General Information of the Cell Line
Cell Line ID
CL000383
Cell Line Name
AR42J
Synonyms
AR4-2J
AR-42J
Category
Cancer cell line
Organism
Rattus norvegicus (Rat)
Cellosaurus ID
CVCL_0143
Tissue Information
Pancreas
Disease
Rat digestive system neoplasms (NCIt: C60682)
Map of Molecular Bioactivity Related to the Cell Line
Map of Molecular Bioactivity Related to the Cell Line

Cell Line
Protein
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Cell Line
Protein ID: PT02587, Gastrin/cholecystokinin type B receptor
Compound ID Compound Name Compound Formula
CP0038292
3-{2-[2-(3-tert-Butoxycarbonylamino-propionylamino)-3-(1H-indol-3-yl)-propionylamino]-4-methylsulfanyl-butyrylamino}-N-(1-carbamoyl-2-phenyl-ethyl)-succinamic acid
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C37H49N7O9S
 1
1
EC50 = 0.43 nM
   TI
   LI
   LO
   TS
CP0906752
2,2',2''-(10-(2-((R)-1-((S)-1-((S)-1-((S)-2-((S)-1-(((S)-1-((S)-1-((S)-1-amino-3-(naphthalen-1-yl)-1-oxopropan-2-ylamino)-3-carboxy-1-oxopropan-2-ylamino)-1-oxohexan-2-yl)(methyl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylcarbamoyl)pyrrolidin-1-yl)-3-(4-hydroxyphenyl)-1-oxopropan-2-ylamino)-1-oxopropan-2-ylamino)-4-carboxy-1-oxobutan-2-ylamino)-2-oxoethyl)-1,4,7,10-tetraazacyclododecane-1,4,7-triyl)triacetic acid
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C73H96N14O20
 1
1
EC50 = 1.27 nM
   TI
   LI
   LO
   TS
CP0962464
2,2',2''-(10-(2-((R)-1-((S)-2-((2S,5S,8S,11S,17S)-11-((1H-indol-3-yl)methyl)-1-amino-8-butyl-5-(carboxymethyl)-18-(4-hydroxyphenyl)-9-methyl-2-(naphthalen-1-ylmethyl)-1,4,7,10,13,16-hexaoxo-3,6,9,12,15-pentaazaoctadecan-17-ylcarbamoyl)pyrrolidin-1-yl)-4-carboxy-1-oxobutan-2-ylamino)-2-oxoethyl)-1,4,7,10-tetraazacyclododecane-1,4,7-triyl)triacetic acid
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C72H94N14O20
 1
1
EC50 = 1.74 nM
   TI
   LI
   LO
   TS
CP0962465
2,2',2''-(10-(2-((R)-1-((S)-1-((S)-2-((4S,7S,10S,13S)-4-((1H-indol-3-yl)methyl)-14-amino-7-butyl-10-(carboxymethyl)-6-methyl-13-(naphthalen-1-ylmethyl)-2,5,8,11,14-pentaoxo-3,6,9,12-tetraazatetradecylcarbamoyl)pyrrolidin-1-yl)-3-(4-hydroxyphenyl)-1-oxopropan-2-ylamino)-4-carboxy-1-oxobutan-2-ylamino)-2-oxoethyl)-1,4,7,10-tetraazacyclododecane-1,4,7-triyl)triacetic acid
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C72H94N14O20
 1
1
EC50 = 1.91 nM
   TI
   LI
   LO
   TS
Protein family and CMB statistics Related to the Cell Line
Cell Lines Derived from the same Tissue Source (Pancreas)
Cell Line Name Organism Disease
PSN1 Homo sapiens (Human) Pancreatic adenocarcinoma
DAN-G Homo sapiens (Human) Pancreatic adenocarcinoma
PANC-1 Homo sapiens (Human) Pancreatic ductal adenocarcinoma
MIA PaCa-2 Homo sapiens (Human) Pancreatic ductal adenocarcinoma
MiaPaCa(BCRP) Homo sapiens (Human) Pancreatic ductal adenocarcinoma
BxPC-3 Homo sapiens (Human) Pancreatic ductal adenocarcinoma
Beta-TC-3 Mus musculus (Mouse) Mouse insulinoma
MIN6 Mus musculus (Mouse) Mouse insulinoma
Beta-TC-6 Mus musculus (Mouse) Mouse insulinoma
Panc02 Mus musculus (Mouse) Mouse pancreatic ductal adenocarcinoma
INS-1 Rattus norvegicus (Rat) Rat insulinoma
INS-1 832/13 Rattus norvegicus (Rat) Rat insulinoma
INS-1E Rattus norvegicus (Rat) Rat insulinoma