Compound ID |
Compound Name |
Compound Formula |
CP0541128
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-pyridin-3-ylmethanesulfonamide
Show/Hide
|
C19H15Br2N5O2S2
|
1
|
1 |
IC50 = 32 nM
|
|
|
CP0102676
|
1-(6-bromoquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C14H12BrNO2S
|
1
|
1 |
IC50 = 33.7 nM
|
|
|
CP0517742
|
1-[2-(4-cyanophenyl)phenyl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C18H15NO2S
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0385475
|
1-[6-(trifluoromethyl)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C15H12F3NO2S
|
1
|
1 |
IC50 = 61.2 nM
|
|
|
CP0547970
|
sodium;2-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate
Show/Hide
|
C15H10Br2N3NaO2S
|
1
|
1 |
IC50 = 94 nM
|
|
|
CP0429844
|
1-[6-[2-(trifluoromethyl)phenyl]quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C21H16F3NO2S
|
1
|
1 |
IC50 = 115.3 nM
|
|
|
CP0375457
|
1-(7-bromoquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C14H12BrNO2S
|
1
|
1 |
IC50 = 129.8 nM
|
|
|
CP0491662
|
US8889724, EG
Show/Hide
|
C18H20N4O
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0463051
|
1-[6-(4-fluorophenyl)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C20H16FNO2S
|
1
|
1 |
IC50 = 158.8 nM
|
|
|
CP0546617
|
sodium;2-[3-(4-cyanonaphthalen-1-yl)pyridin-4-yl]sulfanyl-2-methylpropanoate
Show/Hide
|
C20H15N2NaO2S
|
1
|
1 |
IC50 = 170 nM
|
|
|
CP0463105
|
1-[6-(methoxymethyl)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C16H17NO3S
|
1
|
1 |
IC50 = 197.8 nM
|
|
|
CP0541063
|
1-[6-(2-methoxyethoxy)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C17H19NO4S
|
1
|
1 |
IC50 = 206.9 nM
|
|
|
CP0556249
|
US8889724, EC
Show/Hide
|
C17H18N4O
|
1
|
1 |
IC50 = 240 nM
|
|
|
CP0546619
|
sodium;2-[[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylmethyl]benzoate
Show/Hide
|
C24H16N3NaO2S
|
1
|
1 |
IC50 = 240 nM
|
|
|
CP0491664
|
US8889724, ED
Show/Hide
|
C18H20N4O2
|
1
|
1 |
IC50 = 250 nM
|
|
|
CP0575161
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(2-bromopyridin-3-yl)methanesulfonamide
Show/Hide
|
C19H14Br3N5O2S2
|
1
|
1 |
IC50 = 280 nM
|
|
|
CP0538447
|
1-(6-bromoquinolin-4-yl)sulfanylcyclopentane-1-carboxylic acid
Show/Hide
|
C15H14BrNO2S
|
1
|
1 |
IC50 = 324.3 nM
|
|
|
CP0420503
|
1-[6-(2-fluorophenyl)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C20H16FNO2S
|
1
|
1 |
IC50 = 333.4 nM
|
|
|
CP0434753
|
1-(6-methoxyquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C15H15NO3S
|
1
|
1 |
IC50 = 342.8 nM
|
|
|
CP0538448
|
1-(6-methylquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C15H15NO2S
|
1
|
1 |
IC50 = 343.2 nM
|
|
|
CP0385474
|
1-(6-bromoquinolin-4-yl)sulfanylcyclopropane-1-carboxylic acid
Show/Hide
|
C13H10BrNO2S
|
1
|
1 |
IC50 = 352.3 nM
|
|
|
CP0385473
|
1-[6-[3-(trifluoromethyl)phenyl]quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C21H16F3NO2S
|
1
|
1 |
IC50 = 358.7 nM
|
|
|
CP0417801
|
1-(6-cyanoquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C15H12N2O2S
|
1
|
1 |
IC50 = 398.8 nM
|
|
|
CP0456496
|
1-quinolin-4-ylsulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C14H13NO2S
|
1
|
1 |
IC50 = 448 nM
|
|
|
CP0546618
|
sodium;4-[[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylmethyl]-3-methoxybenzoate
Show/Hide
|
C26H20N3NaO3S
|
1
|
1 |
IC50 = 460 nM
|
|
|
CP0538449
|
1-(6-fluoroquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C14H12FNO2S
|
1
|
1 |
IC50 = 557.6 nM
|
|
|
CP0559979
|
2-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-hydroxyacetamide
Show/Hide
|
C15H12Br2N4O2S
|
1
|
1 |
IC50 = 640 nM
|
|
|
CP0472125
|
1-(6-cyclopropylquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C17H17NO2S
|
1
|
1 |
IC50 = 659.2 nM
|
|
|
CP0406890
|
1-[6-(cyanomethoxy)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C16H14N2O3S
|
1
|
1 |
IC50 = 680.2 nM
|
|
|
CP0491661
|
US8889724, EF
Show/Hide
|
C18H20N4O
|
1
|
1 |
IC50 = 740 nM
|
|
|
CP0041383
|
(3,5-dibromo-4-hydroxyphenyl)(2-ethyl-1-benzofuran-3-yl)methanone
Show/Hide
|
C17H12Br2O3
|
1
|
1 |
IC50 = 750 nM
|
|
|
CP0375456
|
1-(4-cyanonaphthalen-1-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C16H13NO2S
|
1
|
1 |
IC50 = 926.4 nM
|
|
|
CP0527621
|
US8889724, EB
Show/Hide
|
C16H16N4O
|
1
|
1 |
IC50 = 930 nM
|
|
|
CP0559825
|
1-[6-(3-fluorophenyl)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C20H16FNO2S
|
1
|
1 |
IC50 = 1189 nM
|
|
|
CP0571249
|
sodium;4-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylbutanoate
Show/Hide
|
C20H15N2NaO3S
|
1
|
1 |
IC50 = 1230 nM
|
|
|
CP0538106
|
1-[6-(hydroxymethyl)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C15H15NO3S
|
1
|
1 |
IC50 = 1257 nM
|
|
|
CP0568250
|
2-[1-[(4-bromonaphthalen-1-yl)methyl]imidazo[4,5-b]pyridin-2-yl]sulfanyl-2-methylpropanoic acid
Show/Hide
|
C21H18BrN3O2S
|
1
|
1 |
IC50 = 1360 nM
|
|
|
CP0549091
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(6-fluoropyridin-3-yl)methanesulfonamide
Show/Hide
|
C19H14Br2FN5O2S2
|
1
|
1 |
IC50 = 1550 nM
|
|
|
CP0552688
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(2,6-dichloropyridin-3-yl)methanesulfonamide
Show/Hide
|
C19H13Br2Cl2N5O2S2
|
1
|
1 |
IC50 = 1660 nM
|
|
|
CP0570258
|
sodium;4-[[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylmethyl]-3-methoxybenzoate
Show/Hide
|
C25H18N3NaO3S
|
1
|
1 |
IC50 = 1660 nM
|
|
|
CP0472133
|
1-[6-[4-(trifluoromethyl)phenyl]quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C21H16F3NO2S
|
1
|
1 |
IC50 = 1753 nM
|
|
|
CP0385626
|
1-(6-aminoquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C14H14N2O2S
|
1
|
1 |
IC50 = 1787 nM
|
|
|
CP0486629
|
1-[6-(2-hydroxyethoxy)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C16H17NO4S
|
1
|
1 |
IC50 = 1886 nM
|
|
|
CP0375461
|
1-(1,6-naphthyridin-4-ylsulfanyl)cyclobutane-1-carboxylic acid
Show/Hide
|
C13H12N2O2S
|
1
|
1 |
IC50 = 1932 nM
|
|
|
CP0547968
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(6-chloropyridin-3-yl)methanesulfonamide
Show/Hide
|
C19H14Br2ClN5O2S2
|
1
|
1 |
IC50 = 1940 nM
|
|
|
CP0567735
|
sodium;3-[[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylmethyl]benzoate
Show/Hide
|
C24H16N3NaO2S
|
1
|
1 |
IC50 = 1960 nM
|
|
|
CP0555223
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(6-bromopyridin-3-yl)methanesulfonamide
Show/Hide
|
C19H14Br3N5O2S2
|
1
|
1 |
IC50 = 2200 nM
|
|
|
CP0578825
|
sodium;5-[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylpentanoate
Show/Hide
|
C21H18N3NaO2S
|
1
|
1 |
IC50 = 2280 nM
|
|
|
CP0570427
|
3-[1-[(4-cyclopropylnaphthalen-1-yl)methyl]imidazo[4,5-b]pyridin-2-yl]sulfanylpropanoic acid
Show/Hide
|
C23H21N3O2S
|
1
|
1 |
IC50 = 2490 nM
|
|
|
CP0580203
|
sodium;4-[[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylmethyl]benzoate
Show/Hide
|
C24H16N3NaO2S
|
1
|
1 |
IC50 = 2550 nM
|
|
|
CP0578050
|
2-[1-[(4-bromonaphthalen-1-yl)methyl]imidazo[4,5-c]pyridin-2-yl]sulfanyl-2-methylpropanoic acid
Show/Hide
|
C21H18BrN3O2S
|
1
|
1 |
IC50 = 2570 nM
|
|
|
CP0578824
|
sodium;4-[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylbutanoate
Show/Hide
|
C21H18N3NaO2S
|
1
|
1 |
IC50 = 2580 nM
|
|
|
CP0375459
|
1-[6-(2-cyanoethyl)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
Show/Hide
|
C17H16N2O2S
|
1
|
1 |
IC50 = 2757 nM
|
|
|
CP0578907
|
sodium;4-[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylbutanoate
Show/Hide
|
C20H16N3NaO2S
|
1
|
1 |
IC50 = 2780 nM
|
|
|
CP0537985
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(2,5-dichloropyridin-3-yl)methanesulfonamide
Show/Hide
|
C19H13Br2Cl2N5O2S2
|
1
|
1 |
IC50 = 2790 nM
|
|
|
CP0578051
|
2-[1-(4-cyclopropylnaphthalen-1-yl)imidazo[4,5-b]pyridin-2-yl]oxy-2-methylpropanoic acid
Show/Hide
|
C23H21N3O3
|
1
|
1 |
IC50 = 3060 nM
|
|
|
CP0548163
|
sodium;5-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,3-triaza-4-azanidacyclopenta-2,5-diene
Show/Hide
|
C15H10Br2N7NaS
|
1
|
1 |
IC50 = 3240 nM
|
|
|
CP0578826
|
sodium;2-[2-[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanyl-6-nitrophenyl]acetate
Show/Hide
|
C24H15N4NaO4S
|
1
|
1 |
IC50 = 3440 nM
|
|
|
CP0010999
|
4-[2-(5-amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-(1,3-thiazol-4-yl)benzenesulfonamide
Show/Hide
|
C18H12Cl2FN5O3S2
|
1
|
1 |
IC50 = 3500 nM
|
|
|
CP0568249
|
2-[1-[(4-cyclopropylnaphthalen-1-yl)methyl]imidazo[4,5-c]pyridin-2-yl]sulfanylacetic acid
Show/Hide
|
C22H19N3O2S
|
1
|
1 |
IC50 = 3550 nM
|
|
|
CP0580201
|
sodium;3-[[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylmethyl]benzoate
Show/Hide
|
C25H18N3NaO2S
|
1
|
1 |
IC50 = 3570 nM
|
|
|
CP0577433
|
sodium;5-[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylpentanoate
Show/Hide
|
C22H20N3NaO2S
|
1
|
1 |
IC50 = 3580 nM
|
|
|
CP0579517
|
1-[1-(4-cyclopropylnaphthalen-1-yl)imidazo[4,5-b]pyridin-2-yl]oxycyclobutane-1-carboxylic acid
Show/Hide
|
C24H21N3O3
|
1
|
1 |
IC50 = 3670 nM
|
|
|
CP0579209
|
2-[1-(4-cyclopropylnaphthalen-1-yl)imidazo[4,5-b]pyridin-2-yl]oxypropanoic acid
Show/Hide
|
C22H19N3O3
|
1
|
1 |
IC50 = 3700 nM
|
|
|
CP0577111
|
sodium;6-[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylhexanoate
Show/Hide
|
C23H22N3NaO2S
|
1
|
1 |
IC50 = 3760 nM
|
|
|
CP0574280
|
sodium;7-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylheptanoate
Show/Hide
|
C23H21N2NaO3S
|
1
|
1 |
IC50 = 3780 nM
|
|
|
CP0432064
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(2-methoxypyridin-3-yl)methanesulfonamide
Show/Hide
|
C20H17Br2N5O3S2
|
1
|
1 |
IC50 = 4050 nM
|
|
|
CP0576347
|
sodium;2-[5-bromo-2-[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylphenyl]acetate
Show/Hide
|
C24H15BrN3NaO2S
|
1
|
1 |
IC50 = 4120 nM
|
|
|
CP0573739
|
sodium;5-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylpentanoate
Show/Hide
|
C21H17N2NaO3S
|
1
|
1 |
IC50 = 4220 nM
|
|
|
CP0571299
|
sodium;6-[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylhexanoate
Show/Hide
|
C22H20N3NaO2S
|
1
|
1 |
IC50 = 4240 nM
|
|
|
CP0579630
|
sodium;2-[2-[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanyl-5-methoxyphenyl]acetate
Show/Hide
|
C25H18N3NaO3S
|
1
|
1 |
IC50 = 4250 nM
|
|
|
CP0573738
|
sodium;2-[[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylmethyl]benzoate
Show/Hide
|
C25H18N3NaO2S
|
1
|
1 |
IC50 = 4440 nM
|
|
|
CP0580202
|
sodium;2-[4-[[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylmethyl]phenyl]benzoate
Show/Hide
|
C31H22N3NaO2S
|
1
|
1 |
IC50 = 4570 nM
|
|
|
CP0578823
|
sodium;7-[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylheptanoate
Show/Hide
|
C24H24N3NaO2S
|
1
|
1 |
IC50 = 4640 nM
|
|
|
CP0576346
|
sodium;2-[4-[[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylmethyl]phenyl]benzoate
Show/Hide
|
C30H20N3NaO2S
|
1
|
1 |
IC50 = 4680 nM
|
|
|
CP0573740
|
sodium;6-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylhexanoate
Show/Hide
|
C22H19N2NaO3S
|
1
|
1 |
IC50 = 4740 nM
|
|
|
CP0579966
|
3-[1-(4-cyclopropylnaphthalen-1-yl)imidazo[4,5-b]pyridin-2-yl]oxypropanoic acid
Show/Hide
|
C22H19N3O3
|
1
|
1 |
IC50 = 4940 nM
|
|
|
CP0569911
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(2-chloropyridin-3-yl)methanesulfonamide
Show/Hide
|
C19H14Br2ClN5O2S2
|
1
|
1 |
IC50 = 5100 nM
|
|
|
CP0578892
|
sodium;2-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanyl-2-methylpropanoate
Show/Hide
|
C20H15N2NaO3S
|
1
|
1 |
IC50 = 5210 nM
|
|
|
CP0574304
|
sodium;2-[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanyl-2-methylpropanoate
Show/Hide
|
C21H18N3NaO2S
|
1
|
1 |
IC50 = 5360 nM
|
|
|
CP0549191
|
1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(2,6-dibromopyridin-3-yl)methanesulfonamide
Show/Hide
|
C19H13Br4N5O2S2
|
1
|
1 |
IC50 = 5410 nM
|
|
|
CP0674431
|
LESINURAD
Show/Hide
|
C17H14BrN3O2S
|
2
|
1 |
IC50 = 5540 nM
|
|
|
2 |
IC50 = 7200 nM
|
|
|
CP0571298
|
sodium;7-[3-[(4-cyanonaphthalen-1-yl)amino]pyridin-4-yl]sulfanylheptanoate
Show/Hide
|
C23H22N3NaO2S
|
1
|
1 |
IC50 = 5750 nM
|
|
|
CP0550521
|
sodium;4-[[3-[(4-cyanonaphthalen-1-yl)-methylamino]pyridin-4-yl]sulfanylmethyl]benzoate
Show/Hide
|
C25H18N3NaO2S
|
1
|
1 |
IC50 = 6250 nM
|
|
|
CP0558553
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1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[5-(trifluoromethyl)pyridin-3-yl]methanesulfonamide
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C20H14Br2F3N5O2S2
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1
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1 |
IC50 = 6380 nM
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CP0546615
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sodium;3-[[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylmethyl]benzoate
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C24H15N2NaO3S
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1
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1 |
IC50 = 6580 nM
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CP0574293
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sodium;2-[[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylmethyl]benzoate
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C24H15N2NaO3S
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1
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1 |
IC50 = 6860 nM
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CP0546614
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sodium;2-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylacetate
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C18H11N2NaO3S
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1
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1 |
IC50 = 6970 nM
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CP0574294
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sodium;2-[5-bromo-2-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylphenyl]acetate
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C24H14BrN2NaO3S
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1
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1 |
IC50 = 8050 nM
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CP0385482
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1-quinazolin-4-ylsulfanylcyclobutane-1-carboxylic acid
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C13H12N2O2S
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1
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1 |
IC50 > 10000 nM
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CP0403505
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1-(6-hydroxyquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
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C14H13NO3S
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1
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1 |
IC50 > 10000 nM
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CP0403506
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1-[(3-oxo-4H-1,4-benzoxazin-5-yl)sulfanyl]cyclobutane-1-carboxylic acid
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C13H13NO4S
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1
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1 |
IC50 > 10000 nM
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CP0403507
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1-quinazolin-4-yloxycyclobutane-1-carboxylic acid
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C13H12N2O3
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1
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1 |
IC50 > 10000 nM
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CP0406891
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1-(1,6-naphthyridin-5-ylsulfanyl)cyclobutane-1-carboxylic acid
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C13H12N2O2S
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1
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1 |
IC50 > 10000 nM
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CP0417799
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1-[6-[2-(methylamino)-2-oxoethoxy]quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
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C17H18N2O4S
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1
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1 |
IC50 > 10000 nM
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CP0463052
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1-[6-(cyclopropanecarbonylamino)quinolin-4-yl]sulfanylcyclobutane-1-carboxylic acid
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C18H18N2O3S
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1
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1 |
IC50 > 10000 nM
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CP0538441
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1-(1,5-naphthyridin-4-ylsulfanyl)cyclobutane-1-carboxylic acid
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C13H12N2O2S
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1
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1 |
IC50 > 10000 nM
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CP0564207
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1-(6-acetamidoquinolin-4-yl)sulfanylcyclobutane-1-carboxylic acid
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C16H16N2O3S
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1
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1 |
IC50 > 10000 nM
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CP0554602
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1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-[6-(trifluoromethyl)pyridin-3-yl]methanesulfonamide
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C20H14Br2F3N5O2S2
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1
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1 |
IC50 = 10210 nM
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CP0568801
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sodium;4-[[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylmethyl]benzoate
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C24H15N2NaO3S
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1
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1 |
IC50 = 10250 nM
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CP0577104
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sodium;2-[2-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanyl-6-nitrophenyl]acetate
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C24H14N3NaO5S
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1
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1 |
IC50 = 10450 nM
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CP0533504
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1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-(4-iodopyridin-3-yl)methanesulfonamide
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C19H14Br2IN5O2S2
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1
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1 |
IC50 = 10570 nM
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CP0546616
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sodium;2-[2-[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanyl-5-methoxyphenyl]acetate
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C25H17N2NaO4S
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1
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1 |
IC50 = 14180 nM
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CP0554603
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sodium;[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanylmethanesulfonate
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C14H10Br2N3NaO3S2
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1
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1 |
IC50 = 14380 nM
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CP0576348
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sodium;2-[4-[[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylmethyl]phenyl]benzoate
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C30H19N2NaO3S
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1
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1 |
IC50 = 15110 nM
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CP0432021
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1-[[5-bromo-4-[(4-bromonaphthalen-1-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]-N-phenylmethanesulfonamide
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C20H16Br2N4O2S2
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1
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1 |
IC50 = 15780 nM
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CP0575659
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sodium;4-[[3-(4-cyanonaphthalen-1-yl)oxypyridin-4-yl]sulfanylmethyl]-3-methoxybenzoate
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C25H17N2NaO4S
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1
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1 |
IC50 = 16350 nM
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