| Compound ID |
Compound Name |
Compound Formula |
|
CP0471587
|
2-(4-Chlorophenyl)-2-(1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidin-4-ylidene)acetonitrile
Show/Hide
|
C18H19ClN4O2S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0559140
|
2-(4-Chlorophenyl)-2-(1-((1,3,5-trimethyl-1H-pyrazol-4-yl) sulfonyl)piperidin-4-ylidene)acetonitrile
Show/Hide
|
C19H21ClN4O2S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0545986
|
2-(4-Chlorophenyl)-2-(1-((3,5-diethyl-1H-pyrazol-4-yl) sulfonyl)piperidin-4-ylidene)acetonitrile
Show/Hide
|
C20H23ClN4O2S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0548098
|
US10167273, Example 79
Show/Hide
|
C19H26ClN3O3S
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0493341
|
3-((1-(3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)piperidin-4-ylidene) fluoromethyl)quinoline
Show/Hide
|
C20H21FN4O2S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0572273
|
US10167273, Example 99
Show/Hide
|
C19H26ClN3O3S
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0572277
|
US10167273, Example 78
Show/Hide
|
C18H24ClN3O3S
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0500937
|
US10167273, Example 91
Show/Hide
|
C19H25ClFN3O3S
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0467354
|
2-(1-((3,5-Dimethyl-1H-pyrazol-4-yl)sulfonyl)piperidin-4-ylidene)-2-(4-(trifluoromethoxy)phenypacetonitrile
Show/Hide
|
C19H19F3N4O3S
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0551071
|
4-((4-Chlorophenyl)fluoromethylene)-1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C17H19ClFN3O2S
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0481219
|
US10167273, Example 74
Show/Hide
|
C18H24ClN3O4S
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0537358
|
US10167273, Example 90
Show/Hide
|
C18H23ClFN3O3S
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0536439
|
2-(4-Chloro-2-fluorophenyl)-2-(1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidin-4-ylidene)acetonitrile
Show/Hide
|
C18H18ClFN4O2S
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0566092
|
4-((4-Chloro-3-fluorophenyl)fluoromethylene)-1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C17H18ClF2N3O2S
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0537353
|
US10167273, Example 73
Show/Hide
|
C17H22ClN3O4S
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0572278
|
US10167273, Example 88
Show/Hide
|
C19H26ClN3O4S
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0519133
|
2-(4-Chlorophenyl)-2-(1-((1,5-dimethyl-3-(trifluoromethyl)-1H-pyrazol-4-yl) sulfonyl)piperidin-4-ylidene)acetonitrile
Show/Hide
|
C19H18ClF3N4O2S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0544405
|
US10167273, Example 40
Show/Hide
|
C17H19ClF3N3O3S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0574115
|
US10167273, Example 39
Show/Hide
|
C18H21ClF3N3O3S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0475705
|
US10167273, Example 23
Show/Hide
|
C21H25N3O3S
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0536059
|
US10167273, Example 34
Show/Hide
|
C17H19ClN4O3S
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0469162
|
4-((2,4-Dichlorophenyl)fluoromethylene)-1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C17H18Cl2FN3O2S
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0541825
|
[3-(5-chloro-3-methylpyridin-2-yl)-3-fluoropiperidin-1-yl]-[2-(methylamino)pyridin-4-yl]methanone
Show/Hide
|
C18H20ClFN4O
|
1
|
| 1 |
IC50 = 290 nM
|
|
|
|
CP0515717
|
US10167273, Example 31
Show/Hide
|
C18H21ClN4O3S
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0541162
|
[2-(dimethylamino)pyridin-4-yl]-[3-(1-propan-2-ylbenzimidazol-2-yl)piperidin-1-yl]methanone
Show/Hide
|
C23H29N5O
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0519662
|
US10167273, Example 28
Show/Hide
|
C19H25Cl2N3O3S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0528881
|
(1-ethylpyrazol-4-yl)-[3-(1-propan-2-ylindol-2-yl)piperidin-1-yl]methanone
Show/Hide
|
C22H28N4O
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0904519
|
US9475795, 111
Show/Hide
|
C18H22ClF2N3O2S
|
1
|
| 1 |
IC50 = 340 nM
|
|
|
|
CP0551072
|
4-((4-Chloro-2-fluorophenyl)fluoromethylene)-1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C17H18ClF2N3O2S
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0548100
|
US10167273, Example 89
Show/Hide
|
C18H24ClN3O4S
|
1
|
| 1 |
IC50 = 410 nM
|
|
|
|
CP0544409
|
US10167273, Example 72
Show/Hide
|
C18H23ClFN3O2S
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0572268
|
US10167273, Example 33
Show/Hide
|
C20H23N3O3S
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0967192
|
2-(4-Chlorophenyl)-2-(1-((3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl)-3-methylpiperidin-4-ylidene)acetonitrile
Show/Hide
|
C19H21ClN4O2S
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0475710
|
US10167273, Example 14
Show/Hide
|
C17H21BrFN3O3S
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0914835
|
US9475795, 102
Show/Hide
|
C18H24ClN3O2S
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
|
CP0481217
|
US10167273, Example 30
Show/Hide
|
C17H21ClFN3O3S
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
|
CP0461661
|
4-((3,4-Dichlorophenyl)fluoromethylene)-1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C17H18Cl2FN3O2S
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0474877
|
US10167273, Example 55
Show/Hide
|
C18H24ClN3O2S
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0490998
|
US10167273, Example 67
Show/Hide
|
C17H22ClN3O2S
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
|
CP0531514
|
US10167273, Example 5
Show/Hide
|
C17H22ClN3O3S
|
1
|
| 1 |
IC50 = 530 nM
|
|
|
|
CP0566091
|
4-(4-Chloro-2-fluorobenzylidene)-1-((1,3,5-trimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C18H21ClFN3O2S
|
1
|
| 1 |
IC50 = 550 nM
|
|
|
|
CP0455524
|
4-(4-Chloro-2-fluorobenzylidene)-1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C17H19ClFN3O2S
|
1
|
| 1 |
IC50 = 600 nM
|
|
|
|
CP0953593
|
US9475795, 93
Show/Hide
|
C18H21ClN4O2S
|
1
|
| 1 |
IC50 = 610 nM
|
|
|
|
CP0566337
|
US10167273, Example 63
Show/Hide
|
C21H28BrN3O4S
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0423920
|
US10167273, Example 81
Show/Hide
|
C18H22ClF2N3O2S
|
1
|
| 1 |
IC50 = 670 nM
|
|
|
|
CP0544407
|
US10167273, Example 62
Show/Hide
|
C20H26BrN3O4S
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
|
CP0423921
|
US10167273, Example 95
Show/Hide
|
C18H24ClN3O3S
|
1
|
| 1 |
IC50 = 710 nM
|
|
|
|
CP0537357
|
US10167273, Example 84
Show/Hide
|
C17H23ClN4O4S
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0929619
|
US9475795, 104
Show/Hide
|
C19H26ClN3O3S
|
1
|
| 1 |
IC50 = 720 nM
|
|
|
|
CP0572272
|
US10167273, Example 83
Show/Hide
|
C18H23ClFN3O2S
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0545987
|
4-(4-Chlorobenzylidene)-1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C17H20ClN3O2S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0567316
|
4-(1-(4-Chlorophenypethylidene)-1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C18H22ClN3O2S
|
1
|
| 1 |
IC50 = 760 nM
|
|
|
|
CP0515728
|
US10167273, Example 71
Show/Hide
|
C17H21ClFN3O2S
|
1
|
| 1 |
IC50 = 780 nM
|
|
|
|
CP0548090
|
US10167273, Example 13
Show/Hide
|
C17H21Cl2N3O3S
|
1
|
| 1 |
IC50 = 790 nM
|
|
|
|
CP0475713
|
US10167273, Example 80
Show/Hide
|
C17H20ClF2N3O2S
|
1
|
| 1 |
IC50 = 810 nM
|
|
|
|
CP0548102
|
US10167273, Example 4
Show/Hide
|
C18H25N3O3S
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0515716
|
US10167273, Example 11
Show/Hide
|
C17H22ClN3O3S
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0518651
|
US10167273, Example 64
Show/Hide
|
C18H21ClN4O2S
|
1
|
| 1 |
IC50 = 890 nM
|
|
|
|
CP0481218
|
US10167273, Example 60
Show/Hide
|
C20H28ClN3O3S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0566336
|
US10167273, Example 53
Show/Hide
|
C18H25ClN4O2S
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
|
CP0549322
|
(3-amino-1-methylpyrazol-4-yl)-[3-(5-chloro-1-ethylindol-2-yl)piperidin-1-yl]methanone
Show/Hide
|
C20H24ClN5O
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0475709
|
US10167273, Example 65
Show/Hide
|
C18H20Cl2N4O2S
|
1
|
| 1 |
IC50 = 940 nM
|
|
|
|
CP0493478
|
US10167273, Example 56
Show/Hide
|
C18H23Cl2N3O2S
|
1
|
| 1 |
IC50 = 950 nM
|
|
|
|
CP0423926
|
US10167273, Example 46
Show/Hide
|
C17H20ClF2N3O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0519659
|
US10167273, Example 2
Show/Hide
|
C16H19Cl2N3O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0572271
|
US10167273, Example 49
Show/Hide
|
C18H22ClN3O3S
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0486276
|
US10167273, Example 66
Show/Hide
|
C19H26ClN3O2S
|
1
|
| 1 |
IC50 = 1010 nM
|
|
|
|
CP0566343
|
US10167273, Example 82
Show/Hide
|
C17H21ClFN3O2S
|
1
|
| 1 |
IC50 = 1020 nM
|
|
|
|
CP0490997
|
US10167273, Example 61
Show/Hide
|
C21H28ClN3O4S
|
1
|
| 1 |
IC50 = 1080 nM
|
|
|
|
CP0475706
|
US10167273, Example 29
Show/Hide
|
C17H19Cl2F2N3O3S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0475707
|
US10167273, Example 35
Show/Hide
|
C16H19ClFN3O3S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0536060
|
US10167273, Example 36
Show/Hide
|
C16H19Cl2N3O3S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0475711
|
US10167273, Example 22
Show/Hide
|
C16H19Cl2N3O3S
|
1
|
| 1 |
IC50 = 1180 nM
|
|
|
|
CP0515730
|
US10167273, Example 85
Show/Hide
|
C16H21ClN4O4S
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
|
CP0481214
|
US10167273, Example 25
Show/Hide
|
C16H18Cl3N3O3S
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0493340
|
4-(4-Chloro-3-fluorobenzyl)-1-((3-cyclopropyl-5-methyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C19H23ClFN3O2S
|
1
|
| 1 |
IC50 = 1370 nM
|
|
|
|
CP0481212
|
US10167273, Example 1
Show/Hide
|
C17H21Cl2N3O3S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0481213
|
US10167273, Example 3
Show/Hide
|
C18H22F3N3O4S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0515726
|
US10167273, Example 45
Show/Hide
|
C17H21ClFN3O3S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0519660
|
US10167273, Example 8
Show/Hide
|
C16H20ClN3O3S
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
|
CP0423916
|
US10167273, Example 51
Show/Hide
|
C17H23ClN4O2S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0548105
|
US10167273, Example 24
Show/Hide
|
C18H24ClN3O3S
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0548093
|
US10167273, Example 57
Show/Hide
|
C18H24ClN3O3S
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0545988
|
4-((2,4-Difluorophenyl)fluoromethylene)-1-(3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidine
Show/Hide
|
C17H18F3N3O2S
|
1
|
| 1 |
IC50 = 1630 nM
|
|
|
|
CP0566344
|
US10167273, Example 108
Show/Hide
|
C17H22ClN3O3S
|
1
|
| 1 |
IC50 = 1640 nM
|
|
|
|
CP0563168
|
US10167273, Example 26
Show/Hide
|
C17H18Cl2F3N3O3S
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0574118
|
US10167273, Example 10
Show/Hide
|
C18H22F3N3O3S
|
1
|
| 1 |
IC50 = 1700 nM
|
|
|
|
CP0916590
|
US9475795, 94
Show/Hide
|
C17H22ClN3O3S
|
1
|
| 1 |
IC50 = 1740 nM
|
|
|
|
CP0499644
|
US10167273, Example 103
Show/Hide
|
C16H21ClN4O2S
|
1
|
| 1 |
IC50 = 1760 nM
|
|
|
|
CP0913833
|
US9475795, 92
Show/Hide
|
C18H20ClFN4O2S
|
1
|
| 1 |
IC50 = 1850 nM
|
|
|
|
CP0904788
|
US9475795, 109
Show/Hide
|
C19H26ClN3O3S
|
1
|
| 1 |
IC50 = 1860 nM
|
|
|
|
CP0374927
|
4-((3-Chloro-4-fluorophenyl)fluoromethylene)-1-((3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl) piperidine
Show/Hide
|
C17H18ClF2N3O2S
|
1
|
| 1 |
IC50 = 1880 nM
|
|
|
|
CP0490996
|
US10167273, Example 47
Show/Hide
|
C16H19ClFN3O3S
|
1
|
| 1 |
IC50 = 1900 nM
|
|
|
|
CP0537356
|
US10167273, Example 68
Show/Hide
|
C17H21Cl2N3O2S
|
1
|
| 1 |
IC50 = 2020 nM
|
|
|
|
CP0423915
|
US10167273, Example 21
Show/Hide
|
C18H24ClN3O3S
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0544406
|
US10167273, Example 50
Show/Hide
|
C18H21Cl2N3O3S
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0572274
|
US10167273, Example 6
Show/Hide
|
C17H22ClN3O3S
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0515650
|
US10167273, Example 9
Show/Hide
|
C19H27N3O3S
|
1
|
| 1 |
IC50 = 2300 nM
|
|
|
|
CP0943103
|
US9475795, 101
Show/Hide
|
C18H24ClN3O3S
|
1
|
| 1 |
IC50 = 2380 nM
|
|
|
|
CP0515727
|
US10167273, Example 59
Show/Hide
|
C18H23Cl2N3O3S
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0566342
|
US10167273, Example 58
Show/Hide
|
C19H26ClN3O3S
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0537355
|
US10167273, Example 52
Show/Hide
|
C17H22Cl2N4O2S
|
1
|
| 1 |
IC50 = 2700 nM
|
|
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CP0490995
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US10167273, Example 15
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C16H19Cl2N3O3S
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1
|
| 1 |
IC50 = 2900 nM
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CP0904790
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US9475795, 110
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C18H25N3O3S
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1
|
| 1 |
IC50 = 3010 nM
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CP0471586
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Methyl 2-(4-Chlorophenyl)-2-(1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidin-4-ylidene)acetate
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C19H22ClN3O4S
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1
|
| 1 |
IC50 = 3100 nM
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CP0548096
|
US10167273, Example 77
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C16H20ClFN4O3S
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1
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| 1 |
IC50 = 3190 nM
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CP0519663
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US10167273, Example 38
Show/Hide
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C18H25N3O3S
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1
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| 1 |
IC50 = 3200 nM
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CP0577315
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US10167273, Example 32
Show/Hide
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C17H20F3N3O4S
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1
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| 1 |
IC50 = 3400 nM
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CP0490927
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US10167273, Example 20
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C17H22FN3O3S
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1
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| 1 |
IC50 = 3600 nM
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CP0572267
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US10167273, Example 17
Show/Hide
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C18H25N3O4S
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1
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| 1 |
IC50 = 3600 nM
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CP0519148
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2-(2,6-Difluorophenyl)-2-(1-((3,5-dimethyl-1H-pyrazol-4-yl) sulfonyl)piperidin-4-ylidene)acetonitrile
Show/Hide
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C18H18F2N4O2S
|
1
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| 1 |
IC50 = 3680 nM
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CP0475712
|
US10167273, Example 76
Show/Hide
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C16H20FN3O3S
|
1
|
| 1 |
IC50 = 3730 nM
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CP0519664
|
US10167273, Example 48
Show/Hide
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C16H21ClN4O3S
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1
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| 1 |
IC50 = 3800 nM
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CP0493486
|
US10167273, Example 86
Show/Hide
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C19H26ClN3O4S
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1
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| 1 |
IC50 = 4600 nM
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CP0519661
|
US10167273, Example 16
Show/Hide
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C17H19ClF3N3O3S
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1
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| 1 |
IC50 = 4600 nM
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CP0474878
|
US10167273, Example 12
Show/Hide
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C18H22F3N3O3S
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1
|
| 1 |
IC50 = 4700 nM
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CP0486381
|
US10167273, Example 44
Show/Hide
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C18H23F2N3O4S
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1
|
| 1 |
IC50 = 5100 nM
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CP0566341
|
US10167273, Example 54
Show/Hide
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C18H24Cl2N4O2S
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1
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| 1 |
IC50 = 5200 nM
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CP0525445
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2-(2,6-Difluorophenyl)-2-(1-((1,3,5-trimethyl-1H-pyrazol-4-yl) sulfonyl)piperidin-4-ylidene)acetonitrile
Show/Hide
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C19H20F2N4O2S
|
1
|
| 1 |
IC50 = 5430 nM
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CP0475704
|
US10167273, Example 19
Show/Hide
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C17H23N3O3S
|
1
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| 1 |
IC50 = 5600 nM
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CP0481215
|
US10167273, Example 27
Show/Hide
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C16H19Cl2N3O3S
|
1
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| 1 |
IC50 = 5600 nM
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CP0481216
|
US10167273, Example 87
Show/Hide
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C20H28ClN3O4S
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1
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| 1 |
IC50 = 5880 nM
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CP0572269
|
US10167273, Example 41
Show/Hide
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C17H22FN3O4S
|
1
|
| 1 |
IC50 = 5900 nM
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|
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CP0572276
|
US10167273, Example 42
Show/Hide
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C17H21F2N3O4S
|
1
|
| 1 |
IC50 = 5900 nM
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CP0475708
|
US10167273, Example 43
Show/Hide
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C18H24FN3O4S
|
1
|
| 1 |
IC50 = 6300 nM
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CP0548094
|
US10167273, Example 69
Show/Hide
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C18H23Cl2N3O3S
|
1
|
| 1 |
IC50 = 6470 nM
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CP0566338
|
US10167273, Example 75
Show/Hide
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C17H21ClFN3O3S
|
1
|
| 1 |
IC50 = 6980 nM
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CP0499645
|
US10167273, Example 18
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C18H25N3O4S
|
1
|
| 1 |
IC50 = 7000 nM
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CP0572266
|
US10167273, Example 7
Show/Hide
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C18H22N4O3S
|
1
|
| 1 |
IC50 = 7300 nM
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CP0563167
|
US10167273, Example 37
Show/Hide
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C16H20ClN3O3S
|
1
|
| 1 |
IC50 = 7400 nM
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CP0483985
|
[6-(methylamino)pyridazin-4-yl]-[3-(3-methyl-1H-indol-2-yl)piperidin-1-yl]methanone
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|
C20H23N5O
|
1
|
| 1 |
IC50 = 7410 nM
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|
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CP0544408
|
US10167273, Example 70
Show/Hide
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C17H21Cl2N3O3S
|
1
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| 1 |
IC50 = 8620 nM
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CP0908207
|
US9475795, 100
Show/Hide
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C18H24ClN3O3S
|
1
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| 1 |
IC50 = 9420 nM
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CP0457576
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(3-amino-1-methylpyrazol-4-yl)-[3-(5-chloro-3-methylpyridin-2-yl)-3-methoxypiperidin-1-yl]methanone
Show/Hide
|
C17H22ClN5O2
|
1
|
| 1 |
IC50 > 9000 nM
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