Brief Information of the Compound and Protein
Compound Name
(7-(5-chlorothiophen-2-yl)-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl)(4-(4-fluorophenyl)piperazin-1-yl)methanone
    Show/Hide
PubChem ID
CID: 135843976
Canonical SMILES
CC1=C(C(=O)N2CCN(c3ccc(F)cc3)CC2)C(c2ccc(Cl)s2)n2nccc2N1
    Show/Hide
Compound Formula C22H21ClFN5OS
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily A member 5
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Potassium channels
>
Voltage-gated potassium channel
Uniprot ID
P22460
Gene Name
KCNA5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000309 NCTC clone 929 Mus musculus (Mouse)  1
1
IC50 = 230 nM
   TI
   LI
   LO
   TS