7-(3,4-dichlorophenyl)-6-(5-fluoro-1-methyl-1H-benzo[d]imidazol-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

8-methoxy-N-(2-methyl-2-phenylpropyl)isoquinolin-1-amine

5-methoxy-4-[(2-methyl-2-phenylpropyl)amino]-1H-quinazolin-2-one

4-methoxy-N-(2-methyl-2-phenylpropyl)-1,2-benzothiazol-3-amine

2,2,2-trifluoroethyl N-[4-[[(4-methoxy-1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]methyl]-4-phenylcyclohexyl]carbamate

7-(3,4-dichlorophenyl)-6-(5-fluoro-1-methyl-1H-benzo[d]imidazol-2-yl)-5-(methoxymethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

[4-[[(4-methoxy-1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]methyl]-4-phenylcyclohexyl] N-[4-(dimethylamino)phenyl]carbamate

4-methoxy-1,1-dioxo-N-[[1-phenyl-4-(tetrazol-1-yl)cyclohexyl]methyl]-1,2-benzothiazol-3-imine

N-[(2R,3R)-3-[(4-ethylphenyl)sulfonylamino]-2-hydroxy-2,3-dihydro-1H-inden-5-yl]-3-methoxybenzamide

4-[[(4-methoxy-1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]methyl]-4-phenylcyclohexan-1-ol

4-methoxy-3-(2-methyl-2-phenylpropyl)iminoisoindol-1-one

(R)-6-(1-cyclopentyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

4-methoxy-N-(2-methyl-2-phenylpropyl)-1,2-benzoxazol-3-amine

N-[(8S)-8-[(4-ethylphenyl)sulfonylamino]-5,6,7,8-tetrahydronaphthalen-2-yl]-N-[(6-methylpyridin-2-yl)methyl]-3-phenylpropanamide

5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]pyridine-3-sulfonamide

N-[4-[[(4-methoxy-1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]methyl]-4-phenylcyclohexyl]pyrimidin-2-amine

7-(3,4-dichlorophenyl)-6-(5-fluoro-1-propyl-1H-benzo[d]imidazol-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-6-(1-cyclobutyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

((R)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(4-fluorophenyl)pyrrolidin-1-yl)methanone

CHEMBL3622360

3-[[4-(diethylsulfamoylamino)-1-phenylcyclohexyl]methylimino]-4-methoxy-1,1-dioxo-1,2-benzothiazole

ethyl N-[4-[[(4-methoxy-1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]methyl]-4-phenylcyclohexyl]carbamate

(3S,4R)-4-(N-butyl-4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenethylchroman-6-carboxamide

6-(5-chloro-1-ethyl-1H-benzo[d]imidazol-2-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-6-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

N-[(3S,4R)-6-[(2S)-2-[(2,6-dimethylanilino)methyl]pyrrolidine-1-carbonyl]-3-hydroxy-2,2-dimethyl-3,4-dihydrochromen-4-yl]-4-ethylbenzenesulfonamide

N-[4-[[(4-methoxy-1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]methyl]-4-phenylcyclohexyl]ethanesulfonamide

5-phenyl-2-pyridin-3-yl-N-(pyridin-2-ylmethyl)quinazolin-4-amine

7-(3,4-dichlorophenyl)-6-(4-fluoro-1-methyl-1H-benzo[d]imidazol-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

CHEMBL3622348

6-(5-chloro-1-methyl-1H-benzo[d]imidazol-2-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

N-[(7R,8R)-7-hydroxy-8-[(4-pentylphenyl)sulfonylamino]-5,6,7,8-tetrahydronaphthalen-2-yl]-3-methoxybenzamide

[(7R)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone

7-(3,4-dichlorophenyl)-5-methyl-N,N-dipropyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide

((R)-7-(3,4-Dichlorophenyl)-5-(methoxymethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone

6-(7-chloro-1-methyl-1H-benzo[d]imidazol-2-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

((S)-5-Methyl-7-(1-methyl-1H-indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone

2-chloro-5-methoxy-N-(2-methyl-2-phenylpropyl)quinazolin-4-amine

(7R)-7-(3,4-dichlorophenyl)-6-(1-(2-fluorophenyl)-1H-1,2,4-triazol-5-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

7-(3,4-dichlorophenyl)-5-methyl-6-(1-methyl-1H-benzo[d]imidazol-2-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(3S,4R)-N-ethyl-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-(2-(phenylamino)ethyl)-3,4-dihydro-2H-chromene-6-carboxamide

N-[(3S,4R)-6-(5-amino-3-phenylpyrazole-1-carbonyl)-3-hydroxy-2,2-dimethyl-3,4-dihydrochromen-4-yl]-4-ethylbenzenesulfonamide

(R)-7-(3,4-dichlorophenyl)-5-methyl-6-(1-p-tolyl-1H-1,2,4-triazol-5-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

N-(3-morpholin-4-ylsulfonylphenyl)-5-phenyl-2-pyrimidin-5-ylquinazolin-4-amine

((R)-7-(3,4-Dichlorophenyl)-5-methyl-4,7-dihydropyrazolo-[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone

(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-phenylpiperazin-1-yl)methanone

(R)-7-(3,4-dichlorophenyl)-6-(1-(6-methoxypyridin-2-yl)-1H-1,2,4-triazol-5-yl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

[4-[[(4-methoxy-1-methylindazol-3-yl)amino]methyl]-4-phenylcyclohexyl] N-ethylcarbamate

N-[(3R,4S)-6-[(2R)-2-[(2,6-dimethylanilino)methyl]pyrrolidine-1-carbonyl]-3-hydroxy-2,2-dimethyl-3,4-dihydrochromen-4-yl]-4-ethylbenzenesulfonamide

(R)-7-(3,4-dichlorophenyl)-6-(1-isopropyl-1H-1,2,4-triazol-5-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

CHEMBL3622350

N-[(7R,8R)-7-hydroxy-8-[(4-propylphenyl)sulfonylamino]-5,6,7,8-tetrahydronaphthalen-2-yl]-3-methoxybenzamide

5-(1-cyclohexylvinyl)-4-(3,4-dimethylphenyl)-6-methyl-4,7-dihydro-3aH-indene

5-phenyl-N-(pyridin-2-ylmethyl)-2-pyrimidin-5-ylquinazolin-4-amine

[4-[[(4-methoxy-1,1-dioxo-1,2-benzothiazol-3-ylidene)amino]methyl]-4-phenylcyclohexyl] N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)carbamate

6-(5-chloro-1-isopropyl-1H-benzo[d]imidazol-2-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-6-(1-cyclobutyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-2,5-dimethyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-7-(3,4-dichlorophenyl)-5-methyl-2-(trifluoromethyl)-6-(1-(6-(trifluoromethyl)pyridin-2-yl)-1H-1,2,4-triazol-5-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-7-(3,4-dichlorophenyl)-6-(1-(3-fluorophenyl)-1H-1,2,4-triazol-5-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-7-(3,4-dichlorophenyl)-6-(1-(2-ethoxyethyl)-1H-imidazol-2-yl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

7-(3,4-dichlorophenyl)-5-methyl-N-phenethyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide

((R)-7-(3,4-Dichlorophenyl)-2,5-dimethyl-4,7-dihydropyrazolo-[1,5-a]pyrimidin-6-yl)((S)-2-(4-fluorophenyl)pyrrolidin-1-yl)-methanone

2-(2-methoxypyrimidin-5-yl)-5-phenyl-N-(pyridin-2-ylmethyl)quinazolin-4-amine

5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]pyridine-2-carboxamide

N-[5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]pyridin-3-yl]acetamide

((R)-7-(3,4-Dichlorophenyl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone

(R)-7-(3,4-dichlorophenyl)-5-methyl-6-(1-propyl-1H-1,2,4-triazol-5-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-7-(3,4-dichlorophenyl)-5-methyl-6-(1-(4,4,4-trifluorobutyl)-1H-1,2,4-triazol-5-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

N-[(4S)-6-[(2S)-2-[(2,6-dimethylanilino)methyl]pyrrolidine-1-carbonyl]-2,2-dimethyl-3,4-dihydrochromen-4-yl]-4-ethylbenzenesulfonamide

7-(3,4-dichlorophenyl)-6-(1,7-dimethyl-1H-benzo[d]imidazol-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

5-[5-phenyl-4-(pyridin-2-ylmethylamino)quinazolin-2-yl]-1H-pyridin-2-one

(R)-7-(3,4-dichlorophenyl)-6-(1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(7R)-7-(3,4-dichlorophenyl)-6-(1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

5-methoxy-N-(2-methyl-2-phenylpropyl)quinazolin-4-amine

(3S,4R)-4-(4-ethyl-N-(pyridin-2-ylmethyl)phenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenethylchroman-6-carboxamide

(3S,4R)-4-(4-ethyl-N-neopentylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenethylchroman-6-carboxamide

(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone

rac-[7-(3,4-dichlorophenyl)-2,5-dimethyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl]-[4-(4-fluorophenyl)piperazin-1-yl]methanone

(R)-6-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-2,5-dimethyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-7-(3,4-dichlorophenyl)-6-(1-ethyl-1H-imidazol-2-yl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

N-[(3S,4R)-6-[(2R)-2-[(2,6-dimethylanilino)methyl]pyrrolidine-1-carbonyl]-3-hydroxy-2,2-dimethyl-3,4-dihydrochromen-4-yl]-4-ethylbenzenesulfonamide

(3S,4R)-4-(4-ethyl-N-(pyridin-3-ylmethyl)phenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenethylchroman-6-carboxamide

(R)-6-(1-benzyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

[4-[[(4-methoxy-1H-indazol-3-yl)amino]methyl]-4-phenylcyclohexyl] N-ethylcarbamate

N-[(7R,8R)-8-[(4-butylphenyl)sulfonylamino]-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl]-3-methoxybenzamide

(7-(3,5-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone

rac-(7-(3,4-Dichlorophenyl)-2,5-dimethyl-4,7-dihydropyrazolo-[1,5-a]pyrimidin-6-yl)(4-phenylpiperazin-1-yl)methanone

(3S,4R)-3-hydroxy-2,2-dimethyl-N-phenethyl-4-(2-(trifluoromethoxy)phenylsulfonamido)chroman-6-carboxamide

7-(3,4-dichlorophenyl)-5-methyl-6-(7-methyl-1H-benzo[d]imidazol-2-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

7-(3,4-dichlorophenyl)-6-(7-fluoro-1-methyl-1H-benzo[d]imidazol-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(2-phenylpyrrolidin-1-yl)methanone

(2S)-methyl 1-(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carbonyl)pyrrolidine-2-carboxylate

((S)-5-(Methoxymethyl)-7-(1-methyl-1H-indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone

(R)-7-(3,4-dichlorophenyl)-5-methyl-6-(1-(3,3,3-trifluoropropyl)-1H-1,2,4-triazol-5-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-phenylpiperidin-1-yl)methanone

N-[(7R,8R)-8-[(4-tert-butylphenyl)sulfonylamino]-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl]-3-methoxybenzamide

(S)-(7-(2,3-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone

(7-(benzofuran-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone

N-benzyl-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide

(7-(2,3-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone

(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(3-(4-fluorophenyl)pyrrolidin-1-yl)methanone

((R)-7-(3,4-Dichlorophenyl)-2,5-dimethyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)-pyrrolidin-1-yl)methanone

(R)-6-(1-cyclobutyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(3S,4R)-N-((S)-1-benzylpyrrolidin-3-yl)-N-ethyl-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromene-6-carboxamide

(3S,4R)-N-(2-fluorobenzyl)-N-ethyl-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromene-6-carboxamide

7-(3,4-dichlorophenyl)-5-methyl-N-phenyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide

CHEMBL3622349

4-methoxy-N-methyl-N-(2-methyl-2-phenylpropyl)-1,2-benzoxazol-3-amine

(7-(3-chlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone

azepan-1-yl(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)methanone

(R)-6-(1-(6-chloropyridin-2-yl)-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-7-(3,4-dichlorophenyl)-6-(1-ethyl-1H-1,2,4-triazol-5-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

5-methoxy-4-[(2-methyl-2-phenylpropyl)amino]-1,3-benzoxazin-2-one

4-methoxy-1-methyl-N-(2-methyl-2-phenylpropyl)-1H-indazol-3-amine

(E)-N-[(7R,8R)-8-[(4-ethylphenyl)sulfonylamino]-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl]-3-phenylprop-2-enamide

(3R,4S)-N-((S)-1-benzylpyrrolidin-3-yl)-N-ethyl-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromene-6-carboxamide

(3S,4R)-3-hydroxy-2,2-dimethyl-N-phenethyl-4-(4-(trifluoromethyl)phenylsulfonamido)chroman-6-carboxamide

(4-(4-fluorophenyl)piperazin-1-yl)(5-methyl-7-(3-methylbenzo[b]thiophen-2-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)methanone

(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(methoxymethyl)pyrrolidin-1-yl)methanone

7-(3,4-dichlorophenyl)-6-(1,5-dimethyl-1H-benzo[d]imidazol-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

methyl 2-(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)-1-methyl-1H-benzo[d]imidazole-5-carboxylate

(R)-7-(3,4-dichlorophenyl)-5-methyl-6-(1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-7-(3,4-dichlorophenyl)-6-(1-isopropyl-1H-imidazol-2-yl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

rac-(2-Chloro-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo-[1,5-a]pyrimidin-6-yl)(4-fluorophenylpiperazin-1-yl)methanone

(3S,4R)-N-((R)-1-benzylpyrrolidin-3-yl)-N-ethyl-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromene-6-carboxamide

2-chloro-N-(3-morpholin-4-ylsulfonylphenyl)-5-phenylquinazolin-4-amine

(R)-7-(3,4-dichlorophenyl)-5-methyl-6-(1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

4-ethyl-N-(2-methyl-2-phenylpropyl)-1,2-benzoxazol-3-amine

(R)-1-(3-chlorobenzyl)-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl)pyrrolidine-2-carboxamide

(3R,4S)-N-((R)-1-benzylpyrrolidin-3-yl)-N-ethyl-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromene-6-carboxamide

2-(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)-1-methyl-1H-benzo[d]imidazole-5-carbonitrile

(R)-7-(3,4-dichlorophenyl)-6-(1-(6-ethoxypyridin-2-yl)-1H-1,2,4-triazol-5-yl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-6-(1-tert-butyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

((R)-2-Cyclopropyl-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone

(R)-6-(1-(cyclopropylmethyl)-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

benzyl N-[(7R,8R)-8-[(4-ethylphenyl)sulfonylamino]-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl]carbamate

(7-(5-chlorothiophen-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone

4-ethyl-N-((3S,4R)-3-hydroxy-2,2-dimethyl-6-((phenethylamino)methyl)chroman-4-yl)benzenesulfonamide

N-[(7R,8R)-8-[(4-ethylphenyl)sulfonylamino]-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl]-3-phenylpropanamide

(R)-7-(3,4-dichlorophenyl)-6-(1-(6-fluoropyridin-2-yl)-1H-1,2,4-triazol-5-yl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(3S,4R)-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenethyl-3,4-dihydro-2H-chromene-6-carboxamide

N-[(3R,4S)-6-[(2S)-2-[(2,6-dimethylanilino)methyl]pyrrolidine-1-carbonyl]-3-hydroxy-2,2-dimethyl-3,4-dihydrochromen-4-yl]-4-ethylbenzenesulfonamide

(3S,4R)-4-(4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenyl-3,4-dihydro-2H-chromene-6-carboxamide

3-[(2-methyl-2-phenylpropyl)amino]-1,2-benzoxazol-4-ol

(S)-N-(8-(4-ethylphenylsulfonamido)-5,6,7,8-tetrahydronaphthalen-2-yl)-3-phenylpropanamide

(3S,4R)-4-(4-ethylphenylsulfonamido)-3-hydroxy-N,2,2-trimethyl-N-phenyl-3,4-dihydro-2H-chromene-6-carboxamide

(3S,4R)-4-(N-((1H-imidazol-4-yl)methyl)-4-ethylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenethylchroman-6-carboxamide

(7-(2,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone

((S)-7-(Benzo[d]thiazol-2-yl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone

(R)-2-tert-butyl-6-(1-cyclobutyl-1H-1,2,4-triazol-5-yl)-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl)-1-(3-(trifluoromethoxy)benzyl)pyrrolidine-2-carboxamide

N-[(3S,4R)-4-[(4-ethylphenyl)sulfonylamino]-3-hydroxy-2,2-dimethyl-3,4-dihydrochromen-6-yl]-3-methoxybenzamide

7-(3,4-dichlorophenyl)-6-(6-fluoro-1-methyl-1H-benzo[d]imidazol-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine

(R)-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl)-1-(3-methoxybenzyl)pyrrolidine-2-carboxamide

(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)((S)-2-(4,5-dimethylthiazol-2-yl)pyrrolidin-1-yl)methanone

N,N-dibutyl-7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide

(7-(3,4-dichlorophenyl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(2-(pyridin-4-yl)pyrrolidin-1-yl)methanone

(3S,4R)-N-(4-bromophenyl)-4-[(4-ethylphenyl)sulfonylamino]-3-hydroxy-2,2-dimethyl-3,4-dihydrochromene-6-carboxamide

(3S,4R)-4-(4-ethyl-N-isobutylphenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenethylchroman-6-carboxamide

5-[4-(dimethylamino)phenyl]-N-(pyridin-2-ylmethyl)-2-pyrimidin-5-ylquinazolin-4-amine

4-chloro-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl)benzamide

(3S,4R)-3-hydroxy-2,2-dimethyl-4-(3-methylphenylsulfonamido)-N-phenethylchroman-6-carboxamide

(1S,2S)-N-((7R,8R)-8-(4-ethylphenylsulfonamido)-7-hydroxy-5,6,7,8-tetrahydronaphthalen-2-yl)-2-phenylcyclopropanecarboxamide

(3S,4R)-N-ethyl-4-[(4-ethylphenyl)sulfonylamino]-3-hydroxy-2,2-dimethyl-N-phenyl-3,4-dihydropyrano[2,3-b]pyridine-6-carboxamide

(R)-7-(3,4-dichlorophenyl)-5-methyl-6-(1-(5-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

(3S,4R)-3-hydroxy-2,2-dimethyl-4-(4-methylphenylsulfonamido)-N-phenethylchroman-6-carboxamide

(R)-7-(3,4-dichlorophenyl)-5-methyl-6-(1-(4-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine

rac-(7-(3,4-Dichlorophenyl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)-piperazin-1-yl)methanone