| Compound ID |
Compound Name |
Compound Formula |
|
CP0565376
|
N-[2-[(2S)-2-[2-[(3,4-dimethoxyphenyl)methylamino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
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|
C27H28N4O6
|
1
|
| 1 |
IC50 = 0.089 nM
|
|
|
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CP0494210
|
tert-butyl 2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetate
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|
C24H28N4O6
|
1
|
| 1 |
IC50 = 0.13 nM
|
|
|
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CP0444481
|
N-[2-[(2S)-2-[2-[(4-methoxyphenyl)methylamino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
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|
C26H26N4O5
|
1
|
| 1 |
IC50 = 0.18 nM
|
|
|
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CP0487460
|
N-[2-[(2S)-2-[2-[2-(3,4-dimethoxyphenyl)ethylamino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C28H30N4O6
|
1
|
| 1 |
IC50 = 0.19 nM
|
|
|
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CP0565076
|
N-[2-[(2S)-2-[2-[(3-methoxyphenyl)methylamino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C26H26N4O5
|
1
|
| 1 |
IC50 = 0.22 nM
|
|
|
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CP0552719
|
methyl (2S)-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]-6-(phenylmethoxycarbonylamino)hexanoate
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|
C35H40N6O9
|
1
|
| 1 |
IC50 = 0.31 nM
|
|
|
|
CP0494241
|
N-[2-[(2S)-2-[2-[(2-morpholin-4-yl-2-oxoethyl)amino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C24H27N5O6
|
1
|
| 1 |
IC50 = 0.32 nM
|
|
|
|
CP0494240
|
methyl (2S)-5-(benzylamino)-5-oxo-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]pentanoate
Show/Hide
|
C33H36N6O8
|
1
|
| 1 |
IC50 = 0.33 nM
|
|
|
|
CP0422701
|
methyl 4-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]benzoate
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|
C26H24N4O6
|
1
|
| 1 |
IC50 = 0.42 nM
|
|
|
|
CP0559191
|
ethyl 2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetate
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|
C22H24N4O6
|
1
|
| 1 |
IC50 = 0.42 nM
|
|
|
|
CP0444675
|
N-[2-[(2S)-2-[2-[(4-fluorophenyl)methylamino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
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|
C25H23FN4O4
|
1
|
| 1 |
IC50 = 0.44 nM
|
|
|
|
CP0444674
|
methyl (2S)-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]-3-phenylpropanoate
Show/Hide
|
C30H31N5O7
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0471078
|
N-[2-[(2S)-2-[2-[[2-(tert-butylamino)-2-oxoethyl]amino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C24H29N5O5
|
1
|
| 1 |
IC50 = 0.53 nM
|
|
|
|
CP0547959
|
N-[2-oxo-2-[(2S)-2-[2-oxo-2-(pentylamino)acetyl]pyrrolidin-1-yl]ethyl]quinoline-4-carboxamide
Show/Hide
|
C23H28N4O4
|
1
|
| 1 |
IC50 = 0.58 nM
|
|
|
|
CP0422700
|
N-[2-[(2S)-2-[2-[(2,4-dimethylphenyl)methylamino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C27H28N4O4
|
1
|
| 1 |
IC50 = 0.63 nM
|
|
|
|
CP0444482
|
N-[2-oxo-2-[(2S)-2-[2-oxo-2-(2-phenylethylamino)acetyl]pyrrolidin-1-yl]ethyl]quinoline-4-carboxamide
Show/Hide
|
C26H26N4O4
|
1
|
| 1 |
IC50 = 0.63 nM
|
|
|
|
CP0494211
|
5-O-benzyl 1-O-methyl (2S)-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]pentanedioate
Show/Hide
|
C33H35N5O9
|
1
|
| 1 |
IC50 = 0.63 nM
|
|
|
|
CP0422702
|
N-[2-[(2S)-2-[2-(cyclopropylamino)-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
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|
C21H22N4O4
|
1
|
| 1 |
IC50 = 0.64 nM
|
|
|
|
CP0471075
|
N-[2-[(2S)-2-[2-[[2-(hexylamino)-2-oxoethyl]amino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C26H33N5O5
|
1
|
| 1 |
IC50 = 0.67 nM
|
|
|
|
CP0494209
|
N-[2-[(2S)-2-[2-(benzylamino)-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C25H24N4O4
|
1
|
| 1 |
IC50 = 0.77 nM
|
|
|
|
CP0444485
|
methyl 2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetate
Show/Hide
|
C21H22N4O6
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0570593
|
methyl 2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]propanoate
Show/Hide
|
C22H24N4O6
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0570595
|
N-[2-oxo-2-[(2S)-2-[2-oxo-2-[[2-oxo-2-(propan-2-ylamino)ethyl]amino]acetyl]pyrrolidin-1-yl]ethyl]quinoline-4-carboxamide
Show/Hide
|
C23H27N5O5
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0565375
|
N-[2-[(2S)-2-[2-(4-methoxyanilino)-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C25H24N4O5
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0570607
|
N-[2-[(2S)-2-[2-[[2-[(3,4-dimethoxyphenyl)methylamino]-2-oxoethyl]amino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C29H31N5O7
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0471074
|
N-[2-oxo-2-[(2S)-2-[2-oxo-2-[(2-oxo-2-pyrrolidin-1-ylethyl)amino]acetyl]pyrrolidin-1-yl]ethyl]quinoline-4-carboxamide
Show/Hide
|
C24H27N5O5
|
1
|
| 1 |
IC50 = 1.8 nM
|
|
|
|
CP0517076
|
(4S)-5-methoxy-5-oxo-4-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]pentanoic acid
Show/Hide
|
C26H29N5O9
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
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CP0086238
|
N-[2-[(2S)-2-cyano-4,4-difluoropyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C17H14F2N4O2
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
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CP0552716
|
N-[2-[(2S)-2-[2-[[2-(cyclopropylamino)-2-oxoethyl]amino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C23H25N5O5
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
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CP0547957
|
N-[2-[(2S)-2-[2-(benzhydrylamino)-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C31H28N4O4
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
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CP0422703
|
4-O-benzyl 1-O-methyl (2S)-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]butanedioate
Show/Hide
|
C32H33N5O9
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0570606
|
N-[2-[(2S)-2-[2-[[2-(benzylamino)-2-oxoethyl]amino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C27H27N5O5
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
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CP0444483
|
N-[2-oxo-2-[(2S)-2-[2-oxo-2-(propan-2-ylamino)acetyl]pyrrolidin-1-yl]ethyl]quinoline-4-carboxamide
Show/Hide
|
C21H24N4O4
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
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CP0451212
|
methyl (2S)-5-amino-5-oxo-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]pentanoate
Show/Hide
|
C26H30N6O8
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
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CP0570594
|
N-[2-[(2S)-2-[2-[[2-(dimethylamino)-2-oxoethyl]amino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C22H25N5O5
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
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CP0552717
|
N-[2-oxo-2-[(2S)-2-[2-oxo-2-[[2-oxo-2-(2-oxoethylamino)ethyl]amino]acetyl]pyrrolidin-1-yl]ethyl]quinoline-4-carboxamide
Show/Hide
|
C22H23N5O6
|
1
|
| 1 |
IC50 = 5.4 nM
|
|
|
|
CP0552718
|
methyl (2S)-4-methyl-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]pentanoate
Show/Hide
|
C27H33N5O7
|
1
|
| 1 |
IC50 = 6.7 nM
|
|
|
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CP0042682
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N-[2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C17H16N4O2
|
1
|
| 1 |
IC50 = 6.8 nM
|
|
|
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CP0471076
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methyl 2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]acetate
Show/Hide
|
C23H25N5O7
|
1
|
| 1 |
IC50 = 7.2 nM
|
|
|
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CP0451211
|
methyl 3-methyl-2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]butanoate
Show/Hide
|
C24H28N4O6
|
1
|
| 1 |
IC50 = 8.3 nM
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|
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CP0570608
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methyl (2S)-3-hydroxy-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]propanoate
Show/Hide
|
C24H27N5O8
|
1
|
| 1 |
IC50 = 11 nM
|
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CP0552715
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N-[2-[(2S)-2-[2-[[2-(methylamino)-2-oxoethyl]amino]-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C21H23N5O5
|
1
|
| 1 |
IC50 = 13 nM
|
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|
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CP0444484
|
N-[2-[(2S)-2-[2-(cyclohexylamino)-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C24H28N4O4
|
1
|
| 1 |
IC50 = 15 nM
|
|
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CP0471077
|
methyl (2S)-6-amino-2-[[2-[[2-oxo-2-[(2S)-1-[2-(quinoline-4-carbonylamino)acetyl]pyrrolidin-2-yl]acetyl]amino]acetyl]amino]hexanoate
Show/Hide
|
C27H34N6O7
|
1
|
| 1 |
IC50 = 20 nM
|
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CP0471073
|
N-[2-[(2S)-2-[2-(2,2-dimethylpropylamino)-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C23H28N4O4
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
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CP0547961
|
N-[2-[(2S)-2-[2-(1-adamantylamino)-2-oxoacetyl]pyrrolidin-1-yl]-2-oxoethyl]quinoline-4-carboxamide
Show/Hide
|
C28H32N4O4
|
1
|
| 1 |
IC50 = 150 nM
|
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