| Compound ID |
Compound Name |
Compound Formula |
|
CP0510498
|
5-[2-(4-Fluorophenyl)ethyl]-2,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C21H23FN2
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0506291
|
8-Fluoro-2-methyl-5-(2-p-tolylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C21H23FN2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0492826
|
8-Fluoro-5-[2-(4-methoxyphenyl)ethyl]-2-methyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C21H23FN2O
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0498731
|
2-Methyl-5-((Z)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C20H20N2
|
2
|
| 1 |
IC50 = 33 nM
|
|
|
| 2 |
IC50 = 181 nM
|
|
|
|
CP0436736
|
8-Fluoro-2-methyl-5-[2-(4-trifluoromethylphenyl)ethyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C21H20F4N2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0237538
|
2,8-Dimethyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C21H24N2
|
2
|
| 1 |
IC50 = 40 nM
|
|
|
| 2 |
IC50 = 146 nM
|
|
|
|
CP0446549
|
8-Fluoro-2-methyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C20H21FN2
|
2
|
| 1 |
IC50 = 40 nM
|
|
|
| 2 |
IC50 = 131 nM
|
|
|
|
CP0439140
|
5-[2-(4-Methoxyphenyl)ethyl]-2,8-dimethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C22H26N2O
|
1
|
| 1 |
IC50 = 66 nM
|
|
|
|
CP0439139
|
2-Methyl-5-phenethyl-8-trifluoromethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C21H21F3N2
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0150364
|
2,8-Dimethyl-5-((Z)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C21H22N2
|
2
|
| 1 |
IC50 = 70 nM
|
|
|
| 2 |
IC50 = 154 nM
|
|
|
|
CP0453872
|
2,8-Dimethyl-5-[2-(4-trifluoromethylphenyl)ethyl]-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C22H23F3N2
|
1
|
| 1 |
IC50 = 98 nM
|
|
|
|
CP0424945
|
2-methyl-5-(2-(pyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C19H21N3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0446548
|
8-Methoxy-2-methyl-5-phenethyl-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C21H24N2O
|
1
|
| 1 |
IC50 = 104 nM
|
|
|
|
CP0390109
|
8-fluoro-2-methyl-5-(2-(6-methylpyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C20H22FN3
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0353494
|
2,8-Dimethyl-5-(2-p-tolylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C22H26N2
|
1
|
| 1 |
IC50 = 112 nM
|
|
|
|
CP0378179
|
2-methyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C19H21N3
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0378180
|
8-bromo-2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C19H20BrN3
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0478590
|
8-fluoro-2-methyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C19H20FN3
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0017601
|
2,8-dimethyl-5-[2-(6-methylpyridin-3-yl)ethyl]-3,4-dihydro-1H-pyrido[4,3-b]indole
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|
C21H25N3
|
3
|
| 1 |
IC50 = 158 nM
|
|
|
| 2 |
IC50 = 160 nM
|
|
|
| 3 |
IC50 = 1580 nM
|
|
|
|
CP0375182
|
2,8-dimethyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C20H23N3
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0390108
|
2-methyl-5-(2-(pyridin-4-yl)ethyl)-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C20H20F3N3
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0524738
|
2,8-dimethyl-5-(2-pyrazine-2-ylethyl)-gamma-carboline
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|
C19H22N4
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0430385
|
2-Methyl-5-((E)-styryl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C20H22N2
|
2
|
| 1 |
IC50 = 345 nM
|
|
|
| 2 |
IC50 = 2130 nM
|
|
|
|
CP0524739
|
8-methoxy-2-methyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
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|
C20H23N3O
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0494107
|
2,8-dimethyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H23N3
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0501165
|
2,8-dimethyl-5-(2-(pyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H23N3
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0460301
|
2-methyl-5-(2-(pyridin-2-yl)ethyl)-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H20F3N3
|
1
|
| 1 |
IC50 = 560 nM
|
|
|
|
CP0389115
|
8-fluoro-2-methyl-5-(2-(pyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C19H20FN3
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0378181
|
8-fluoro-2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C19H20FN3
|
1
|
| 1 |
IC50 = 940 nM
|
|
|
|
CP0524747
|
2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole-8-carbonitrile
Show/Hide
|
C20H20N4
|
1
|
| 1 |
IC50 = 1290 nM
|
|
|
|
CP0377931
|
2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C19H21N3
|
1
|
| 1 |
IC50 = 1820 nM
|
|
|
|
CP0375183
|
8-methyl-2-(1-methylpiperidin-4-yl)-5-(2-(pyridin-3-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C25H32N4
|
1
|
| 1 |
IC50 = 2790 nM
|
|
|
|
CP0524501
|
8-methoxy-2-methyl-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H23N3O
|
1
|
| 1 |
IC50 = 4670 nM
|
|
|
|
CP0377930
|
2-methyl-8-pyridin-3-yl-5-(2-pyridin-2-ylethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C24H24N4
|
1
|
| 1 |
IC50 = 7160 nM
|
|
|
|
CP0507760
|
8-methyl-2-(1-methylpiperidin-4-yl)-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C25H32N4
|
1
|
| 1 |
IC50 = 7570 nM
|
|
|
|
CP0377932
|
2-methyl-5-(2-(pyridin-4-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole-8-carboxylic acid
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|
C20H21N3O2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0390107
|
2-methyl-5-(2-(pyridin-3-yl)ethyl)-8-(trifluoromethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C20H20F3N3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0503462
|
8-methyl-2-(1-methylpiperidin-4-yl)-5-(2-(pyridin-2-yl)ethyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole
Show/Hide
|
C25H32N4
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
