| Compound ID |
Compound Name |
Compound Formula |
|
CP0413654
|
6-phenyl-N-[(3-phenylphenyl)methyl]-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C27H21N5
|
3
|
| 1 |
EC50 = 500 nM
|
|
|
| 2 |
EC50 = 2490 nM
|
|
|
| 3 |
EC50 = 2570 nM
|
|
|
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CP0279103
|
N-[(4-tert-butylphenyl)methyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C25H25N5
|
3
|
| 1 |
EC50 = 600 nM
|
|
|
| 2 |
EC50 = 1120 nM
|
|
|
| 3 |
EC50 = 1710 nM
|
|
|
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CP0159682
|
6-phenyl-N-[(4-phenylphenyl)methyl]-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C27H21N5
|
5
|
| 1 |
EC50 = 1120 nM
|
|
|
| 2 |
EC50 = 1400 nM
|
|
|
| 3 |
EC50 = 1630 nM
|
|
|
| 4 |
EC50 = 5010 nM
|
|
|
| 5 |
EC50 = 15600 nM
|
|
|
|
CP0446194
|
N-[(4-methylphenyl)methyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C22H19N5
|
3
|
| 1 |
EC50 = 1190 nM
|
|
|
| 2 |
EC50 = 2600 nM
|
|
|
| 3 |
EC50 = 4580 nM
|
|
|
|
CP0381227
|
N-[(1R)-1-cyclohexylethyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C22H25N5
|
3
|
| 1 |
EC50 = 1200 nM
|
|
|
| 2 |
EC50 = 1880 nM
|
|
|
| 3 |
EC50 = 6730 nM
|
|
|
|
CP0486983
|
N-[(3-chlorophenyl)methyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C21H16ClN5
|
3
|
| 1 |
EC50 = 1490 nM
|
|
|
| 2 |
EC50 = 2330 nM
|
|
|
| 3 |
EC50 = 2770 nM
|
|
|
|
CP0381226
|
N-[(3,4-dimethylphenyl)methyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C23H21N5
|
3
|
| 1 |
EC50 = 1850 nM
|
|
|
| 2 |
EC50 = 2300 nM
|
|
|
| 3 |
EC50 = 2960 nM
|
|
|
|
CP0404918
|
N-[(1S)-1-cyclohexylethyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C22H25N5
|
3
|
| 1 |
EC50 = 2060 nM
|
|
|
| 2 |
EC50 = 2550 nM
|
|
|
| 3 |
EC50 = 4170 nM
|
|
|
|
CP0449465
|
N-[(3-methylphenyl)methyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C22H19N5
|
3
|
| 1 |
EC50 = 2390 nM
|
|
|
| 2 |
EC50 = 2910 nM
|
|
|
| 3 |
EC50 = 5410 nM
|
|
|
|
CP0493992
|
N-(cyclohexylmethyl)-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C21H23N5
|
3
|
| 1 |
EC50 = 2460 nM
|
|
|
| 2 |
EC50 = 3450 nM
|
|
|
| 3 |
EC50 = 4740 nM
|
|
|
|
CP0413652
|
N-(3,3-dimethylbutyl)-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C20H23N5
|
3
|
| 1 |
EC50 = 2480 nM
|
|
|
| 2 |
EC50 = 2970 nM
|
|
|
| 3 |
EC50 = 3820 nM
|
|
|
|
CP0271056
|
N-(4-hydroxybutyl)-5-phenyl-1,2-oxazole-3-carboxamide
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|
C14H16N2O3
|
3
|
| 1 |
EC50 = 3040 nM
|
|
|
| 2 |
EC50 = 7570 nM
|
|
|
| 3 |
EC50 = 22000 nM
|
|
|
|
CP0445339
|
N-[(2-methylphenyl)methyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C22H19N5
|
3
|
| 1 |
EC50 = 3080 nM
|
|
|
| 2 |
EC50 = 6670 nM
|
|
|
| 3 |
EC50 = 9540 nM
|
|
|
|
CP0413653
|
N-(6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-yl)quinoxalin-2-amine
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|
C22H15N7
|
3
|
| 1 |
EC50 = 3260 nM
|
|
|
| 2 |
EC50 = 4460 nM
|
|
|
| 3 |
EC50 = 7640 nM
|
|
|
|
CP0493993
|
6-phenyl-N-(2-phenylethyl)-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C22H19N5
|
3
|
| 1 |
EC50 = 3630 nM
|
|
|
| 2 |
EC50 = 8720 nM
|
|
|
| 3 |
EC50 = 9820 nM
|
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|
|
CP0446189
|
N-[(4-methoxyphenyl)methyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C22H19N5O
|
3
|
| 1 |
EC50 = 3670 nM
|
|
|
| 2 |
EC50 = 3730 nM
|
|
|
| 3 |
EC50 = 4740 nM
|
|
|
|
CP0514514
|
N-[(3-methoxyphenyl)methyl]-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C22H19N5O
|
3
|
| 1 |
EC50 = 3920 nM
|
|
|
| 2 |
EC50 = 4150 nM
|
|
|
| 3 |
EC50 = 6270 nM
|
|
|
|
CP0435573
|
N-(cyclopropylmethyl)-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C18H17N5
|
3
|
| 1 |
EC50 = 4270 nM
|
|
|
| 2 |
EC50 = 6210 nM
|
|
|
| 3 |
EC50 = 12700 nM
|
|
|
|
CP0435572
|
6-phenyl-3-pyridin-2-yl-N-(pyridin-3-ylmethyl)-1,2,4-triazin-5-amine
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|
C20H16N6
|
3
|
| 1 |
EC50 = 4350 nM
|
|
|
| 2 |
EC50 = 5020 nM
|
|
|
| 3 |
EC50 = 26000 nM
|
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|
|
CP0435574
|
N-benzyl-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C21H17N5
|
3
|
| 1 |
EC50 = 4480 nM
|
|
|
| 2 |
EC50 = 4800 nM
|
|
|
| 3 |
EC50 = 7740 nM
|
|
|
|
CP0113585
|
6-phenyl-N-prop-2-enyl-3-(2-pyridinyl)-1,2,4-triazin-5-amine
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|
C17H15N5
|
3
|
| 1 |
EC50 = 4620 nM
|
|
|
| 2 |
EC50 = 6150 nM
|
|
|
| 3 |
EC50 = 7130 nM
|
|
|
|
CP0446192
|
N-(6-methylpyridin-2-yl)-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C20H16N6
|
3
|
| 1 |
EC50 = 5410 nM
|
|
|
| 2 |
EC50 = 7550 nM
|
|
|
| 3 |
EC50 = 22400 nM
|
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|
CP0554441
|
N-(3-morpholin-4-ylpropyl)-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C21H24N6O
|
3
|
| 1 |
EC50 = 6270 nM
|
|
|
| 2 |
EC50 = 8120 nM
|
|
|
| 3 |
EC50 = 14200 nM
|
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|
|
CP0449552
|
6-phenyl-3-pyridin-2-yl-N-(pyridin-2-ylmethyl)-1,2,4-triazin-5-amine
Show/Hide
|
C20H16N6
|
3
|
| 1 |
EC50 = 6450 nM
|
|
|
| 2 |
EC50 = 7620 nM
|
|
|
| 3 |
EC50 = 27800 nM
|
|
|
|
CP0166390
|
MLS000541553
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|
C16H15N5
|
3
|
| 1 |
EC50 = 7460 nM
|
|
|
| 2 |
EC50 = 9060 nM
|
|
|
| 3 |
EC50 = 9820 nM
|
|
|
|
CP0449551
|
N-(oxan-4-ylmethyl)-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C20H21N5O
|
3
|
| 1 |
EC50 = 7670 nM
|
|
|
| 2 |
EC50 = 8380 nM
|
|
|
| 3 |
EC50 = 29500 nM
|
|
|
|
CP0186574
|
MLS000708948
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|
C16H16N4O2
|
3
|
| 1 |
EC50 = 7720 nM
|
|
|
| 2 |
EC50 = 8670 nM
|
|
|
| 3 |
EC50 = 15800 nM
|
|
|
|
CP0486984
|
5-(4-methylpiperazin-1-yl)-6-phenyl-3-pyridin-2-yl-1,2,4-triazine
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|
C19H20N6
|
3
|
| 1 |
EC50 = 8690 nM
|
|
|
| 2 |
EC50 = 10200 nM
|
|
|
| 3 |
EC50 = 21900 nM
|
|
|
|
CP0339667
|
N-butyl-5-(4-fluorophenyl)-1,2-oxazole-3-carboxamide
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|
C14H15FN2O2
|
1
|
| 1 |
EC50 = 8850 nM
|
|
|
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CP0446188
|
N-(2-morpholin-4-ylethyl)-6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-amine
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|
C20H22N6O
|
3
|
| 1 |
EC50 = 9080 nM
|
|
|
| 2 |
EC50 = 10000 nM
|
|
|
| 3 |
EC50 = 20800 nM
|
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CP0513236
|
6-phenyl-3-pyridin-2-yl-N-(2-pyridin-2-ylethyl)-1,2,4-triazin-5-amine
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|
C21H18N6
|
3
|
| 1 |
EC50 = 9600 nM
|
|
|
| 2 |
EC50 = 9840 nM
|
|
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| 3 |
EC50 = 17500 nM
|
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|
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CP0486067
|
3-[(6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-yl)amino]propan-1-ol
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|
C17H17N5O
|
3
|
| 1 |
EC50 = 10500 nM
|
|
|
| 2 |
EC50 = 10600 nM
|
|
|
| 3 |
EC50 = 25000 nM
|
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|
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CP0413655
|
[1-(6-phenyl-3-pyridin-2-yl-1,2,4-triazin-5-yl)piperidin-4-yl]methanol
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|
C20H21N5O
|
3
|
| 1 |
EC50 = 11600 nM
|
|
|
| 2 |
EC50 = 12100 nM
|
|
|
| 3 |
EC50 = 22900 nM
|
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CP0260429
|
N-(cyclopropylmethyl)-5-phenyl-1,2-oxazole-3-carboxamide
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|
C14H14N2O2
|
3
|
| 1 |
EC50 = 16600 nM
|
|
|
| 2 |
EC50 = 21500 nM
|
|
|
| 3 |
EC50 = 24900 nM
|
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|
CP0075152
|
DEFEROXAMINE
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|
C25H48N6O8
|
1
|
| 1 |
EC50 = 17800 nM
|
|
|
|
CP0316928
|
N-(3-morpholin-4-ylpropyl)-5-phenyl-1,2-oxazole-3-carboxamide
Show/Hide
|
C17H21N3O3
|
3
|
| 1 |
EC50 = 20000 nM
|
|
|
| 2 |
EC50 = 23900 nM
|
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| 3 |
EC50 = 28000 nM
|
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|
