| Compound ID |
Compound Name |
Compound Formula |
|
CP0505006
|
(2S,3R,4R,5S,6R)-2-(3-(4-ethoxybenzyl)-4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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|
C22H28O6
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0444289
|
(2R,3R,4S,5S,6R)-2-(3-(4-cyclopropylbenzyl)-4-fluoro-1H-indol-1-yl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H26FNO5
|
2
|
| 1 |
EC50 = 1.9 nM
|
|
|
| 2 |
IC50 = 1.4 nM
|
|
|
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CP0462381
|
(2R,3R,4S,5S,6R)-2-(4-chloro-3-(4-cyclopropylbenzyl)-1H-indol-1-yl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H26ClNO5
|
2
|
| 1 |
EC50 = 2.3 nM
|
|
|
| 2 |
EC50 = 14 nM
|
|
|
|
CP0198642
|
(2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl}-6-(hydroxymethyl)oxane-3,4,5-triol
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|
C21H25ClO6
|
3
|
| 1 |
EC50 = 2.4 nM
|
|
|
| 2 |
IC50 = 1 nM
|
|
|
| 3 |
IC50 = 1.3 nM
|
|
|
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CP0441419
|
(2R,3R,4S,5S,6R)-2-(3-(4-cyclopropylbenzyl)-4,6-difluoro-1H-indol-1-yl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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|
C24H25F2NO5
|
1
|
| 1 |
EC50 = 2.8 nM
|
|
|
|
CP0438225
|
(2R,3S,4S,5R,6S)-2-Hydroxymethyl-6-[2-(4-methyl-benzyl)-phenoxy]-tetrahydro-pyran-3,4,5-triol
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|
C20H24O6
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0490987
|
(2S,3R,4R,5S,6R)-2-(3-(4-ethylbenzyl)-4-methylphenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
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|
C22H28O5
|
1
|
| 1 |
EC50 = 12 nM
|
|
|
|
CP0407868
|
(2S,3R,4S,5S,6R)-2-(3-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C24H27NO7
|
2
|
| 1 |
EC50 = 24 nM
|
|
|
| 2 |
IC50 = 24 nM
|
|
|
|
CP0478508
|
methyl 3-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylamino]-3-oxopropanoate
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|
C28H31ClN2O7
|
1
|
| 1 |
EC50 = 39 nM
|
|
|
|
CP0863178
|
1-[6-(Acetylamino)-6-deoxy-beta-D-glucopyranosyl]-4-chloro-3-(4-cyclopropylbenzyl)-1H-indole
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|
C26H29ClN2O5
|
1
|
| 1 |
EC50 = 42 nM
|
|
|
|
CP0507349
|
(2S,3R,4S,5R)-2-[1-[(4-cyclopropylphenyl)methyl]-7-fluoroindol-3-yl]oxane-3,4,5-triol
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|
C23H24FNO4
|
1
|
| 1 |
EC50 = 47 nM
|
|
|
|
CP0439723
|
(2S,3R,4S,5R)-2-[1-[(4-cyclopropylphenyl)methyl]-7-methylindol-3-yl]oxane-3,4,5-triol
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|
C24H27NO4
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0499634
|
(2S,3R,4S,5S,6R)-2-(3-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)-1-methyl-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
|
C25H29NO7
|
2
|
| 1 |
EC50 = 67 nM
|
|
|
| 2 |
IC50 = 67 nM
|
|
|
|
CP0050531
|
1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}phenyl)-3-(4-hydroxyphenyl)propan-1-one
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|
C21H24O10
|
4
|
| 1 |
EC50 = 77 nM
|
|
|
| 2 |
EC50 = 123 nM
|
|
|
| 3 |
IC50 = 16 nM
|
|
|
| 4 |
IC50 = 27.8 nM
|
|
|
|
CP0415955
|
(2S,3R,4S,5R)-2-[1-[(4-cyclopropylphenyl)methyl]indol-3-yl]oxane-3,4,5-triol
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|
C23H25NO4
|
1
|
| 1 |
EC50 = 87 nM
|
|
|
|
CP0462391
|
2-chloro-N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]acetamide
Show/Hide
|
C26H28Cl2N2O5
|
1
|
| 1 |
EC50 = 113 nM
|
|
|
|
CP0532366
|
ethyl 3-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylamino]-3-oxopropanoate
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|
C29H33ClN2O7
|
1
|
| 1 |
EC50 = 118 nM
|
|
|
|
CP0386077
|
methyl 1-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]triazole-4-carboxylate
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|
C28H29ClN4O6
|
1
|
| 1 |
EC50 = 119 nM
|
|
|
|
CP0504874
|
(2S,3R,4S,5R)-2-[7-fluoro-1-[(4-methoxyphenyl)methyl]indol-3-yl]oxane-3,4,5-triol
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|
C21H22FNO5
|
1
|
| 1 |
EC50 = 151 nM
|
|
|
|
CP0409800
|
1-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-3-(3-chloropropyl)urea
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|
C28H33Cl2N3O5
|
1
|
| 1 |
EC50 = 151 nM
|
|
|
|
CP0409804
|
3-bromo-N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]propanamide
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|
C27H30BrClN2O5
|
1
|
| 1 |
EC50 = 151 nM
|
|
|
|
CP0508518
|
3-chloro-N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]propanamide
Show/Hide
|
C27H30Cl2N2O5
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0386075
|
2,2-dichloro-N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]acetamide
Show/Hide
|
C26H27Cl3N2O5
|
1
|
| 1 |
EC50 = 184 nM
|
|
|
|
CP0409806
|
4-Chloro-3-(4-cyclopropylbenzyl)-1-(beta-D-xylopyranosyl)-1Hindole
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|
C23H24ClNO4
|
2
|
| 1 |
EC50 = 203 nM
|
|
|
| 2 |
EC50 = 205 nM
|
|
|
|
CP0386076
|
(2R,3S,4S,5R,6R)-2-(aminomethyl)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]oxane-3,4,5-triol
Show/Hide
|
C24H27ClN2O4
|
1
|
| 1 |
EC50 = 237 nM
|
|
|
|
CP0478509
|
ethyl 2-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylamino]-2-oxoacetate
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|
C28H31ClN2O7
|
1
|
| 1 |
EC50 = 249 nM
|
|
|
|
CP0478510
|
methyl 2-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylamino]-2-oxoacetate
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|
C27H29ClN2O7
|
1
|
| 1 |
EC50 = 284 nM
|
|
|
|
CP0409805
|
ethyl 2-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylcarbamothioylamino]acetate
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|
C29H34ClN3O6S
|
1
|
| 1 |
EC50 = 286 nM
|
|
|
|
CP0462383
|
1-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-3-methylthiourea
Show/Hide
|
C26H30ClN3O4S
|
1
|
| 1 |
EC50 = 315 nM
|
|
|
|
CP0566897
|
(2R,3R,4S,5S,6R)-2-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-6-[(4-cyclopropyltriazol-1-yl)methyl]oxane-3,4,5-triol
Show/Hide
|
C29H31ClN4O4
|
1
|
| 1 |
EC50 = 359 nM
|
|
|
|
CP0409803
|
N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-1,2-oxazole-5-carboxamide
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|
C28H28ClN3O6
|
1
|
| 1 |
EC50 = 387 nM
|
|
|
|
CP0462382
|
1-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-3-(4-chlorophenyl)thiourea
Show/Hide
|
C31H31Cl2N3O4S
|
1
|
| 1 |
EC50 = 485 nM
|
|
|
|
CP0409801
|
N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-2-thiophen-2-ylacetamide
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|
C30H31ClN2O5S
|
1
|
| 1 |
EC50 = 499 nM
|
|
|
|
CP0493937
|
ethyl 2-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylcarbamoylamino]acetate
Show/Hide
|
C29H34ClN3O7
|
1
|
| 1 |
EC50 = 515 nM
|
|
|
|
CP0566894
|
N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]cyclopropanecarboxamide
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|
C28H31ClN2O5
|
1
|
| 1 |
EC50 = 552 nM
|
|
|
|
CP0491282
|
1-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-3-(3-methoxypropyl)thiourea
Show/Hide
|
C29H36ClN3O5S
|
1
|
| 1 |
EC50 = 586 nM
|
|
|
|
CP0409136
|
(2S,3R,4S,5R)-2-[1-[(4-propylphenyl)methyl]indol-3-yl]oxane-3,4,5-triol
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|
C23H27NO4
|
1
|
| 1 |
EC50 = 588 nM
|
|
|
|
CP0566893
|
ethyl 4-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylamino]-4-oxobutanoate
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|
C30H35ClN2O7
|
1
|
| 1 |
EC50 = 588 nM
|
|
|
|
CP0483534
|
1-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-3-(2-chloroethyl)urea
Show/Hide
|
C27H31Cl2N3O5
|
1
|
| 1 |
EC50 = 598 nM
|
|
|
|
CP0434466
|
(2S,3R,4R,5R)-2-[4-chloro-5-[(4-ethylphenyl)methyl]-2-methoxyphenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C22H27ClO6
|
1
|
| 1 |
EC50 = 620 nM
|
|
|
|
CP0508517
|
N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-2-methylpropanamide
Show/Hide
|
C28H33ClN2O5
|
1
|
| 1 |
EC50 = 649 nM
|
|
|
|
CP0532367
|
(2R,3R,4S,5S,6R)-2-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-6-[(4-ethoxytriazol-1-yl)methyl]oxane-3,4,5-triol
Show/Hide
|
C28H31ClN4O5
|
1
|
| 1 |
EC50 = 655 nM
|
|
|
|
CP0386074
|
1-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-3-ethylthiourea
Show/Hide
|
C27H32ClN3O4S
|
1
|
| 1 |
EC50 = 716 nM
|
|
|
|
CP0415965
|
(2S,3R,4S,5R)-2-[1-(naphthalen-2-ylmethyl)indol-3-yl]oxane-3,4,5-triol
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|
C24H23NO4
|
1
|
| 1 |
EC50 = 722 nM
|
|
|
|
CP0443586
|
(2S,3R,4S,5R)-2-[1-[(4-methoxyphenyl)methyl]indol-3-yl]oxane-3,4,5-triol
Show/Hide
|
C21H23NO5
|
1
|
| 1 |
EC50 = 736 nM
|
|
|
|
CP0462385
|
ethyl N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylcarbamoyl]carbamate
Show/Hide
|
C28H32ClN3O7
|
1
|
| 1 |
EC50 = 1004 nM
|
|
|
|
CP0481438
|
(2S,3R,4S,5R)-2-[4-fluoro-1-[(4-methoxyphenyl)methyl]indol-3-yl]oxane-3,4,5-triol
Show/Hide
|
C21H22FNO5
|
1
|
| 1 |
EC50 = 1110 nM
|
|
|
|
CP0462393
|
(2R,3R,4S,5S,6R)-2-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-6-[(4-cyclopentyltriazol-1-yl)methyl]oxane-3,4,5-triol
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|
C31H35ClN4O4
|
1
|
| 1 |
EC50 = 1585 nM
|
|
|
|
CP0462387
|
N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-2-phenylsulfanylacetamide
Show/Hide
|
C32H33ClN2O5S
|
1
|
| 1 |
EC50 = 2091 nM
|
|
|
|
CP0508516
|
N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-4-methoxybenzamide
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|
C32H33ClN2O6
|
1
|
| 1 |
EC50 = 2367 nM
|
|
|
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CP0434531
|
(2R,3R,4R,5S)-2-[(1R)-1,2-dihydroxyethyl]-5-[3-[(4-ethylphenyl)methyl]-4-methylphenyl]oxolane-3,4-diol
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|
C22H28O5
|
1
|
| 1 |
EC50 = 2500 nM
|
|
|
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CP0462389
|
N-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]-4-(chloromethyl)benzamide
Show/Hide
|
C32H32Cl2N2O5
|
1
|
| 1 |
EC50 = 2591 nM
|
|
|
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CP0566895
|
1-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methyl]triazole-4-carboxylic acid
Show/Hide
|
C27H27ClN4O6
|
1
|
| 1 |
EC50 = 2723 nM
|
|
|
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CP0483535
|
3-[[(2R,3S,4S,5R,6R)-6-[4-chloro-3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-3,4,5-trihydroxyoxan-2-yl]methylamino]-3-oxopropanoic acid
Show/Hide
|
C27H29ClN2O7
|
1
|
| 1 |
EC50 = 3441 nM
|
|
|
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CP0507338
|
(2S,3R,4S,5R)-2-[1-[(4-tert-butylphenyl)methyl]indol-3-yl]oxane-3,4,5-triol
Show/Hide
|
C24H29NO4
|
1
|
| 1 |
EC50 = 3632 nM
|
|
|
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CP0525556
|
(2S,3R,4R,5R)-2-[4-chloro-3-[(4-methylsulfanylphenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C20H23ClO5S
|
1
|
| 1 |
EC50 = 3700 nM
|
|
|
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CP0465074
|
1-(3-benzyl-2-imino-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-3,3-dimethylbutan-2-ol
Show/Hide
|
C20H25N3O
|
1
|
| 1 |
EC50 = 3850 nM
|
|
|
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CP0439724
|
(2S,3R,4S,5R)-2-(1-benzylindol-3-yl)oxane-3,4,5-triol
Show/Hide
|
C20H21NO4
|
1
|
| 1 |
EC50 = 4153 nM
|
|
|
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CP0505813
|
1-(3-benzyl-2-imino-benzimidazol-1-yl)-3-phenoxy-propan-2-ol;hydrochloride
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|
C23H23N3O2
|
1
|
| 1 |
EC50 = 4600 nM
|
|
|
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CP0508823
|
(2S,3R,4R,5R)-2-[4-chloro-3-[(6-methoxynaphthalen-2-yl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C24H25ClO6
|
1
|
| 1 |
EC50 = 5100 nM
|
|
|
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CP0494110
|
2-methyl-7-((6-methylpyridin-2-ylamino)(3,4,5-trimethoxyphenyl)methyl)quinolin-8-ol
Show/Hide
|
C26H27N3O4
|
1
|
| 1 |
EC50 = 5920 nM
|
|
|
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CP0441418
|
2-(2-amino-5-phenylthiophene-3-carbonyl)-N-(4-methoxyphenyl)hydrazinecarbothioamide
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|
C19H18N4O2S2
|
1
|
| 1 |
EC50 = 8980 nM
|
|
|
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CP0459251
|
2-[2-azanylidene-3-[(4-chlorophenyl)methyl]benzimidazol-1-yl]-1-(furan-2-yl)ethanol;hydrochloride
Show/Hide
|
C20H18ClN3O2
|
1
|
| 1 |
EC50 = 11000 nM
|
|
|
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CP0432895
|
(2R,3R,4R,5S)-2-[(1R)-1,2-dihydroxyethyl]-5-[4-methyl-3-[(4-propan-2-ylphenyl)methyl]phenyl]oxolane-3,4-diol
Show/Hide
|
C23H30O5
|
1
|
| 1 |
EC50 = 11000 nM
|
|
|
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CP0486692
|
2-(3-benzyl-2-imino-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-1-(4-methoxyphenyl)ethanol
Show/Hide
|
C23H23N3O2
|
1
|
| 1 |
EC50 = 16200 nM
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CP0459252
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2-(3-benzyl-2-imino-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-1-(thiophen-2-yl)ethanol
Show/Hide
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C20H19N3OS
|
1
|
| 1 |
EC50 = 19100 nM
|
|
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CP0469213
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(2S,3R,4R,5R)-2-[4-chloro-2-methoxy-5-[(4-propan-2-ylphenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C23H29ClO6
|
1
|
| 1 |
EC50 = 21000 nM
|
|
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CP0462102
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(2S,3R,4R,5R)-2-[3-[(4-tert-butylphenyl)methyl]-4-chlorophenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C23H29ClO5
|
1
|
| 1 |
EC50 = 24000 nM
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|
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CP0515459
|
(2S,3R,4S,5R)-2-[1-[(4-fluorophenyl)methyl]indol-3-yl]oxane-3,4,5-triol
Show/Hide
|
C20H20FNO4
|
1
|
| 1 |
EC50 = 25505 nM
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CP0520950
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2-(3-(4-chlorobenzyl)-2-imino-2,3-dihydro-1H-benzo[d]imidazol-1-yl)ethanol
Show/Hide
|
C16H16ClN3O
|
1
|
| 1 |
EC50 = 31100 nM
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|
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CP0434465
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(2S,3R,4R,5R)-2-[4-chloro-3-[(4-propan-2-ylphenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C22H27ClO5
|
1
|
| 1 |
EC50 = 33000 nM
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|
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CP0462100
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(2R,3R,4R,5S)-2-[(1R)-1,2-dihydroxyethyl]-5-[3-[(4-ethoxyphenyl)methyl]-4-methylphenyl]oxolane-3,4-diol
Show/Hide
|
C22H28O6
|
1
|
| 1 |
EC50 = 34000 nM
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|
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CP0441417
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1-(2-furanyl)-2-[2-imino-3-(phenylmethyl)-1-benzimidazolyl]ethanol;hydrochloride
Show/Hide
|
C20H19N3O2
|
1
|
| 1 |
EC50 = 34700 nM
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|
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CP0462101
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(2S,3R,4R,5R)-2-[4-chloro-3-[(4-methoxyphenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C20H23ClO6
|
1
|
| 1 |
EC50 = 35000 nM
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|
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CP0459253
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1-(3-allyl-2-imino-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-3,3-dimethylbutan-2-ol
Show/Hide
|
C16H23N3O
|
1
|
| 1 |
EC50 = 40400 nM
|
|
|
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CP0462099
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(2S,3R,4R,5R)-2-[4-chloro-5-[(4-ethoxyphenyl)methyl]-2-methoxyphenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
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C22H27ClO7
|
1
|
| 1 |
EC50 = 46000 nM
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|
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CP0374985
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2-(3-(4-chlorobenzyl)-2-imino-2,3-dihydro-1H-benzo[d]imidazol-1-yl)acetic acid
Show/Hide
|
C16H14ClN3O2
|
1
|
| 1 |
EC50 > 50000 nM
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|
|
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CP0488403
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2-(3-Benzyl-2-imino-2,3-dihydro-benzoimidazol-1-yl)-ethanol
Show/Hide
|
C16H17N3O
|
1
|
| 1 |
EC50 > 50000 nM
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|
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CP0494111
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1-(2-imino-3-(2-(piperidin-1-yl)ethyl)-2,3-dihydro-1H-benzo[d]imidazol-1-yl)-3,3-dimethylbutan-2-ol
Show/Hide
|
C20H32N4O
|
1
|
| 1 |
EC50 > 50000 nM
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|
|
|
CP0375175
|
(2S,3R,4R,5R)-2-[3-(1,3-benzodioxol-5-ylmethyl)-4-chlorophenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C20H21ClO7
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0443656
|
(2S,3R,4R,5R)-2-[4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C21H25ClO6
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0443657
|
(2S,3R,4R,5R)-2-[4-chloro-3-[(4-phenoxyphenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C25H25ClO6
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0443751
|
(2S,3R,4R,5R)-2-[4-chloro-3-[(2-methoxyphenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C20H23ClO6
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0462098
|
(2S,3R,4R,5R)-2-[4-chloro-3-[(3-methoxyphenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C20H23ClO6
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0508822
|
(2S,3R,4R,5R)-2-[4-chloro-3-[(4-fluorophenyl)methyl]phenyl]-5-[(1R)-1,2-dihydroxyethyl]oxolane-3,4-diol
Show/Hide
|
C19H20ClFO5
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0397523
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(5-pyridin-3-ylthiophen-2-yl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H22ClNO5S
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0541252
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[4-methyl-3-[(5-pyridin-3-ylthiophen-2-yl)methyl]phenyl]oxane-3,4,5-triol
Show/Hide
|
C23H25NO5S
|
1
|
| 1 |
IC50 = 1 nM
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|
|
|
CP0405566
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-2-hydroxy-4-methylphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H26O6
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0405567
|
(2S,3R,4R,5S,6R)-2-[3-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-methylphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H26O5
|
1
|
| 1 |
IC50 = 1 nM
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|
|
|
CP0444393
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-chloro-2-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H25ClO6
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0444396
|
(2S,3R,4R,5S,6R)-2-[3-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-chlorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H23ClO5
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0457145
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-ethyl-2-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C24H30O6
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0466056
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-2,4-dimethoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C23H28O7
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0514927
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-2-hydroxy-4-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H26O7
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0515978
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-2-methoxy-4-methylphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C23H28O6
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0547143
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-chloro-2-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H23ClO6
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0395631
|
(2R,3R,4S,5S,6R)-2-[3-[(4-ethylphenyl)methyl]-4-methylindol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C24H29NO5
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0507297
|
(1S)-1,5-Anhydro-1-[4-chloro-3-[4-(methylsulfanyl)benzyl]phenyl]-1-thio-D-glucitol
Show/Hide
|
C20H23ClO4S2
|
1
|
| 1 |
IC50 = 1.16 nM
|
|
|
|
CP0406312
|
(1S)-1,5-Anhydro-1-[4-chloro-3-(4-methylbenzyl)phenyl]-1-thio-D-glucitol
Show/Hide
|
C20H23ClO4S
|
1
|
| 1 |
IC50 = 1.37 nM
|
|
|
|
CP0526188
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(5-pyrazol-1-ylthiophen-2-yl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C20H21ClN2O5S
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0479981
|
(1S)-1,5-Anhydro-1-[4-chloro-5-(4-ethylbenzyl)-2-methoxyphenyl]-1-thio-D-glucitol
Show/Hide
|
C22H27ClO5S
|
1
|
| 1 |
IC50 = 1.51 nM
|
|
|
|
CP0444290
|
(2R,3R,4S,5S,6R)-2-[3-[(4-cyclopropylphenyl)methyl]-4-methylindol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C25H29NO5
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0479978
|
(1S)-1,5-Anhydro-1-[4-chloro-3-(4-methoxybenzyl)phenyl]-1-thio-D-glucitol
Show/Hide
|
C20H23ClO5S
|
1
|
| 1 |
IC50 = 1.68 nM
|
|
|
|
CP0508556
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[4-methyl-3-[(5-pyrimidin-2-ylthiophen-2-yl)methyl]phenyl]oxane-3,4,5-triol
Show/Hide
|
C22H24N2O5S
|
1
|
| 1 |
IC50 = 1.7 nM
|
|
|
|
CP0462892
|
(1S)-1,5-Anhydro-1-[5-(4-ethylbenzyl)-2-methoxy-4-methylphenyl]-1-thio-D-glucitol
Show/Hide
|
C23H30O5S
|
1
|
| 1 |
IC50 = 1.71 nM
|
|
|
|
CP0479982
|
(1S)-1,5-Anhydro-1-[4-chloro-3-(4-ethoxybenzyl)phenyl]-1-thio-D-glucitol
Show/Hide
|
C21H25ClO5S
|
1
|
| 1 |
IC50 = 1.77 nM
|
|
|
|
CP0513985
|
(1S)-1,5-Anhydro-1-[4-chloro-3-(4-ethylbenzyl)phenyl]-1-thio-D-glucitol
Show/Hide
|
C21H25ClO4S
|
1
|
| 1 |
IC50 = 1.78 nM
|
|
|
|
CP0508555
|
(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[5-(6-fluoropyridin-3-yl)thiophen-2-yl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H21ClFNO5S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0514928
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-ethyl-2-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C23H28O6
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0493036
|
(2S,3R,4R,5S,6R)-2-[3-chloro-4-[(4-ethoxyphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H25ClO6
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0392697
|
(2S,3R,4R,5S,6R)-2-[5-[(4-ethylphenyl)methyl]-2-hydroxy-4-methylphenyl]-6-(hydroxymethyl)thiane-3,4,5-triol
Show/Hide
|
C22H28O5S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0411696
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[2-hydroxy-4-methyl-5-[(4-methylphenyl)methyl]phenyl]thiane-3,4,5-triol
Show/Hide
|
C21H26O5S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0834420
|
Canagliflozin
Show/Hide
|
C48H52F2O11S2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0420661
|
(2R,3R,4S,5S,6R)-2-[3-[(4-cyclopropylphenyl)methyl]indol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C24H27NO5
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0076250
|
(1S)-1,5-Anhydro-1-[5-(4-ethoxybenzyl)-2-methoxy-4-methylphenyl]-1-thio-D-glucitol
Show/Hide
|
C23H30O6S
|
1
|
| 1 |
IC50 = 2.26 nM
|
|
|
|
CP0495877
|
(1S)-1,5-Anhydro-1-[3-(4-ethoxybenzyl)-4-methylphenyl]-1-thio-D-glucitol
Show/Hide
|
C22H28O5S
|
1
|
| 1 |
IC50 = 2.29 nM
|
|
|
|
CP0561033
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[4-methyl-3-[[5-(1,3-thiazol-5-yl)thiophen-2-yl]methyl]phenyl]oxane-3,4,5-triol
Show/Hide
|
C21H23NO5S2
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0393316
|
2-[[5-[(2S,3R,4R,5S,6R)-5-fluoro-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-4-hydroxy-2-methylphenyl]methyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carbonitrile
Show/Hide
|
C22H25FN2O5S
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0470293
|
(1S)-1,5-Anhydro-1-[2-methoxy-4-methyl-5-[4-(propan-2-yl)-benzyl]phenyl]-1-thio-D-glucitol
Show/Hide
|
C24H32O5S
|
1
|
| 1 |
IC50 = 2.68 nM
|
|
|
|
CP0444394
|
(2S,3R,4R,5S,6R)-2-[3-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-ethylphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C23H28O5
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0444395
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-2-fluoro-4-methylphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H25FO5
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0547145
|
(2S,3R,4R,5S,6R)-2-[3-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C22H26O6
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0564226
|
(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-chloro-2-fluorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H22ClFO5
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0471886
|
(2S,3R,4R,5S,6R)-2-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-hydroxy-2,3-dihydro-1-benzofuran-5-yl]-5-fluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
|
C23H25FO8
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0389349
|
(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[2-hydroxy-4-methyl-5-[(4-propan-2-yloxyphenyl)methyl]phenyl]thiane-3,4,5-triol
Show/Hide
|
C23H30O6S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0440178
|
(2S,3R,4R,5S,6R)-2-[5-[(4-ethoxyphenyl)methyl]-2-hydroxy-4-methylphenyl]-6-(hydroxymethyl)thiane-3,4,5-triol
Show/Hide
|
C22H28O6S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0487386
|
(2R,3R,4S,5S,6R)-2-[2-[(4-ethylphenyl)methyl]anilino]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C21H27NO5
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0434622
|
2-[[(E)-4-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)thian-2-yl]phenyl]methyl]phenyl]but-3-enoyl]amino]-2-methylpropanamide
Show/Hide
|
C28H36N2O7S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0440176
|
1-(1-hydroxy-2-methylpropan-2-yl)-3-[2-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]ethyl]urea
Show/Hide
|
C27H38N2O8
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0543910
|
(1S)-1,5-Anhydro-1-[4-chloro-3-[4-(propan-2-yl)benzyl]phenyl]-1-thio-D-glucitol
Show/Hide
|
C22H27ClO4S
|
1
|
| 1 |
IC50 = 4.01 nM
|
|
|
|
CP0165583
|
(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-{2-[(4-methoxyphenyl)methyl]phenoxy}oxane-3,4,5-triol
Show/Hide
|
C20H24O7
|
1
|
| 1 |
IC50 = 4.8 nM
|
|
|
|
CP0522997
|
(2R,3R,4S,5S,6R)-2-[3-[(4-ethoxyphenyl)methyl]-4-fluoroindol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C23H26FNO6
|
1
|
| 1 |
IC50 = 4.8 nM
|
|
|
|
CP0405568
|
(2S,3R,4R,5S,6R)-2-[3-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-cyclopropylphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
|
C24H28O5
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0411695
|
(E)-N-(1,3-dihydroxy-2-methylpropan-2-yl)-4-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)thian-2-yl]phenyl]methyl]phenyl]but-3-enamide
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C28H37NO8S
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1
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| 1 |
IC50 = 5 nM
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CP0426535
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N-[3-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]propyl]-4-methylpiperazine-1-carboxamide
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C29H41N3O7
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1
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| 1 |
IC50 = 5 nM
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CP0476741
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1-(1-hydroxy-2-methylpropan-2-yl)-3-[3-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]propyl]urea
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C28H40N2O8
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1
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| 1 |
IC50 = 5 nM
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CP0262485
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(2S,3R,4R,5S,6R)-2-[3-[(4-ethylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C21H26O5
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1
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| 1 |
IC50 = 5.1 nM
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CP0420663
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(2R,3R,4S,5S,6R)-2-[3-[(4-ethylphenyl)methyl]-4-fluoroindol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C23H26FNO5
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1
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| 1 |
IC50 = 5.2 nM
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CP0405782
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2-[[5-[(2S,3R,4R,5S,6R)-5-fluoro-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-4-methoxy-2-methylphenyl]methyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carbonitrile
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C23H27FN2O5S
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1
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| 1 |
IC50 = 5.3 nM
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CP0518786
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(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-4-cyclopropyl-2-hydroxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C24H28O6
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1
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| 1 |
IC50 = 6 nM
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CP0178282
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CANAGLIFLOZIN
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C24H25FO5S
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1
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| 1 |
IC50 = 6.7 nM
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CP0389347
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1-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-3-[3-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]propyl]urea
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C28H40N2O10
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1
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| 1 |
IC50 = 7 nM
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CP0389348
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2-[[(E)-4-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]but-3-enoyl]amino]-2-methylpropanamide
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C28H36N2O8
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1
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| 1 |
IC50 = 7 nM
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CP0411780
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1-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-3-[2-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]ethyl]urea
Show/Hide
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C27H38N2O10
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1
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| 1 |
IC50 = 7 nM
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CP0395632
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(2R,3R,4S,5S,6R)-2-[3-[(4-ethylphenyl)methyl]indol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C23H27NO5
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1
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| 1 |
IC50 = 7.1 nM
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CP0561034
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(2R,3S,4R,5R,6S)-2-(hydroxymethyl)-6-[4-methyl-3-[(5-pyrimidin-5-ylthiophen-2-yl)methyl]phenyl]oxane-3,4,5-triol
Show/Hide
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C22H24N2O5S
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1
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| 1 |
IC50 = 7.3 nM
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CP0514139
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(2S,3R,4R,5S,6R)-2-[5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-methoxy-2,3-dihydro-1-benzofuran-7-yl]-5-fluoro-6-(hydroxymethyl)oxane-3,4-diol
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C24H27FO8
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1
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| 1 |
IC50 = 7.5 nM
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CP0253223
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(1R,2R,3S,4S,6R)-4-[3-[(4-ethylphenyl)methyl]-4-methoxyphenyl]-6-(hydroxymethyl)cyclohexane-1,2,3-triol
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C23H30O5
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1
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| 1 |
IC50 = 8.3 nM
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CP0431878
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(2S,3R,4R,5S,6R)-2-[7-(2,3-dihydro-1,4-benzoxathiin-6-ylmethyl)-4-methoxy-2,3-dihydro-1-benzofuran-5-yl]-5-fluoro-6-(hydroxymethyl)oxane-3,4-diol
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C24H27FO7S
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1
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| 1 |
IC50 = 8.3 nM
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CP0295291
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(1R,2R,3S,4S,6R)-4-[5-[(4-ethylphenyl)methyl]-2,4-dimethoxyphenyl]-6-(hydroxymethyl)cyclohexane-1,2,3-triol
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C24H32O6
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1
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| 1 |
IC50 = 8.5 nM
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CP0179227
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(2S,3R,4R,5S,6R)-2-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-methoxy-2,3-dihydro-1-benzofuran-5-yl]-5-fluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
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C24H27FO8
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1
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| 1 |
IC50 = 9 nM
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CP0440177
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(E)-N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-4-[4-[[4-hydroxy-2-methyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)thian-2-yl]phenyl]methyl]phenyl]but-3-enamide
Show/Hide
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C28H37NO9S
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1
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| 1 |
IC50 = 9 nM
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CP0479979
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(1S)-1,5-Anhydro-1-[3-(4-ethoxybenzyl)-4-fluorophenyl]-1-thio-D-glucitol
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C21H25FO5S
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1
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| 1 |
IC50 = 9.4 nM
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CP0304363
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(1R,2R,3S,4R,5R)-1-[2-ethoxy-5-[(4-ethylphenyl)methyl]phenyl]-5-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol
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C24H32O6
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1
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| 1 |
IC50 = 9.9 nM
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CP0271163
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(1R,2R,3S,4R,5R)-1-[5-[(4-ethylphenyl)methyl]-2,4-dimethoxyphenyl]-5-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol
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C24H32O7
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1
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| 1 |
IC50 = 10 nM
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CP0550429
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(2S,3R,4R,5S,6R)-2-[5-(3-bicyclo[4.2.0]octa-1(6),2,4-trienylmethyl)-2-fluoro-4-methoxyphenyl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C22H25FO6
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1
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| 1 |
IC50 = 10 nM
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CP0432924
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(E)-4-[4-[[2,4-dimethyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-N-(1-hydroxy-2-methylpropan-2-yl)-2,2-dimethylbut-3-enamide
Show/Hide
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C31H43NO7
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1
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| 1 |
IC50 = 10 nM
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CP0447633
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(1S)-1,5-Anhydro-1-[2,4-dimethoxy-5-(4-ethoxybenzyl)phenyl]-1-thio-D-glucitol
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C23H30O7S
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1
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| 1 |
IC50 = 10.8 nM
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CP0123977
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1-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-3-ethylimidazolidine-2,4-dione
Show/Hide
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C24H27ClN2O7
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1
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| 1 |
IC50 = 10.9 nM
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CP0042564
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3-(1-benzofuran-5-yl)-1-(2-hydroxy-4-methyl-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}phenyl)propan-1-one
Show/Hide
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C24H26O9
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2
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| 1 |
IC50 = 11 nM
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| 2 |
Ki = 4 nM
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CP0238425
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(1R,2R,3S,4S,6R)-4-[3-[(4-cyclopropylphenyl)methyl]phenyl]-6-(hydroxymethyl)cyclohexane-1,2,3-triol
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C23H28O4
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1
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| 1 |
IC50 = 11 nM
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CP0420658
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(2R,3R,4S,5S,6R)-2-[3-[(4-cyclobutylphenyl)methyl]indol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C25H29NO5
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1
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| 1 |
IC50 = 11 nM
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CP0257117
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(1R,2R,3S,4S,6R)-4-[5-[(4-ethylphenyl)methyl]-2-methoxyphenyl]-6-(hydroxymethyl)cyclohexane-1,2,3-triol
Show/Hide
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C23H30O5
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1
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| 1 |
IC50 = 12 nM
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CP0406313
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(1S)-1,5-Anhydro-1-[3-(4-ethoxybenzyl)-4-methoxyphenyl]-1-thio-D-glucitol
Show/Hide
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C22H28O6S
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1
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| 1 |
IC50 = 13.4 nM
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CP0514140
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[2-[[5-[(2S,3R,4R,5S,6R)-5-fluoro-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-4-hydroxy-2-methylphenyl]methyl]-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-pyrrolidin-1-ylmethanone
Show/Hide
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C26H33FN2O6S
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1
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| 1 |
IC50 = 13.6 nM
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CP0257119
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(1R,2R,3S,4R,5R)-1-[5-[(4-ethylphenyl)methyl]-2-methoxyphenyl]-5-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol
Show/Hide
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C23H30O6
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1
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| 1 |
IC50 = 14 nM
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CP0438151
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(E)-4-[4-[[4-methoxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-2,2-dimethyl-N-(2-methyl-1-oxo-1-piperazin-1-ylpropan-2-yl)but-3-enamide
Show/Hide
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C37H53N3O8
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1
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| 1 |
IC50 = 17 nM
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CP0455864
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(E)-4-[4-[[2,4-dimethyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-fluorophenyl]-N-(1-hydroxy-2-methylpropan-2-yl)-2,2-dimethylbut-3-enamide
Show/Hide
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C31H42FNO7
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1
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| 1 |
IC50 = 17 nM
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CP0507296
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(1S)-1,5-Anhydro-1-[5-(4-ethoxybenzyl)-2-hydroxyphenyl]-1-thio-D-glucitol
Show/Hide
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C21H26O6S
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1
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| 1 |
IC50 = 17.4 nM
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CP0483825
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(2R,3R,4S,5S,6R)-2-[3-[(4-chlorophenyl)methyl]-4-fluoroindol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C21H21ClFNO5
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1
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| 1 |
IC50 = 18 nM
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CP0479977
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(1S)-1,5-Anhydro-1-[3-(4-tert-butylbenzyl)-4-chlorophenyl]-1-thio-D-glucitol
Show/Hide
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C23H29ClO4S
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1
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| 1 |
IC50 = 18.8 nM
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CP0257120
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(1R,2R,3S,4S,6R)-4-[2-ethoxy-5-[(4-ethylphenyl)methyl]phenyl]-6-(hydroxymethyl)cyclohexane-1,2,3-triol
Show/Hide
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C24H32O5
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1
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| 1 |
IC50 = 19 nM
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CP0438152
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(E)-N-(1-hydroxy-2-methylpropan-2-yl)-4-[4-[[4-hydroxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-2,2-dimethylbut-3-enamide
Show/Hide
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C32H45NO8
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1
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| 1 |
IC50 = 19 nM
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CP0476998
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(E)-N-[1-[2-(dimethylamino)ethylamino]-2-methyl-1-oxopropan-2-yl]-4-[4-[[4-methoxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-2,2-dimethylbut-3-enamide
Show/Hide
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C37H55N3O8
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1
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| 1 |
IC50 = 20 nM
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CP0393318
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[2-[[5-[(2S,3R,4R,5S,6R)-5-fluoro-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-4-methoxy-2-methylphenyl]methyl]-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-(1,3-thiazol-2-yl)methanone
Show/Hide
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C26H29FN2O6S2
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1
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| 1 |
IC50 = 23.2 nM
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CP0440246
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1-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-3-propan-2-ylimidazolidine-2,4-dione
Show/Hide
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C25H29ClN2O7
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1
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| 1 |
IC50 = 23.6 nM
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CP0483824
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(2R,3R,4S,5S,6R)-2-[3-[(4-cyclopentylphenyl)methyl]-4-fluoroindol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C26H30FNO5
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1
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| 1 |
IC50 = 24 nM
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CP0422370
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(E)-4-[4-[[4-methoxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-2,2-dimethyl-N-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]but-3-enamide
Show/Hide
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C38H55N3O8
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1
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| 1 |
IC50 = 26 nM
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CP0432748
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(2S,3R,4S,5S,6R)-2-(3-(4-ethylbenzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C23H27NO6
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1
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| 1 |
IC50 = 28 nM
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CP0462150
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(E)-4-[4-[[4-hydroxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethyl-N-(2-methyl-1-oxo-1-piperazin-1-ylpropan-2-yl)but-3-enamide
Show/Hide
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C37H53N3O8
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1
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| 1 |
IC50 = 28 nM
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CP0116142
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US8575114, I-12
Show/Hide
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C20H21Cl2N3O6
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1
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| 1 |
IC50 = 33 nM
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CP0427045
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(E)-N-(1-hydroxy-2-methylpropan-2-yl)-4-[4-[[4-methoxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-2,2-dimethylbut-3-enamide
Show/Hide
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C33H47NO8
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1
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| 1 |
IC50 = 34 nM
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CP0393317
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[2-[[5-[(2S,3R,4R,5S,6R)-5-fluoro-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-4-hydroxy-2-methylphenyl]methyl]-6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl]-(1,3-thiazol-2-yl)methanone
Show/Hide
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C25H27FN2O6S2
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1
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| 1 |
IC50 = 36 nM
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CP0523522
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ethyl 2-[[5-[(2S,3R,4R,5S,6R)-5-fluoro-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-4-hydroxy-2-methylphenyl]methyl]-6,7-dihydro-4H-thieno[3,2-c]pyridine-5-carboxylate
Show/Hide
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C24H30FNO7S
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1
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| 1 |
IC50 = 36 nM
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CP0470295
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(1S)-1,5-Anhydro-1-[5-(4-ethoxybenzyl)-2-methoxyphenyl]-1-thio-D-glucitol
Show/Hide
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C22H28O6S
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1
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| 1 |
IC50 = 37.9 nM
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CP0394714
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(2S,3R,4S,5S,6R)-2-(3-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)-3H-benzo[d]imidazol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C23H26N2O7
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1
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| 1 |
IC50 = 39 nM
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CP0278902
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(1R,2R,3S,4S,6R)-4-[3-[(4-ethylphenyl)methyl]phenyl]-6-(hydroxymethyl)cyclohexane-1,2,3-triol
Show/Hide
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C22H28O4
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1
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| 1 |
IC50 = 49 nM
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CP0529776
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(2S,3R,4S,5S,6R)-2-(3-(4-(thiophen-3-yl)benzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H25NO6S
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1
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| 1 |
IC50 = 50 nM
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CP0525132
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(2S,3R,4S,5S,6R)-2-(3-(4-(methylthio)benzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C22H25NO6S
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1
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| 1 |
IC50 = 52 nM
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CP0238422
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(1R,2R,3S,4S,6R)-4-[5-[(4-ethylphenyl)methyl]-2-methylphenyl]-6-(hydroxymethyl)cyclohexane-1,2,3-triol
Show/Hide
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C23H30O4
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1
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| 1 |
IC50 = 52 nM
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CP0508309
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(2S,3R,4R,5S,6R)-2-[5-(2,3-dihydro-1,4-benzoxathiin-6-ylmethyl)-4-methoxy-2,3-dihydro-1-benzofuran-7-yl]-5-fluoro-6-(hydroxymethyl)oxane-3,4-diol
Show/Hide
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C24H27FO7S
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1
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| 1 |
IC50 = 62.3 nM
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CP0490840
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(E)-N-[1-[(2-amino-2-methylpropyl)amino]-2-methyl-1-oxopropan-2-yl]-4-[4-[[4-hydroxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethylbut-3-enamide
Show/Hide
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C37H55N3O8
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1
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| 1 |
IC50 = 64 nM
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CP0382434
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(2R,3S,4S,5R,6S)-2-Hydroxymethyl-6-[3-(4-methyl-benzyl)-1H-indol-4-yloxy]-tetrahydro-pyran-3,4,5-triol
Show/Hide
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C22H25NO6
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1
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| 1 |
IC50 = 66 nM
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CP0490019
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(2R,3R,4S,5S,6R)-2-[3-[(4-ethylphenyl)methyl]indazol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
Show/Hide
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C22H26N2O5
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1
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| 1 |
IC50 = 69 nM
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CP0438141
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(E)-N-(1-hydroxy-2-methylpropan-2-yl)-4-[4-[[4-hydroxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethylbut-3-enamide
Show/Hide
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C33H47NO8
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1
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| 1 |
IC50 = 69 nM
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CP0295288
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(1S,2R,3R,4R,6S)-4-(hydroxymethyl)-6-[3-[(4-methoxyphenyl)methyl]phenyl]cyclohexane-1,2,3-triol
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C21H26O5
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1
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| 1 |
IC50 = 73 nM
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CP0414915
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(1S)-1,5-Anhydro-1-[3-(4-ethoxybenzyl)phenyl]-1-thio-D-glucitol
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C21H26O5S
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1
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| 1 |
IC50 = 73.6 nM
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CP0462149
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(E)-N-[1-[2-(dimethylamino)ethylamino]-2-methyl-1-oxopropan-2-yl]-4-[4-[[4-hydroxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethylbut-3-enamide
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C37H55N3O8
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1
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| 1 |
IC50 = 74 nM
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CP0144510
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US8575114, I-8
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C19H19Cl2N3O6
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1
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| 1 |
IC50 = 80 nM
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CP0432923
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(E)-4-[4-[[4-hydroxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethyl-N-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl]but-3-enamide
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C38H55N3O8
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1
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| 1 |
IC50 = 81 nM
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CP0168979
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US8575114, I-1
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C19H20ClN3O6
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1
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| 1 |
IC50 = 83 nM
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CP0477000
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(E)-4-[4-[[2,4-dimethyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-N-(1-hydroxy-2-methylpropan-2-yl)-2,2-dimethylbut-3-enamide
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C32H45NO7
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1
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| 1 |
IC50 = 84 nM
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CP0439466
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(2S,3R,4S,5S,6R)-2-(3-Biphenyl-4-ylmethyl-1H-indol-4-yloxy)-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol
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C27H27NO6
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1
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| 1 |
IC50 = 89 nM
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CP0064929
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US8575114, I-4
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C19H19Cl2N3O6
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1
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| 1 |
IC50 = 89 nM
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CP0395629
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(2R,3R,4S,5S,6R)-2-[3-[(4-cyclopentylphenyl)methyl]indol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C26H31NO5
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1
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| 1 |
IC50 = 93 nM
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CP0376615
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(2S,3R,4S,5S,6R)-2-(3-(4-ethoxybenzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H27NO7
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1
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| 1 |
IC50 = 94 nM
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CP0439468
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(2S,3R,4S,5S,6R)-2-(3-(3-fluoro-4-methylbenzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C22H24FNO6
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1
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| 1 |
IC50 = 99 nM
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CP0333794
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(1R,2R,3S,4R,5R)-1-[3-[(4-ethylphenyl)methyl]-4-methoxyphenyl]-5-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol
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C23H30O6
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1
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| 1 |
IC50 = 100 nM
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CP0147994
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US8575114, I-10
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C19H19BrClN3O6
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1
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| 1 |
IC50 = 107 nM
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CP0306169
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US8575114, I-9
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C20H22ClN3O6
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1
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| 1 |
IC50 = 110 nM
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CP0446642
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(2S,3R,4S,5S,6R)-2-(3-(4-propylbenzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C24H29NO6
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1
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| 1 |
IC50 = 119 nM
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CP0440236
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US8575114, I-2
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C20H22ClN3O6
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1
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| 1 |
IC50 = 120 nM
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CP0467646
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(2S,3R,4S,5S,6R)-2-(3-(2-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)ethyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C24H27NO8
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1
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| 1 |
IC50 = 121 nM
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CP0501947
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(2S,3R,4S,5S,6R)-2-(3-(4-methoxybenzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C22H25NO7
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1
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| 1 |
IC50 = 121 nM
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CP0376616
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(2S,3R,4R,5S,6R)-2-(3-(4-ethylbenzyl)-1H-indol-5-yl)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H27NO5
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1
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| 1 |
IC50 = 132 nM
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CP0210606
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US8575114, I-6
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C20H22ClN3O7
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1
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| 1 |
IC50 = 141 nM
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CP0436988
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(2S,3R,4S,5S,6R)-2-(3-(4-(pyridin-3-yl)benzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C26H26N2O6
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1
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| 1 |
IC50 = 143 nM
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CP0508169
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(2S,3R,4S,5S,6R)-2-(3-(3-fluoro-4-methoxybenzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C22H24FNO7
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1
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| 1 |
IC50 = 143 nM
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CP0424982
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(2S,3R,4S,5S,6R)-2-(3-(4-methoxyphenethyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C23H27NO7
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1
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| 1 |
IC50 = 163 nM
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CP0411611
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5-[(4-ethylphenyl)methyl]-1-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]pyridin-2-one
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C20H25NO6
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1
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| 1 |
IC50 = 163 nM
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CP0178283
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(1R,2R,3S,4R,5R)-1-[5-[(4-ethylphenyl)methyl]-2-methylphenyl]-5-(hydroxymethyl)cyclohexane-1,2,3,4-tetrol
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C23H30O5
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1
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| 1 |
IC50 = 170 nM
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CP0497497
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(2S,3R,4S,5S,6R)-2-[3-(2-Fluoro-biphenyl-4-ylmethyl)-1H-indol-4-yloxy]-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol
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C27H26FNO6
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1
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| 1 |
IC50 = 182 nM
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CP0493902
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(E)-4-[4-[[4-methoxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethyl-N-[2-methyl-1-oxo-1-(2-piperazin-1-ylethylamino)propan-2-yl]but-3-enamide
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C40H60N4O8
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1
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| 1 |
IC50 = 200 nM
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CP0382435
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-(3-(2-(naphthalen-2-yl)ethyl)-1H-indol-4-yloxy)-tetrahydro-2H-pyran-3,4,5-triol
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C26H27NO6
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1
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| 1 |
IC50 = 201 nM
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CP0501948
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(2S,3R,4S,5S,6R)-2-(3-(4-ethoxyphenethyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C24H29NO7
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1
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| 1 |
IC50 = 202 nM
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CP0057639
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US8575114, I-11
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C19H19ClFN3O6
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1
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| 1 |
IC50 = 222 nM
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CP0510246
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1-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-3,5,5-trimethylimidazolidine-2,4-dione
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C25H29ClN2O7
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1
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| 1 |
IC50 = 248 nM
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CP0148733
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US8575114, I-3
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C20H19ClF3N3O6
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1
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| 1 |
IC50 = 252 nM
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CP0767289
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Sergliflozin
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C23H28O9
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1
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| 1 |
IC50 = 260 nM
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CP0473812
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(E)-4-[4-[[4-methoxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethyl-N-[2-methyl-1-[2-(4-methylpiperazin-1-yl)ethylamino]-1-oxopropan-2-yl]but-3-enamide
Show/Hide
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C41H62N4O8
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1
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| 1 |
IC50 = 281 nM
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CP0479980
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(1S)-1,5-Anhydro-1-[3-(4-ethoxybenzyl)-4-hydroxyphenyl]-1-thio-D-glucitol
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C21H26O6S
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1
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| 1 |
IC50 = 283 nM
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CP0439465
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(2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-(3-(naphthalen-2-ylmethyl)-1H-indol-4-yloxy)-tetrahydro-2H-pyran-3,4,5-triol
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C25H25NO6
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1
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| 1 |
IC50 = 293 nM
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CP0436617
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(2S,3R,4S,5S,6R)-2-(3-(4-chlorobenzyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H22ClNO6
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1
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| 1 |
IC50 = 296 nM
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CP0551300
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(E)-N-[1-[(2-amino-2-methylpropyl)amino]-2-methyl-1-oxopropan-2-yl]-4-[4-[[4-methoxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethylbut-3-enamide
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C38H57N3O8
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1
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| 1 |
IC50 = 322 nM
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CP0506662
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1-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-3-tritylimidazolidine-2,4-dione
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C41H37ClN2O7
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1
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| 1 |
IC50 = 328 nM
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CP0455863
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(E)-N-(1-hydroxy-2-methylpropan-2-yl)-4-[4-[[4-methoxy-2-propan-2-yl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methylphenyl]-2,2-dimethylbut-3-enamide
Show/Hide
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C34H49NO8
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1
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| 1 |
IC50 = 354 nM
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CP0485880
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(2S,3R,4S,5S,6R)-2-(3-(4-methoxyphenethyl)-3H-benzo[d][1,2,3]triazol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
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C21H25N3O7
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1
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| 1 |
IC50 = 380 nM
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CP0510439
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(2R,3R,4S,5S,6R)-2-[4-[(4-ethylphenyl)methyl]pyrazol-1-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C18H24N2O5
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1
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| 1 |
IC50 = 381 nM
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CP0401541
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(2S,3R,4S,5S,6R)-2-(3-(4-methoxyphenethyl)-6-methyl-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H29NO7
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1
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| 1 |
IC50 = 394 nM
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CP0422234
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(2S,3R,4S,5S,6R)-2-(3-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)-6-methyl-1H-indazol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H28N2O7
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1
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| 1 |
IC50 = 458 nM
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CP0440247
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1-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]-3-methylimidazolidine-2,4-dione
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C23H25ClN2O7
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1
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| 1 |
IC50 = 489 nM
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CP0485878
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(2S,3R,4S,5S,6R)-2-(3-(2-(benzofuran-5-yl)ethyl)-6-methyl-1H-indazol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C24H26N2O7
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1
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| 1 |
IC50 = 491 nM
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CP0428314
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(2S,3R,4S,5S,6R)-2-(3-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)-6-ethyl-1H-indazol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H30N2O7
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1
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| 1 |
IC50 = 532 nM
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CP0485879
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(2S,3R,4S,5S,6R)-2-(3-(2-(2,3-dihydrobenzofuran-5-yl)ethyl)-1,6-dimethyl-1H-indazol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C25H30N2O7
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1
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| 1 |
IC50 = 754 nM
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CP0120490
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US8575114, I-5
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C20H19ClF3N3O6
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1
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| 1 |
IC50 = 762 nM
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CP0424398
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(E)-4-[4-[[2,4-dimethyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-methoxyphenyl]-N-(1-hydroxy-2-methylpropan-2-yl)-2,2-dimethylbut-3-enamide
Show/Hide
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C32H45NO8
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1
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| 1 |
IC50 = 798 nM
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CP0566839
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(2R,3R,4S,5S,6R)-2-[3-[(4-ethylphenyl)methyl]indazol-2-yl]-6-(hydroxymethyl)oxane-3,4,5-triol
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C22H26N2O5
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1
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| 1 |
IC50 = 1098 nM
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CP0446646
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(2S,3R,4S,5S,6R)-2-(3-((2,3-dihydrobenzofuran-6-yl)methyl)-1H-indol-4-yloxy)-6-(hydroxymethyl)-tetrahydro-2H-pyran-3,4,5-triol
Show/Hide
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C23H25NO7
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1
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| 1 |
IC50 = 1870 nM
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CP0476997
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(E)-4-[4-[[2,4-dimethyl-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-3-propan-2-ylphenyl]-N-(1-hydroxy-2-methylpropan-2-yl)-2,2-dimethylbut-3-enamide
Show/Hide
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C34H49NO7
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1
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| 1 |
IC50 = 2126 nM
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CP0440235
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2-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-8-fluoro-[1,2,4]triazolo[4,3-a]pyridin-3-one
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C19H19ClFN3O6
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1
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| 1 |
IC50 = 3296 nM
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CP0541001
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2-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-7-methoxy-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
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C20H22ClN3O7
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1
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| 1 |
IC50 = 5478 nM
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CP0399424
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2-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-7-(2,2,2-trifluoroethoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
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C21H21ClF3N3O7
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1
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| 1 |
IC50 = 5699 nM
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CP0566840
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3-[(4-ethylphenyl)methyl]-1-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]pyridin-2-one
Show/Hide
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C20H25NO6
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1
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| 1 |
IC50 = 6671 nM
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CP0415674
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8-chloro-2-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
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C19H19Cl2N3O6
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1
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| 1 |
IC50 = 9000 nM
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CP0440245
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2-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]-5-methyl-[1,2,4]triazolo[4,3-a]pyridin-3-one
Show/Hide
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C20H22ClN3O6
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1
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| 1 |
IC50 = 9916 nM
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CP0379164
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3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-1-[2-hydroxy-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-propan-1-one
Show/Hide
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C24H28O10
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1
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| 1 |
Ki = 9 nM
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CP0379163
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1-[2-Hydroxy-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-naphthalen-2-yl-propan-1-one
Show/Hide
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C26H28O8
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1
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| 1 |
Ki = 10 nM
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CP0442226
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3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-1-[4-ethyl-2-hydroxy-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-propan-1-one
Show/Hide
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C25H30O10
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1
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| 1 |
Ki = 10 nM
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CP0445528
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1-[4-Ethyl-2-hydroxy-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-naphthalen-2-yl-propan-1-one
Show/Hide
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C27H30O8
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1
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| 1 |
Ki = 10 nM
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CP0445585
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3-(4-Ethoxy-phenyl)-1-[2-hydroxy-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-propan-1-one
Show/Hide
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C24H30O9
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1
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| 1 |
Ki = 10 nM
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CP0469285
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1-[4-Chloro-2-hydroxy-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-propan-1-one
Show/Hide
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C23H25ClO10
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1
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| 1 |
Ki = 20 nM
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CP0486396
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3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-1-[2-hydroxy-4-isopropyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-propan-1-one
Show/Hide
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C26H32O10
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1
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| 1 |
Ki = 20 nM
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CP0451815
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1-[4-Chloro-2-hydroxy-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-naphthalen-2-yl-propan-1-one
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C25H25ClO8
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1
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| 1 |
Ki = 30 nM
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CP0485717
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3-(4-Ethoxy-phenyl)-1-[4-ethyl-2-hydroxy-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-propan-1-one
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C25H32O9
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1
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| 1 |
Ki = 30 nM
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CP0420102
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3-Cyclohexyl-1-[2-hydroxy-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-propan-1-one
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C22H32O8
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1
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| 1 |
Ki = 40 nM
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CP0435397
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1-[2-Hydroxy-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-thiophen-3-yl-propan-1-one
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C20H24O8S
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1
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| 1 |
Ki = 70 nM
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CP0451816
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1-[4-Fluoro-2-hydroxy-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-naphthalen-2-yl-propan-1-one
Show/Hide
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C25H25FO8
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1
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| 1 |
Ki = 70 nM
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CP0435324
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1-[4-Chloro-2-hydroxy-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-(4-ethoxy-phenyl)-propan-1-one
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C23H27ClO9
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1
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| 1 |
Ki = 80 nM
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CP0496909
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3-(4-Ethoxy-phenyl)-1-[2-hydroxy-4-isopropyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-propan-1-one
Show/Hide
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C26H34O9
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1
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| 1 |
Ki = 110 nM
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CP0448886
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1-[2-Hydroxy-4-isopropyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-naphthalen-2-yl-propan-1-one
Show/Hide
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C28H32O8
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1
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| 1 |
Ki = 150 nM
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CP0442218
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3-Furan-3-yl-1-[2-hydroxy-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-propan-1-one
Show/Hide
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C20H24O9
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1
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| 1 |
Ki = 230 nM
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CP0551768
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1-[2-Amino-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-propan-1-one
Show/Hide
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C24H29NO9
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1
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| 1 |
Ki = 290 nM
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CP0485716
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1-[2-Amino-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-naphthalen-2-yl-propan-1-one
Show/Hide
|
C26H29NO7
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1
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| 1 |
Ki = 520 nM
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CP0551760
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1-[2-Amino-4-methyl-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-(4-ethoxy-phenyl)-propan-1-one
Show/Hide
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C24H31NO8
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1
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| 1 |
Ki = 1280 nM
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CP0420103
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1-[2-Chloro-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-(4-ethoxy-phenyl)-propan-1-one
Show/Hide
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C23H27ClO8
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1
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| 1 |
Ki > 1700 nM
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CP0464620
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1-[2-Chloro-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-naphthalen-2-yl-propan-1-one
Show/Hide
|
C25H25ClO7
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1
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| 1 |
Ki > 1700 nM
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CP0485709
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1-[2-Chloro-6-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yloxy)-phenyl]-3-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-propan-1-one
Show/Hide
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C23H25ClO9
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1
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| 1 |
Ki > 1700 nM
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