General Information of the Compound
Compound ID
CP0383812
Compound Name
4-(4-chlorophenyl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
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Structure
Formula
C15H18ClN5
Molecular Weight
303.797
Canonical SMILES
CN1CCN(CC1)c1cc(nc(N)n1)-c1ccc(Cl)cc1
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InChI
InChI=1S/C15H18ClN5/c1-20-6-8-21(9-7-20)14-10-13(18-15(17)19-14)11-2-4-12(16)5-3-11/h2-5,10H,6-9H2,1H3,(H2,17,18,19)
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InChIKey
YYUPHZVTHXGIJI-UHFFFAOYSA-N
Physicochemical Property
logP
2.131
Rotatable Bonds
2
Heavy Atom Count
21
Polar Areas
58.28
Hydrogen Bond Donor Count
1
Hydrogen Bond Acceptor Count
5
Complexity
21

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 25129527
SID: 56453873
ChEMBL ID
CHEMBL493720
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT02519, Histamine H4 receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 37.15 nM
   TI
   LI
   LO
   TS
Protein ID: PT01711, Histamine H4 receptor
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  3
1
Ki = 1.995 nM
   TI
   LI
   LO
   TS
2
Ki = 63.1 nM
   TI
   LI
   LO
   TS
3
Ki = 199.53 nM
   TI
   LI
   LO
   TS
CL000074 SK-N-MC Homo sapiens (Human)  1
1
Ki = 3.162 nM
   TI
   LI
   LO
   TS