Brief Information of the Compound and Protein
| Compound Name |
2-[3-[3-[[2-chloro-3-(trifluoromethyl)phenyl]methyl-[2,2-di(phenyl)ethyl]amino]propoxy]phenyl]acetic acid
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
Oxysterols receptor LXR-beta
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Protein Classification |
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group H
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Nuclear hormone receptor subfamily 1 group H member 3
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| Uniprot ID | Gene Name | NR1H2 |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Biochemical Assays
| 1 | EC50 = 4 nM | ||
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| 2 | EC50 = 5 nM | ||
| 3 | EC50 = 20 nM | ||
| 4 | EC50 = 40 nM | ||
| 5 | EC50 = 78 nM | ||
| 6 | EC50 = 390 nM | ||
| 7 | EC50 = 400 nM | ||
| 8 | IC50 = 7.943 nM | ||
| 9 | IC50 = 12 nM | ||
| 10 | IC50 = 30 nM | ||