oxane-4-carbonyl)-3,6-dihydro-2H-pyridin-4-yl]-11-oxo-5H-benzo[b]carbazole-3-carbonitrile
Show/Hide
|
C32H33N3O3
|
1
|
1 |
IC50 = 126 nM
|
|
|