Brief Information of the Compound and Protein
Compound Name
2,8-dimethyl-5-(2-pyrazine-2-ylethyl)-gamma-carboline
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PubChem ID
CID: 54583938
Canonical SMILES
CN1CCc2c(C1)c1cc(C)ccc1n2CCc1cnccn1
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Compound Formula C19H22N4
Compound Structure
Protein Name
Histamine H1 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
P35367
Gene Name
HRH1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000289 SK-N-SH Homo sapiens (Human)  1
1
IC50 = 320 nM
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