Brief Information of the Cell Line and Protein
Cell Line ID: CL000389 , CHO-DXB11
Synonyms
CHO DXB11
DXB11-CHO
CHO-DUX-B11
CHO (Dux B11)
CHO-DUK-XB11
DUK-XB11
CHO-DUKX B11
CHO-DUKXB11
DUKX-B11
DUX B11
DUXB11
DXB-11
DXB11
CHO-DUKX
DUKX-CHO
DUKX
CHO-DHFR -
CHO/dhFr-
CHO/dhfr-
CHO(dhfr-)
CHO duk-
CHOd-
CHO B11
B11
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_1977
Protein ID: PT02392 , B2 bradykinin receptor
Gene Name BDKRB2
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID P30411
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000389  Protein ID: PT02392
 
Compound ID Compound Name Compound Formula
CP0172614
(S)-4-amino-5-(4-(4-(2,4-dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2H-pyran-4-carbonyl)piperazin-1-yl)-N,N,N-trimethyl-5-oxopentan-1-aminium chloride
   Show/Hide
C36H49Cl2N6O6S+
 1
1
Kd = 0.05012 nM
   TI
   LI
   LO
   TS
CP0892092
(S)-N-(4-(4-(2-amino-5-(dimethylamino)pentanoyl)piperazine-1-carbonyl)tetrahydro-2H-pyran-4-yl)-2,4-dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)benzenesulfonamide trifluoroacetate salt
   Show/Hide
C37H47Cl2F3N6O8S
 1
1
Kd = 0.123 nM
   TI
   LI
   LO
   TS
CP0839078
[(S)-4-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-thiopyran-4-carbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium
   Show/Hide
C36H49Cl2N6O5S2+
 1
1
Kd = 0.1585 nM
   TI
   LI
   LO
   TS
CP0789365
N-{1-[4-((S)-2-amino-6-guanidino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C35H46Cl2N8O5S
 1
1
Kd = 0.2512 nM
   TI
   LI
   LO
   TS
CP0839077
[(S)-4-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-1-methyl-piperidine-4-carbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium
   Show/Hide
C37H52Cl2N7O5S+
 1
1
Kd = 0.2512 nM
   TI
   LI
   LO
   TS
CP0682478
[(S)-4-amino-5-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium
   Show/Hide
C36H49Cl2N6O5S+
 1
1
Kd = 0.3162 nM
   TI
   LI
   LO
   TS
CP0893994
[5-(4-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium trifluoroacetate salt
   Show/Hide
C38H48Cl2F3N5O8S
 1
1
Kd = 0.3162 nM
   TI
   LI
   LO
   TS
CP0789361
LF16-0687
   Show/Hide
C34H36Cl2N6O5S
 1
1
Kd = 0.3981 nM
   TI
   LI
   LO
   TS
CP0867622
(S)-5-Amino-6-(4-(4-(2,4-dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2Hpyran-4-carbonyl)piperazin-1-yl)-N,N,N-trimethyl-6-oxohexan-1-aminium trifluoroacetate salt
   Show/Hide
C39H51Cl2F3N6O8S
 1
1
Kd = 0.3981 nM
   TI
   LI
   LO
   TS
CP0896456
(S)-2,4-dichloro-N-(4-(4-(2,6-diaminohexanoyl)piperazine-1-carbonyl)tetrahydro-2H-pyran-4-yl)-3-((2,4-dimethylquinolin-8-yloxy)methyl)benzenesulfonamide trifluoroacetate salt
   Show/Hide
C36H45Cl2F3N6O8S
 1
1
Kd = 0.3981 nM
   TI
   LI
   LO
   TS
CP0917488
2,4-Dichloro-N-{4-[4-(5-dimethylamino-pentanoyl)-piperazine-1-carbonyl]-tetrahydro-pyran-4-yl}-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide trifluoroacetate salt
   Show/Hide
C37H46Cl2F3N5O8S
 1
1
Kd = 0.4365 nM
   TI
   LI
   LO
   TS
CP0916503
N-{4-[4-(5-Amino-pentanoyl)-piperazine-1-carbonyl]-tetrahydro-pyran-4-yl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide trifluoroacetate salt
   Show/Hide
C35H42Cl2F3N5O8S
 1
1
Kd = 0.4786 nM
   TI
   LI
   LO
   TS
CP0682476
[(S)-4-amino-1-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazine-1-carbonyl)-butyl]-trimethyl-ammonium
   Show/Hide
C36H49Cl2N6O5S+
 1
1
Kd = 0.5012 nM
   TI
   LI
   LO
   TS
CP0682481
2,4-dichloro-N-{1-[4-((S)-3,6-diamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C34H44Cl2N6O5S
 1
1
Kd = 0.5012 nM
   TI
   LI
   LO
   TS
CP0789364
4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-N-(3-dimethylamino-propyl)-piperazine-1-carboxamidine
   Show/Hide
C34H45Cl2N7O4S
 1
1
Kd = 0.5012 nM
   TI
   LI
   LO
   TS
CP0829543
[(S)-1-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazine-1-carbonyl)-5-guanidino-pentyl]-trimethyl-ammonium
   Show/Hide
C38H53Cl2N8O5S+
 1
1
Kd = 0.631 nM
   TI
   LI
   LO
   TS
CP0851981
2,4-Dichloro-N-{4-[4-((S)-2,5-diamino-pentanoyl)-piperazine-1-carbonyl]-tetrahydro-pyran-4-yl}-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide trifluoroacetate salt
   Show/Hide
C35H43Cl2F3N6O8S
 1
1
Kd = 0.7244 nM
   TI
   LI
   LO
   TS
CP0682479
N-{1-[4-((S)-3-amino-6-guanidino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C35H46Cl2N8O5S
 1
1
Kd = 0.7943 nM
   TI
   LI
   LO
   TS
CP0720693
N-{2-[4-((S)-2-amino-5-(dimethylamino)pentanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonamide
   Show/Hide
C33H44Cl2N6O5S
 1
1
Kd = 0.7943 nM
   TI
   LI
   LO
   TS
CP0829545
N-{2-[4-((S)-2-amino-6-guanidino-hexanoyl)-piperazin-1-yl]-1,1-dimethyl-2-oxo-ethyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C33H44Cl2N8O5S
 1
1
Kd = 0.7943 nM
   TI
   LI
   LO
   TS
CP0871079
N-{1-[4-((S)-2-amino-6-dimethylamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C36H48Cl2N6O5S
 1
1
Kd = 0.7943 nM
   TI
   LI
   LO
   TS
CP0847132
[6-(4-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperazin-1-yl)-hexyl]-trimethyl-ammonium trifluoroacetate salt
   Show/Hide
C39H52Cl2F3N5O7S
 1
1
Kd = 0.7943 nM
   TI
   LI
   LO
   TS
CP0851980
[4-(4-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperazin-1-yl)-4-oxo-butyl]-trimethyl-ammonium trifluoroacetate salt
   Show/Hide
C37H46Cl2F3N5O8S
 1
1
Kd = 0.7943 nM
   TI
   LI
   LO
   TS
CP0851983
[2-(4-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperazin-1-yl)-2-oxo-ethyl]-trimethylammonium trifluoroacetate salt
   Show/Hide
C35H42Cl2F3N5O8S
 1
1
Kd = 0.7943 nM
   TI
   LI
   LO
   TS
CP0853240
[6-(4-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperazin-1-yl)-6-oxo-hexyl]-trimethyl-ammonium trifluoroacetate salt
   Show/Hide
C39H50Cl2F3N5O8S
 1
1
Kd = 0.7943 nM
   TI
   LI
   LO
   TS
CP0892090
4-(4-(2,4-Dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2H-pyran-4-carbonyl)-1-methyl-1-(3-(trimethylammonio)propyl)piperazin-1-ium trifluoroacetate salt
   Show/Hide
C39H49Cl2F6N5O9S
 1
1
Kd = 1 nM
   TI
   LI
   LO
   TS
CP0779070
{(S)-4-amino-1-[2-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-2-oxo-ethyl]-butyl}-trimethyl-ammonium
   Show/Hide
C37H51Cl2N6O5S+
 1
1
Kd = 1.259 nM
   TI
   LI
   LO
   TS
CP0789362
[(S)-5-(4-{1-acetyl-4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-piperidine-4-carbonyl}-piperazin-1-yl)-4-amino-5-oxo-pentyl]-trimethyl-ammonium
   Show/Hide
C38H52Cl2N7O6S+
 1
1
Kd = 1.259 nM
   TI
   LI
   LO
   TS
CP0800201
[(S)-5-amino-6-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-6-oxo-hexyl]-trimethyl-ammonium
   Show/Hide
C37H51Cl2N6O5S+
 1
1
Kd = 1.259 nM
   TI
   LI
   LO
   TS
CP0917487
7-(4-(4-(2,4-dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2H-pyran-4-carbonyl)piperazin-1-yl)-N,N,N-trimethyl-7-oxoheptan-1-aminium trifluoroacetate salt
   Show/Hide
C40H52Cl2F3N5O8S
 1
1
Kd = 1.259 nM
   TI
   LI
   LO
   TS
CP0711137
{3-[(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazine-1-carboximidoyl)-amino]-propyl}-trimethyl-ammonium
   Show/Hide
C35H48Cl2N7O4S+
 1
1
Kd = 1.585 nM
   TI
   LI
   LO
   TS
CP0711141
[(S)-4-amino-6-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-6-oxo-hexyl]-trimethyl-ammonium
   Show/Hide
C37H51Cl2N6O5S+
 1
1
Kd = 1.585 nM
   TI
   LI
   LO
   TS
CP0789363
[(S)-4-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-piperidine-4-carbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium
   Show/Hide
C36H50Cl2N7O5S+
 1
1
Kd = 1.585 nM
   TI
   LI
   LO
   TS
CP0829540
[5-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-5-oxo-pentyl]-trimethyl-ammonium
   Show/Hide
C36H48Cl2N5O5S+
 1
1
Kd = 1.585 nM
   TI
   LI
   LO
   TS
CP0829542
[(S)-5-amino-1-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazine-1-carbonyl)-pentyl]-trimethyl-ammonium
   Show/Hide
C37H51Cl2N6O5S+
 1
1
Kd = 1.585 nM
   TI
   LI
   LO
   TS
CP0829544
N-{1-[4-((S)-3-amino-6-dimethylamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C36H48Cl2N6O5S
 1
1
Kd = 1.585 nM
   TI
   LI
   LO
   TS
CP0847106
3-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-9-methyl-3,9-diaza-6-azonia-spiro[5.5]undecane trifluoroacetate salt
   Show/Hide
C35H42Cl2F3N5O7S
 1
1
Kd = 1.585 nM
   TI
   LI
   LO
   TS
CP0847137
[3-(1-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperidin-4-yl)-propyl]-trimethyl-ammonium trilfuoroacetate salt
   Show/Hide
C37H47Cl2F3N4O7S
 1
1
Kd = 1.585 nM
   TI
   LI
   LO
   TS
CP0711142
2,4-dichloro-N-{1-[4-((S)-2,6-diamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C34H44Cl2N6O5S
 1
1
Kd = 1.995 nM
   TI
   LI
   LO
   TS
CP0800200
2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-N-{1-[4-(6-guanidino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-benzenesulfonamide
   Show/Hide
C35H45Cl2N7O5S
 1
1
Kd = 1.995 nM
   TI
   LI
   LO
   TS
CP0829541
[(S)-3-amino-4-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-4-oxo-butyl]-trimethyl-ammonium
   Show/Hide
C35H47Cl2N6O5S+
 1
1
Kd = 1.995 nM
   TI
   LI
   LO
   TS
CP0860944
[4-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-4-oxo-butyl]-trimethyl-ammonium
   Show/Hide
C35H46Cl2N5O5S+
 1
1
Kd = 1.995 nM
   TI
   LI
   LO
   TS
CP0847133
4-(4-(2,4-dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2H-pyran-4-carbonyl)-1-methyl-1-(4-(trimethylammonio)butyl)piperazin-1-ium 2,2,2-trifluoroacetate
   Show/Hide
C40H51Cl2F6N5O9S
 1
1
Kd = 1.995 nM
   TI
   LI
   LO
   TS
CP0682483
N-{2-[4-((S)-3-amino-6-(dimethylamino)hexanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonamide
   Show/Hide
C34H46Cl2N6O5S
 1
1
Kd = 2.512 nM
   TI
   LI
   LO
   TS
CP0702267
[5-(4-(1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl]-piperazin-1-yl)-4(S)-trimethylammonio-5-oxo-pentyl]trimethyl-ammonium
   Show/Hide
C39H56Cl2N6O5S+2
 1
1
Kd = 2.512 nM
   TI
   LI
   LO
   TS
CP0847134
4-(4-(2,4-Dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2H-pyran-4-carbonyl)-1-methyl-1-(5-(trimethylammonio)pentyl)piperazin-1-ium trifluoroacetate salt
   Show/Hide
C41H53Cl2F6N5O9S
 1
1
Kd = 2.512 nM
   TI
   LI
   LO
   TS
CP0853852
{3-[(1-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperidin-4-ylmethyl)-amino]-propyl}-trimethylammonium trifluoroacetate salt
   Show/Hide
C38H50Cl2F3N5O7S
 1
1
Kd = 2.512 nM
   TI
   LI
   LO
   TS
CP0892093
{4-[(1-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperidin-4-ylmethyl)-amino]-butyl}-trimethylammonium trifluoroacetate salt
   Show/Hide
C39H52Cl2F3N5O7S
 1
1
Kd = 2.512 nM
   TI
   LI
   LO
   TS
CP0916501
{2-[(1-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperidin-4-ylmethyl)-amino]-ethyl}-trimethylammonium trifluoroacetate salt
   Show/Hide
C37H48Cl2F3N5O7S
 1
1
Kd = 2.512 nM
   TI
   LI
   LO
   TS
CP0847138
3-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-3-aza-6-azonia-spiro[5.5]undecane trifluoroacetate salt
   Show/Hide
C35H41Cl2F3N4O7S
 1
1
Kd = 2.63 nM
   TI
   LI
   LO
   TS
CP0800202
N-{1-[4-((S)-2,6-bis-dimethylamino-hexanoyl)-piperazine-1-carbonyl]-cyclopentyl}-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C38H52Cl2N6O5S
 1
1
Kd = 3.162 nM
   TI
   LI
   LO
   TS
CP0800203
N-{2-[4-((S)-2-amino-6-(dimethylamino)hexanoyl)piperazin-1-yl]-1,1-dimethyl-2-oxoethyl}-2,4-dichloro-3-(2,4-dimethylquinolin-8-yloxymethyl)benzenesulfonamide
   Show/Hide
C34H46Cl2N6O5S
 1
1
Kd = 3.162 nM
   TI
   LI
   LO
   TS
CP0847105
4-(4-(2,4-Dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2H-pyran-4-carbonyl)-1-methyl-1-(2-(trimethylammonio)ethyl)piperazin-1-ium trifluoroacetate salt
   Show/Hide
C38H47Cl2F6N5O9S
 1
1
Kd = 3.162 nM
   TI
   LI
   LO
   TS
CP0847135
8-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-8-aza-5-azonia-spiro[4.5]decane trifluoroacetate salt
   Show/Hide
C34H39Cl2F3N4O7S
 1
1
Kd = 3.162 nM
   TI
   LI
   LO
   TS
CP0874519
4-(4-(2,4-Dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2H-pyran-4-carbonyl)-1-methyl-1-(6-(trimethylammonio)hexyl)piperazin-1-ium trifluoroacetate salt
   Show/Hide
C42H55Cl2F6N5O9S
 1
1
Kd = 3.162 nM
   TI
   LI
   LO
   TS
CP0847136
[2-(1-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperidin-4-yl)-ethyl]-trimethyl-ammonium trilfuoroacetate salt
   Show/Hide
C36H45Cl2F3N4O7S
 1
1
Kd = 3.981 nM
   TI
   LI
   LO
   TS
CP0859150
[4-(1-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperidin-4-yl)-butyl]-trimethyl-ammonium trilfuoroacetate salt
   Show/Hide
C38H49Cl2F3N4O7S
 1
1
Kd = 3.981 nM
   TI
   LI
   LO
   TS
CP0711139
[2-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-2-oxo-ethyl]-trimethyl-ammonium
   Show/Hide
C33H42Cl2N5O5S+
 1
1
Kd = 5.012 nM
   TI
   LI
   LO
   TS
CP0800199
[6-(4-{1-[2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-cyclopentanecarbonyl}-piperazin-1-yl)-6-oxo-hexyl]-trimethyl-ammonium
   Show/Hide
C37H50Cl2N5O5S+
 1
1
Kd = 5.012 nM
   TI
   LI
   LO
   TS
CP0853853
9-(4-(2,4-Dichloro-3-((2,4-dimethylquinolin-8-yloxy)methyl)phenylsulfonamido)tetrahydro-2H-pyran-4-carbonyl)-3,3-dimethyl-9-aza-3,6-diazoniaspiro[5.5]undecane trifluoroacetate salt
   Show/Hide
C38H45Cl2F6N5O9S
 1
1
Kd = 5.012 nM
   TI
   LI
   LO
   TS
CP0894500
(1-{4-[2,4-Dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonylamino]-tetrahydro-pyran-4-carbonyl}-piperidin-4-ylmethyl)-trimethyl-ammonium trifluoroacetate salt
   Show/Hide
C35H43Cl2F3N4O7S
 1
1
Kd = 5.012 nM
   TI
   LI
   LO
   TS
CP0702268
N-[1-[4-(2-(S)-trimethylammonium-6-trimethylammoniumhexanoyl)-piperazin-1-yl]-cyclopentyl]-2,4-dichloro-3-(2,4-dimethyl-quinolin-8-yloxymethyl)-benzenesulfonamide
   Show/Hide
C40H58Cl2N6O5S+2
 1
1
Kd = 6.31 nM
   TI
   LI
   LO
   TS