Brief Information of the Cell Line and Protein
Cell Line ID: CL000383 , AR42J
Synonyms
AR4-2J
AR-42J
Category Cancer cell line
Organism
Rattus norvegicus (Rat)
Cellosaurus ID
CVCL_0143
Protein ID: PT01505 , Somatostatin receptor type 2
Gene Name SSTR2
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P30874
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000383  Protein ID: PT01505
 
Compound ID Compound Name Compound Formula
CP0522300
(3R,6S,9S,12S,15S,18S,21S,24S,27S,30S,33S,36R)-21-((1H-indol-3-yl)methyl)-30-(2-amino-2-oxoethyl)-18,33-bis(4-aminobutyl)-36-(2-((S)-2-aminopropanamido)acetamido)-12,24,27-tribenzyl-9,15-bis((R)-1-hydroxyethyl)-6-(hydroxymethyl)-5,8,11,14,17,20,23,26,29,32,35-undecaoxo-1,2-dithia-4,7,10,13,16,19,22,25,28,31,34-undecaazacycloheptatriacontane-3-carboxylic acid
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C75H102N18O19S2
 1
1
IC50 = 0.4 nM
   TI
   LI
   LO
   TS
CP0845169
(2E,8S,11S,14S,17S,20S,23S,26S,29S,32S,35S,38S,41S)-23,38-bis(4-aminobutyl)-41-{2-[(2S)-2-aminopropanamido]acetamido}-17,29,32-tribenzyl-35-(carbamoylmethyl)-49-hydroxy-14,20-bis[(1R)-1-hydroxyethyl]-11-(hydroxymethyl)-26-(1H-indol-3-ylmethyl)-10,13,16,19,22,25,28,31,34,37,40-undecaoxo-2,3,9,12,15,18,21,24,27,30,33,36,39-tridecaazatricyclo[41.2.2.2^{4,7}]nonatetraconta-1(45),2,4,6,43,46,48-heptaene-8-carboxylic acid
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C87H110N20O20
 1
1
IC50 > 600 nM
   TI
   LI
   LO
   TS