Brief Information of the Compound and Protein
Compound Name
(2R,3R)-N-(1,3-dimethylpyrazol-4-yl)-3-[2-fluoro-4-(1H-pyrazol-5-yl)benzoyl]bicyclo[2.2.2]octane-2-carboxamide
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Canonical SMILES
Cc1nn(C)cc1NC(=O)[C@@H]1[C@H]2CC[C@H](CC2)[C@H]1C(=O)c1ccc(cc1F)-c1cc[nH]n1
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Compound Formula C24H26FN5O2
Compound Structure
Protein Name
Arachidonate 5-lipoxygenase-activating protein
Protein Classification
Other cytosolic protein
Uniprot ID
P20292
Gene Name
ALOX5AP
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000053 COS-7 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 63.1 nM
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