Brief Information of the Compound and Protein
Compound Name
1-methyl-4-[[(1S,3R,4R,6R)-4-[6-(5-methyl-1H-pyrazol-3-yl)-1,2-benzoxazol-3-yl]bicyclo[4.1.0]heptane-3-carbonyl]amino]pyrazole-3-carboxamide
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PubChem ID
CID: 155558755
Canonical SMILES
Cc1cc(n[nH]1)-c1ccc2c(noc2c1)[C@@H]1C[C@H]2C[C@H]2C[C@H]1C(=O)Nc1cn(C)nc1C(N)=O
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Compound Formula C24H25N7O3
Compound Structure
Protein Name
Arachidonate 5-lipoxygenase-activating protein
Protein Classification
Other cytosolic protein
Uniprot ID
P20292
Gene Name
ALOX5AP
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000053 COS-7 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 39.81 nM
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