| Compound ID |
Compound Name |
Compound Formula |
|
CP0208256
|
N-[5-[(2-acetamido-[1,3]thiazolo[5,4-b]pyridin-5-yl)-methylamino]-2-fluorophenyl]-2-chloro-3-(2-cyanopropan-2-yloxy)benzamide
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|
C26H22ClFN6O3S
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0744518
|
N-{7-Cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]-carbamoyl}amino)phenoxy]-1,3-benzothiazol-2-yl}-cyclopropanecarboxamide
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|
C26H17F4N5O3S
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0699586
|
Methyl 6-[3-({[3-(1-Cyano-1-methylethyl)phenyl]carbonyl}-amino)phenoxy]-2-[(cyclopropylcarbonyl)amino]-1,3-benzothiazole-7-carboxylate
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|
C30H26N4O5S
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0829202
|
3-(1-Cyano-1-methylethyl)-N-[3-({2-[(cyclopropylcarbonyl)-amino]-7-nitro-1,3-benzothiazol-6-yl}oxy)phenyl]benzamide
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|
C28H23N5O5S
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0238393
|
N-[5-[(2-acetamido-[1,3]thiazolo[5,4-b]pyridin-5-yl)-methylamino]-2-fluorophenyl]-3-(2-cyanopropan-2-yloxy)benzamide
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|
C26H23FN6O3S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0807256
|
N-[3-({7-Cyano-2-[(cyclopropylcarbonyl)amino]-1,3-benzothiazol-6-yl}oxy)phenyl]-3-(1-cyano-1-methylethyl)benzamide
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|
C29H23N5O3S
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0057236
|
2-chloro-3-(2-cyanopropan-2-yloxy)-N-[5-[[2-(cyclopropanecarbonylamino)-[1,3]thiazolo[5,4-b]pyridin-5-yl]-methylamino]-2-fluorophenyl]benzamide
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|
C28H24ClFN6O3S
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0029366
|
US8497274, 32
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|
C27H18F4N4O3S
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0672244
|
N-{7-Cyano-6-[3-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)-phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide
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|
C26H18F3N5O3S
|
1
|
| 1 |
IC50 = 75 nM
|
|
|
|
CP0056606
|
US8497274, 53
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|
C26H17F4N5O3S
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0169800
|
2-chloro-3-(2-cyanopropan-2-yloxy)-N-[5-[[2-(cyclopropanecarbonylamino)-[1,3]thiazolo[5,4-b]pyridin-5-yl]amino]-2-fluorophenyl]benzamide
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|
C27H22ClFN6O3S
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0057239
|
N-[3-[(2-acetamido-[1,3]thiazolo[5,4-d]pyrimidin-5-yl)amino]-4-methylphenyl]-3-(2-cyanopropan-2-yloxy)benzamide
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|
C25H23N7O3S
|
1
|
| 1 |
IC50 = 88 nM
|
|
|
|
CP0707799
|
N-{7-Cyano-6-[3-({[4-(trifluoromethyl)phenyl]carbamoyl}amino)-phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide
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|
C26H18F3N5O3S
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0145560
|
N-[3-[(2-acetamido-[1,3]thiazolo[5,4-d]pyrimidin-5-yl)amino]-4-methylphenyl]-2-chloro-3-(1-cyanocyclopropyl)benzamide
Show/Hide
|
C25H20ClN7O2S
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0286275
|
N-[3-[(2-acetamido-[1,3]thiazolo[5,4-d]pyrimidin-5-yl)amino]-4-methylphenyl]-3-(2-cyano-2-methylpropyl)benzamide
Show/Hide
|
C26H25N7O2S
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0699584
|
3-(1-Cyano-1-methylethyl)-N-[3-({2-[(cyclopropylcarbonyl)-amino]-7-(hydroxymethyl)-1,3-benzothiazol-6-yl}oxy)phenyl]-benzamide
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|
C29H26N4O4S
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0672243
|
N-{7-Cyano-6-[3-({[4-(trifluoromethyl)phenyl]acetyl}amino)-phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide
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|
C27H19F3N4O3S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
|
CP0829201
|
N-{7-Cyano-6-[3-({[3-(trifluoromethyl)phenyl]acetyl}amino)-phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide
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|
C27H19F3N4O3S
|
1
|
| 1 |
IC50 = 360 nM
|
|
|
|
CP0279558
|
N-[3-[(2-acetamido-[1,3]thiazolo[5,4-d]pyrimidin-5-yl)amino]-4-methylphenyl]-3-(2-cyanoethyl)benzamide
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|
C24H21N7O2S
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0672245
|
N-{7-Cyano-6-[3-({[2-(trifluoromethyl)phenyl]carbamoyl}amino)-phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide
Show/Hide
|
C26H18F3N5O3S
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
|
CP0699581
|
N-{7-Cyano-6-[3-({[2-(trifluoromethyl)phenyl]acetyl}amino)-phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide
Show/Hide
|
C27H19F3N4O3S
|
1
|
| 1 |
IC50 > 500 nM
|
|
|
