Compound ID |
Compound Name |
Compound Formula |
CP0943716
|
3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-(3-(trifluoromethyl)phenyl)benzamide
Show/Hide
|
C20H15F3N6O
|
1
|
1 |
EC50 = 0.05 nM
|
|
|
CP0525627
|
2-[5-[[[5-butyl-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carbonyl]amino]methyl]imidazol-1-yl]acetic acid
Show/Hide
|
C23H25N7O3S
|
1
|
1 |
EC50 = 0.2 nM
|
|
|
CP0887620
|
N-(3-chlorophenyl)-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C19H15ClN6O
|
1
|
1 |
EC50 = 0.21 nM
|
|
|
CP0965988
|
4-methyl-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-(3-(trifluoromethoxy)phenyl)benzamide
Show/Hide
|
C21H17F3N6O2
|
1
|
1 |
EC50 = 0.21 nM
|
|
|
CP0887621
|
3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-m-tolylbenzamide
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|
C20H18N6O
|
1
|
1 |
EC50 = 0.37 nM
|
|
|
CP0903216
|
N-(3-chlorophenyl)-4-methyl-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C20H17ClN6O
|
1
|
1 |
EC50 = 0.37 nM
|
|
|
CP0903297
|
N-(3-fluoro-5-(trifluoromethyl)phenyl)-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C20H14F4N6O
|
1
|
1 |
EC50 < 0.38 nM
|
|
|
CP0943718
|
3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-(3-nitrophenyl)benzamide
Show/Hide
|
C19H15N7O3
|
1
|
1 |
EC50 < 0.38 nM
|
|
|
CP0958685
|
N-(3-(difluoromethoxy)phenyl)-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C20H16F2N6O2
|
1
|
1 |
EC50 < 0.38 nM
|
|
|
CP0969091
|
N-(3-bromo-5-methylphenyl)-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C20H17BrN6O
|
1
|
1 |
EC50 < 0.38 nM
|
|
|
CP0969090
|
4-methyl-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-(3-(trifluoromethyl)phenyl)benzamide
Show/Hide
|
C21H17F3N6O
|
1
|
1 |
EC50 = 0.4 nM
|
|
|
CP0943717
|
N-(2-fluoro-3-(trifluoromethyl)phenyl)-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C20H14F4N6O
|
1
|
1 |
EC50 = 0.45 nM
|
|
|
CP0965900
|
3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-(3-(trifluoromethoxy)phenyl)benzamide
Show/Hide
|
C20H15F3N6O2
|
1
|
1 |
EC50 = 0.47 nM
|
|
|
CP0965901
|
3-(4-(1,4-dimethyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-(3-(trifluoromethyl)phenyl)benzamide
Show/Hide
|
C21H17F3N6O
|
1
|
1 |
EC50 = 0.63 nM
|
|
|
CP0887622
|
3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-(3-(1,1,2,2-tetrafluoroethoxy)phenyl)benzamide
Show/Hide
|
C21H16F4N6O2
|
1
|
1 |
EC50 = 0.64 nM
|
|
|
CP0956051
|
3-(4-(1,4-dimethyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)-N-(3-(trifluoromethoxy)phenyl)benzamide
Show/Hide
|
C21H17F3N6O2
|
1
|
1 |
EC50 = 0.64 nM
|
|
|
CP0965989
|
methyl 3-(3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamido)benzoate
Show/Hide
|
C21H18N6O3
|
1
|
1 |
EC50 = 0.73 nM
|
|
|
CP0903299
|
N-(3-cyanophenyl)-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C20H15N7O
|
1
|
1 |
EC50 = 0.74 nM
|
|
|
CP0903301
|
N-(3-(dimethylamino)phenyl)-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C21H21N7O
|
1
|
1 |
EC50 = 0.85 nM
|
|
|
CP0962197
|
N-(3-methoxyphenyl)-3-(4-(1-methyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C20H18N6O2
|
1
|
1 |
EC50 = 0.86 nM
|
|
|
CP0965902
|
N-(3-chlorophenyl)-3-(4-(1,4-dimethyl-1H-imidazol-5-yl)-1H-1,2,3-triazol-1-yl)benzamide
Show/Hide
|
C20H17ClN6O
|
1
|
1 |
EC50 = 0.95 nM
|
|
|
CP0489368
|
5-butyl-N-[(3,5-dimethylimidazol-4-yl)methyl]-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C23H27N7OS
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0489369
|
5-butyl-N-[(3-methylimidazol-4-yl)methyl]-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C22H25N7OS
|
1
|
1 |
EC50 = 1 nM
|
|
|
CP0554561
|
5-(ethoxymethyl)-N-[(3-methylimidazol-4-yl)methyl]-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C21H23N7O2S
|
1
|
1 |
EC50 = 1.3 nM
|
|
|
CP0404590
|
1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-5-propyl-N-(2-pyridin-4-ylpropan-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C24H26N6OS
|
1
|
1 |
EC50 = 5 nM
|
|
|
CP0525625
|
5-butyl-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-N-(pyridin-4-ylmethyl)pyrazole-4-carboxamide
Show/Hide
|
C23H24N6OS
|
1
|
1 |
EC50 = 7 nM
|
|
|
CP0859662
|
N-((1R,3S)-3-(5-(1,4-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C22H25F3N6O
|
2
|
1 |
EC50 = 11 nM
|
|
|
2 |
EC50 < 120 nM
|
|
|
CP0449774
|
5-(ethoxymethyl)-N-[(3-methylimidazol-4-yl)methyl]-1-(5-methyl-4-pyrrolidin-1-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C21H28N8O2
|
1
|
1 |
EC50 = 14 nM
|
|
|
CP0701745
|
3-chloro-N-((1R,3S)-3-(5-(1,4-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methylbenzamide
Show/Hide
|
C21H25ClN6O
|
2
|
1 |
EC50 = 14 nM
|
|
|
2 |
EC50 = 14.4 nM
|
|
|
CP0943180
|
N-((2S,4R)-2-(5-(1-(cyclopropylmethyl)-4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)tetrahydro-2H-pyran-4-yl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C24H27F3N6O2
|
1
|
1 |
EC50 = 14 nM
|
|
|
CP0914179
|
N-((2S,4R)-2-(5-(1-cyclobutyl-4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)tetrahydro-2H-pyran-4-yl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C24H27F3N6O2
|
1
|
1 |
EC50 = 16 nM
|
|
|
CP0339388
|
5-(ethoxymethyl)-N-[(3-methylimidazol-4-yl)methyl]-1-(5-methyl-4-piperidin-1-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C22H30N8O2
|
1
|
1 |
EC50 = 22 nM
|
|
|
CP0525624
|
1-[4-(cyclobutylamino)-5-methylpyrimidin-2-yl]-5-(ethoxymethyl)-N-[(3-methylimidazol-4-yl)methyl]pyrazole-4-carboxamide
Show/Hide
|
C21H28N8O2
|
1
|
1 |
EC50 = 25 nM
|
|
|
CP0374931
|
(2S)-3-(4-fluorophenyl)-N-[2-methyl-5-[2-(methylamino)pyridin-4-yl]pyrazol-3-yl]-2-(2H-triazol-4-ylmethylamino)propanamide
Show/Hide
|
C22H24FN9O
|
1
|
1 |
EC50 = 26 nM
|
|
|
CP0939972
|
3-chloro-N-((2S,4R)-2-(5-(1,4-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)tetrahydro-2H-pyran-4-yl)-N-methylbenzamide
Show/Hide
|
C20H23ClN6O2
|
1
|
1 |
EC50 = 27 nM
|
|
|
CP0489367
|
1-[4-(azetidin-1-yl)-5-methylpyrimidin-2-yl]-5-(ethoxymethyl)-N-[(3-methylimidazol-4-yl)methyl]pyrazole-4-carboxamide
Show/Hide
|
C20H26N8O2
|
1
|
1 |
EC50 = 28 nM
|
|
|
CP0387774
|
5-(ethoxymethyl)-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-N-(pyridin-4-ylmethyl)pyrazole-4-carboxamide
Show/Hide
|
C22H22N6O2S
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0487839
|
5-butyl-N-[(2,3-dimethylimidazol-4-yl)methyl]-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C23H27N7OS
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0121654
|
N-[(1R,3S)-3-[(3,5-dimethylimidazol-4-yl)carbamoyl]cyclohexyl]-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C21H25F3N4O2
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0961053
|
N-((2S,4R)-2-(5-(1,4-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)tetrahydro-2H-pyran-4-yl)-N-methyl-3-(trifluoromethoxy)benzamide
Show/Hide
|
C21H23F3N6O3
|
1
|
1 |
EC50 = 30 nM
|
|
|
CP0859663
|
N-((1R,3S)-3-(5-(6,8-dihydro-5H-imidazo[2,1-c][1,4]oxazin-3-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C23H25F3N6O2
|
2
|
1 |
EC50 = 32 nM
|
|
|
2 |
EC50 < 120 nM
|
|
|
CP0939973
|
3-chloro-N-((2S,4R)-2-(5-(imidazo[1,2-a]pyridin-3-yl)-4H-1,2,4-triazol-3-yl)tetrahydro-2H-pyran-4-yl)-N-methylbenzamide
Show/Hide
|
C22H21ClN6O2
|
1
|
1 |
EC50 = 35 nM
|
|
|
CP0480716
|
(2S)-N-[5-[2-(methylamino)pyridin-4-yl]-1,3,4-thiadiazol-2-yl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C21H21N7OS2
|
1
|
1 |
EC50 = 36 nM
|
|
|
CP0249490
|
(2S)-N-[2-methyl-5-[2-(methylamino)pyridin-4-yl]pyrazol-3-yl]-3-phenyl-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C23H25N7OS
|
1
|
1 |
EC50 = 37 nM
|
|
|
CP0369079
|
(2S)-N-(2-methyl-5-pyridin-4-ylpyrazol-3-yl)-3-phenyl-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C22H22N6OS
|
1
|
1 |
EC50 = 37 nM
|
|
|
CP0870287
|
N-((1R,3S)-3-(5-(1-(2,2-difluoroethyl)-4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C23H25F5N6O
|
2
|
1 |
EC50 = 41 nM
|
|
|
2 |
EC50 < 120 nM
|
|
|
CP0526730
|
2-[[(2S)-3-(4-fluorophenyl)-1-[[2-methyl-5-[2-(methylamino)pyridin-4-yl]pyrazol-3-yl]amino]-1-oxopropan-2-yl]amino]acetic acid
Show/Hide
|
C21H23FN6O3
|
1
|
1 |
EC50 = 42 nM
|
|
|
CP0678057
|
N-((2S,4R)-2-(5-(1,4-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)tetrahydro-2H-pyran-4-yl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C21H23F3N6O2
|
1
|
1 |
EC50 = 43 nM
|
|
|
CP0924820
|
N-((1R,3S)-3-(5-(1,2-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C22H25F3N6O
|
2
|
1 |
EC50 = 46 nM
|
|
|
2 |
EC50 < 120 nM
|
|
|
CP0369078
|
(2S)-3-(4-fluorophenyl)-N-[2-methyl-5-[2-(methylamino)pyridin-4-yl]pyrazol-3-yl]-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C23H24FN7OS
|
1
|
1 |
EC50 = 49 nM
|
|
|
CP0569457
|
N-methyl-N-[(1R,3S)-3-[[5-methyl-3-(2-morpholin-4-ylethyl)imidazol-4-yl]carbamoyl]cyclohexyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C26H34F3N5O3
|
1
|
1 |
EC50 = 51 nM
|
|
|
CP0047893
|
(2S)-N-[3-(2-methylpyridin-4-yl)phenyl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C25H24N4OS
|
1
|
1 |
EC50 = 52 nM
|
|
|
CP0042063
|
2-[[(2S)-1-[(2-methyl-5-pyridin-4-ylpyrazol-3-yl)amino]-1-oxo-3-phenylpropan-2-yl]amino]acetic acid
Show/Hide
|
C20H21N5O3
|
1
|
1 |
EC50 = 52 nM
|
|
|
CP0402163
|
N-[(1R,3S)-3-[[3-(cyclopropylmethyl)-5-methylimidazol-4-yl]carbamoyl]cyclohexyl]-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C24H29F3N4O2
|
1
|
1 |
EC50 = 52 nM
|
|
|
CP0526853
|
(2S)-N-(3-methoxy-5-pyridin-4-ylphenyl)-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C25H24N4O2S
|
2
|
1 |
EC50 = 53 nM
|
|
|
2 |
EC50 = 810 nM
|
|
|
CP0939971
|
N-((2S,4R)-2-(5-(6,7-dihydro-5H-pyrrolo[1,2-a]imidazol-3-yl)-4H-1,2,4-triazol-3-yl)tetrahydro-2H-pyran-4-yl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C22H23F3N6O2
|
1
|
1 |
EC50 = 53 nM
|
|
|
CP0513075
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-[(1-pyridin-2-ylcyclopropyl)amino]propanamide
Show/Hide
|
C27H25N5O2
|
1
|
1 |
EC50 = 54 nM
|
|
|
CP0402164
|
N-[(1R,3S)-3-[[3-(2,2-difluoroethyl)-5-methylimidazol-4-yl]carbamoyl]cyclohexyl]-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C22H25F5N4O2
|
1
|
1 |
EC50 = 63 nM
|
|
|
CP0247821
|
(2S)-N-[5-(2-methylpyridin-4-yl)-2-oxo-1H-pyridin-3-yl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C24H23N5O2S
|
2
|
1 |
EC50 = 67 nM
|
|
|
2 |
EC50 = 290 nM
|
|
|
CP0301279
|
(2S)-3-phenyl-N-(3-pyridin-4-ylphenyl)-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C24H22N4OS
|
2
|
1 |
EC50 = 67 nM
|
|
|
2 |
EC50 = 970 nM
|
|
|
CP0341788
|
(2S)-3-phenyl-N-[3-(1H-pyrazol-5-yl)phenyl]-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C22H21N5OS
|
1
|
1 |
EC50 = 67 nM
|
|
|
CP0395512
|
(2S)-3-(4-fluorophenyl)-N-[2-methyl-5-[2-(methylamino)pyridin-4-yl]pyrazol-3-yl]-2-(2H-tetrazol-5-ylmethylamino)propanamide
Show/Hide
|
C21H23FN10O
|
1
|
1 |
EC50 = 71 nM
|
|
|
CP0402166
|
N-[(1R,3S)-3-[(3,5-dimethylimidazol-4-yl)carbamoyl]cyclohexyl]-N-methyl-3-(trifluoromethoxy)benzamide
Show/Hide
|
C21H25F3N4O3
|
1
|
1 |
EC50 = 71 nM
|
|
|
CP0869212
|
N-methyl-N-((1R,3S)-3-(5-(4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-3-(trifluoromethyl)benzamide
Show/Hide
|
C21H23F3N6O
|
2
|
1 |
EC50 = 76 nM
|
|
|
2 |
EC50 < 120 nM
|
|
|
CP0406758
|
(2S)-2-[(2-amino-2-oxoethyl)amino]-3-(4-fluorophenyl)-N-[2-methyl-5-[2-(methylamino)pyridin-4-yl]pyrazol-3-yl]propanamide
Show/Hide
|
C21H24FN7O2
|
1
|
1 |
EC50 = 78 nM
|
|
|
CP0564644
|
N-methyl-N-[(1R,3S)-3-[[5-methyl-3-(2,2,2-trifluoroethyl)imidazol-4-yl]carbamoyl]cyclohexyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C22H24F6N4O2
|
1
|
1 |
EC50 = 81 nM
|
|
|
CP0452217
|
(2S)-3-phenyl-N-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C20H18N6OS2
|
1
|
1 |
EC50 = 86 nM
|
|
|
CP0481725
|
(2S)-N-(2-methoxy-5-pyridin-4-ylphenyl)-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C25H24N4O2S
|
2
|
1 |
EC50 = 89 nM
|
|
|
2 |
EC50 = 1000 nM
|
|
|
CP0470413
|
5-butyl-N-[(2-methylpyrazol-3-yl)methyl]-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C22H25N7OS
|
1
|
1 |
EC50 = 90 nM
|
|
|
CP0374930
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C23H21N5O2S
|
2
|
1 |
EC50 = 90 nM
|
|
|
2 |
EC50 = 502 nM
|
|
|
CP0395510
|
(2S)-3-phenyl-N-(2-pyridin-4-yl-1,3-thiazol-5-yl)-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C21H19N5OS2
|
2
|
1 |
EC50 = 90 nM
|
|
|
2 |
EC50 = 161 nM
|
|
|
CP0360743
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C23H21N5O2S
|
3
|
1 |
EC50 = 93 nM
|
|
|
2 |
EC50 = 500 nM
|
|
|
3 |
EC50 = 930 nM
|
|
|
CP0423881
|
N-[(1R,3S)-3-[[3-(cyanomethyl)-5-methylimidazol-4-yl]carbamoyl]cyclohexyl]-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C22H24F3N5O2
|
1
|
1 |
EC50 = 93 nM
|
|
|
CP0488631
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-(pyridin-2-ylmethylamino)propanamide
Show/Hide
|
C25H23N5O2
|
1
|
1 |
EC50 = 95 nM
|
|
|
CP0403868
|
(2S)-3-phenyl-N-(5-pyridin-4-yl-1H-pyrazol-3-yl)-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C21H20N6OS
|
2
|
1 |
EC50 = 95 nM
|
|
|
2 |
EC50 = 164 nM
|
|
|
CP0526729
|
ethyl 2-[[(2S)-1-[(2-methyl-5-pyridin-4-ylpyrazol-3-yl)amino]-1-oxo-3-phenylpropan-2-yl]amino]acetate
Show/Hide
|
C22H25N5O3
|
1
|
1 |
EC50 = 95 nM
|
|
|
CP0376015
|
5-(ethoxymethyl)-1-(4-ethoxy-5-methylpyrimidin-2-yl)-N-[(3-methylimidazol-4-yl)methyl]pyrazole-4-carboxamide
Show/Hide
|
C19H25N7O3
|
1
|
1 |
EC50 = 96 nM
|
|
|
CP0413885
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-[(1-pyrimidin-2-ylcyclopropyl)amino]propanamide
Show/Hide
|
C26H24N6O2
|
1
|
1 |
EC50 = 99 nM
|
|
|
CP0554560
|
5-butyl-N-(3-methyl-4,5,6,7-tetrahydrobenzimidazol-4-yl)-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C25H29N7OS
|
1
|
1 |
EC50 = 100 nM
|
|
|
CP0965062
|
N-((2S,4R)-2-(5-(6,8-dihydro-5H-imidazo[2,1-c][1,4]oxazin-3-yl)-4H-1,2,4-triazol-3-yl)tetrahydro-2H-pyran-4-yl)-N-methyl-3-(trifluoromethyl)benzamide
Show/Hide
|
C22H23F3N6O3
|
1
|
1 |
EC50 = 102 nM
|
|
|
CP0423883
|
3-chloro-N-[(1R,3S)-3-[[3-(2,2-difluoroethyl)-5-methylimidazol-4-yl]carbamoyl]cyclohexyl]-N-methylbenzamide
Show/Hide
|
C21H25ClF2N4O2
|
1
|
1 |
EC50 = 104 nM
|
|
|
CP0349499
|
3-[[(2S)-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanoyl]amino]-5-pyridin-4-ylbenzoic acid
Show/Hide
|
C25H22N4O3S
|
2
|
1 |
EC50 = 110 nM
|
|
|
2 |
EC50 = 480 nM
|
|
|
CP0486940
|
(2S)-2-(1H-imidazol-5-ylmethylamino)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C23H22N6O2
|
1
|
1 |
EC50 = 110 nM
|
|
|
CP0548909
|
N-methyl-N-[(1R,3S)-3-[[5-methyl-3-(2,2,2-trifluoroethyl)imidazol-4-yl]carbamoyl]cyclohexyl]-3-(trifluoromethoxy)benzamide
Show/Hide
|
C22H24F6N4O3
|
1
|
1 |
EC50 = 110 nM
|
|
|
CP0374933
|
2-[[(2S)-3-phenyl-2-(1,3-thiazol-5-ylmethylamino)propanoyl]amino]-5-pyridin-4-ylthiophene-3-carboxylic acid
Show/Hide
|
C23H20N4O3S2
|
2
|
1 |
EC50 = 121 nM
|
|
|
2 |
EC50 = 1250 nM
|
|
|
CP0525573
|
N-methyl-N-[(1R,3S)-3-[(5-methyl-3-propan-2-ylimidazol-4-yl)carbamoyl]cyclohexyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C23H29F3N4O2
|
1
|
1 |
EC50 = 131 nM
|
|
|
CP0423882
|
N-methyl-N-[(1R,3S)-3-[[5-methyl-3-[(1-methylazetidin-3-yl)methyl]imidazol-4-yl]carbamoyl]cyclohexyl]-3-(trifluoromethyl)benzamide
Show/Hide
|
C25H32F3N5O2
|
1
|
1 |
EC50 = 147 nM
|
|
|
CP0047894
|
(2S)-N-[3-(1-methylpyrazol-4-yl)phenyl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C23H23N5OS
|
1
|
1 |
EC50 = 180 nM
|
|
|
CP0093721
|
(2S)-3-phenyl-N-[3-(1H-pyrazol-4-yl)phenyl]-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C22H21N5OS
|
1
|
1 |
EC50 = 180 nM
|
|
|
CP0413922
|
(2S)-N-[5-(3-methylimidazol-4-yl)-1,3,4-thiadiazol-2-yl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C19H19N7OS2
|
1
|
1 |
EC50 = 180 nM
|
|
|
CP0566813
|
(2S)-3-phenyl-N-[5-pyridin-4-yl-2-(2,2,2-trifluoroethyl)pyrazol-3-yl]-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C23H21F3N6OS
|
1
|
1 |
EC50 = 180 nM
|
|
|
CP0349498
|
(2S)-N-[2-oxo-5-(1H-pyrazol-5-yl)-1H-pyridin-3-yl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C21H20N6O2S
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0476872
|
(2S)-2-[[1-(2-methyl-1,3-thiazol-4-yl)cyclopropyl]amino]-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C26H25N5O2S
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0387773
|
5-butyl-N-[(2,4-dimethyl-1,3-thiazol-5-yl)methyl]-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C23H26N6OS2
|
1
|
1 |
EC50 = 200 nM
|
|
|
CP0331814
|
(2S)-N-[3-(2-aminopyridin-4-yl)phenyl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C24H23N5OS
|
1
|
1 |
EC50 = 210 nM
|
|
|
CP0413886
|
(2S)-2-[(1-methylpyrazol-3-yl)methylamino]-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C24H24N6O2
|
1
|
1 |
EC50 = 210 nM
|
|
|
CP0452215
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-[[(1S)-1-pyridin-2-ylethyl]amino]propanamide
Show/Hide
|
C26H25N5O2
|
1
|
1 |
EC50 = 220 nM
|
|
|
CP0114936
|
(2S)-N-[5-(1-methylpyrazol-4-yl)-2-oxo-1H-pyridin-3-yl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C22H22N6O2S
|
1
|
1 |
EC50 = 230 nM
|
|
|
CP0410728
|
(2S)-N-(4-methoxy-3-pyridin-4-ylphenyl)-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C25H24N4O2S
|
2
|
1 |
EC50 = 240 nM
|
|
|
2 |
EC50 = 980 nM
|
|
|
CP0489735
|
1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-5-propyl-N-(pyridin-4-ylmethyl)pyrazole-4-carboxamide
Show/Hide
|
C22H22N6OS
|
1
|
1 |
EC50 = 250 nM
|
|
|
CP0452218
|
2-[2-oxo-3-[[(2S)-3-phenyl-2-[(1-pyridin-2-ylcyclopropyl)amino]propanoyl]amino]-5-pyridin-4-ylpyridin-1-yl]acetic acid
Show/Hide
|
C29H27N5O4
|
1
|
1 |
EC50 = 260 nM
|
|
|
CP0406428
|
(2S)-3-phenyl-N-(3-pyridin-4-yl-1,2-oxazol-5-yl)-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C21H19N5O2S
|
2
|
1 |
EC50 = 263 nM
|
|
|
2 |
EC50 = 306 nM
|
|
|
CP0413884
|
(2S)-N-[1-[2-(dimethylamino)ethyl]-2-oxo-5-pyridin-4-ylpyridin-3-yl]-3-phenyl-2-[(1-pyridin-2-ylcyclopropyl)amino]propanamide
Show/Hide
|
C31H34N6O2
|
1
|
1 |
EC50 = 280 nM
|
|
|
CP0397601
|
(2S)-3-phenyl-N-(2-pyridin-4-yl-1,3-thiazol-4-yl)-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C21H19N5OS2
|
2
|
1 |
EC50 = 287 nM
|
|
|
2 |
EC50 = 452 nM
|
|
|
CP0507370
|
(2S)-3-phenyl-N-(4-pyridin-4-ylpyrimidin-2-yl)-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C22H20N6OS
|
2
|
1 |
EC50 = 290 nM
|
|
|
2 |
EC50 = 360 nM
|
|
|
CP0480717
|
(2S)-N-(2-methoxy-5-pyridin-4-ylpyridin-3-yl)-3-phenyl-2-[(1-pyridin-2-ylcyclopropyl)amino]propanamide
Show/Hide
|
C28H27N5O2
|
1
|
1 |
EC50 = 350 nM
|
|
|
CP0452208
|
(2S)-2-[[(2R)-oxolan-2-yl]methylamino]-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C24H26N4O3
|
1
|
1 |
EC50 = 390 nM
|
|
|
CP0513072
|
(2S)-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)-N-[5-(1,3-thiazol-5-yl)-1,3,4-thiadiazol-2-yl]propanamide
Show/Hide
|
C18H16N6OS3
|
1
|
1 |
EC50 = 390 nM
|
|
|
CP0513073
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-(pyrimidin-2-ylmethylamino)propanamide
Show/Hide
|
C24H22N6O2
|
1
|
1 |
EC50 = 440 nM
|
|
|
CP0482488
|
2-[5-[[(2S)-3-phenyl-2-(1,3-thiazol-5-ylmethylamino)propanoyl]amino]-3-pyridin-4-ylpyrazol-1-yl]acetic acid
Show/Hide
|
C23H22N6O3S
|
1
|
1 |
EC50 = 516 nM
|
|
|
CP0341789
|
(2S)-3-phenyl-N-(3-phenylphenyl)-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C25H23N3OS
|
1
|
1 |
EC50 = 640 nM
|
|
|
CP0481701
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-(1-pyridin-2-ylpropylamino)propanamide
Show/Hide
|
C27H27N5O2
|
1
|
1 |
EC50 = 730 nM
|
|
|
CP0397599
|
(2S)-3-phenyl-N-(5-pyridin-4-yl-1,3-thiazol-2-yl)-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C21H19N5OS2
|
2
|
1 |
EC50 = 734 nM
|
|
|
2 |
EC50 = 1040 nM
|
|
|
CP0481726
|
(2S)-2-(cyclopropylmethylamino)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C23H24N4O2
|
1
|
1 |
EC50 = 760 nM
|
|
|
CP0377336
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-(2-phenylethylamino)propanamide
Show/Hide
|
C27H26N4O2
|
1
|
1 |
EC50 = 780 nM
|
|
|
CP0497660
|
(2S)-2-(benzylamino)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C26H24N4O2
|
1
|
1 |
EC50 = 830 nM
|
|
|
CP0489734
|
5-ethyl-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-N-(pyridin-4-ylmethyl)pyrazole-4-carboxamide
Show/Hide
|
C21H20N6OS
|
1
|
1 |
EC50 = 1000 nM
|
|
|
CP0525623
|
1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-5-pentyl-N-(pyridin-4-ylmethyl)pyrazole-4-carboxamide
Show/Hide
|
C24H26N6OS
|
1
|
1 |
EC50 = 1000 nM
|
|
|
CP0476873
|
(2S)-2-[2-(oxan-4-yl)ethylamino]-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C26H30N4O3
|
1
|
1 |
EC50 = 1060 nM
|
|
|
CP0414754
|
(2S)-3-phenyl-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C21H19N5OS2
|
2
|
1 |
EC50 = 1081 nM
|
|
|
2 |
EC50 = 1110 nM
|
|
|
CP0500981
|
5-butan-2-yl-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-N-(pyridin-4-ylmethyl)pyrazole-4-carboxamide
Show/Hide
|
C23H24N6OS
|
1
|
1 |
EC50 = 1200 nM
|
|
|
CP0476874
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-(2-pyridin-2-ylethylamino)propanamide
Show/Hide
|
C26H25N5O2
|
1
|
1 |
EC50 = 1320 nM
|
|
|
CP0253142
|
5-(methoxymethyl)-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-N-(pyridin-4-ylmethyl)pyrazole-4-carboxamide
Show/Hide
|
C21H20N6O2S
|
1
|
1 |
EC50 = 1500 nM
|
|
|
CP0114935
|
(2S)-N-[3-(1-methylpyrazol-3-yl)phenyl]-3-phenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C23H23N5OS
|
1
|
1 |
EC50 = 1900 nM
|
|
|
CP0520368
|
(2S)-3-phenyl-N-(5-pyridin-4-yl-1H-1,2,4-triazol-3-yl)-2-(1,3-thiazol-5-ylmethylamino)propanamide
Show/Hide
|
C20H19N7OS
|
1
|
1 |
EC50 = 2170 nM
|
|
|
CP0452209
|
(2S)-2-[(5-methyl-1,2-oxazol-3-yl)methylamino]-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C24H23N5O3
|
1
|
1 |
EC50 = 2200 nM
|
|
|
CP0452219
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-2-[[(2R)-5-oxopyrrolidin-2-yl]methylamino]-3-phenylpropanamide
Show/Hide
|
C24H25N5O3
|
1
|
1 |
EC50 = 2230 nM
|
|
|
CP0542235
|
(2S)-3-phenyl-1-(6-pyridin-4-yl-2,3-dihydroimidazo[1,2-b]pyrazol-1-yl)-2-(1,3-thiazol-5-ylmethylamino)propan-1-one
Show/Hide
|
C23H22N6OS
|
1
|
1 |
EC50 = 2780 nM
|
|
|
CP0407848
|
N-ethyl-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-5-propyl-N-(pyridin-4-ylmethyl)pyrazole-4-carboxamide
Show/Hide
|
C24H26N6OS
|
1
|
1 |
EC50 = 3000 nM
|
|
|
CP0125163
|
(2S)-N,3-diphenyl-2-(1,3-thiazol-4-ylmethylamino)propanamide
Show/Hide
|
C19H19N3OS
|
1
|
1 |
EC50 = 3300 nM
|
|
|
CP0400660
|
(2S)-2-amino-3-(4-chlorophenyl)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)propanamide
Show/Hide
|
C19H17ClN4O2
|
1
|
1 |
EC50 = 3800 nM
|
|
|
CP0526855
|
(2S)-2-amino-3-(4-fluorophenyl)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)propanamide
Show/Hide
|
C19H17FN4O2
|
1
|
1 |
EC50 = 4200 nM
|
|
|
CP0526856
|
(2S)-2-amino-3-(4-cyanophenyl)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)propanamide
Show/Hide
|
C20H17N5O2
|
1
|
1 |
EC50 = 4600 nM
|
|
|
CP0383672
|
(2S)-2-amino-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C19H18N4O2
|
1
|
1 |
EC50 = 4800 nM
|
|
|
CP0486941
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-[[(1R)-1-pyridin-2-ylethyl]amino]propanamide
Show/Hide
|
C26H25N5O2
|
1
|
1 |
EC50 = 6000 nM
|
|
|
CP0536577
|
(2S)-2-amino-3-(4-methylphenyl)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)propanamide
Show/Hide
|
C20H20N4O2
|
1
|
1 |
EC50 = 6600 nM
|
|
|
CP0452214
|
(2S)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenyl-2-(2-pyridin-2-ylpropan-2-ylamino)propanamide
Show/Hide
|
C27H27N5O2
|
1
|
1 |
EC50 = 9450 nM
|
|
|
CP0526854
|
(2R)-2-amino-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C19H18N4O2
|
1
|
1 |
EC50 = 13000 nM
|
|
|
CP0491804
|
N-[(1-methylimidazol-4-yl)methyl]-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-5-propylpyrazole-4-carboxamide
Show/Hide
|
C21H23N7OS
|
1
|
1 |
EC50 = 15000 nM
|
|
|
CP0452216
|
(2S)-2-[(1,1-dioxothian-4-yl)methylamino]-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
Show/Hide
|
C25H28N4O4S
|
1
|
1 |
EC50 = 20000 nM
|
|
|
CP0407844
|
5-butyl-N-(1H-indol-3-ylmethyl)-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)pyrazole-4-carboxamide
Show/Hide
|
C26H26N6OS
|
1
|
1 |
EC50 > 20000 nM
|
|
|
CP0407845
|
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(5-methyl-4-thiophen-2-ylpyrimidin-2-yl)-5-propylpyrazole-4-carboxamide
Show/Hide
|
C21H22N6O2S
|
1
|
1 |
EC50 > 20000 nM
|
|
|
CP0383694
|
(2S)-2-amino-3-(4-methoxyphenyl)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)propanamide
Show/Hide
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C20H20N4O3
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1
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1 |
EC50 = 25000 nM
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CP0400658
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2-amino-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)acetamide
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C12H12N4O2
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1
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1 |
EC50 > 33000 nM
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CP0416289
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(2S)-2-amino-3-(2-chlorophenyl)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)propanamide
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C19H17ClN4O2
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1
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1 |
EC50 > 33000 nM
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CP0416290
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(2S)-2-amino-3-(3-chlorophenyl)-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)propanamide
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C19H17ClN4O2
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1
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1 |
EC50 > 33000 nM
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CP0481724
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(2S)-2-amino-3-cyclohexyl-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)propanamide
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C19H24N4O2
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1
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1 |
EC50 > 33000 nM
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CP0497659
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(2S)-2-amino-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-2-phenylacetamide
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C18H16N4O2
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1
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1 |
EC50 > 33000 nM
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CP0536578
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(2S)-2-acetamido-N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
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C21H20N4O3
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1
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1 |
EC50 > 33000 nM
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CP0544660
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N-(2-oxo-5-pyridin-4-yl-1H-pyridin-3-yl)-3-phenylpropanamide
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C19H17N3O2
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1
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1 |
EC50 > 33000 nM
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CP0374929
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(2S)-3-phenyl-N-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)-2-(1,3-thiazol-5-ylmethylamino)propanamide
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C20H18N6O2S
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1
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1 |
EC50 > 33000 nM
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CP0942968
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Cis-3-chloro-N-((1R,3S)-3-(5-(1,2-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methylbenzamide
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C21H25ClN6O
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1
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1 |
EC50 < 120 nM
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CP0956139
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Cis-3-chloro-N-((1R,3S)-3-(5-(1-(2-methoxyethyl)-4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methylbenzamide
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C23H29ClN6O2
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1
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1 |
EC50 < 120 nM
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CP0958176
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Cis-rac-3-chloro-N-((1S,3R)-3-(5-(1,4-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methylbenzamide
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C21H25ClN6O
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1
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1 |
EC50 < 120 nM
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CP0961952
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Cis-3-chloro-N-methyl-N-((1R,3S)-3-(5-(4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)benzamide
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C20H23ClN6O
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1
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1 |
EC50 < 120 nM
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CP0962744
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Cis-N-methyl-N-((1R,3S)-3-(5-(2-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-3-(trifluoromethyl)benzamide
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C21H23F3N6O
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1
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1 |
EC50 < 120 nM
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CP0965850
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N-methyl-N-((1R,3S)-3-(5-(4-methyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-3-(trifluoromethoxy)benzamide
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C21H23F3N6O2
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1
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1 |
EC50 < 120 nM
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