| Compound ID |
Compound Name |
Compound Formula |
|
CP0060212
|
N-[(3-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 < 1 nM
|
|
|
|
CP0074413
|
N-[(1R)-1-(3-methoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
Show/Hide
|
C20H19N5O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0094071
|
N-[(1R)-1-(3-methoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
|
C21H20N4O2
|
1
|
| 1 |
IC50 < 1 nM
|
|
|
|
CP0127884
|
2-[(3S,4R)-4-(4-chlorophenyl)pyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C21H18ClN5O
|
1
|
| 1 |
IC50 < 1 nM
|
|
|
|
CP0128777
|
N-[(4-chlorophenyl)-[4-oxo-6-(1H-pyrazol-4-yl)-3H-quinazolin-2-yl]methyl]-2-(dimethylamino)acetamide
Show/Hide
|
C22H21ClN6O2
|
1
|
| 1 |
IC50 < 1 nM
|
|
|
|
CP0185392
|
2-[(3S,4R)-4-phenylpyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C21H19N5O
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0140194
|
N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-ylbenzamide
Show/Hide
|
C21H20N2O2
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0070702
|
N-[(3-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine-3-carboxamide
Show/Hide
|
C19H17N5O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0077151
|
N-[(3-methoxyphenyl)methyl]-6-pyridin-4-yl-1H-indole-3-carboxamide
Show/Hide
|
C22H19N3O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0083275
|
N-[(3-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
Show/Hide
|
C19H17N5O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0130674
|
N-[(3-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-indole-2-carboxamide
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0474120
|
6-(1H-pyrazol-4-yl)-2-[(3S,4R)-4-[4-(trifluoromethyl)phenyl]pyrrolidin-3-yl]-3H-quinazolin-4-one
Show/Hide
|
C22H18F3N5O
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0474121
|
2-[(3S,4R)-4-(4-fluorophenyl)pyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C21H18FN5O
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0579459
|
(2R)-4-(3-fluoropyridin-4-yl)-2-methyl-N-[(1R)-1-pyrazolo[1,5-a]pyridin-4-ylethyl]piperazine-1-carboxamide
Show/Hide
|
C20H23FN6O
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0144110
|
N,N-dimethyl-2-[(3S,4R)-4-phenylpyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)quinazolin-4-amine
Show/Hide
|
C23H24N6
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0221985
|
6-(1H-pyrazol-4-yl)-N-(2-thiophen-2-ylethyl)-1H-indole-3-carboxamide
Show/Hide
|
C18H16N4OS
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0544232
|
(2R)-4-(3-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methylpiperazine-1-carboxamide
Show/Hide
|
C20H25FN4O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0546163
|
(2R)-N-[(1R)-1-(4-fluoro-3-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
Show/Hide
|
C20H24F2N4O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0571313
|
(2R)-N-[(1R)-1-(2-chloro-5-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
Show/Hide
|
C20H24ClFN4O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0574451
|
(2R)-N-[(1R)-1-(3-fluoro-5-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
Show/Hide
|
C20H24F2N4O2
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0186050
|
2-[(1S)-1-amino-2-(4-methoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C20H19N5O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0418029
|
2-[(3S,4R)-1,1-dimethyl-4-phenylpyrrolidin-1-ium-3-yl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C23H24N5O+
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0543995
|
2-[(1R)-1-amino-2-(4-chlorophenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H16ClN5O
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0542771
|
4-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]benzamide
Show/Hide
|
C21H19FN2O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0546999
|
N-[(1R)-1-(3-methoxyphenyl)ethyl]-6-pyridin-4-ylpyridine-3-carboxamide
Show/Hide
|
C20H19N3O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0071398
|
N-[(3-methoxyphenyl)methyl]-6-(5-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
Show/Hide
|
C20H19N5O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0094144
|
N-[(2-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
Show/Hide
|
C19H17N5O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0066776
|
2-[(3S,4R)-4-(4-methoxyphenyl)-1-methylpyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C23H23N5O2
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0576775
|
(2R)-4-(3-fluoropyridin-4-yl)-N-[(1R)-1-imidazo[1,2-a]pyridin-5-ylethyl]-2-methylpiperazine-1-carboxamide
Show/Hide
|
C20H23FN6O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0114828
|
2-[(1S)-1-amino-2-(4-chlorophenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H16ClN5O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0558438
|
6-(2-aminopyrimidin-4-yl)-2-[(3S,4R)-4-phenylpyrrolidin-3-yl]-3H-quinazolin-4-one
Show/Hide
|
C22H20N6O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0574113
|
3-amino-N-[(4-chlorophenyl)-[4-oxo-6-(1H-pyrazol-4-yl)-3H-quinazolin-2-yl]methyl]propanamide
Show/Hide
|
C21H19ClN6O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0579036
|
(2R)-4-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methylpiperazine-1-carboxamide
Show/Hide
|
C20H25FN4O2
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0282637
|
N-[(3-methoxyphenyl)methyl]-6-pyridin-4-yl-1H-pyrrolo[2,3-b]pyridine-3-carboxamide
Show/Hide
|
C21H18N4O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0131319
|
2-[(1R)-1-amino-2-(3-fluorophenyl)ethyl]-8-methoxy-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C20H18FN5O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0513229
|
2-[(1R)-1-amino-2-(3,4-difluorophenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H15F2N5O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0543996
|
6-(5-methyl-1H-pyrazol-4-yl)-2-[(3S,4R)-4-phenylpyrrolidin-3-yl]-3H-quinazolin-4-one
Show/Hide
|
C22H21N5O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0569283
|
(2R)-N-[(1R)-1-(2-fluoro-5-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
Show/Hide
|
C20H24F2N4O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0574450
|
4-(3-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]piperazine-1-carboxamide
Show/Hide
|
C19H23FN4O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0238447
|
N-[(3,4-difluorophenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
|
C19H14F2N4O
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0076870
|
2-[amino-(3-chlorophenyl)methyl]-8-methoxy-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H16ClN5O2
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0131316
|
2-[(1R)-1-amino-2-(4-fluorophenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H16FN5O
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0513231
|
2-[(1S)-1-amino-2-(3-fluorophenyl)ethyl]-8-methoxy-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C20H18FN5O2
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0094069
|
N-[(2-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
|
C20H18N4O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0127883
|
2-[(1S)-1-amino-2-(4-fluorophenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H16FN5O
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0572645
|
2-[amino-(4-chlorophenyl)methyl]-8-methoxy-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H16ClN5O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0572222
|
(2R,4S)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylpiperidine-1-carboxamide
Show/Hide
|
C21H27N3O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0483756
|
2-[amino-(4-chlorophenyl)methyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C18H14ClN5O
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0483757
|
2-[(1R)-1-amino-2-(3-fluorophenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H16FN5O
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0071893
|
N-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-[3-(methanesulfonamido)phenyl]acetamide
Show/Hide
|
C18H16FN3O3S2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0418032
|
2-[(1S)-1-amino-2-phenylethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H17N5O
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0128778
|
2-[amino-(3-chlorophenyl)methyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C18H14ClN5O
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0499274
|
2-[(1R)-1-amino-2-(3-chlorophenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H16ClN5O
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0474119
|
2-[(1R)-2-(4-chlorophenyl)-1-(ethylamino)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C21H20ClN5O
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0119276
|
N-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-(3-methoxyphenyl)acetamide
Show/Hide
|
C18H15FN2O2S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0507843
|
2-[(1R)-1-amino-2-[3-(trifluoromethyl)phenyl]ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C20H16F3N5O
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0154919
|
N-[(3-methoxyphenyl)methyl]-5-(1H-pyrazol-5-yl)-1,3-benzothiazole-2-carboxamide
Show/Hide
|
C19H16N4O2S
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0076871
|
4-(aminomethyl)-N-[(4-chlorophenyl)-[4-oxo-6-(1H-pyrazol-4-yl)-3H-quinazolin-2-yl]methyl]benzamide
Show/Hide
|
C26H21ClN6O2
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0558437
|
2-[(1S)-1-amino-2-(4-ethoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C21H21N5O2
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0574112
|
3-(aminomethyl)-N-[(4-chlorophenyl)-[4-oxo-6-(1H-pyrazol-4-yl)-3H-quinazolin-2-yl]methyl]benzamide
Show/Hide
|
C26H21ClN6O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0543997
|
2-[(3S,4R)-4-phenylpyrrolidin-3-yl]-6-pyridin-4-yl-3H-quinazolin-4-one
Show/Hide
|
C23H20N4O
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0547001
|
(2R)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyrimidin-4-ylpiperazine-1-carboxamide
Show/Hide
|
C19H25N5O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0572223
|
(2R)-N-[(1R)-1-(2-fluoro-3-methoxyphenyl)ethyl]-4-(3-fluoropyridin-4-yl)-2-methylpiperazine-1-carboxamide
Show/Hide
|
C20H24F2N4O2
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0576408
|
6-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]pyridine-3-carboxamide
Show/Hide
|
C20H18FN3O2
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0574108
|
2-[[2-[(1S)-1-amino-2-(3-fluorophenyl)ethyl]-6-(1H-pyrazol-4-yl)quinazolin-4-yl]-methylamino]ethanol
Show/Hide
|
C22H23FN6O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0574110
|
2-[[2-[(1R)-1-amino-2-(3-fluorophenyl)ethyl]-6-(1H-pyrazol-4-yl)quinazolin-4-yl]-methylamino]ethanol
Show/Hide
|
C22H23FN6O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0551241
|
(2R,4R)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylpiperidine-1-carboxamide
Show/Hide
|
C21H27N3O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0071386
|
6-(2-aminopyrimidin-4-yl)-N-[(3-methoxyphenyl)methyl]-1H-indole-2-carboxamide
Show/Hide
|
C21H19N5O2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0558436
|
2-[(1S)-1-amino-2-(3,4-dimethoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C21H21N5O3
|
1
|
| 1 |
IC50 = 39 nM
|
|
|
|
CP0128779
|
2-[amino-(4-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C19H17N5O2
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0542773
|
4-(3-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]piperidine-1-carboxamide
Show/Hide
|
C20H24FN3O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0551242
|
(1S,2R,4S)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylcyclohexane-1-carboxamide
Show/Hide
|
C22H28N2O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0574088
|
2-[(3S,4R)-1-benzyl-4-(2-fluorophenyl)pyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
|
C28H24FN5O
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0569252
|
5-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]pyridine-2-carboxamide
Show/Hide
|
C20H18FN3O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0541711
|
2-[(1S)-1-amino-2-phenylethyl]-6-pyridin-4-yl-3H-quinazolin-4-one
Show/Hide
|
C21H18N4O
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0543994
|
2-[(1S)-1-amino-2-(3-fluorophenyl)ethyl]-N,N-dimethyl-6-(1H-pyrazol-4-yl)quinazolin-4-amine
Show/Hide
|
C21H21FN6
|
1
|
| 1 |
IC50 = 67 nM
|
|
|
|
CP0543993
|
4-(azetidin-1-yl)-2-[(3S,4R)-4-(4-fluorophenyl)pyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)quinazoline
Show/Hide
|
C24H23FN6
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0542772
|
N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-ylpiperidine-1-carboxamide
Show/Hide
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C20H25N3O2
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1
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| 1 |
IC50 = 74 nM
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CP0354408
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N-(cyclohexylmethyl)-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
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C19H22N4O
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1
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| 1 |
IC50 = 76 nM
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CP0505450
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2-[(3S,4R)-1-benzyl-4-(4-methoxyphenyl)pyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
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C29H27N5O2
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1
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| 1 |
IC50 = 88 nM
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CP0565942
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2-[amino-(4-methoxyphenyl)methyl]-6-(5-methyl-1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
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C20H19N5O2
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1
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| 1 |
IC50 = 98 nM
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CP0547000
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CHEMBL5184099
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C21H26N2O2
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1
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| 1 |
IC50 = 98 nM
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CP0282639
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N-[(1S)-1-(3-methoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
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C21H20N4O2
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1
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| 1 |
IC50 = 130 nM
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CP0016240
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(R)-TRANS-4-(1-AMINOETHYL)-N-(4-PYRIDYL) CYCLOHEXANECARBOXAMIDE
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C14H21N3O
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1
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| 1 |
IC50 = 143 nM
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CP0443227
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3-[[2-[(1R)-1-amino-2-(3-fluorophenyl)ethyl]-6-(1H-pyrazol-4-yl)quinazolin-4-yl]-methylamino]propan-1-ol
Show/Hide
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C23H25FN6O
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1
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| 1 |
IC50 = 159 nM
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CP0203790
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N-[(3-methoxyphenyl)methyl]-6-pyridin-4-yl-1H-indole-2-carboxamide
Show/Hide
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C22H19N3O2
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1
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| 1 |
IC50 = 160 nM
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CP0253342
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N-[2-(3-methoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
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C21H20N4O2
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1
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| 1 |
IC50 = 170 nM
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CP0282640
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N-[(4-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
Show/Hide
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C19H17N5O2
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1
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| 1 |
IC50 = 180 nM
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CP0094079
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N-[(3-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-pyrrolo[3,2-c]pyridine-2-carboxamide
Show/Hide
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C19H17N5O2
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1
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| 1 |
IC50 = 190 nM
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CP0231361
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5-(1,4-diazepane-1-sulfonyl)-1,2-dihydroisoquinolin-1-one
Show/Hide
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C14H17N3O3S
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1
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| 1 |
IC50 = 194 nM
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CP0221987
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6-(1H-pyrazol-4-yl)-N-[[3-(trifluoromethoxy)phenyl]methyl]-1H-indole-3-carboxamide
Show/Hide
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C20H15F3N4O2
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1
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| 1 |
IC50 = 220 nM
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CP0221989
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N-[(3-methoxyphenyl)methyl]-6-pyridin-4-yl-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
Show/Hide
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C21H18N4O2
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1
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| 1 |
IC50 = 220 nM
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CP0418030
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2-[(3S,4R)-1-benzyl-4-(3-fluorophenyl)pyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)-3H-quinazolin-4-one
Show/Hide
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C28H24FN5O
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1
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| 1 |
IC50 = 225 nM
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|
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CP0565964
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N-[(1R)-2-(4-chlorophenyl)-1-[4-oxo-6-(1H-pyrazol-4-yl)-3H-quinazolin-2-yl]ethyl]-2-pyridin-3-ylacetamide
Show/Hide
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C26H21ClN6O2
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1
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| 1 |
IC50 = 239 nM
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CP0571159
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6-(2-fluoropyridin-4-yl)-N-[(1R)-1-(3-methoxyphenyl)ethyl]pyridazine-3-carboxamide
Show/Hide
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C19H17FN4O2
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1
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| 1 |
IC50 = 280 nM
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CP0282641
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N-[(1S)-1-(3-methoxyphenyl)ethyl]-6-(1H-pyrazol-4-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
Show/Hide
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C20H19N5O2
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1
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| 1 |
IC50 = 290 nM
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|
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CP0565963
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N-[2-[(3S,4R)-4-(4-fluorophenyl)pyrrolidin-3-yl]-6-(1H-pyrazol-4-yl)quinazolin-4-yl]-N',N'-dimethylethane-1,2-diamine
Show/Hide
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C25H28FN7
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1
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| 1 |
IC50 = 371 nM
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CP0094078
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N-[(3-methoxyphenyl)methyl]-6-pyridin-4-yl-1H-pyrrolo[3,2-c]pyridine-2-carboxamide
Show/Hide
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C21H18N4O2
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1
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| 1 |
IC50 = 420 nM
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CP0210283
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N-[(3-methoxyphenyl)methyl]-6-(5-methyl-1H-pyrazol-4-yl)-1H-pyrrolo[3,2-c]pyridine-2-carboxamide
Show/Hide
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C20H19N5O2
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1
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| 1 |
IC50 = 530 nM
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CP0569683
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N-[(1R)-1-(3-methoxyphenyl)ethyl]-3-oxo-4-pyridin-4-ylpiperazine-1-carboxamide
Show/Hide
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C19H22N4O3
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1
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| 1 |
IC50 = 534 nM
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CP0513230
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N'-[2-[(1R)-1-amino-2-(3-fluorophenyl)ethyl]-6-(1H-pyrazol-4-yl)quinazolin-4-yl]-N,N,N'-trimethylethane-1,2-diamine
Show/Hide
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C24H28FN7
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1
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| 1 |
IC50 = 627 nM
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CP0094844
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N-[(2,5-dimethoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
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C21H20N4O3
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1
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| 1 |
IC50 = 740 nM
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CP0248168
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N-[(4-methoxyphenyl)methyl]-6-(1H-pyrazol-4-yl)-1H-indole-3-carboxamide
Show/Hide
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C20H18N4O2
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1
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| 1 |
IC50 = 750 nM
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CP0576683
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(1R,2S,4R)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylcyclohexane-1-carboxamide
Show/Hide
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C22H28N2O2
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1
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| 1 |
IC50 = 851 nM
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CP0210282
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6-(2-aminopyridin-4-yl)-N-[(3-methoxyphenyl)methyl]-1H-indole-2-carboxamide
Show/Hide
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C22H20N4O2
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1
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| 1 |
IC50 = 1200 nM
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CP0574619
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(2S,4R)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylpiperidine-1-carboxamide
Show/Hide
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C21H27N3O2
|
1
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| 1 |
IC50 = 1300 nM
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CP0576682
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(2S,4S)-N-[(1R)-1-(3-methoxyphenyl)ethyl]-2-methyl-4-pyridin-4-ylpiperidine-1-carboxamide
Show/Hide
|
C21H27N3O2
|
1
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| 1 |
IC50 = 1640 nM
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CP0576410
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N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-ylcyclohexane-1-carboxamide
Show/Hide
|
C21H26N2O2
|
1
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| 1 |
IC50 = 4330 nM
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|
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CP0576412
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N-[(1R)-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-ylpiperazine-1-carboxamide
Show/Hide
|
C19H24N4O2
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1
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| 1 |
IC50 = 4790 nM
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CP0382649
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3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-methylamino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
Show/Hide
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C50H56BF2N7O7
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1
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| 1 |
Kd = 16 nM
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CP0382724
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3-(2,2-difluoro-10,12-dimethyl-1-aza-3-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-3,5,7,9,11-pentaen-4-yl)-N-[2-[2-[2-[2-[[(2S,3R,4R,6R)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]amino]ethoxy]ethoxy]ethoxy]ethyl]propanamide
Show/Hide
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C49H54BF2N7O7
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1
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| 1 |
Kd = 23 nM
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