| Compound ID |
Compound Name |
Compound Formula |
|
CP0065724
|
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
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|
C22H19N5O4
|
3
|
| 1 |
EC50 > 12500 nM
|
|
|
| 2 |
EC50 > 25000 nM
|
|
|
| 3 |
IC50 > 8000 nM
|
|
|
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CP0088338
|
(1R,2S,4R,5R,6R)-2-amino-4-(1H-1,2,4-triazol-5-ylsulfanyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C10H12N4O4S
|
2
|
| 1 |
EC50 > 25000 nM
|
|
|
| 2 |
IC50 > 12500 nM
|
|
|
|
CP0067673
|
(1S,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C15H15Cl2NO6
|
2
|
| 1 |
EC50 > 25000 nM
|
|
|
| 2 |
IC50 > 12500 nM
|
|
|
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CP0356641
|
(1S,2S,4S,5R,6S)-2-amino-4-[(3-methoxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C16H18N2O6
|
2
|
| 1 |
EC50 > 25000 nM
|
|
|
| 2 |
IC50 > 12500 nM
|
|
|
|
CP0492194
|
(1R,2R)-N-[3-(4-bromophenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C15H15BrN2OS
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0530223
|
(1R,2R)-N-[3-(3-fluoro-4-methoxyphenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C16H17FN2O2S
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0535542
|
(1R,2R)-N-[3-(4-chlorophenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C15H15ClN2OS
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0400064
|
(1R,2R)-N-[3-(4-methoxyphenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C16H18N2O2S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0482876
|
(1R,2R)-N-[3-(3,4-dichlorophenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C15H14Cl2N2OS
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0425303
|
(1R,2R)-2-methyl-N-(4-methyl-3-phenyl-1,2-thiazol-5-yl)cyclopropane-1-carboxamide
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|
C15H16N2OS
|
1
|
| 1 |
IC50 = 65 nM
|
|
|
|
CP0535543
|
(1R,2R)-N-[3-[4-(1,1-difluoroethyl)phenyl]-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C17H18F2N2OS
|
1
|
| 1 |
IC50 = 67 nM
|
|
|
|
CP0530222
|
(1R,2R)-N-[3-(4-ethoxyphenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C17H20N2O2S
|
1
|
| 1 |
IC50 = 92 nM
|
|
|
|
CP0482875
|
(1R,2R)-N-[3-(4-fluorophenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C15H15FN2OS
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0437683
|
(1S,2S)-N-[3-(4-methoxyphenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C16H18N2O2S
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0437684
|
(1R,2R)-N-[3-(4-hydroxyphenyl)-4-methyl-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C15H16N2O2S
|
1
|
| 1 |
IC50 = 138 nM
|
|
|
|
CP0425771
|
(1R,2R)-N-[4-(6-methoxypyridin-2-yl)-3-(2-methylindazol-5-yl)-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C22H21N5O2S
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0851137
|
(1R,2R)-2-methyl-N-(3-(2-methyl-2H-indazol-5-yl)-4-(pyridin-2-yl)isothiazol-5-yl)cyclopropanecarboxamide hydrochloride
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|
C21H20ClN5OS
|
1
|
| 1 |
IC50 = 238 nM
|
|
|
|
CP0864305
|
(1R,2R)-N-(4-(6-ethylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide hydrochloride
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|
C23H24ClN5OS
|
1
|
| 1 |
IC50 = 279 nM
|
|
|
|
CP0857084
|
N-(4-(6-isopropylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)cyclopropanecarboxamide hydrochloride
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|
C23H24ClN5OS
|
1
|
| 1 |
IC50 = 397 nM
|
|
|
|
CP0411064
|
(1R,2R)-2-methyl-N-[3-(2-methylindazol-5-yl)-4-(6-propylpyridin-2-yl)-1,2-thiazol-5-yl]cyclopropane-1-carboxamide
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|
C24H25N5OS
|
1
|
| 1 |
IC50 = 409 nM
|
|
|
|
CP0662728
|
(1R,2R)-N-(4-(6-isopropylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide hydrochloride
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|
C24H26ClN5OS
|
1
|
| 1 |
IC50 = 644 nM
|
|
|
|
CP0857085
|
(1R,2R)-N-(4-(6-cyclobutylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide hydrochloride
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|
C25H26ClN5OS
|
1
|
| 1 |
IC50 = 687 nM
|
|
|
|
CP0871658
|
(1R,2R)-N-(4-(6-cyclopropylpyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide hydrochloride
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|
C24H24ClN5OS
|
1
|
| 1 |
IC50 = 735 nM
|
|
|
|
CP0440836
|
(1R,2R)-N-[4-(6-cyclopentylpyridin-2-yl)-3-(2-methylindazol-5-yl)-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C26H27N5OS
|
1
|
| 1 |
IC50 = 891 nM
|
|
|
|
CP0452632
|
(1R,2R)-N-[4-[6-(difluoromethyl)pyridin-2-yl]-3-(2-methylindazol-5-yl)-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C22H19F2N5OS
|
1
|
| 1 |
IC50 = 1020 nM
|
|
|
|
CP0411065
|
(1R,2R)-N-[4-[6-(fluoromethyl)pyridin-2-yl]-3-(2-methylindazol-5-yl)-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C22H20FN5OS
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0888585
|
(1R,2R)-2-methyl-N-(3-(2-methyl-2H-indazol-5-yl)-4-(6-(methylamino)pyridin-2-yl)isothiazol-5-yl)cyclopropanecarboxamide hydrochloride
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|
C22H23ClN6OS
|
1
|
| 1 |
IC50 = 1590 nM
|
|
|
|
CP0894675
|
(1R,2R)-2-methyl-N-(3-(2-methyl-2H-indazol-5-yl)-4-(6-methylpyridin-2-yl)isothiazol-5-yl)cyclopropanecarboxamide hydrochloride
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|
C22H22ClN5OS
|
1
|
| 1 |
IC50 = 2210 nM
|
|
|
|
CP0864303
|
(1R,2R)-N-(4-(6-ethylpyridin-2-yl)-3-(2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide hydrochloride
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|
C22H22ClN5OS
|
1
|
| 1 |
IC50 = 3110 nM
|
|
|
|
CP0864302
|
(1R,2R)-N-(3-(2H-indazol-5-yl)-4-(6-isopropylpyridin-2-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide hydrochloride
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|
C23H24ClN5OS
|
1
|
| 1 |
IC50 = 4570 nM
|
|
|
|
CP0386245
|
(1R,2R)-N-[4-[6-(dimethylamino)pyridin-2-yl]-3-(2-methylindazol-5-yl)-1,2-thiazol-5-yl]-2-methylcyclopropane-1-carboxamide
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|
C23H24N6OS
|
1
|
| 1 |
IC50 = 9540 nM
|
|
|
|
CP0857086
|
(1R,2R)-N-(4-(6-(dimethylamino)pyridin-2-yl)-3-(2H-indazol-5-yl)isothiazol-5-yl)-2-methylcyclopropanecarboxamide hydrochloride
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|
C22H23ClN6OS
|
1
|
| 1 |
IC50 > 12500 nM
|
|
|
|
CP0871659
|
(1R,2R)-N-(4-(6-(dimethylamino)pyridin-2-yl)-3-(2-methyl-2H-indazol-5-yl)isothiazol-5-yl)-2-ethylcyclopropanecarboxamide hydrochloride
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|
C24H27ClN6OS
|
1
|
| 1 |
IC50 > 12500 nM
|
|
|
