Brief Information of the Compound and Protein
Compound Name
2-[[(2S)-3-phenyl-2-(1,3-thiazol-5-ylmethylamino)propanoyl]amino]-5-pyridin-4-ylthiophene-3-carboxylic acid
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PubChem ID
CID: 72945365
Canonical SMILES
OC(=O)c1cc(sc1NC(=O)[C@H](Cc1ccccc1)NCc1cncs1)-c1ccncc1
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Compound Formula C23H20N4O3S2
Compound Structure
Protein Name
Probable G-protein coupled receptor 142
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
Q7Z601
Gene Name
GPR142
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 121 nM
   TI
   LI
   LO
   TS
2
EC50 = 1250 nM
   TI
   LI
   LO
   TS