Brief Information of the Compound and Protein
Compound Name
(R)-7-(3,4-dichlorophenyl)-6-(1-(6-fluoropyridin-2-yl)-1H-1,2,4-triazol-5-yl)-5-methyl-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine
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PubChem ID
CID: 136226195
SID: 163594540
Canonical SMILES
CC1=C(c2ncnn2-c2cccc(F)n2)[C@@H](c2ccc(Cl)c(Cl)c2)n2nc(C(F)(F)F)cc2N1
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Compound Formula C21H13Cl2F4N7
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily A member 5
Protein Classification
Ion channel
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Voltage-gated ion channel
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Potassium channels
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Voltage-gated potassium channel
Uniprot ID
P22460
Gene Name
KCNA5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000309 NCTC clone 929 Mus musculus (Mouse)  1
1
IC50 = 256 nM
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