| Compound ID |
Compound Name |
Compound Formula |
|
CP0098465
|
2-methyl-N-[(2-methylpropan-2-yl)oxy]-4-[[(1R,2R)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexanecarbonyl]amino]pyrazole-3-carboxamide
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|
C27H34N6O4
|
1
|
| 1 |
IC50 = 5.8 nM
|
|
|
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CP0063832
|
(1R,2R)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]-N-(4-oxo-6,7-dihydro-5H-pyrazolo[1,5-a]pyrazin-3-yl)cyclohexane-1-carboxamide
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|
C24H26N6O3
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
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CP0534508
|
(1R,2R)-N-[3-(difluoromethyl)-1-methylpyrazol-4-yl]-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexane-1-carboxamide
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|
C23H25F2N5O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
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CP0356625
|
(1S,3R,4R,6R)-N-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-4-[4-(1H-pyrazol-5-yl)benzoyl]bicyclo[4.1.0]heptane-3-carboxamide
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|
C23H22F3N5O2
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
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CP0534510
|
(1S,3R,4R,6R)-N-[1-methyl-5-(trifluoromethyl)pyrazol-4-yl]-4-[4-(1H-pyrazol-5-yl)benzoyl]bicyclo[4.1.0]heptane-3-carboxamide
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|
C23H22F3N5O2
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
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CP0149564
|
(1R,2R)-N-(6-methoxypyrimidin-4-yl)-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
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|
C22H23N5O3
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
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CP0238638
|
N-(2-hydroxy-2-methylpropyl)-5-[[(1R,2R)-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexanecarbonyl]amino]pyrazine-2-carboxamide
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|
C26H30N6O4
|
1
|
| 1 |
IC50 = 15.85 nM
|
|
|
|
CP0426861
|
2-methyl-4-[[(1R,2R)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexanecarbonyl]amino]pyrazole-3-carboxylic acid
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|
C23H25N5O4
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0476659
|
(1R,2R)-N-(3-cyano-1-methylpyrazol-4-yl)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexane-1-carboxamide
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|
C23H24N6O2
|
1
|
| 1 |
IC50 = 19.95 nM
|
|
|
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CP0564783
|
5-methyl-4-[[(1R,2R)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexanecarbonyl]amino]-1H-pyrazole-3-carboxamide
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|
C23H26N6O3
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0139650
|
(1R,2R)-N-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
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|
C22H22F3N5O2
|
1
|
| 1 |
IC50 = 25.12 nM
|
|
|
|
CP0960908
|
1-ethyl-4-((1R,2R)-2-(4-(3-methyl-1H-pyrazol-5-yl)benzoyl)cyclohexanecarboxamido)-1H-pyrazole-5-carboxamide
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|
C24H28N6O3
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0238652
|
(1R,2R)-N-pyrazolo[1,5-a]pyrimidin-3-yl-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
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|
C23H22N6O2
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0534697
|
(1R,2R)-N-[3-(difluoromethoxy)-1-methylpyrazol-4-yl]-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
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|
C22H23F2N5O3
|
1
|
| 1 |
IC50 = 31.62 nM
|
|
|
|
CP0098466
|
(1R,2R)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]-N-(1-methyl-5-sulfamoylpyrazol-4-yl)cyclohexane-1-carboxamide
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|
C22H26N6O4S
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0959472
|
1-methyl-4-((1R,2R)-2-(4-(3-methyl-1H-pyrazol-5-yl)benzoyl)cyclohexanecarboxamido)-1H-pyrazole-5-carboxamide
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|
C23H26N6O3
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0149566
|
1-methyl-4-[[(1R,2R)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexanecarbonyl]amino]pyrazole-3-carboxamide
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|
C23H26N6O3
|
2
|
| 1 |
IC50 = 36 nM
|
|
|
| 2 |
IC50 = 39.81 nM
|
|
|
|
CP0347329
|
1-methyl-4-[[(1S,3R,4R,6R)-4-[6-(5-methyl-1H-pyrazol-3-yl)-1,2-benzoxazol-3-yl]bicyclo[4.1.0]heptane-3-carbonyl]amino]pyrazole-3-carboxamide
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|
C24H25N7O3
|
1
|
| 1 |
IC50 = 39.81 nM
|
|
|
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CP0532531
|
(1R,2R)-N-[1-methyl-5-(trifluoromethyl)pyrazol-4-yl]-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
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|
C22H22F3N5O2
|
1
|
| 1 |
IC50 = 39.81 nM
|
|
|
|
CP0575284
|
N-hydroxy-2-methyl-4-[[(1R,2R)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexanecarbonyl]amino]pyrazole-3-carboxamide
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|
C23H26N6O4
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0028152
|
(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexane-1-carboxamide
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|
C23H27N5O2
|
2
|
| 1 |
IC50 = 59 nM
|
|
|
| 2 |
IC50 = 63.1 nM
|
|
|
|
CP0493797
|
(2R,3R)-N-(1,3-dimethylpyrazol-4-yl)-3-[2-fluoro-4-(1H-pyrazol-5-yl)benzoyl]bicyclo[2.2.2]octane-2-carboxamide
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|
C24H26FN5O2
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
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CP0534414
|
(1R,2R)-N-(2-methyl-2-methylsulfonylpropyl)-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
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|
C22H29N3O4S
|
1
|
| 1 |
IC50 = 63.1 nM
|
|
|
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CP0238653
|
1-methyl-4-[[(1R,2R)-2-[6-(5-methyl-1H-pyrazol-3-yl)-1,2-benzoxazol-3-yl]cyclohexanecarbonyl]amino]pyrazole-3-carboxamide
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|
C23H25N7O3
|
1
|
| 1 |
IC50 = 79.43 nM
|
|
|
|
CP0356624
|
4-[[(1R,2R)-2-[2-fluoro-4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexanecarbonyl]amino]-1-methylpyrazole-3-carboxamide
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|
C23H25FN6O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
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CP0564782
|
2,5-dimethyl-4-[[(1R,2R)-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexanecarbonyl]amino]pyrazole-3-carboxamide
Show/Hide
|
C24H28N6O3
|
1
|
| 1 |
IC50 = 101 nM
|
|
|
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CP0476658
|
(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-2-[2-fluoro-4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
Show/Hide
|
C22H24FN5O2
|
1
|
| 1 |
IC50 = 125.89 nM
|
|
|
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CP0476660
|
(1R,2R)-N-(3,5-dimethyl-1,2-oxazol-4-yl)-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
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|
C22H24N4O3
|
1
|
| 1 |
IC50 = 199.53 nM
|
|
|
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CP0517700
|
(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-N-methyl-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
Show/Hide
|
C23H27N5O2
|
1
|
| 1 |
IC50 = 199.53 nM
|
|
|
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CP0569617
|
(1R,2R)-N-[1-(2-amino-2-oxoethyl)pyrazol-4-yl]-2-[4-(5-methyl-1H-pyrazol-3-yl)benzoyl]cyclohexane-1-carboxamide
Show/Hide
|
C23H26N6O3
|
1
|
| 1 |
IC50 = 241 nM
|
|
|
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CP0482640
|
(1R,2R)-2-[4-(1H-pyrazol-5-yl)benzoyl]-N-(2-pyridin-2-ylethyl)cyclohexane-1-carboxamide
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|
C24H26N4O2
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
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CP0534415
|
3-[[(1R,2R)-2-[4-(4-methylpyrazol-1-yl)benzoyl]cyclohexanecarbonyl]amino]benzamide
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|
C25H26N4O3
|
1
|
| 1 |
IC50 = 316.23 nM
|
|
|
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CP0532530
|
(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-2-(4-pyridin-2-ylbenzoyl)cyclohexane-1-carboxamide
Show/Hide
|
C24H26N4O2
|
1
|
| 1 |
IC50 = 501.19 nM
|
|
|
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CP0438857
|
(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-2-[4-(4-methyl-1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
Show/Hide
|
C23H27N5O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
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CP0517701
|
(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-2-[4-(1H-pyrrol-2-yl)benzoyl]cyclohexane-1-carboxamide
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|
C23H26N4O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
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CP0570263
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(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-2-[6-(1H-pyrazol-5-yl)pyridine-3-carbonyl]cyclohexane-1-carboxamide
Show/Hide
|
C21H24N6O2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
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CP0574082
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(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-2-[2-methyl-4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
Show/Hide
|
C23H27N5O2
|
1
|
| 1 |
IC50 = 1000 nM
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CP0529545
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(1S,2S)-N-(1,3-dimethylpyrazol-4-yl)-2-[4-(1H-pyrazol-5-yl)benzoyl]cyclohexane-1-carboxamide
Show/Hide
|
C22H25N5O2
|
1
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| 1 |
IC50 = 1995.26 nM
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CP0441041
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(1R,2R)-2-[4-(3-acetylphenyl)benzoyl]-N-(3,5-dimethyl-1,2-oxazol-4-yl)cyclohexane-1-carboxamide
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|
C27H28N2O4
|
1
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| 1 |
IC50 = 2511.89 nM
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CP0441040
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(1R,2R)-N-(1,3-dimethylpyrazol-4-yl)-2-[4-(2-methylpyrazol-3-yl)benzoyl]cyclohexane-1-carboxamide
Show/Hide
|
C23H27N5O2
|
1
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| 1 |
IC50 = 25118.86 nM
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