CHEMBL4799793

CHEMBL5070261

(5S)-8-chloro-1-(4-pyridin-2-yloxycyclohexyl)-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepin-5-ol

8-bromo-1-(4-pyridin-2-yloxycyclohexyl)-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepine

3-[4-(8-bromo-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepin-1-yl)cyclohexyl]-5-methyl-1,2-oxazole

CHEMBL5070075

CHEMBL5081323

[6-chloro-1-[2-(dimethylamino)ethyl]indol-3-yl]-spiro[1H-2-benzofuran-3,4'-piperidine]-1'-ylmethanone

3-[4-(8-chloro-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepin-1-yl)cyclohexyl]-5-methyl-1,2-oxazole

[(3S)-6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydro-2H-quinolin-3-yl]-pyrrolidin-1-ylmethanone

[(3S)-6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydro-2H-quinolin-3-yl]-cyclopentylmethanone

8-ethynyl-1-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepine

Balovaptan

8-chloro-1-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepine

[6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,4-dihydroquinazolin-3-yl]-cyclopropylmethanone

[6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,4-dihydroquinazolin-3-yl]-cyclopentylmethanone

1-[6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,4-dihydroquinazolin-3-yl]-2-methylpropan-1-one

8-bromo-1-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepine

1-(4-pyridin-2-yloxycyclohexyl)-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepine

(6-chloro-3-methylsulfonyl-2,4-dihydroquinazolin-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

3-[4-(5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepin-1-yl)cyclohexyl]-5-methyl-1,2-oxazole

[(3R)-6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydro-2H-quinolin-3-yl]-cyclopentylmethanone

8-chloro-5-methyl-1-(1-pyridin-2-ylpiperidin-4-yl)-4,6-dihydro-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine

1-[6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,4-dihydroquinazolin-3-yl]-2-hydroxyethanone

[7-chloro-4-[4-(2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydro-1H-isoquinolin-2-yl]-cyclopentylmethanone

[6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,4-dihydroquinazolin-3-yl]-phenylmethanone

(2R)-4-oxo-2-[(3S,4R)-2-oxo-3-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]-4-[(E)-2-phenylethenyl]azetidin-1-yl]-N-[(1S)-1-phenylethyl]-4-(4-piperidin-1-ylpiperidin-1-yl)butanamide

(6-chloro-3,4-dihydro-2H-quinazolin-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

1-[6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,4-dihydroquinazolin-3-yl]ethanone

(6-chloro-4-methyl-2,3-dihydroquinoxalin-1-yl)-[4-(3-chloropyridin-2-yl)piperazin-1-yl]methanone

7-chloro-1-(4-pyridin-2-yloxycyclohexyl)-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoline

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

(6-chloro-3-methyl-2,4-dihydroquinazolin-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

3-[4-(7-chloro-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinolin-1-yl)cyclohexyl]-5-methyl-1,2-oxazole

1-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepine

1-[7-chloro-4-[4-(2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydro-1H-isoquinolin-2-yl]-2-methylpropan-1-one

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-[4-(3-chloropyridin-2-yl)piperazin-1-yl]methanone

[7-chloro-4-[4-(2-methylphenyl)piperazine-1-carbonyl]-3,4-dihydro-1H-isoquinolin-2-yl]-cyclopropylmethanone

(6-chloro-3,4-dihydro-2H-quinolin-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

methyl 2-[7-chloro-1-(4-pyridin-2-yloxycyclohexyl)-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinolin-4-yl]acetate

8-ethyl-1-(1-pyridin-2-ylpiperidin-4-yl)-5,6-dihydro-4H-[1,2,4]triazolo[4,3-a][1]benzazepine

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-(1-pyridin-2-ylpiperidin-4-yl)methanone

(6-chloro-4-methyl-2,3-dihydroquinoxalin-1-yl)-(1-pyridin-2-ylpiperidin-4-yl)methanone

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-spiro[1H-2-benzofuran-3,4'-piperidine]-1'-ylmethanone

(6-chloro-4-methyl-2,3-dihydroquinoxalin-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-[4-(2-methylphenyl)piperidin-1-yl]methanone

(7-chloro-2,3,4,5-tetrahydro-1-benzazepin-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

CHEMBL5085869

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-[4-(3-methylpyridin-2-yl)piperazin-1-yl]methanone

N-[4-(7-chloro-5-hydroxy-2,3,4,5-tetrahydro-1-benzazepine-1-carbonyl)-3-methylphenyl]-2-methylbenzamide

3-[4-(13-chloro-6,7,9-triazatetracyclo[8.4.0.02,4.05,9]tetradeca-1(10),5,7,11,13-pentaen-8-yl)cyclohexyl]-5-methyl-1,2-oxazole

3-[4-[(2S,4R)-13-chloro-6,7,9-triazatetracyclo[8.4.0.02,4.05,9]tetradeca-1(10),5,7,11,13-pentaen-8-yl]cyclohexyl]-5-methyl-1,2-oxazole

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-[(2R)-2-methyl-4-(3-methylpyridin-2-yl)piperazin-1-yl]methanone

N-[2-chloro-5-[4-(2-methylphenyl)piperazine-1-carbonyl]phenyl]thiophene-2-carboxamide

(5-chloro-2,3-dihydroindol-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-[(3S)-3-methyl-4-pyridin-2-ylpiperazin-1-yl]methanone

7-chloro-1-(1-pyridin-2-ylpiperidin-4-yl)-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoline

1-[7-chloro-4-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,3-dihydroquinoxalin-1-yl]ethanone

(7-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-[4-(2-methylphenyl)piperazin-1-yl]methanone

3,4-dihydro-2H-quinoxalin-1-yl-[4-(2-methylphenyl)piperazin-1-yl]methanone

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-(4-pyridin-2-ylpiperazin-1-yl)methanone

(4-benzylpiperazin-1-yl)-(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)methanone

[6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,4-dihydroquinazolin-3-yl]-cyclohexylmethanone

[6-chloro-1-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,4-dihydroquinazolin-3-yl]-[1-(4-fluorophenyl)cyclopropyl]methanone

13-chloro-8-(4-pyridin-2-yloxycyclohexyl)-6,7,9-triazatetracyclo[8.4.0.02,4.05,9]tetradeca-1(10),5,7,11,13-pentaene

13-chloro-8-(1-pyridin-2-ylpiperidin-4-yl)-6,7,9-triazatetracyclo[8.4.0.02,4.05,9]tetradeca-1(10),5,7,11,13-pentaene

(6-chloro-3,4-dihydro-2H-quinoxalin-1-yl)-[(3R)-3-methyl-4-pyridin-2-ylpiperazin-1-yl]methanone

methyl 13-chloro-8-(4-pyridin-2-yloxycyclohexyl)-6,7,9-triazatetracyclo[8.4.0.02,4.05,9]tetradeca-1(10),5,7,11,13-pentaene-4-carboxylate

1-[7-fluoro-4-[4-(2-methylphenyl)piperazine-1-carbonyl]-2,3-dihydroquinoxalin-1-yl]ethanone

3-[4-[(2R,4S)-13-chloro-6,7,9-triazatetracyclo[8.4.0.02,4.05,9]tetradeca-1(10),5,7,11,13-pentaen-8-yl]cyclohexyl]-5-methyl-1,2-oxazole

7-chloro-4-methoxy-1-(1-pyridin-2-ylpiperidin-4-yl)-[1,2,4]triazolo[4,3-a]quinoxaline

7-chloro-4,4-dimethyl-1-(1-pyridin-2-ylpiperidin-4-yl)-5H-[1,2,4]triazolo[4,3-a]quinoxaline

1-[7-chloro-4,4-dimethyl-1-(1-pyridin-2-ylpiperidin-4-yl)-[1,2,4]triazolo[4,3-a]quinoxalin-5-yl]ethanone

6-chloro-1-(1-pyridin-2-ylpiperidin-4-yl)-3H-[1,2,4]triazolo[4,3-a]benzimidazole