| Compound ID |
Compound Name |
Compound Formula |
|
CP0271903
|
(S)-1-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-5-(2-((pyridin-3-yloxy)methyl)pyrrolidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C23H23FN6O5S
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0050269
|
(S)-1-(4-(2-fluoroethoxy)benzyl)-5-(2-((pyridin-3-yloxy)methyl)azetidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C26H24FN3O6S
|
1
|
| 1 |
EC50 = 380 nM
|
|
|
|
CP0036627
|
(S)-1-(4-(2-fluoroethoxy)benzyl)-5-(2-((pyridin-3-yloxy)methyl)pyrrolidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C27H26FN3O6S
|
1
|
| 1 |
EC50 = 390 nM
|
|
|
|
CP0297684
|
(S)-1-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-5-(2-((pyridin-3-yloxy)methyl)azetidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C22H21FN6O5S
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0050270
|
(S)-1-(4-methoxybenzyl)-5-(2-((pyridin-3-yloxy)methyl)azetidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C25H23N3O6S
|
1
|
| 1 |
EC50 = 450 nM
|
|
|
|
CP0202684
|
1-(4-Methoxybenzyl)-5-(2-(pyridin-3-yl-oxymethyl)-pyrolidine-1-sulfonyl)-1H-indole-2,3-dione
Show/Hide
|
C26H25N3O6S
|
1
|
| 1 |
EC50 = 450 nM
|
|
|
|
CP0166997
|
1-Benzyl-5-(2-(pyridin-3-yl-oxymethyl)-pyrrolidine-1-sulfonyl)-1H-indole-2,3-dione
Show/Hide
|
C25H23N3O5S
|
1
|
| 1 |
EC50 = 650 nM
|
|
|
|
CP0050273
|
(S)-1-((1-(2-Fluoroethyl)-1H-[1,2,3]-triazol-4-yl)methyl)-5-(2(2,4-difluorophenoxymethyl)-pyrrolidine-1-sulfonyl)isatin
Show/Hide
|
C24H22F3N5O5S
|
1
|
| 1 |
EC50 = 680 nM
|
|
|
|
CP0050278
|
(S)-1-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)-5-(2-(phenoxymethyl)azetidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C23H22FN5O5S
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0138925
|
(S)-1-((1-(2-Fluoroethyl)-1H-[1,2,3]-triazol-4-yl)methyl)-5-(2-phenoxymethyl-pyrrolidine-1-sulfonyl)isatin
Show/Hide
|
C24H24FN5O5S
|
1
|
| 1 |
EC50 = 930 nM
|
|
|
|
CP0050282
|
(S)-5-(2-((2,4-difluorophenoxy)methyl)azetidin-1-ylsulfonyl)-1-((1-(2-fluoroethyl)-1H-1,2,3-triazol-4-yl)methyl)indoline-2,3-dione
Show/Hide
|
C23H20F3N5O5S
|
1
|
| 1 |
EC50 = 1060 nM
|
|
|
|
CP0050272
|
(S)-1-(4-(2-(2-(2-fluoroethoxy)ethoxy)ethoxy)benzyl)-5-(2-(phenoxymethyl)pyrrolidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C32H35FN2O8S
|
1
|
| 1 |
EC50 = 1300 nM
|
|
|
|
CP0050280
|
(S)-5-(2-((2,4-difluorophenoxy)methyl)azetidin-1-ylsulfonyl)-1-(4-(2-fluoroethoxy)benzyl)indoline-2,3-dione
Show/Hide
|
C27H23F3N2O6S
|
1
|
| 1 |
EC50 = 1390 nM
|
|
|
|
CP0160303
|
(S)-1-(4-(2-(2-fluoroethoxy)ethoxy)benzyl)-5-(2-(phenoxymethyl)pyrrolidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C30H31FN2O7S
|
1
|
| 1 |
EC50 = 1690 nM
|
|
|
|
CP0109320
|
1-Methyl-5-(2-(pyridin-3-yl-oxymethyl)-pyrrolidine-1-sulfonyl)--1H-indole-2,3-dione
Show/Hide
|
C19H19N3O5S
|
1
|
| 1 |
EC50 = 1800 nM
|
|
|
|
CP0109321
|
5-(2-(Pyridin-3-yl-oxymethyl)-pyrrolidine-1-sulfonyl)-1H-indole-2,3-dione
Show/Hide
|
C18H17N3O5S
|
1
|
| 1 |
EC50 = 1830 nM
|
|
|
|
CP0219109
|
(S)-1-(4-(2-fluoroethoxy)benzyl)-5-(2-(phenoxymethyl)azetidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C27H25FN2O6S
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
|
CP0050268
|
(S)-1-(4-(2-(2-fluoroethoxy)ethoxy)benzyl)-5-(2-(phenoxymethyl)azetidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C29H29FN2O7S
|
1
|
| 1 |
EC50 = 2150 nM
|
|
|
|
CP0050281
|
(S)-5-(2-((2,4-difluorophenoxy)methyl)pyrrolidin-1-ylsulfonyl)-1-(4-(2-fluoroethoxy)benzyl)indoline-2,3-dione
Show/Hide
|
C28H25F3N2O6S
|
1
|
| 1 |
EC50 = 2500 nM
|
|
|
|
CP0057625
|
(S)-1-Benzyl-5-(2-phenoxymethyl-azetidine-1-sulfonyl)-1H-indole-2,3-dione
Show/Hide
|
C25H22N2O5S
|
1
|
| 1 |
EC50 = 2800 nM
|
|
|
|
CP0061807
|
(S)-1-(4-Methoxybenzyl)-5-(2-phenoxymethyl-azetidine-1-sulfonyl)-1H-indole-2,3-dione
Show/Hide
|
C26H24N2O6S
|
1
|
| 1 |
EC50 = 3070 nM
|
|
|
|
CP0136663
|
(S)-1-Methyl-5-(2-phenoxymethyl-azetidine-1-sulfonyl)-1H-indole-2,3-dione
Show/Hide
|
C19H18N2O5S
|
1
|
| 1 |
EC50 = 3250 nM
|
|
|
|
CP0096205
|
(S)-1-Benzyl-5-{1-[2-(phenoxymethyl)pyrrolidinyl]sulfonyl}isatin
Show/Hide
|
C26H24N2O5S
|
1
|
| 1 |
EC50 = 3670 nM
|
|
|
|
CP0045095
|
(S)-1-(4-(2-fluoroethoxy)benzyl)-5-(2-(phenoxymethyl)pyrrolidin-1-ylsulfonyl)indoline-2,3-dione
Show/Hide
|
C28H27FN2O6S
|
1
|
| 1 |
EC50 = 4500 nM
|
|
|
|
CP0057628
|
(S)-1-Methyl-5-{1-[2-(phenoxymethyl)pyrrolidinyl]sulfonyl}isatin
Show/Hide
|
C20H20N2O5S
|
1
|
| 1 |
EC50 = 7670 nM
|
|
|
|
CP0255351
|
(S)-5-(2-Phenoxymethyl-azetidine-1-sulfonyl)-1H-indole-2,3-dione
Show/Hide
|
C18H16N2O5S
|
1
|
| 1 |
EC50 = 9570 nM
|
|
|
|
CP0040399
|
(S)-5-{1-[2-(Phenoxymethyl)pyrrolidinyl]sulfonyl}isatin
Show/Hide
|
C19H18N2O5S
|
1
|
| 1 |
EC50 = 11500 nM
|
|
|
|
CP0108917
|
US10167313, Compound 65
Show/Hide
|
C40H43N5O12S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0108924
|
US10167313, Compound 55
Show/Hide
|
C35H41N5O11S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0450808
|
US10167313, Compound 48
Show/Hide
|
C35H40ClN5O11S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0204032
|
US10167313, Compound 59
Show/Hide
|
C28H38N4O13S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0116022
|
US10167313, Compound 85
Show/Hide
|
C36H41N5O11S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0148760
|
US10167313, Compound 76
Show/Hide
|
C32H40N4O12S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0169022
|
US10167313, Compound 57
Show/Hide
|
C34H42N4O11S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0206708
|
US10167313, Compound 63
Show/Hide
|
C40H43N5O11S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0700327
|
US9045524, 88
Show/Hide
|
C34H41N5O11S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0041050
|
US10167313, Compound 53
Show/Hide
|
C31H38N4O11S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0094271
|
US9045524, 71
Show/Hide
|
C35H41N5O11S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0153303
|
US10167313, Compound 69
Show/Hide
|
C36H40N4O11S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0113334
|
US10167313, Compound 66
Show/Hide
|
C46H62N6O12S
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0115533
|
US10167313, Compound 68
Show/Hide
|
C36H46N4O11S
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0066458
|
US9045524, 70
Show/Hide
|
C40H43N5O11S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0128430
|
US10167313, Compound 82
Show/Hide
|
C33H42N4O12S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0128368
|
US10167313, Compound 51
Show/Hide
|
C36H46N4O11S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0066497
|
US10167313, Compound 96
Show/Hide
|
C36H42N4O10S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0066892
|
US10167313, Compound 93
Show/Hide
|
C6H11NO4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0158506
|
US10167313, Compound 33
Show/Hide
|
C10H19NO4S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0066027
|
US10167313, Compound 37
Show/Hide
|
C15H21NO4S
|
1
|
| 1 |
IC50 > 2000 nM
|
|
|
|
CP0122107
|
US10167313, Compound 36
Show/Hide
|
C20H29NO6S
|
1
|
| 1 |
IC50 > 2000 nM
|
|
|
|
CP0227050
|
US10167313, Compound 16
Show/Hide
|
C29H37N3O8
|
1
|
| 1 |
IC50 > 2000 nM
|
|
|
|
CP0066480
|
US10167313, Compound 50
Show/Hide
|
C30H35ClN4O8S2
|
1
|
| 1 |
IC50 > 3330 nM
|
|
|
|
CP0104497
|
US10167313, Compound 61
Show/Hide
|
C19H26N2O7S
|
1
|
| 1 |
IC50 > 3330 nM
|
|
|
|
CP0158973
|
US9045524, 101
Show/Hide
|
C33H42N4O11S
|
1
|
| 1 |
IC50 > 3330 nM
|
|
|
