US9447038, 9

US9073853, 12

US9073853, 5

(S)-3-(4-Chloro-3-fluoro-phenyl)-3-(cyclopropylmethyl-{4-[2-(2,5-dioxo-pyrrolidin-1-yl)-ethoxy]-3-methoxy-benzyl}-amino)-propionic acid hydrochloride

3-(4-chlorophenyl)-3-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methylphenyl]methyl-propylamino]propanoic acid

US9073853, 88

US9447038, 5

US9073853, 10

US9073853, 14

US9073853, 148

US9447038, 28

(S)-3-(4-Chloro-3-fluoro-phenyl)-3-({4-[2-(2,5-dioxo-pyrrolidin-1-yl)-ethoxy]-3-methylbenzyl}-isobutyl-amino)-propionic acid hydrochloride

US9447038, 2

US9073853, 16

(3S)-3-(4-chlorophenyl)-3-[cyclopentylmethyl-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methylphenyl]methyl]amino]propanoic acid

US9073853, 15

US9073853, 7

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)propyl-(2-methylpropyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

(3S)-3-(4-chlorophenyl)-3-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methylphenyl]methyl-(2-methylpropyl)amino]propanoic acid

(S)-3-({3-Chloro-4-[2-(2,5-dioxo-pyrrolidin-1-yl)-ethoxy]-benzyl}-cyclopropylmethylamino)-3-(4-chloro-3-fluoro-phenyl)-propionic acid hydrochloride

US9447038, 1

US9447038, 23

US9073853, 17

US9447038, 4

3-(4-chloro-3-fluorophenyl)-3-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methylphenyl]methyl-(2-methylpropyl)amino]propanoic acid

1-[2-[4-[[cyclohexylmethyl-[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl]amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9073853, 30

US9447038, 17

US9073853, 19

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-(2-methylpropyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

(S)-3-(4-chloro-3-fluorophenyl)-3-((cyclopropylmethyl)(4-(2-(2,5-dioxopyrrolidin-1-yl)ethoxy)-3-fluorobenzyl)amino)propanoic acid

CHEMBL3965002

(3S)-3-(4-chloro-3-fluorophenyl)-3-[cyclopentylmethyl-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methylphenyl]methyl]amino]propanoic acid;hydrochloride

US9447038, 70

3-(4-chlorophenyl)-3-[cyclopropylmethyl-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methylphenyl]methyl]amino]propanoic acid

US9447038, 118

1-[2-[4-[[2,3-dihydro-1-benzofuran-5-ylmethyl(2-methylpropyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9447038, 42

US9447038, 72

US9447038, 186

US9447038, 69

US9073853, 37

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-(2-hydroxypropyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

3-(4-Chloro-phenyl)-3-[{4-[2-(2,5-dioxo-pyrrolidin-1-yl)-ethoxy]-3-methyl-benzyl}-(4-fluoro-benzyl)-amino]-propionic acid hydrochloride

US9447038, 144

US9447038, 80

US9447038, 73

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-(2-hydroxyethyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9447038, 114

US9447038, 116

US9447038, 7

US9447038, 120

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-[(4-fluorophenyl)methyl]amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

(S)-3-(Cyclopropylmethyl-{4-[2-(2,5-dioxo-pyrrolidin-1-yl)-ethoxy]-3-fluoro-benzyl}-amino)-3-(3,4-dichloro-phenyl)-propionic acid hydrochloride

CHEMBL3970774

3-(5-Chloro-thiophen-2-yl)-3-({4-[2-(2,5-dioxo-pyrrolidin-1-yl)-ethoxy]-3-methylbenzyl}-propyl-amino)-propionic acid hydrochloride

US9447038, 6

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)propyl-ethylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)butyl-methylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9447038, 151

US9447038, 68

4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methoxyphenyl]methyl]amino]methyl]benzoic acid

3-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-methylamino]methyl]-2-methoxyphenoxy]ethyl]-1,3-thiazolidine-2,4-dione

N-[(1R)-1-[3-(4-ethoxyphenyl)-4-oxo-1,2-dihydropyrido[2,3-d]pyrimidin-2-yl]ethyl]-N-(pyridin-3-ylmethyl)-2-[4-(trifluoromethoxy)phenyl]acetamide

US9447038, 122

US9447038, 113

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-[[4-(2H-tetrazol-5-yl)phenyl]methyl]amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-(pyridin-4-ylmethyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9447038, 10

US9447038, 117

(E)-3-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methoxyphenyl]methyl]amino]methyl]phenyl]prop-2-enoic acid

US9447038, 47

US9447038, 121

US9447038, 119

1-[2-[4-[[[(1S)-1-(2,3-dihydro-1-benzofuran-5-yl)ethyl]-methylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9447038, 123

4-[[1-(2,3-dihydro-1-benzofuran-5-yl)propyl-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methoxyphenyl]methyl]amino]methyl]benzoic acid

US9073853, 71

1-[2-[2-chloro-4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-methylamino]methyl]phenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-(pyridin-3-ylmethyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9073853, 11

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-(2-oxopropyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

3-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-methylamino]methyl]-2-methoxyphenoxy]ethyl]-1-methylimidazolidine-2,4-dione

4-[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methoxyphenyl]methyl]amino]butanoic acid

4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methoxyphenyl]methyl]amino]methyl]bicyclo[2.2.2]octane-1-carboxylic acid

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-methylamino]methyl]-2-methylphenoxy]ethyl]pyrrolidine-2,5-dione

3-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-methylamino]methyl]-2-methoxyphenoxy]ethyl]imidazolidine-2,4-dione

US9447038, 183

US9447038, 162

1-[2-[4-[(2,3-dihydro-1-benzofuran-5-ylmethylamino)methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[[1-(2,3-dihydro-1-benzofuran-5-yl)-3-methylbutyl]-methylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

4-[[[(1R)-1-(4-chlorophenyl)ethyl]-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methoxyphenyl]methyl]amino]methyl]benzoic acid

4-[[cyclopentyl(2,3-dihydro-1-benzofuran-5-yl)methyl]-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methoxyphenyl]methyl]amino]butanoic acid

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-methylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9447038, 67

US9447038, 112

US9447038, 115

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl-methylamino]methyl]-2-methoxyanilino]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)ethylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

US9447038, 157

US9447038, 8

US9073853, 2

1-[2-[4-[[2-(2,3-dihydro-1-benzofuran-5-yl)propan-2-ylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[[(1R)-1-(2,3-dihydro-1-benzofuran-5-yl)ethyl]-methylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

CHEMBL3932217

US9073853, 45

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)propylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[1-(2,3-dihydro-1-benzofuran-5-yl)butylamino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

3-(4-chlorophenyl)-3-[methyl-[[3-methyl-4-[2-(3-methyl-2,6-dioxopyrimidin-1-yl)ethoxy]phenyl]methyl]amino]propanoic acid

US9447038, 172

US9073853, 13

1-[2-[4-[[[1-(2,3-dihydro-1-benzofuran-5-yl)-3-methylbutyl]amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[2-aminoethyl-[1-(2,3-dihydro-1-benzofuran-5-yl)ethyl]amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

1-[2-[4-[[[cyclopentyl(2,3-dihydro-1-benzofuran-5-yl)methyl]amino]methyl]-2-methoxyphenoxy]ethyl]pyrrolidine-2,5-dione

4-[[[cyclopentyl(2,3-dihydro-1-benzofuran-5-yl)methyl]-[[4-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]-3-methoxyphenyl]methyl]amino]methyl]benzoic acid

5-[[[(1S)-1-(4-chlorophenyl)ethyl]-(cyclopentylmethyl)amino]methyl]-2-[2-(2,5-dioxopyrrolidin-1-yl)ethoxy]benzoic acid