Compound ID |
Compound Name |
Compound Formula |
CP0168917
|
Omidenepag
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|
C23H22N6O4S
|
2
|
1 |
EC50 = 1.1 nM
|
|
|
2 |
IC50 = 10 nM
|
|
|
CP0847243
|
5-{(R)-1-[4-(1-Hydroxy-heptyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
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|
C24H31NO5S
|
3
|
1 |
EC50 = 1.6 nM
|
|
|
2 |
Ki = 10 nM
|
|
|
3 |
Ki = 190 nM
|
|
|
CP0870431
|
5-(3-{(S)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-yl}-propyl)-thiophene-2-carboxylic acid
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|
C24H31NO4S
|
2
|
1 |
EC50 = 1.6 nM
|
|
|
2 |
Ki = 15 nM
|
|
|
CP0394034
|
2-[[6-[[(4-pyridin-2-ylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid
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|
C25H23N5O4S
|
1
|
1 |
EC50 = 1.6 nM
|
|
|
CP0870239
|
5-(3-((1R,2S)-2-(4-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)propyl)thiophene-2-carboxylic acid
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|
C25H32O4S
|
2
|
1 |
EC50 = 2 nM
|
|
|
2 |
Ki = 54 nM
|
|
|
CP0946462
|
(6-((Biphenyl-4-ylmethyl)(pyridin-3-ylsulfonyl)aminomethyl)-pyridin-2-ylamino)acetic Acid Hydrochloride
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|
C26H25ClN4O4S
|
1
|
1 |
EC50 = 2 nM
|
|
|
CP0401695
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[(2,3,4-trichlorophenoxy)methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
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|
C19H18Cl3NO5S
|
1
|
1 |
EC50 = 2.3 nM
|
|
|
CP0401697
|
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3,5-dimethylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H24ClNO5S
|
1
|
1 |
EC50 = 2.3 nM
|
|
|
CP0468701
|
2-[[6-[[[4-(1-methylcyclopropyl)phenyl]methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C24H27ClN4O4S
|
1
|
1 |
EC50 = 2.6 nM
|
|
|
CP0539129
|
2-[[6-[[(4-tert-butylphenyl)methyl-(4-fluorophenyl)sulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C25H29ClFN3O4S
|
1
|
1 |
EC50 = 2.7 nM
|
|
|
CP0575238
|
2-[[6-[[(4-tert-butylphenyl)methyl-pyridin-2-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C24H29ClN4O4S
|
1
|
1 |
EC50 = 2.7 nM
|
|
|
CP0538158
|
2-[[6-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C24H29ClN4O4S
|
1
|
1 |
EC50 = 2.8 nM
|
|
|
CP0538161
|
2-[[6-[[1-benzothiophen-2-ylmethyl(pyridin-3-ylsulfonyl)amino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C22H21ClN4O4S2
|
1
|
1 |
EC50 = 3.4 nM
|
|
|
CP0401696
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[(2,4,5-trichlorophenoxy)methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H18Cl3NO5S
|
1
|
1 |
EC50 = 3.7 nM
|
|
|
CP0434757
|
2-[[6-[[benzenesulfonyl-[(4-tert-butylphenyl)methyl]amino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C25H30ClN3O4S
|
1
|
1 |
EC50 = 4.3 nM
|
|
|
CP0436871
|
2-[[6-[[(4-tert-butylphenyl)methyl-(4-chlorophenyl)sulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C25H29Cl2N3O4S
|
1
|
1 |
EC50 = 4.4 nM
|
|
|
CP0482823
|
2-[[6-[[[4-(1-ethylcyclopropyl)phenyl]methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid
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|
C25H28N4O4S
|
1
|
1 |
EC50 = 4.5 nM
|
|
|
CP0866241
|
5-(3-{(S)-1-[4-(1-Hydroxy-heptyl)-phenyl]-5-oxo-pyrrolidin-2-yl}-propyl)-thiophene-2-carboxylic acid
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|
C25H33NO4S
|
2
|
1 |
EC50 = 5 nM
|
|
|
2 |
Ki = 8 nM
|
|
|
CP0440481
|
2-[[6-[[1-benzofuran-2-ylmethyl(pyridin-3-ylsulfonyl)amino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C22H21ClN4O5S
|
1
|
1 |
EC50 = 5.6 nM
|
|
|
CP0468700
|
2-[[6-[[(4-tert-butylphenyl)methyl-(3-fluorophenyl)sulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C25H29ClFN3O4S
|
1
|
1 |
EC50 = 6.1 nM
|
|
|
CP0847236
|
5-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
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|
C23H29NO5S
|
2
|
1 |
EC50 = 8 nM
|
|
|
2 |
Ki = 115 nM
|
|
|
CP0377164
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[[3-(trifluoromethyl)phenoxy]methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H20F3NO5S
|
1
|
1 |
EC50 = 9 nM
|
|
|
CP0377163
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[[2-(trifluoromethyl)phenoxy]methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H20F3NO5S
|
1
|
1 |
EC50 = 11 nM
|
|
|
CP0482824
|
2-[[6-[[[4-(1-ethylcyclobutyl)phenyl]methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid
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|
C26H30N4O4S
|
1
|
1 |
EC50 = 13 nM
|
|
|
CP0870434
|
7-((1R,2S,3R,5R)-3,5-dichloro-2-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)hept-5-enoic acid
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|
C24H34Cl2O3
|
2
|
1 |
EC50 = 15 nM
|
|
|
2 |
Ki = 25 nM
|
|
|
CP0080235
|
4-(2-((R)-2-((S)-3-hydroxyhept-1-enyl)-5-oxopyrrolidin-1-yl)ethyl)benzoate
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|
C20H27NO4
|
2
|
1 |
EC50 = 16 nM
|
|
|
2 |
Ki = 125.5 nM
|
|
|
CP0847237
|
5-{3-[(S)-1-(4-Hexanoyl-phenyl)-5-oxo-pyrrolidin-2-yl]-propyl}-thiophene-2-carboxylic acid
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|
C24H29NO4S
|
2
|
1 |
EC50 = 16 nM
|
|
|
2 |
Ki = 31 nM
|
|
|
CP0539128
|
C-533,536-02
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|
C25H27N2NaO5S
|
2
|
1 |
EC50 = 17 nM
|
|
|
2 |
Ki = 16 nM
|
|
|
CP0466688
|
2-[[6-[[[4-(1-propan-2-ylcyclopropyl)phenyl]methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid
Show/Hide
|
C26H30N4O4S
|
1
|
1 |
EC50 = 18 nM
|
|
|
CP0458129
|
2-[[6-[[(4-tert-butylphenyl)methyl-(4-methoxyphenyl)sulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C26H32ClN3O5S
|
1
|
1 |
EC50 = 19 nM
|
|
|
CP0452767
|
4-(2-((R)-2-(3-methylocta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
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|
C22H29NO3
|
2
|
1 |
EC50 = 23 nM
|
|
|
2 |
Ki = 29 nM
|
|
|
CP0847242
|
5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-thiophene-2-carboxylic acid
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|
C21H25NO4S
|
4
|
1 |
EC50 = 27 nM
|
|
|
2 |
EC50 = 1343 nM
|
|
|
3 |
Ki = 27 nM
|
|
|
4 |
Ki = 501 nM
|
|
|
CP0539130
|
2-[[6-[[(4-cyclohexylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid
Show/Hide
|
C26H30N4O4S
|
1
|
1 |
EC50 = 29 nM
|
|
|
CP0866746
|
7-((1R,2S,3R)-2-(4-hexanoylphenyl)-3-hydroxy-5-oxocyclopentyl)hept-5-enoic acid
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|
C24H32O5
|
2
|
1 |
EC50 = 31 nM
|
|
|
2 |
Ki = 111 nM
|
|
|
CP0899507
|
7-((1S,2S,3R,5R)-5-cyano-3-hydroxy-2-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)hept-5-enoic acid
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|
C25H35NO4
|
2
|
1 |
EC50 = 34 nM
|
|
|
2 |
Ki = 1252 nM
|
|
|
CP0452766
|
4-(2-((R)-2-(4-methylocta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
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|
C22H29NO3
|
2
|
1 |
EC50 = 35 nM
|
|
|
2 |
Ki = 60 nM
|
|
|
CP0901193
|
(6-((4'-Fluorobiphenyl-4-ylmethyl)(pyridin-3-ylsulfonyl)-aminomethyl)pyridin-2-ylamino)acetic Acid Hydrochloride
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|
C26H24ClFN4O4S
|
1
|
1 |
EC50 = 35 nM
|
|
|
CP0468695
|
2-[[6-[[pyridin-3-ylsulfonyl-[[4-(1,2,4-triazol-1-yl)phenyl]methyl]amino]methyl]pyridin-2-yl]amino]acetic acid
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|
C22H21N7O4S
|
1
|
1 |
EC50 = 43 nM
|
|
|
CP0394031
|
2-[[6-[[(4-tert-butylphenyl)methyl-(2-fluorophenyl)sulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
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|
C25H29ClFN3O4S
|
1
|
1 |
EC50 = 45 nM
|
|
|
CP0377162
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[[3-(trifluoromethoxy)phenoxy]methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H20F3NO6S
|
1
|
1 |
EC50 = 69 nM
|
|
|
CP0882301
|
(6-((4'-Chlorobiphenyl-4-ylmethyl)(pyridin-3-ylsulfonyl)-aminomethyl)pyridin-2-ylamino)acetic Acid Hydrochloride
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|
C26H24Cl2N4O4S
|
1
|
1 |
EC50 = 75 nM
|
|
|
CP0434756
|
3-[[6-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]propanoic acid;hydrochloride
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|
C25H31ClN4O4S
|
1
|
1 |
EC50 = 83 nM
|
|
|
CP0458128
|
2-[[6-[[(4-tert-butylphenyl)methyl-methylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
|
C20H28ClN3O4S
|
1
|
1 |
EC50 = 91 nM
|
|
|
CP0924067
|
7-((1R,2S,3R)-2-(4-tert-butylphenyl)-3-hydroxy-5-oxocyclopentyl)heptanoic acid
Show/Hide
|
C22H32O4
|
1
|
1 |
EC50 = 102 nM
|
|
|
CP0558990
|
2-[[6-[[(3-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
|
C24H29ClN4O4S
|
1
|
1 |
EC50 = 109 nM
|
|
|
CP0866254
|
7-((1R,2S,3R,5R)-2-(4-tert-butylphenyl)-5-chloro-3-hydroxycyclopentyl)hept-5-enoic acid
Show/Hide
|
C22H31ClO3
|
1
|
1 |
EC50 = 118 nM
|
|
|
CP0574584
|
2-[[6-[[5-phenylpentyl(pyridin-3-ylsulfonyl)amino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
|
C24H29ClN4O4S
|
1
|
1 |
EC50 = 118 nM
|
|
|
CP0394032
|
2-[[6-[[pyridin-3-ylsulfonyl-[[4-(trifluoromethyl)phenyl]methyl]amino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
|
C21H20ClF3N4O4S
|
1
|
1 |
EC50 = 119 nM
|
|
|
CP0885328
|
5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-furan-2-carboxylic acid
Show/Hide
|
C21H25NO5
|
4
|
1 |
EC50 = 189 nM
|
|
|
2 |
EC50 = 442 nM
|
|
|
3 |
Ki = 189 nM
|
|
|
4 |
Ki = 4000 nM
|
|
|
CP0483781
|
4-(2-((R)-2-(octa-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
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|
C21H27NO3
|
2
|
1 |
EC50 = 197 nM
|
|
|
2 |
Ki = 88 nM
|
|
|
CP0380277
|
2-[(2R,4aR,5S,6R,7aS)-5-[(2-chlorophenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H20ClNO5S
|
1
|
1 |
EC50 = 203 nM
|
|
|
CP0850988
|
5-{(R)-1-[4-(1-Hydroxy-pentyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
Show/Hide
|
C22H27NO5S
|
2
|
1 |
EC50 = 212 nM
|
|
|
2 |
Ki = 387 nM
|
|
|
CP0847238
|
5-[(R)-1-(4-Hexanoyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-thiophene-2-carboxylic acid
Show/Hide
|
C23H27NO5S
|
2
|
1 |
EC50 = 215 nM
|
|
|
2 |
Ki = 163 nM
|
|
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CP0464527
|
4-(2-((R)-2-(4-methylocta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C22H29NO3
|
2
|
1 |
EC50 = 222 nM
|
|
|
2 |
Ki = 134 nM
|
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|
CP0895715
|
5-(3-((2R)-1-(4-(1-hydroxyhexyl)phenyl)-5-oxopyrrolidin-2-yl)allyl)thiophene-2-carboxylic acid
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|
C24H29NO4S
|
2
|
1 |
EC50 = 226 nM
|
|
|
2 |
Ki = 1382 nM
|
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CP0866433
|
7-((1R,2S,3R,5R)-2-(4-tert-butylphenyl)-5-chloro-3-hydroxycyclopentyl)heptanoic acid
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|
C22H33ClO3
|
1
|
1 |
EC50 = 264 nM
|
|
|
CP0863098
|
2-(3-(((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)cyclopentyl)methyl)phenoxy)acetic acid
Show/Hide
|
C28H35ClO5
|
2
|
1 |
EC50 = 266 nM
|
|
|
2 |
IC50 = 5200 nM
|
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|
CP0387031
|
2-[[6-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]-methylamino]acetic acid;hydrochloride
Show/Hide
|
C25H31ClN4O4S
|
1
|
1 |
EC50 = 283 nM
|
|
|
CP0174264
|
7-[(1R,2S)-2-[4-(1-hydroxyhexyl)phenyl]-5-oxocyclopentyl]heptanoic acid
Show/Hide
|
C24H36O4
|
2
|
1 |
EC50 = 284 nM
|
|
|
2 |
Ki = 871 nM
|
|
|
CP0538160
|
2-[[6-[[(4-pyridazin-4-ylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
|
C24H23ClN6O4S
|
1
|
1 |
EC50 = 307 nM
|
|
|
CP0869429
|
7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
|
C26H37ClO4
|
1
|
1 |
EC50 = 322 nM
|
|
|
CP0888285
|
7-((1R,2S)-2-(4-(2-hydroxyhexyl)phenyl)-5-oxocyclopentyl)heptanoic acid
Show/Hide
|
C24H36O4
|
2
|
1 |
EC50 = 343 nM
|
|
|
2 |
Ki = 700 nM
|
|
|
CP0055947
|
(15S)-prostaglandin E2
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|
C20H32O5
|
5
|
1 |
EC50 = 346 nM
|
|
|
2 |
IC50 = 2.6 nM
|
|
|
3 |
IC50 = 4 nM
|
|
|
4 |
Ki = 1.03 nM
|
|
|
5 |
Ki = 4.9 nM
|
|
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CP0558989
|
2-[[4-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]-1,3-thiazol-2-yl]amino]acetic acid;hydrochloride
Show/Hide
|
C22H27ClN4O4S2
|
1
|
1 |
EC50 = 360 nM
|
|
|
CP0850987
|
5-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-furan-2-carboxylic acid
Show/Hide
|
C23H29NO6
|
2
|
1 |
EC50 = 388 nM
|
|
|
2 |
Ki = 2028 nM
|
|
|
CP0866434
|
7-((1R,2S,3R,5R)-5-chloro-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxycyclopentyl)hept-5-enoic acid
Show/Hide
|
C25H35ClO4
|
1
|
1 |
EC50 = 392 nM
|
|
|
CP0866283
|
7-((1R,2S,3R)-3-hydroxy-2-(1-hydroxy-2,3-dihydro-1H-inden-5-yl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
|
C21H26O5
|
2
|
1 |
EC50 = 405 nM
|
|
|
2 |
IC50 = 2281 nM
|
|
|
CP0847234
|
5-{(R)-1-[4-(1-Hydroxy-butyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
Show/Hide
|
C21H25NO5S
|
2
|
1 |
EC50 = 426 nM
|
|
|
2 |
Ki = 1639 nM
|
|
|
CP0866287
|
7-((1R,2S,3S,5R)-3,5-dichloro-2-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
|
C24H34Cl2O3
|
2
|
1 |
EC50 = 427 nM
|
|
|
2 |
Ki = 504 nM
|
|
|
CP0856816
|
7-((1R,2S,3R)-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxy-5-oxocyclopentyl)heptanoic acid
Show/Hide
|
C25H36O5
|
1
|
1 |
EC50 = 450 nM
|
|
|
CP0866427
|
7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
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C22H31ClO4
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1
|
1 |
EC50 = 497 nM
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CP0852835
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxycyclobutyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
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C22H29ClO4
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1
|
1 |
EC50 = 513 nM
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CP0866768
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7-((1R,2S,3R)-3-hydroxy-2-(4-(1-hydroxy-2-methylpropan-2-yl)phenyl)-5-oxocyclopentyl)heptanoic acid
Show/Hide
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C22H32O5
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2
|
1 |
EC50 = 526 nM
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2 |
IC50 = 18735 nM
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CP0852857
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(1-hydroxy-2,3-dihydro-1H-inden-5-yl)cyclopentyl)heptanoic acid
Show/Hide
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C21H29ClO4
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2
|
1 |
EC50 = 529 nM
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2 |
IC50 = 13139 nM
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CP0852840
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C26H39ClO4
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1
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1 |
EC50 = 546 nM
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CP0552130
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2-[[6-[[(4-tert-butylphenyl)methyl-(3-chlorophenyl)sulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
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C25H29Cl2N3O4S
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1
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1 |
EC50 = 620 nM
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CP0866252
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7-((1R,2S,3R)-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)heptanoic acid
Show/Hide
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C26H38O5
|
1
|
1 |
EC50 = 635 nM
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CP0468691
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2-[[6-[[(4-tert-butylcyclohexyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
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C24H35ClN4O4S
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1
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1 |
EC50 = 649 nM
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CP0895714
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropan-2-yl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C22H33ClO4
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2
|
1 |
EC50 = 708 nM
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2 |
IC50 = 8950 nM
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CP0866243
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4-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxy}-benzoic acid
Show/Hide
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C24H29NO5
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2
|
1 |
EC50 = 728 nM
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|
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2 |
Ki = 22726 nM
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CP0900745
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxycyclobutyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C22H31ClO4
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1
|
1 |
EC50 = 743 nM
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CP0869414
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7-((1R,2R,5S)-2-chloro-5-(5-(1-hydroxyhexyl)thiophen-2-yl)cyclopentyl)heptanoic acid
Show/Hide
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C22H35ClO3S
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2
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1 |
EC50 = 769 nM
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|
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2 |
Ki = 600 nM
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CP0888315
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2,2-dimethylpropyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
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C23H33ClO4
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2
|
1 |
EC50 = 779 nM
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|
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2 |
IC50 = 1537 nM
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CP0938030
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7-((1R,2S,3R,5R)-5-chloro-2-(2,3-dihydro-1H-inden-5-yl)-3-hydroxycyclopentyl)heptanoic acid
Show/Hide
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C21H29ClO3
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2
|
1 |
EC50 = 818 nM
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|
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2 |
IC50 = 6251 nM
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CP0866431
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methyl 7-((1R,2S,3R)-2-(4-tert-butylphenyl)-3-hydroxy-5-oxocyclopentyl)heptanoate
Show/Hide
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C23H34O4
|
1
|
1 |
EC50 = 936 nM
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CP0852855
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7-((1R,2S)-2-(4-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
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C24H34O4
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2
|
1 |
EC50 = 1011 nM
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|
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2 |
Ki = 700 nM
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CP0866286
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7-((1R,2S)-2-(4-tert-butylphenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
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C22H30O3
|
1
|
1 |
EC50 = 1050 nM
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CP0847240
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5-{(R)-1-[4-(1-Hydroxy-2-phenyl-ethyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-furan-2-carboxylic acid
Show/Hide
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C25H25NO6
|
2
|
1 |
EC50 = 1228 nM
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|
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2 |
Ki = 2293 nM
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CP0856827
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2,2-dimethylpropyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C23H35ClO4
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2
|
1 |
EC50 = 1265 nM
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|
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2 |
IC50 = 3630 nM
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CP0921736
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7-((1R,2R,5S)-2-chloro-5-(4-(1-hydroxypentyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C23H35ClO3
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2
|
1 |
EC50 = 1409 nM
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|
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2 |
Ki = 1400 nM
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CP0423796
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4-[2-[3,5-dichloro-2-(3-hydroxyoctyl)-6-oxopyridin-1-yl]ethyl]benzoic acid
Show/Hide
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C22H27Cl2NO4
|
1
|
1 |
EC50 = 1500 nM
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|
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CP0863099
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2-(4-((2S,3R,5R)-5-chloro-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxycyclopentyl)but-2-ynyloxy)acetic acid
Show/Hide
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C24H31ClO5
|
1
|
1 |
EC50 = 1550 nM
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|
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CP0870234
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7-((1R,2S)-2-(4-((R)-cyclohexyl(hydroxy)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
|
C25H34O4
|
1
|
1 |
EC50 = 1640 nM
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|
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CP0866304
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7-((1R,2S,3R)-2-(4-tert-butylphenyl)-3-hydroxy-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
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C22H30O4
|
1
|
1 |
EC50 = 1709 nM
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|
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CP0847239
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5-{(R)-1-[4-(1-Hydroxy-propyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-thiophene-2-carboxylic acid
Show/Hide
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C20H23NO5S
|
2
|
1 |
EC50 = 1812 nM
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|
|
2 |
Ki = 5731 nM
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CP0866249
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7-((1R,2S)-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
|
C25H34O4
|
1
|
1 |
EC50 = 2101 nM
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|
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CP0856833
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methyl 7-((1R,2S)-2-(4-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)heptanoate
Show/Hide
|
C25H38O4
|
2
|
1 |
EC50 = 2162 nM
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|
|
2 |
Ki = 4677 nM
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CP0870418
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(hydroxy(1-propylcyclobutyl)methyl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
|
C26H37ClO4
|
1
|
1 |
EC50 = 2270 nM
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|
|
CP0870435
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7-((1R,2S)-2-(3-((R)-hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
|
C26H36O4
|
1
|
1 |
EC50 = 2657 nM
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|
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CP0866258
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7-((1R,2S,3R,5R)-5-chloro-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxycyclopentyl)heptanoic acid
Show/Hide
|
C25H37ClO4
|
1
|
1 |
EC50 = 2813 nM
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|
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CP0866395
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7-((1R,2S,3R)-3-hydroxy-5-oxo-2-p-tolylcyclopentyl)heptanoic acid
Show/Hide
|
C19H26O4
|
1
|
1 |
EC50 = 3128 nM
|
|
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CP0888298
|
7-((1R,2S)-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)heptanoic acid
Show/Hide
|
C26H38O4
|
1
|
1 |
EC50 = 3407 nM
|
|
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CP0852831
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7-((1R,2S,3R,5R)-5-chloro-2-(4-(cyclohexylmethyl)phenyl)-3-hydroxycyclopentyl)heptanoic acid
Show/Hide
|
C25H37ClO3
|
1
|
1 |
EC50 = 3445 nM
|
|
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CP0856836
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7-((1R,2S,3R)-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
|
C26H36O5
|
1
|
1 |
EC50 = 3723 nM
|
|
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CP0866278
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2-(4-((1R,2S,3R,5R)-5-chloro-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxycyclopentyl)but-2-enyloxy)acetic acid
Show/Hide
|
C24H33ClO5
|
1
|
1 |
EC50 = 3844 nM
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|
|
CP0866744
|
7-[(S)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-yl]-heptanoic acid
Show/Hide
|
C21H31NO3
|
2
|
1 |
EC50 = 4121 nM
|
|
|
2 |
Ki > 10000 nM
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|
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CP0380281
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[[4-(trifluoromethoxy)phenoxy]methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H20F3NO6S
|
1
|
1 |
EC50 = 4500 nM
|
|
|
CP0437308
|
4-[2-[3,5-dichloro-2-[(E)-3-hydroxy-3-methyloct-1-enyl]-6-oxopyridin-1-yl]ethyl]benzoic acid
Show/Hide
|
C23H27Cl2NO4
|
1
|
1 |
EC50 = 4700 nM
|
|
|
CP0957655
|
7-((5S)-5-(4-(1-hydroxyhexyl)phenyl)cyclopent-1-enyl)heptanoic acid
Show/Hide
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C24H36O3
|
2
|
1 |
EC50 = 4877 nM
|
|
|
2 |
Ki = 2811 nM
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CP0866285
|
methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2,2-dimethylpropyl)phenyl)cyclopentyl)heptanoate
Show/Hide
|
C24H37ClO4
|
1
|
1 |
EC50 = 4995 nM
|
|
|
CP0888286
|
methyl 7-((1R,2R,5S)-2-chloro-5-(5-(1-hydroxyhexyl)thiophen-2-yl)cyclopentyl)heptanoate
Show/Hide
|
C23H37ClO3S
|
2
|
1 |
EC50 = 7100 nM
|
|
|
2 |
Ki = 7100 nM
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|
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CP0870416
|
5-{(R)-1-[4-(1-Hydroxy-2-methyl-propyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-furan-2-carboxylic acid
Show/Hide
|
C21H25NO6
|
2
|
1 |
EC50 = 7669 nM
|
|
|
2 |
Ki > 10000 nM
|
|
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CP0457559
|
4-(2-((R)-2-oxo-5-(4-phenylpenta-1,3-dienyl)pyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
|
C24H25NO3
|
2
|
1 |
EC50 > 10000 nM
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|
|
2 |
Ki = 749 nM
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|
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CP0380278
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-(phenoxymethyl)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H21NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0380280
|
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chlorophenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H20ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0391092
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2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-oxazole-4-carboxylic acid
Show/Hide
|
C20H22ClNO6
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0391098
|
4-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]thiophene-2-carboxylic acid
Show/Hide
|
C21H23ClO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0401698
|
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-methoxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H24ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0401699
|
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H22ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0401700
|
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H22ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0401702
|
2-[(2R,4aR,5S,6S,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-fluoro-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H21ClFNO4S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0407410
|
4-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]furan-2-carboxylic acid
Show/Hide
|
C21H23ClO6
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0407431
|
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methoxyphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H22ClNO6S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0414542
|
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-propan-2-ylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C22H26ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0414599
|
2-[(2R,4aR,5S,6R,7aS)-5-[(3,4-dimethylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H25NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0434442
|
2-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-ethylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H24ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0434444
|
5-[(2R,4aR,5S,6R,7aS)-5-[(4-chloro-3-methylphenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]furan-2-carboxylic acid
Show/Hide
|
C21H23ClO6
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0483476
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[[3-methyl-4-(trifluoromethyl)phenoxy]methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H22F3NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0498080
|
2-[(2R,4aR,5S,6R,7aS)-5-[(3,4-dichlorophenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H19Cl2NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0508797
|
2-[(2R,4aR,5S,6R,7aS)-5-[[4-chloro-3-(trifluoromethyl)phenoxy]methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H19ClF3NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0377166
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[(4-methylphenoxy)methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H23NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0380283
|
2-[(2R,4aR,5S,6R,7aS)-5-[(2-fluorophenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H20FNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0380284
|
2-[(2R,4aR,5S,6R,7aS)-5-[(3-chlorophenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H20ClNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0409741
|
2-[(2R,4aR,5R,6R,7aS)-6-hydroxy-5-(5-phenoxypentyl)-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C23H29NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0424625
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[[4-(trifluoromethyl)phenoxy]methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C20H20F3NO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0428589
|
2-[(2R,4aR,5S,6R,7aS)-5-[(3-fluorophenoxy)methyl]-6-hydroxy-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C19H20FNO5S
|
1
|
1 |
EC50 > 10000 nM
|
|
|
CP0452553
|
2-[(2R,4aR,5S,6R,7aS)-6-hydroxy-5-[(3-methylphenoxy)methyl]-2,3,4,4a,5,6,7,7a-octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
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C20H23NO5S
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1
|
1 |
EC50 > 10000 nM
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|
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CP0847318
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2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-3-phenoxy-1-propen-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
Show/Hide
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C21H23NO5S
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1
|
1 |
EC50 > 10000 nM
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CP0847319
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2-{(2R,4aR,5R,6R,7aS)-5-[(4-fluorophenoxy)methyl]-6-hydroxyoctahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
Show/Hide
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C19H20FNO5S
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1
|
1 |
EC50 > 10000 nM
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CP0847320
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2-[(2R,4aR,5R,6R,7aS)-6-hydroxy-5-(2-phenoxyethyl)octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
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C20H23NO5S
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1
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1 |
EC50 > 10000 nM
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CP0847322
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2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-5-phenoxy-1-penten-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
Show/Hide
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C23H27NO5S
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1
|
1 |
EC50 > 10000 nM
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CP0862926
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2-{(2R,4aR,5R,6R,7aS)-6-hydroxy-5-[(1E)-4-phenoxy-1-buten-1-yl]octahydrocyclopenta[b]pyran-2-yl}-1,3-thiazole-4-carboxylic acid
Show/Hide
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C22H25NO5S
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1
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1 |
EC50 > 10000 nM
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CP0870958
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2-[(2R,4aR,5R,6R,7aS)-6-hydroxy-5-(3-phenoxypropyl)octahydrocyclopenta[b]pyran-2-yl]-1,3-thiazole-4-carboxylic acid
Show/Hide
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C21H25NO5S
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1
|
1 |
EC50 > 10000 nM
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CP0847233
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3-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-ylmethoxymethyl}-benzoic acid
Show/Hide
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C25H31NO5
|
1
|
1 |
EC50 > 10000 nM
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CP0847241
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3-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxymethyl]-benzoic acid
Show/Hide
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C23H27NO4
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1
|
1 |
EC50 > 10000 nM
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CP0852829
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methyl 7-((1R,2S,3R,5R)-2-(4-tert-butylphenyl)-5-chloro-3-hydroxycyclopentyl)hept-5-enoate
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C23H33ClO3
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1
|
1 |
EC50 > 10000 nM
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CP0852830
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methyl 7-((1R,2S,3R,5R)-2-(4-tert-butylphenyl)-5-chloro-3-hydroxycyclopentyl)heptanoate
Show/Hide
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C23H35ClO3
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1
|
1 |
EC50 > 10000 nM
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|
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CP0852841
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methyl 7-((1R,2S,3R)-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)heptanoate
Show/Hide
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C27H40O5
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1
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1 |
EC50 > 10000 nM
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|
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CP0856820
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7-((1R,2S,3R)-3-hydroxy-2-(4-(1-hydroxycyclobutyl)phenyl)-5-oxocyclopentyl)heptanoic acid
Show/Hide
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C22H30O5
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1
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1 |
EC50 > 10000 nM
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|
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CP0856822
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methyl 7-((1R,2S,3R)-3-hydroxy-5-oxo-2-p-tolylcyclopentyl)heptanoate
Show/Hide
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C20H28O4
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1
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1 |
EC50 > 10000 nM
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|
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CP0863084
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methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)cyclopentyl)hept-5-enoate
Show/Hide
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C27H39ClO4
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1
|
1 |
EC50 > 10000 nM
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|
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CP0863766
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methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxycyclobutyl)phenyl)cyclopentyl)hept-5-enoate
Show/Hide
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C23H31ClO4
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1
|
1 |
EC50 > 10000 nM
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|
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CP0866245
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7-((1R,2S)-2-(4-((R)-hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
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C26H36O4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0866247
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methyl 7-((1R,2S)-2-(4-((R)-cyclohexyl(hydroxy)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoate
Show/Hide
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C26H36O4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0866253
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N-ethyl-7-((1R,2S,3R)-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)hept-5-enamide
Show/Hide
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C26H37NO4
|
1
|
1 |
EC50 > 10000 nM
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CP0866291
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7-((1R,2S,3R)-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxy-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
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C25H34O5
|
1
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1 |
EC50 > 10000 nM
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|
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CP0866292
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methyl 7-((1R,2S,3R)-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxy-5-oxocyclopentyl)heptanoate
Show/Hide
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C26H38O5
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0866303
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7-((1R,2S,3R)-3-hydroxy-2-(4-(1-hydroxycyclobutyl)phenyl)-5-oxocyclopentyl)hept-5-enoic acid
Show/Hide
|
C22H28O5
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0866394
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methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropan-2-yl)phenyl)cyclopentyl)hept-5-enoate
Show/Hide
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C23H33ClO4
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2
|
1 |
EC50 > 10000 nM
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2 |
IC50 = 48765 nM
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CP0866430
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methyl 7-((1R,2S,3R)-2-(4-tert-butylphenyl)-3-hydroxy-5-oxocyclopentyl)hept-5-enoate
Show/Hide
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C23H32O4
|
1
|
1 |
EC50 > 10000 nM
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CP0870436
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methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxycyclobutyl)phenyl)cyclopentyl)heptanoate
Show/Hide
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C23H33ClO4
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1
|
1 |
EC50 > 10000 nM
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|
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CP0882892
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methyl 7-((1R,2S,3R)-2-(2,3-dihydro-1H-inden-5-yl)-3-hydroxy-5-oxocyclopentyl)heptanoate
Show/Hide
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C22H30O4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0883084
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5-[(R)-1-(4-tert-Butyl-phenyl)-5-oxo-pyrrolidin-2-ylmethoxy]-pentanoic acid
Show/Hide
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C20H29NO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0888283
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(hydroxymethyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C19H27ClO4
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1
|
1 |
EC50 > 10000 nM
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|
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CP0888287
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7-((1R,2S)-2-(4-(1-hydroxycyclobutyl)phenyl)-5-oxocyclopentyl)heptanoic acid
Show/Hide
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C22H30O4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0888294
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methyl 7-((1R,2S,3R)-3-hydroxy-2-(3-(hydroxy(1-propylcyclobutyl)methyl)phenyl)-5-oxocyclopentyl)hept-5-enoate
Show/Hide
|
C27H38O5
|
1
|
1 |
EC50 > 10000 nM
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|
|
CP0888316
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methyl 7-((1R,2S)-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-5-oxocyclopentyl)heptanoate
Show/Hide
|
C26H38O4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0899422
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methyl 7-((1R,2S,3R)-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxy-5-oxocyclopentyl)hept-5-enoate
Show/Hide
|
C26H36O5
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0900747
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C22H33ClO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0920861
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methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(hydroxymethyl)phenyl)cyclopentyl)hept-5-enoate
Show/Hide
|
C20H27ClO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0920862
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methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropyl)phenyl)cyclopentyl)hept-5-enoate
Show/Hide
|
C23H33ClO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0928827
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methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropan-2-yl)phenyl)cyclopentyl)heptanoate
Show/Hide
|
C23H35ClO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0966505
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methyl 7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropyl)phenyl)cyclopentyl)heptanoate
Show/Hide
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C23H35ClO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0420325
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4-[2-[3,5-dichloro-2-[(E)-3-hydroxyoct-1-enyl]-6-oxopyridin-1-yl]ethyl]benzoic acid
Show/Hide
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C22H25Cl2NO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0437306
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7-[2-(3-hydroxyoctyl)-6-oxopyridin-1-yl]heptanoic acid
Show/Hide
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C20H33NO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0487510
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7-[3,5-dibromo-2-[(E)-3-hydroxyoct-1-enyl]-6-oxopyridin-1-yl]heptanoic acid
Show/Hide
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C20H29Br2NO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0525833
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7-[3,5-dichloro-2-[(E)-3-hydroxyoct-1-enyl]-6-oxopyridin-1-yl]heptanoic acid
Show/Hide
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C20H29Cl2NO4
|
1
|
1 |
EC50 > 10000 nM
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|
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CP0852856
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methyl 7-((1R,2R,5S)-2-chloro-5-(4-(1-hydroxypentyl)phenyl)cyclopentyl)heptanoate
Show/Hide
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C24H37ClO3
|
2
|
1 |
EC50 = 15000 nM
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|
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2 |
Ki = 15000 nM
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CP0863699
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methyl 7-((1R,2S)-2-(4-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)hept-5-enoate
Show/Hide
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C25H36O4
|
2
|
1 |
EC50 = 15000 nM
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|
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2 |
Ki = 15000 nM
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CP0867160
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methyl 7-((1R,2S)-2-(4-(2-hydroxyhexyl)phenyl)-5-oxocyclopentyl)heptanoate
Show/Hide
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C25H38O4
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2
|
1 |
EC50 = 15000 nM
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|
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2 |
Ki = 4600 nM
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CP0926161
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7-((1R,2R,5S)-2-fluoro-5-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C24H37FO3
|
2
|
1 |
EC50 = 15000 nM
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|
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2 |
Ki = 600 nM
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CP0947233
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7-((1R,2R,5S)-2-chloro-5-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)heptanoic acid
Show/Hide
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C24H37ClO3
|
2
|
1 |
EC50 = 15000 nM
|
|
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2 |
Ki = 1900 nM
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CP0867141
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2-(4-((1R,2S,3R,5R)-5-chloro-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-3-hydroxycyclopentyl)butoxy)acetic acid
Show/Hide
|
C24H35ClO5
|
1
|
1 |
EC50 = 20773 nM
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|
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CP0893966
|
7-((1R,2R,5S)-2-chloro-5-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)heptan-1-ol
Show/Hide
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C24H39ClO2
|
2
|
1 |
EC50 = 50000 nM
|
|
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2 |
Ki = 50000 nM
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CP0921737
|
methyl 7-((5S)-5-(4-(1-hydroxyhexyl)phenyl)cyclopent-1-enyl)heptanoate
Show/Hide
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C25H38O3
|
2
|
1 |
EC50 = 50000 nM
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|
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2 |
Ki = 50000 nM
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CP0926160
|
methyl 7-((1R,2S)-2-(3-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)heptanoate
Show/Hide
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C25H38O4
|
2
|
1 |
EC50 = 50000 nM
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|
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2 |
Ki = 50000 nM
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CP0930472
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7-((1R,2S)-2-(3-(1-hydroxyhexyl)phenyl)-5-oxocyclopentyl)heptanoic acid
Show/Hide
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C24H36O4
|
2
|
1 |
EC50 = 50000 nM
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|
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2 |
Ki = 15000 nM
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CP0942915
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methyl 7-((1R,2R,5S)-2-fluoro-5-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)heptanoate
Show/Hide
|
C25H39FO3
|
2
|
1 |
EC50 = 50000 nM
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|
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2 |
Ki = 50000 nM
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CP0942917
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methyl 7-((1R,2R,5S)-2-chloro-5-(4-(1-hydroxyhexyl)phenyl)cyclopentyl)heptanoate
Show/Hide
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C25H39ClO3
|
2
|
1 |
EC50 = 50000 nM
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|
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2 |
Ki = 50000 nM
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CP0866760
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(1-hydroxy-2-methylpropan-2-yl)phenyl)cyclopentyl)hept-5-enoic acid
Show/Hide
|
C22H31ClO4
|
2
|
1 |
EC50 >= 173 nM
|
|
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2 |
IC50 = 4185 nM
|
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CP0394028
|
2-[[4-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
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C24H29ClN4O4S
|
1
|
1 |
EC50 > 1000 nM
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|
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CP0394030
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2-[[2-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]pyridin-4-yl]amino]acetic acid;hydrochloride
Show/Hide
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C24H29ClN4O4S
|
1
|
1 |
EC50 > 1000 nM
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|
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CP0468699
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2-[6-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]indol-1-yl]acetic acid;2,2,2-trifluoroacetic acid
Show/Hide
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C29H30F3N3O6S
|
1
|
1 |
EC50 > 1000 nM
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|
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CP0538159
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2-[[6-[[(4-tert-butylphenyl)methyl-(2-chlorophenyl)sulfonylamino]methyl]pyridin-2-yl]amino]acetic acid;hydrochloride
Show/Hide
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C25H29Cl2N3O4S
|
1
|
1 |
EC50 > 1000 nM
|
|
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CP0882894
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7-((1R,2S)-2-(4-(cyclohexyl(hydroxy)methyl)phenyl)-5-oxocyclopentyl)heptanoic acid
Show/Hide
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C25H36O4
|
1
|
1 |
EC50 >= 2047 nM
|
|
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CP0087804
|
ACT-129968
Show/Hide
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C24H19FN2O3
|
1
|
1 |
IC50 = 2600 nM
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|
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CP0156868
|
2-[6-chloro-8-fluoro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C24H18ClFN2O3
|
1
|
1 |
IC50 = 2700 nM
|
|
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CP0440482
|
De-117
Show/Hide
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C26H28N6O4S
|
1
|
1 |
IC50 = 4180 nM
|
|
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CP0471861
|
6-bromo-3-methyl-N-(2-pyridin-3-ylethyl)-2-thiophen-2-ylquinoline-4-carboxamide
Show/Hide
|
C22H18BrN3OS
|
1
|
1 |
IC50 = 4400 nM
|
|
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CP0042409
|
2-[2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C28H26N2O3
|
1
|
1 |
IC50 = 6400 nM
|
|
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CP0055416
|
2-[2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C24H20N2O3
|
1
|
1 |
IC50 = 6600 nM
|
|
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CP0042410
|
2-[8-chloro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C24H19ClN2O3
|
1
|
1 |
IC50 = 7400 nM
|
|
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CP0083568
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2-[8-fluoro-2-(3-naphthalen-1-ylpropanoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C26H23FN2O3
|
1
|
1 |
IC50 = 9500 nM
|
|
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CP0045673
|
2-[2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H16ClFN2O3
|
1
|
1 |
IC50 > 10000 nM
|
|
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CP0055418
|
2-[6-chloro-2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H15Cl2FN2O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0055420
|
2-[2-(3-chlorobenzoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H17ClN2O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0055873
|
2-[8-fluoro-2-[2-(1H-indol-3-yl)acetyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C23H20FN3O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0055874
|
2-[8-fluoro-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C18H15FN2O3S
|
1
|
1 |
IC50 > 10000 nM
|
|
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CP0055877
|
2-[2-benzoyl-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C21H17F3N2O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0070143
|
2-(2-benzoyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C20H18N2O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0086399
|
2-[6-chloro-2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C28H25ClN2O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0086409
|
2-[8-fluoro-2-(2-naphthalen-1-ylacetyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C25H21FN2O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0130562
|
2-[8-methyl-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C25H22N2O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0261961
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2-[2-(naphthalene-1-carbonyl)-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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C25H19F3N2O3
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1
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1 |
IC50 > 10000 nM
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CP0272414
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US11149018, Example 34
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C26H27BrClN3O3
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1
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1 |
IC50 > 10000 nM
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CP0863769
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7-((1R,2S,3R,5R)-5-chloro-3-hydroxy-2-(4-(hydroxymethyl)phenyl)cyclopentyl)hept-5-enoic acid
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C19H25ClO4
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1
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1 |
IC50 = 13150 nM
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CP0060087
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4-[(1S)-1-[[3-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzoxepine-10-carbonyl]amino]ethyl]benzoic acid
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C25H20F3NO4
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1
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1 |
IC50 > 1000 nM
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CP0060088
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4-[1-[[2-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzoxepine-10-carbonyl]amino]cyclopropyl]benzoic acid
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C26H20F3NO4
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1
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1 |
IC50 > 1000 nM
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CP0060089
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4-[1-[[3-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzoxepine-10-carbonyl]amino]cyclopropyl]benzoic acid
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C26H20F3NO4
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1
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1 |
IC50 > 1000 nM
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CP0091346
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4-[(1S)-1-[[2-(trifluoromethyl)-5,6-dihydrobenzo[b][1]benzoxepine-10-carbonyl]amino]ethyl]benzoic acid
Show/Hide
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C25H20F3NO4
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1
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1 |
IC50 > 1000 nM
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CP0092571
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4-[(1S)-1-[[5-chloro-2-(4-fluorophenoxy)benzoyl]amino]ethyl]benzoic acid
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C22H17ClFNO4
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1
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1 |
IC50 > 1000 nM
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CP0443957
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4-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]-1-benzofuran-2-carboxylic acid
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C26H26N2O5S
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1
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1 |
Ki = 15 nM
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CP0536164
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4-(2-((R)-2-(4-(cyclopentylmethyl)penta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
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C24H31NO3
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1
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1 |
Ki = 60 nM
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CP0343798
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2-[(3R)-4-[(4-chlorophenyl)methyl]-7-fluoro-5-methylsulfonyl-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acid
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C21H19ClFNO4S
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1
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1 |
Ki = 136 nM
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CP0441655
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4-[3-(2-Benzyloxy-phenyl)-propyl]-benzoic acid
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C23H22O3
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1
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1 |
Ki = 150 nM
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CP0457560
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4-(2-((R)-2-(4-methylhexa-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
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C20H25NO3
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1
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1 |
Ki = 173 nM
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CP0108218
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(R)-2-(4-(4-chlorobenzyl)-5-acetyl-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid
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C23H22ClNO5S
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1
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1 |
Ki = 230 nM
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CP0422463
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1-(2,6-dimethoxyphenyl)-N-[[3-methyl-4-[6-oxo-5,9-bis(2,2,2-trifluoroethoxy)-8H-pyrrolo[3,4-g]quinolin-7-yl]phenyl]methylsulfonyl]cyclopropane-1-carboxamide
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C35H31F6N3O8S
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1
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1 |
Ki = 300 nM
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CP0372074
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2-[(3R)-5-acetyl-4-[(4-chlorophenyl)methyl]-7-fluoro-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acid
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C22H19ClFNO3
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1
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1 |
Ki = 310 nM
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CP0426597
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US9180116, 9C
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C19H31F2NO4
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1
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1 |
Ki = 329 nM
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CP0041889
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2-((R)-4-(4-chlorobenzyl)-5-(1-hydroxyethyl)-7-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid
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C23H24ClNO5S
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1
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1 |
Ki = 390 nM
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CP0374187
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2-[(3R)-5-bromo-4-[(4-chlorophenyl)methyl]-7-fluoro-2,3-dihydro-1H-cyclopenta[b]indol-3-yl]acetic acid
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C20H16BrClFNO2
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1
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1 |
Ki = 410 nM
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CP0574605
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6-[[(4-tert-butylphenyl)methyl-pyridin-3-ylsulfonylamino]methyl]-1-benzofuran-2-carboxylic acid
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C26H26N2O5S
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1
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1 |
Ki = 433 nM
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CP0112284
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CHEMBL3933704
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C23H26FNO5
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1
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1 |
Ki = 570 nM
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CP0112283
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APD-811
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C23H26ClNO5
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1
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1 |
Ki = 610 nM
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CP0457558
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4-[2-[(2R)-2-[(1Z,3E)-3-methylocta-1,3-dienyl]-5-oxopyrrolidin-1-yl]ethyl]benzoic acid
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C22H29NO3
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1
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1 |
Ki = 802 nM
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CP0496137
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(E)-3-(2-Benzyloxy-[1,1';3',1'']terphenyl-2''-yl)-acrylic acid
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C28H22O3
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1
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1 |
Ki = 830 nM
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CP0847235
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5-((E/Z)-3-{(R)-1-[4-(1-Hydroxy-hexyl)-phenyl]-5-oxo-pyrrolidin-2-yl}-allyl)-thiophene-2-carboxylic acid
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C24H29NO4S
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1
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1 |
Ki = 1382 nM
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CP0144553
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7-[(R)-2-((E)-(S)-3-Hydroxy-oct-1-enyl)-5-oxo-pyrrolidin-1-yl]-heptanoic acid
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C19H33NO4
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1
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1 |
Ki = 1459 nM
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CP0404585
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3-[2-[3-(2-phenylmethoxyphenyl)phenyl]phenyl]-N-thiophen-2-ylsulfonylpropanamide
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C32H27NO4S2
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1
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1 |
Ki = 1600 nM
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CP0464526
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(R)-4-(2-(2-(4-methylpenta-1,3-dienyl)-5-oxopyrrolidin-1-yl)ethyl)benzoic acid
Show/Hide
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C19H23NO3
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1
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1 |
Ki = 1850 nM
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CP0393748
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N-[[4-(5,9-diethoxy-6-oxo-8H-pyrrolo[3,4-g]quinolin-7-yl)-3-methylphenyl]methylsulfonyl]-2-(2-methoxyphenyl)acetamide
Show/Hide
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C32H33N3O7S
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1
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1 |
Ki = 1900 nM
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CP0181173
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2-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl}-cyclopropanecarboxylic acid
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C27H22O3S
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1
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1 |
Ki = 2300 nM
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CP0381724
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3-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl}-propionic acid
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C26H22O3S
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1
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1 |
Ki = 2500 nM
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CP0466746
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2-[2-[5-(2-phenylmethoxyphenyl)thiophen-3-yl]anilino]acetic acid
Show/Hide
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C25H21NO3S
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1
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1 |
Ki = 2500 nM
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CP0404232
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3-(2-Phenoxymethyl-[1,1';3',1'']terphenyl-2''-yl)-propionic acid
Show/Hide
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C28H24O3
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1
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1 |
Ki = 2900 nM
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CP0424293
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3-{2-[4-(2-Benzyloxy-phenyl)-thiophen-2-yl]-phenyl}-propionic acid
Show/Hide
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C26H22O3S
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1
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1 |
Ki = 2900 nM
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CP0437614
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4-(2-Benzyloxy-[1,1';3',1'']terphenyl-2''-yl)-butyric acid
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C29H26O3
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1
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1 |
Ki = 3500 nM
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CP0406374
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3-(2''-Benzyloxy-[1,1';3',1'']terphenyl-2-yl)-2-methyl-propionic acid
Show/Hide
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C29H26O3
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1
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1 |
Ki = 3600 nM
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CP0441093
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(2''-Benzyloxy-[1,1';3',1'']terphenyl-2-yl)-acetic acid
Show/Hide
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C27H22O3
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1
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1 |
Ki = 3600 nM
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CP0436538
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3-(2-Benzyloxy-[1,1';3',1'']terphenyl-2''-yl)-propionic acid
Show/Hide
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C28H24O3
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1
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1 |
Ki = 3700 nM
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CP0466770
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3-{2-[5-(2-Benzyloxy-phenyl)-thiophen-2-yl]-phenyl}-propionic acid
Show/Hide
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C26H22O3S
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1
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1 |
Ki = 4100 nM
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CP0372972
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3-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl}-butyric acid
Show/Hide
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C27H24O3S
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1
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1 |
Ki = 4600 nM
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CP0404532
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3-[2''-(2,6-Dichloro-benzyloxy)-[1,1';3',1'']terphenyl-2-yl]-propionic acid
Show/Hide
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C28H22Cl2O3
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1
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1 |
Ki = 4600 nM
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CP0426640
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US9180116, 2C
Show/Hide
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C21H31F2NO4
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1
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1 |
Ki = 4971 nM
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CP0430206
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3-{2-[5-(2-Benzyloxy-phenyl)-thiophen-3-yl]-phenyl}-2-methyl-propionic acid
Show/Hide
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C27H24O3S
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1
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1 |
Ki = 5500 nM
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CP0415118
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(E)-3-(3',4'-Dichloro-biphenyl-2-yl)-acrylic acid
Show/Hide
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C15H10Cl2O2
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1
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1 |
Ki = 7500 nM
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CP0277044
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(E)-3-{2-[(E)-3-(2-Benzyloxy-3-methyl-phenyl)-allyl]-phenyl}-acrylic acid
Show/Hide
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C26H24O3
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1
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1 |
Ki = 8100 nM
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CP0381706
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3-[1,1';3',1'']Terphenyl-2-yl-propionic acid
Show/Hide
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C21H18O2
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1
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1 |
Ki = 8100 nM
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CP0160939
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(E)-3-[2-(3,4-dichlorophenyl)phenyl]-N-thiophen-2-ylsulfonylprop-2-enamide
Show/Hide
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C19H13Cl2NO3S2
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1
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1 |
Ki = 10000 nM
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CP0417632
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7-[(2R)-2-[(E,3S,4S)-3-hydroxy-4-methylnon-1-en-6-ynyl]-5-oxopyrrolidin-1-yl]heptanoic acid
Show/Hide
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C21H33NO4
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1
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1 |
Ki = 12173 nM
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CP0388282
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2-(4-(4-(butylcarbamoyl)-2-(2,4-dichlorophenylsulfonamido)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
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C26H26Cl2N2O7S
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1
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1 |
Ki = 44000 nM
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CP0404233
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3-(4''-Benzyloxy-[1,1';3',1'']terphenyl-2-yl)-propionic acid
Show/Hide
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C28H24O3
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1
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1 |
Ki > 97000 nM
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