| Compound ID |
Compound Name |
Compound Formula |
|
CP0548642
|
N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-4-(propan-2-ylamino)-6-(pyrazolo[1,5-a]pyrimidin-5-ylamino)pyridine-3-carboxamide
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|
C20H26FN7O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0136727
|
US9546153, ex. 42
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|
C21H24FN5O2S
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0133598
|
US9546153, ex. 9
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|
C21H25N5O2S
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0139167
|
US9546153, ex. 8
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|
C21H27N5O2S
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0218453
|
US9546153, ex. 143
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|
C23H23N5O3S
|
1
|
| 1 |
IC50 = 300 nM
|
|
|
|
CP0553657
|
US9546153, ex. 41
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|
C20H25FN6O2S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0531465
|
US9546153, ex. 367
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|
C20H25F2N7O2
|
1
|
| 1 |
IC50 = 370 nM
|
|
|
|
CP0233072
|
US9546153, ex. 286
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|
C21H27FN6O2
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0233047
|
US9546153, ex. 35
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|
C21H26FN5O2S
|
1
|
| 1 |
IC50 = 480 nM
|
|
|
|
CP0341632
|
US9546153, ex. 171
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|
C21H25F2N5O2S
|
1
|
| 1 |
IC50 = 570 nM
|
|
|
|
CP0351775
|
US9546153, ex. 45
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|
C20H25FN6O3
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0531787
|
US9546153, ex. 366
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|
C21H24FN5O2S
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0136722
|
6-(1,3-benzothiazol-6-ylamino)-4-(propan-2-ylamino)-N-[2-(4-sulfamoylphenyl)ethyl]pyridine-3-carboxamide
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|
C24H26N6O3S2
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0422246
|
N-[(2R)-2-fluoro-3-hydroxy-3-methylbutyl]-6-[(2-methyl-1,3-benzothiazol-6-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamide
Show/Hide
|
C22H28FN5O2S
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0153113
|
6-(1,3-benzothiazol-6-ylamino)-4-[[(2S)-1-hydroxy-3-phenylpropan-2-yl]amino]-N-methylpyridine-3-carboxamide
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|
C23H23N5O2S
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0321333
|
6-(1,3-benzothiazol-6-ylamino)-N-[(2R)-3-hydroxy-2,3-dimethylbutyl]-4-(propan-2-ylamino)pyridine-3-carboxamide
Show/Hide
|
C22H29N5O2S
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0534231
|
6-(1,3-benzothiazol-6-ylamino)-N-methyl-4-(propan-2-ylamino)pyridine-3-carboxamide
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|
C17H19N5OS
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
|
CP0422244
|
6-(1,3-benzothiazol-6-ylamino)-N-(3-hydroxypropyl)-4-(propan-2-ylamino)pyridine-3-carboxamide
Show/Hide
|
C19H23N5O2S
|
1
|
| 1 |
IC50 = 6900 nM
|
|
|
