Brief Information of the Compound and Protein
| Compound Name |
1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piperidine
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
Histamine H3 receptor
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Protein Classification |
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
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| Uniprot ID | Gene Name | HRH3 |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Biochemical Assays
| 1 | IC50 = 0.53 nM | ||
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| 2 | Kd = 0.1445 nM | ||
| 3 | Ki = 0.2754 nM | ||
| 4 | Ki = 0.5754 nM | ||
| 5 | Ki = 0.6 nM | ||
| 6 | Ki = 0.97 nM | ||
| 7 | Ki = 1 nM | ||
| 8 | Ki = 9.24 nM | ||