Brief Information of the Compound and Protein
Compound Name
N-((1R,3S)-3-(5-(1,2-dimethyl-1H-imidazol-5-yl)-4H-1,2,4-triazol-3-yl)cyclohexyl)-N-methyl-3-(trifluoromethyl)benzamide
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PubChem ID
CID: 134194661
Canonical SMILES
Cc1ncc(-c2nnc([C@H]3CCC[C@@H](N(C)C(=O)c4cccc(C(F)(F)F)c4)C3)[nH]2)n1C
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Compound Formula C22H25F3N6O
Compound Structure
Protein Name
Probable G-protein coupled receptor 142
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
Q7Z601
Gene Name
GPR142
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 46 nM
   TI
   LI
   LO
   TS
2
EC50 < 120 nM
   TI
   LI
   LO
   TS