Brief Information of the Cell Line and Protein
Cell Line ID: CL001042 , HEK293/Gal4
 Cell Line Info 
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT00889 , Estrogen receptor beta
 Protein Info 
Gene Name ESR2
Organism Homo sapiens, Human
Protein Classification Transcription factor
Uniprot ID Q92731
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL001042
 Cell Line Info 
 Protein ID: PT00889
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0043589
 Compound Info 
(13S,17S)-13-Methyl-7-[9-(4,4,5,5,5-pentafluoro-pentane-1-sulfinyl)-nonyl]-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthrene-3,17-diol
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C32H47F5O3S
  1
1
IC50 = 0.3 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0546743
 Compound Info 
N-[4-[[2-[4-chloro-2-(1,1-difluoroethyl)phenyl]-6H-thieno[2,3-e]indazol-3-yl]oxy]phenyl]-1-(3-fluoropropyl)azetidin-3-amine
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C29H26ClF3N4OS
  1
1
IC50 = 2 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0545000
 Compound Info 
2-[4-chloro-2-(1,1-difluoroethyl)phenyl]-3-[4-[1-(3-fluoropropyl)azetidin-3-yl]oxyphenoxy]-6H-thieno[2,3-e]indazole
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C29H25ClF3N3O2S
  1
1
IC50 = 2.3 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0491461
 Compound Info 
6-(2,4-dichlorophenyl)-5-[4-[(3S)-1-(3-fluoropropyl)pyrrolidin-3-yl]oxyphenyl]-8,9-dihydro-7H-benzo[7]annulene-2-carboxylic acid
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C31H30Cl2FNO3
  1
1
IC50 = 8.6 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS