| Compound ID |
Compound Name |
Compound Formula |
|
CP0477098
|
1-[3-(2-methoxyethoxy)-4-phenoxyphenyl]-3-(4-methylphenyl)-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C25H23N3O6
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0538381
|
1-[3-(2-methoxyethoxy)-4-phenoxyphenyl]-3-(3-methylphenyl)-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C25H23N3O6
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0536435
|
1-(3-chlorophenyl)-3-[3-(2-methoxyethoxy)-4-phenoxyphenyl]-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C24H20ClN3O6
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0434610
|
1-(3-bromo-4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C21H14BrN3O4
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0485950
|
1-(2-methoxy-4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C22H17N3O5
|
1
|
| 1 |
EC50 = 270 nM
|
|
|
|
CP0455522
|
1-(4-phenoxy-3-propan-2-yloxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C24H21N3O5
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0536434
|
1-(3-ethoxy-4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C23H19N3O5
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0537014
|
1-(3-methyl-4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C22H17N3O4
|
1
|
| 1 |
EC50 = 390 nM
|
|
|
|
CP0545871
|
1-(3-methoxy-4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C22H17N3O5
|
1
|
| 1 |
EC50 = 450 nM
|
|
|
|
CP0434609
|
1-(4-chlorophenyl)-3-[3-(2-methoxyethoxy)-4-phenoxyphenyl]-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C24H20ClN3O6
|
1
|
| 1 |
EC50 = 460 nM
|
|
|
|
CP0538383
|
1-methyl-3-[3-(oxetan-3-ylmethoxy)-4-phenoxyphenyl]-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C20H19N3O6
|
1
|
| 1 |
EC50 = 610 nM
|
|
|
|
CP0440106
|
1-[3-(oxolan-3-yloxy)-4-phenoxyphenyl]-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C25H21N3O6
|
1
|
| 1 |
EC50 = 750 nM
|
|
|
|
CP0545872
|
1-[3-(oxetan-3-ylmethoxy)-4-phenoxyphenyl]-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C25H21N3O6
|
1
|
| 1 |
EC50 = 790 nM
|
|
|
|
CP0440109
|
1-(3-methoxyphenyl)-3-(4-phenoxyphenyl)-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C22H17N3O5
|
1
|
| 1 |
EC50 = 950 nM
|
|
|
|
CP0485953
|
1-(4-phenoxyphenyl)-3-phenyl-1,3,5-triazinane-2,4,6-trione
Show/Hide
|
C21H15N3O4
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0274475
|
N-[5-(4-amino-7-propan-2-ylpyrrolo[2,3-d]pyrimidine-5-carbonyl)pyridin-3-yl]-2-(4-chlorophenyl)acetamide
Show/Hide
|
C23H21ClN6O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0284251
|
US8846698, 250
Show/Hide
|
C23H21ClN6O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0514698
|
N-[5-[2-amino-7-(1-hydroxy-2-methylpropan-2-yl)pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl]-2-(4-chlorophenyl)acetamide
Show/Hide
|
C24H23ClN6O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0123936
|
2-[(3R,4S)-3-fluoro-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxy-5-(1-methylimidazol-4-yl)pyridine-3-carboxamide
Show/Hide
|
C24H23F4N5O4
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0480003
|
6-(1-methylpyrazol-4-yl)-3-[(3R)-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]pyrrolidin-3-yl]oxypyridine-2-carboxamide
Show/Hide
|
C23H22F3N5O4
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
|
CP0188940
|
US8846698, 69
Show/Hide
|
C23H20ClN5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0261329
|
PF06273340
Show/Hide
|
C23H22ClN7O3
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0367394
|
US8846698, 90
Show/Hide
|
C23H23N7O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0335186
|
5-(1-methylpyrazol-4-yl)-2-[1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxybenzamide
Show/Hide
|
C25H25F3N4O4
|
1
|
| 1 |
IC50 = 4.2 nM
|
|
|
|
CP0323559
|
US9163021, 26
Show/Hide
|
C24H24N6O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0514699
|
US8846698, 253
Show/Hide
|
C23H24N8O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0540119
|
1-[4-(4-amino-7-propan-2-ylpyrrolo[2,3-d]pyrimidine-5-carbonyl)pyridin-2-yl]-3-(2,4-difluorophenyl)urea
Show/Hide
|
C22H19F2N7O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0456114
|
5-(1-methylimidazol-4-yl)-2-[1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxybenzamide
Show/Hide
|
C25H25F3N4O4
|
1
|
| 1 |
IC50 = 6.1 nM
|
|
|
|
CP0198981
|
6-amino-5-[(3S)-4,4-difluoro-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]pyrrolidin-3-yl]oxy-N-methylpyridine-3-carboxamide
Show/Hide
|
C20H19F5N4O4
|
1
|
| 1 |
IC50 = 6.2 nM
|
|
|
|
CP0245291
|
6-(1-methylpyrazol-4-yl)-3-[1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxypyridine-2-carboxamide
Show/Hide
|
C24H24F3N5O4
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
|
CP0142175
|
US9163021, 90
Show/Hide
|
C24H23FN6O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0322061
|
US9163021, 21
Show/Hide
|
C22H19F3N6O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0317452
|
N-[5-(4-amino-7-propan-2-ylpyrrolo[2,3-d]pyrimidine-5-carbonyl)pyridin-3-yl]-2-(4-cyanophenyl)acetamide
Show/Hide
|
C24H21N7O2
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0198982
|
2-[(3R,4S)-3-fluoro-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]piperidin-4-yl]oxy-4-(2-hydroxy-2-methylpropoxy)benzamide
Show/Hide
|
C25H28F4N2O6
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0245290
|
4-[2-carbamoyl-4-(1-methylpyrazol-4-yl)phenoxy]-N-[4-(trifluoromethoxy)phenyl]piperidine-1-carboxamide
Show/Hide
|
C24H24F3N5O4
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0317451
|
US8846698, 71
Show/Hide
|
C24H20N6O2
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0415710
|
6-(1-methylpyrazol-4-yl)-3-[(3S)-1-[2-[4-(trifluoromethoxy)phenyl]acetyl]pyrrolidin-3-yl]oxypyridine-2-carboxamide
Show/Hide
|
C23H22F3N5O4
|
1
|
| 1 |
IC50 = 900 nM
|
|
|
