General Information of the Protein
Protein ID
PT05219
Protein Name
P2Y purinoceptor 4
Secondarily
Protein Name
P2P
Uridine nucleotide receptor
Gene Name
P2RY4
Secondarily
Gene Name
NRU
Sequence
MASTESSLLRSLGLSPGPGSSEVELDCWFDEDFKFILLPVSYAVVFVLGLGLNAPTLWLFIFRLRPWDATATYMFHLALSDTLYVLSLPTLIYYYAAHNHWPFGTEICKFVRFLFYWNLYCSVLFLTCISVHRYLGICHPLRALRWGRPRLAGLLCLAVWLVVAGCLVPNLFFVTTSNKGTTVLCHDTTRPEEFDHYVHFSSAVMGLLFGVPCLVTLVCYGLMARRLYQPLPGSAQSSSRLRSLRTIAVVLTVFAVCFVPFHITRTIYYLARLLEADCRVLNIVNVVYKVTRPLASANSCLDPVLYLLTGDKYRRQLRQLCGGGKPQPRTAASSLALVSLPEDSSCRWAATPQDSSCSTPRADRL
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Organism
Homo sapiens, Human
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Nucleotide-like receptor (family A GPCR)
>
Purine receptor
Function
Receptor for UTP and UDP coupled to G-proteins that activate a phosphatidylinositol-calcium second messenger system. Not activated by ATP or ADP.
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Uniprot ID
Primary ID:
P51582

Secondarily ID:
Q4VBB7
Q4VBB8
Q502W2
Q5JT22
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Ensembl ID
ENSG00000186912
HGNC ID
HGNC:8542
Subcellular Location
Cell membrane
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000094 , 1321N1
Compound ID Compound Name Compound Formula
CP0464732
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(3-thiophen-3-ylpropoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C16H24N3O15P3S
 1
1
EC50 = 20 nM
   TI
   LI
   LO
   TS
CP0460363
((2R,3S,4R,5R)-3,4-dihydroxy-5-(2-oxo-4-thioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-2-yl)methyl triphosphate
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C9H15N2O14P3S
 1
1
EC50 = 23 nM
   TI
   LI
   LO
   TS
CP0494118
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(3-phenylpropoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C18H26N3O15P3
 1
1
EC50 = 23 nM
   TI
   LI
   LO
   TS
CP0464730
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-[3-(4-methoxyphenyl)propoxyamino]-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C19H28N3O16P3
 1
1
EC50 = 23 nM
   TI
   LI
   LO
   TS
CP0440668
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C10H18N3O15P3
 1
1
EC50 = 25 nM
   TI
   LI
   LO
   TS
CP0382300
[[(2R,3S,4R,5R)-5-[4-[3-[4-[2-(but-3-ynylamino)-2-oxoethoxy]phenyl]propoxyamino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C24H33N4O17P3
 1
1
EC50 = 40 nM
   TI
   LI
   LO
   TS
CP0401596
[[(2R,3S,4R,5R)-5-[4-[(3-cyano-3,3-diphenylpropoxy)amino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C25H29N4O15P3
 1
1
EC50 = 47 nM
   TI
   LI
   LO
   TS
CP0844899
N4-Methoxycytidine 5'-Triphosphate triethylammonium Salt
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C16H33N4O15P3
 1
1
EC50 = 50 nM
   TI
   LI
   LO
   TS
CP0487206
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(4-phenylbutoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C19H28N3O15P3
 1
1
EC50 = 54 nM
   TI
   LI
   LO
   TS
CP0503203
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4S,5R,6R)-4-fluoro-3,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
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C15H25FN2O22P4
 1
1
EC50 = 62 nM
   TI
   LI
   LO
   TS
CP0382361
[[(2R,3S,4R,5R)-5-[4-[3-[4-[2-[2-[1-[3-[6-[[2-[4-[(E)-2-(2,2-difluoro-12-thiophen-2-yl-3-aza-1-azonia-2-boranuidatricyclo[7.3.0.03,7]dodeca-1(12),4,6,8,10-pentaen-4-yl)ethenyl]phenoxy]acetyl]amino]hexanoylamino]propyl]triazol-4-yl]ethylamino]-2-oxoethoxy]phenyl]propoxyamino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C56H67BF2N11O20P3S
 1
1
EC50 = 70 nM
   TI
   LI
   LO
   TS
CP0133127
5'-UTP
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C9H15N2O15P3
 9
1
EC50 = 73 nM
   TI
   LI
   LO
   TS
2
EC50 = 80 nM
   TI
   LI
   LO
   TS
3
EC50 = 87 nM
   TI
   LI
   LO
   TS
4
EC50 = 88.4 nM
   TI
   LI
   LO
   TS
5
EC50 = 90 nM
   TI
   LI
   LO
   TS
6
EC50 = 100 nM
   TI
   LI
   LO
   TS
7
EC50 = 480 nM
   TI
   LI
   LO
   TS
8
EC50 = 500 nM
   TI
   LI
   LO
   TS
9
EC50 = 900 nM
   TI
   LI
   LO
   TS
CP0473567
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(2-phenylethoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C17H24N3O15P3
 1
1
EC50 = 73 nM
   TI
   LI
   LO
   TS
CP0525923
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-(2-oxo-4-sulfanylidenepyrimidin-1-yl)oxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4R,5R)-3,4-dihydroxy-5-(2-oxo-4-sulfanylidenepyrimidin-1-yl)oxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
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C18H26N4O21P4S2
 1
1
EC50 = 80 nM
   TI
   LI
   LO
   TS
CP0382306
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-[3-(4-nitrophenyl)propoxyamino]-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C18H25N4O17P3
 1
1
EC50 = 84 nM
   TI
   LI
   LO
   TS
CP0406773
((1S,2S,4S,5S)-4-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-2-hydroxybicyclo[3.1.0]hexan-1-yl)methyl tetrahydrogen triphosphate
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C11H17N2O13P3
 1
1
EC50 = 85 nM
   TI
   LI
   LO
   TS
CP0415529
[dichloro-[[[(2R,3S,4R,5R)-3,4-dihydroxy-5-(4-oxo-2-sulfanylidenepyrimidin-1-yl)oxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]methyl]phosphonic acid
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C10H15Cl2N2O13P3S
 2
1
EC50 = 90 nM
   TI
   LI
   LO
   TS
2
EC50 = 3850 nM
   TI
   LI
   LO
   TS
CP0473872
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-[3-(4-iodophenyl)propoxyamino]-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C18H25IN3O15P3
 1
1
EC50 = 91 nM
   TI
   LI
   LO
   TS
CP0473875
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(3-phenylpropoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
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C27H37N5O23P4
 1
1
EC50 = 93 nM
   TI
   LI
   LO
   TS
CP0499369
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-[3-(3-nitrophenyl)propoxyamino]-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C18H25N4O17P3
 1
1
EC50 = 95 nM
   TI
   LI
   LO
   TS
CP0401584
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(phenylmethoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C16H22N3O15P3
 1
1
EC50 = 97 nM
   TI
   LI
   LO
   TS
CP0524488
[[(2R,3S,4R,5R)-5-[4-[3-(3-fluorophenyl)propoxyamino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C18H25FN3O15P3
 1
1
EC50 = 100 nM
   TI
   LI
   LO
   TS
CP0487207
[[(2R,3S,4R,5R)-5-[4-[3-(4-fluorophenyl)propoxyamino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C18H25FN3O15P3
 1
1
EC50 = 105 nM
   TI
   LI
   LO
   TS
CP0473870
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-[3-(3-iodophenyl)propoxyamino]-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C18H25IN3O15P3
 1
1
EC50 = 114 nM
   TI
   LI
   LO
   TS
CP0401539
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-(3-naphthalen-2-ylpropoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
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C22H28N3O15P3
 1
1
EC50 = 128 nM
   TI
   LI
   LO
   TS
CP0170354
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
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C18H26N4O23P4
 1
1
EC50 = 130 nM
   TI
   LI
   LO
   TS
CP0826611
Diquafosol
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C18H22N4Na4O23P4
 1
1
EC50 = 130 nM
   TI
   LI
   LO
   TS
CP0439410
[[(2R,3S,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C18H27N5O21P4
 1
1
EC50 = 140 nM
   TI
   LI
   LO
   TS
CP0524489
[[(2R,3S,4R,5R)-5-[4-[3-(4-bromophenyl)propoxyamino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C18H25BrN3O15P3
 1
1
EC50 = 141 nM
   TI
   LI
   LO
   TS
CP0852224
N4-Ethoxycytidine 5'-Diphosphate triethylAmmonium Salt
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C17H34N4O12P2
 1
1
EC50 = 180 nM
   TI
   LI
   LO
   TS
CP0390701
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[(2R,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H26N2O23P4
 1
1
EC50 = 183 nM
   TI
   LI
   LO
   TS
CP0382301
3-amino-9-[2-carboxy-4-[6-[4-[2-[[2-[4-[3-[[1-[(2R,3R,4S,5R)-3,4-dihydroxy-5-[[hydroxy-[hydroxy(phosphonooxy)phosphoryl]oxyphosphoryl]oxymethyl]oxolan-2-yl]-2-oxopyrimidin-4-yl]amino]oxypropyl]phenoxy]acetyl]amino]ethyl]triazol-1-yl]hexylcarbamoyl]phenyl]-6-iminoxanthene-4,5-disulfonate;triethylazanium
   Show/Hide
C51H57N10O27P3S2-2
 1
1
EC50 = 200 nM
   TI
   LI
   LO
   TS
CP0441701
[[(2R,3S,4R,5R)-5-[4-(ethoxyamino)-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C11H20N3O15P3
 1
1
EC50 = 210 nM
   TI
   LI
   LO
   TS
CP0520896
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3R,4R,5S,6R)-5-fluoro-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H25FN2O22P4
 1
1
EC50 = 220 nM
   TI
   LI
   LO
   TS
CP0375621
(2S,3S,4S,5R,6R)-6-[[[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-3,4,5-trihydroxyoxane-2-carboxylic acid
   Show/Hide
C15H24N2O24P4
 1
1
EC50 = 227 nM
   TI
   LI
   LO
   TS
CP0412775
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(3-pyridin-4-ylpropoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C17H25N4O15P3
 1
1
EC50 = 250 nM
   TI
   LI
   LO
   TS
CP0465710
4-Thio-uridine-5'-tetraphosphate
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C9H16N2O17P4S
 1
1
EC50 = 280 nM
   TI
   LI
   LO
   TS
CP0889562
(S)-Methanocarbauridine5'-Triphosphate Triethylammonium salt
   Show/Hide
C17H32N3O14P3
 1
1
EC50 = 300 nM
   TI
   LI
   LO
   TS
CP0499368
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(3-pyridin-3-ylpropoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C17H25N4O15P3
 1
1
EC50 = 300 nM
   TI
   LI
   LO
   TS
CP0473562
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4S,5R,6R)-4-fluoro-3,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C16H28FN3O22P4
 1
1
EC50 = 310 nM
   TI
   LI
   LO
   TS
CP0382357
2-thio-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-dione 5'-triphosphate
   Show/Hide
C9H15N2O14P3S
 2
1
EC50 = 350 nM
   TI
   LI
   LO
   TS
2
EC50 = 1770 nM
   TI
   LI
   LO
   TS
CP0541754
[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-[(3-iodophenyl)methoxyamino]-2-oxopyrimidin-1-yl]oxolan-2-yl]methyl phosphono hydrogen phosphate
   Show/Hide
C16H20IN3O12P2
 1
1
EC50 = 352 nM
   TI
   LI
   LO
   TS
CP0375237
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2S,3R,4S,5S)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C18H26N4O23P4
 1
1
EC50 = 400 nM
   TI
   LI
   LO
   TS
CP0382360
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(pent-4-ynoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C14H22N3O15P3
 1
1
EC50 = 410 nM
   TI
   LI
   LO
   TS
CP0488193
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(2-phenoxyethoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C17H24N3O16P3
 1
1
EC50 = 430 nM
   TI
   LI
   LO
   TS
CP0382305
4-[[1-[(2R,3R,4S,5R)-3,4-dihydroxy-5-[[hydroxy-[hydroxy(phosphonooxy)phosphoryl]oxyphosphoryl]oxymethyl]oxolan-2-yl]-2-oxopyrimidin-4-yl]amino]oxybutanoic acid
   Show/Hide
C13H22N3O17P3
 1
1
EC50 = 470 nM
   TI
   LI
   LO
   TS
CP0485934
[[(2R,3S,5R)-5-(2-amino-6-oxo-1H-purin-9-yl)-3-hydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C19H27N7O21P4
 1
1
EC50 = 540 nM
   TI
   LI
   LO
   TS
CP0388696
((((2R,3S,4R,5R)-3,4-dihydroxy-5-((E)-4-(methoxyimino)-2-oxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-2-yl)methoxy)(hydroxy)phosphoryl)methylphosphonic(((2R,3S,4R,5R)-3,4-dihydroxy-5-(4-(methoxyamino)-2-oxopyrimidin-1(2H)-yl)tetrahydrofuran-2-yl)methyl phosphoric)anhydride
   Show/Hide
C20H31N6O20P3
 1
1
EC50 = 560 nM
   TI
   LI
   LO
   TS
CP0421613
((2R,3S,4R,5R)-5-(5-fluoro-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl tetrahydrogen triphosphate
   Show/Hide
C9H14FN2O15P3
 1
1
EC50 = 600 nM
   TI
   LI
   LO
   TS
CP0441715
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[(2R,3R,4S,5R)-3,4,5-trihydroxyoxan-2-yl]oxyphosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C14H24N2O22P4
 1
1
EC50 = 620 nM
   TI
   LI
   LO
   TS
CP0401583
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(phenylmethoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C25H32N5O20P3
 1
1
EC50 = 636 nM
   TI
   LI
   LO
   TS
CP0375615
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(phenylmethoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4S,5R,6R)-4-fluoro-3,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C22H32FN3O22P4
 1
1
EC50 = 670 nM
   TI
   LI
   LO
   TS
CP0463240
[[(2R,3S,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4R,5R)-3,4-dihydroxy-5-(4-oxo-2-sulfanylidenepyrimidin-1-yl)oxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C18H27N5O20P4S
 1
1
EC50 = 710 nM
   TI
   LI
   LO
   TS
CP0866902
P1-Uridine5'-P3-Cyclohexyltriphosphate Triethylammonium salt
   Show/Hide
C25H43N6O20P3
 1
1
EC50 = 790 nM
   TI
   LI
   LO
   TS
CP0418143
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-(methoxyamino)-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C19H28N5O20P3
 1
1
EC50 = 790 nM
   TI
   LI
   LO
   TS
CP0401582
bis[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C18H25N4O20P3
 1
1
EC50 = 870 nM
   TI
   LI
   LO
   TS
CP0473549
[(2R,3R,4R,5S,6R)-3-acetamido-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl] [[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C17H29N3O23P4
 1
1
EC50 = 910 nM
   TI
   LI
   LO
   TS
CP0562508
[(2R,3S,4R,5R)-5-[4-[(3-hexa-1,5-diynylphenyl)methoxyamino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methyl phosphono hydrogen phosphate
   Show/Hide
C22H25N3O12P2
 1
1
EC50 = 952 nM
   TI
   LI
   LO
   TS
CP0515397
[2,3-dihydroxypropoxy(hydroxy)phosphoryl] [[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C12H22N2O20P4
 1
1
EC50 = 1120 nM
   TI
   LI
   LO
   TS
CP0852222
N4-Benzyloxycytidine 5'-Diphosphate triethylammonium Salt
   Show/Hide
C22H36N4O12P2
 1
1
EC50 = 1150 nM
   TI
   LI
   LO
   TS
CP0435254
[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(phenylmethoxyamino)pyrimidin-1-yl]oxolan-2-yl]methyl phosphono hydrogen phosphate
   Show/Hide
C16H21N3O12P2
 1
1
EC50 = 1150 nM
   TI
   LI
   LO
   TS
CP0415558
({[({[(2R,3S,4R,5R)-4-amino-5-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy](hydroxy)phosphoryl}oxy)phosphonic acid
   Show/Hide
C9H16N3O14P3
 1
1
EC50 = 1200 nM
   TI
   LI
   LO
   TS
CP0064491
2'-C-Methyl-uridine-5'-triphosphate
   Show/Hide
C10H17N2O15P3
 1
1
EC50 = 1260 nM
   TI
   LI
   LO
   TS
CP0487210
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(3-phenylpropoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(3-phenylpropoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C36H48N6O23P4
 1
1
EC50 = 1330 nM
   TI
   LI
   LO
   TS
CP0287402
2-methylthio-1-beta-D-ribofuranosylpyrimidine-4-one-5'-diphosphate
   Show/Hide
C10H16N2O11P2S
 1
1
EC50 = 1520 nM
   TI
   LI
   LO
   TS
CP0375618
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[(2R,3R,4S,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H26N2O23P4
 1
1
EC50 = 1770 nM
   TI
   LI
   LO
   TS
CP0415526
[2-cyanoethoxy(hydroxy)phosphoryl] [[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C12H19N3O18P4
 1
1
EC50 = 1960 nM
   TI
   LI
   LO
   TS
CP0460271
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H26N2O23P4
 1
1
EC50 = 2060 nM
   TI
   LI
   LO
   TS
CP0479444
[[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-[(2-methylpropan-2-yl)oxyamino]-2-oxopyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] phosphono hydrogen phosphate
   Show/Hide
C13H24N3O15P3
 1
1
EC50 = 2110 nM
   TI
   LI
   LO
   TS
CP0435255
[(2R,3S,4R,5R)-3,4-dihydroxy-5-[4-[(4-nitrophenyl)methoxyamino]-2-oxopyrimidin-1-yl]oxolan-2-yl]methyl phosphono hydrogen phosphate
   Show/Hide
C16H20N4O14P2
 1
1
EC50 = 2200 nM
   TI
   LI
   LO
   TS
CP0378857
((2R,3S,4R,5R)-4-amino-3-hydroxy-5-(4-oxo-2-thioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-2-yl)methyl tetrahydrogen triphosphate
   Show/Hide
C9H16N3O13P3S
 1
1
EC50 = 2400 nM
   TI
   LI
   LO
   TS
CP0484603
[[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-methylphosphinic acid
   Show/Hide
C10H18N2O17P4
 1
1
EC50 = 2530 nM
   TI
   LI
   LO
   TS
CP0390702
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-(3-nitrophenoxy)phosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H19N3O20P4
 1
1
EC50 = 2540 nM
   TI
   LI
   LO
   TS
CP0375616
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy(methoxy)phosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C10H18N2O18P4
 1
1
EC50 = 2700 nM
   TI
   LI
   LO
   TS
CP0394411
3-methyl-1-beta-D-ribofuranosylpyrimidine-2,4-dione 5'-triphosphate
   Show/Hide
C10H17N2O15P3
 1
1
EC50 = 2920 nM
   TI
   LI
   LO
   TS
CP0849212
(2R,3R,5S)-1-(5-(diphosphoryloxymethyl)-3-hydroxytetrahydrofuran-2-yl)pyrimidine-2,4(1H,3H)-dione triethylammonium salt
   Show/Hide
C15H29N3O11P2
 1
1
EC50 = 3100 nM
   TI
   LI
   LO
   TS
CP0440666
[2-[1-(2-acetamidoethyl)triazol-4-yl]ethoxy-hydroxyphosphoryl] [[(2R,3S,4R,5R)-3,4-dihydroxy-5-[2-oxo-4-(phenylmethoxyamino)pyrimidin-1-yl]oxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C24H34N7O16P3
 1
1
EC50 = 3300 nM
   TI
   LI
   LO
   TS
CP0387447
((2R,3S,4R,5R)-5-(5-bromo-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl tetrahydrogen triphosphate
   Show/Hide
C9H14BrN2O15P3
 2
1
EC50 = 3460 nM
   TI
   LI
   LO
   TS
2
EC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0488963
((2R,3S,4R,5R)-5-(5-fluoro-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl trihydrogen diphosphate
   Show/Hide
C9H13FN2O12P2
 1
1
EC50 = 3500 nM
   TI
   LI
   LO
   TS
CP0043938
({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)oxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy](hydroxy)phosphoryl}oxy)phosphonic acid
   Show/Hide
C10H17N2O15P3
 1
1
EC50 = 3900 nM
   TI
   LI
   LO
   TS
CP0498980
3-Phenacyl-5'-uridylic Acid(1,1-Difluoro-1-phosphonomethyl-1-phosphonyl)anhydride
   Show/Hide
C18H21F2N2O15P3
 1
1
EC50 = 3930 nM
   TI
   LI
   LO
   TS
CP0394415
5-bromouridine-5'-uridylic acid (1,1-dichloro-1-phosphonomethyl-1-phosphonyl)anhydride
   Show/Hide
C10H14BrCl2N2O14P3
 1
1
EC50 = 3990 nM
   TI
   LI
   LO
   TS
CP0439412
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[[(2R,3S,4R)-3,4,6-trihydroxyoxan-2-yl]methoxy]phosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H26N2O22P4
 1
1
EC50 = 4320 nM
   TI
   LI
   LO
   TS
CP0462944
2-Ethylthio-1-beta-D-ribofuranosylpyrimidine-4-one-5'-monophosphate
   Show/Hide
C11H17N2O8PS
 1
1
EC50 = 4330 nM
   TI
   LI
   LO
   TS
CP0473561
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[(2R,3S,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H26N2O23P4
 1
1
EC50 = 4480 nM
   TI
   LI
   LO
   TS
CP0466211
2-methoxy-1-beta-D-ribofuranosylpyrimidine-4-one-5'-diphosphate
   Show/Hide
C10H16N2O12P2
 1
1
EC50 = 4490 nM
   TI
   LI
   LO
   TS
CP0415525
({[({[(2R,3S,4R,5R)-4-(carbamoylamino)-5-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy](hydroxy)phosphoryl}oxy)phosphonic acid
   Show/Hide
C10H17N4O15P3
 1
1
EC50 = 4640 nM
   TI
   LI
   LO
   TS
CP0463237
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy(phosphonooxy)phosphoryl] hydrogen phosphate
   Show/Hide
C9H16N2O18P4
 2
1
EC50 = 4640 nM
   TI
   LI
   LO
   TS
2
EC50 = 7300 nM
   TI
   LI
   LO
   TS
CP0460272
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[[(2S,3R,4S)-3,4,5-trihydroxyoxolan-2-yl]methoxy]phosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C14H24N2O22P4
 1
1
EC50 = 4780 nM
   TI
   LI
   LO
   TS
CP0460358
2-propylthio-1-beta-D-ribofuranosylpyramidine-4-one-5'-diphosphate
   Show/Hide
C12H20N2O11P2S
 1
1
EC50 = 4900 nM
   TI
   LI
   LO
   TS
CP0503315
((2R,3S,4R,5R)-5-(2-amino-4-oxopyrimidin-1(4H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl dihydrogen phosphate
   Show/Hide
C9H14N3O8P
 1
1
EC50 = 4980 nM
   TI
   LI
   LO
   TS
CP0415527
2-Thio-uridine-5'-pentaphosphate
   Show/Hide
C9H17N2O20P5S
 1
1
EC50 = 5270 nM
   TI
   LI
   LO
   TS
CP0509989
2-Thio-4-methylthio-uridine-5'-triphosphate
   Show/Hide
C10H17N2O13P3S2
 1
1
EC50 = 5350 nM
   TI
   LI
   LO
   TS
CP0501815
2-Thio-uridine-5'-tetraphosphate
   Show/Hide
C9H16N2O17P4S
 1
1
EC50 = 5520 nM
   TI
   LI
   LO
   TS
CP0425860
2-benzylthio-1-beta-D-ribofuranosylpyrimidine-4-one-5'-diphosphate
   Show/Hide
C16H20N2O11P2S
 1
1
EC50 = 5980 nM
   TI
   LI
   LO
   TS
CP0861285
N4-tert-Butyloxycytidine 5'-Diphosphate triethylammonium Salt
   Show/Hide
C19H38N4O12P2
 1
1
EC50 = 6230 nM
   TI
   LI
   LO
   TS
CP0460275
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[(2S,3R,4R,5S)-5-ethyl-3,4,5-trihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C16H28N2O22P4
 1
1
EC50 = 6300 nM
   TI
   LI
   LO
   TS
CP0844902
N4-Methoxycytidine 5'-Diphosphate triethylammonium Salt
   Show/Hide
C16H32N4O12P2
 1
1
EC50 = 6450 nM
   TI
   LI
   LO
   TS
CP0467232
((2R,3S,4R,5R)-5-(5-bromo-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl trihydrogen diphosphate
   Show/Hide
C9H13BrN2O12P2
 1
1
EC50 = 7200 nM
   TI
   LI
   LO
   TS
CP0438973
3-Phenacyl-5'-uridylic Acid(1,1-Chloro-1-phosphonomethyl-1-phosphonyl)anhydride
   Show/Hide
C18H21Cl2N2O15P3
 1
1
EC50 = 7300 nM
   TI
   LI
   LO
   TS
CP0440667
[(2R,3S,4R,5R)-5-[4-[(4-bromophenyl)methoxyamino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methyl phosphono hydrogen phosphate
   Show/Hide
C16H20BrN3O12P2
 1
1
EC50 = 7440 nM
   TI
   LI
   LO
   TS
CP0466207
4-Thio-5'-uridylic Acid(1,1-Chloro-1-phosphonomethyl-1-phosphonyl)anhydride
   Show/Hide
C10H15Cl2N2O13P3S
 1
1
EC50 = 7870 nM
   TI
   LI
   LO
   TS
CP0415528
({[({[(2R,3S,4S,5R)-3,4-dihydroxy-5-(4-oxo-2-sulfanylidene-1,2,3,4-tetrahydropyrimidin-1-yl)oxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy](hydroxy)phosphoryl}oxy)phosphonic acid
   Show/Hide
C9H15N2O14P3S
 1
1
EC50 = 7930 nM
   TI
   LI
   LO
   TS
CP0384365
({[({[(2R,3S,4R,5R)-3,4-dihydroxy-5-(4-oxo-2-sulfanylidene-1,2,3,4-tetrahydropyrimidin-1-yl)oxolan-2-yl]methoxy}(hydroxy)phosphoryl)oxy](hydroxy)phosphoryl}difluoromethyl)phosphonic acid
   Show/Hide
C10H15F2N2O13P3S
 1
1
EC50 = 8110 nM
   TI
   LI
   LO
   TS
CP0529670
2'-trifluoroacetylamino-2'-deoxy-2-thiouridine 5'-triphosphate
   Show/Hide
C14H24N3O14P3S
 1
1
EC50 = 8300 nM
   TI
   LI
   LO
   TS
CP0438970
4-Thio-5'-uridylic Acid(1,1-Difluoro-1-phosphonomethyl-1-phosphonyl)anhydride
   Show/Hide
C10H15F2N2O13P3S
 1
1
EC50 = 9300 nM
   TI
   LI
   LO
   TS
CP0460273
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-[[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]-difluoromethyl]phosphinic acid
   Show/Hide
C19H26F2N4O22P4
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0474397
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [hydroxy-[hydroxy-[[(2R,3S,4S,5S)-3,4,5,6-tetrahydroxyoxan-2-yl]methoxy]phosphoryl]oxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H26N2O23P4
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0484602
cyclohexyl [[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C15H26N2O18P4
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0435256
[(2R,3S,4R,5R)-5-[4-[(3-bromophenyl)methoxyamino]-2-oxopyrimidin-1-yl]-3,4-dihydroxyoxolan-2-yl]methyl phosphono hydrogen phosphate
   Show/Hide
C16H20BrN3O12P2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0063449
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dioxoniooxolan-2-yl]methoxy-oxidophosphoryl] hydrogen phosphate
   Show/Hide
C9H14N2O12P2
 1
1
EC50 = 14000 nM
   TI
   LI
   LO
   TS
CP0444113
[[(2S,3R,4S,5S)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C18H27N4O26P5
 1
1
EC50 > 20000 nM
   TI
   LI
   LO
   TS
CP0202705
((2R,3S,4R,5R)-3,4-dihydroxy-5-(5-methoxy-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-2-yl)methyl trihydrogen diphosphate
   Show/Hide
C10H16N2O13P2
 1
1
EC50 >= 20000 nM
   TI
   LI
   LO
   TS
CP0416043
[[(2S,3R,4S,5S)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C18H29N4O32P7
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0453221
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[[[[(2S,3R,4S,5S)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C18H28N4O29P6
 1
1
EC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0453217
[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] [[(2S,3R,4S,5S)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl] hydrogen phosphate
   Show/Hide
C18H25N4O20P3
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0224867
1-beta-D-ribofuranosyl(3H)pyrimidine-2,4,6-trione 5'-monophosphate
   Show/Hide
C9H13N2O10P
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376323
6-methyl-3-beta-D-ribofuranosyl(1H)pyrimidine-2,4-dione 5'-triphosphate
   Show/Hide
C10H17N2O15P3
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376324
6-propyl-3-beta-D-ribofuranosyl(1H)pyrimidine-2,4-dione 5'-diphosphate
   Show/Hide
C12H20N2O12P2
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376575
1-beta-D-ribofuranosyl(3H)pyrimidine-2,4,6-trione 5'-triphosphate
   Show/Hide
C9H15N2O16P3
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376577
((2R,3S,4R,5R)-5-(2,4-dioxo-3-(2-oxo-2-phenylethyl)-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methyl trihydrogen diphosphate
   Show/Hide
C17H20N2O13P2
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376578
3-methyl-1-beta-D-ribofuranosylpyrimidine-2,4-dione 5'-diphosphate
   Show/Hide
C10H16N2O12P2
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376579
1-(BETA-D-RIBOFURANOSYL)-2-THIO-URACIL-5'-PHOSPHATE
   Show/Hide
C9H13N2O8PS
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0382316
6-propyl-3-beta-D-ribofuranosyl(1H)pyrimidine-2,4-dione 5'-monophosphate
   Show/Hide
C12H19N2O9P
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0394410
5-BROMO-URIDINE-5'-MONOPHOSPHATE
   Show/Hide
C9H12BrN2O9P
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0394414
6-propyl-3-beta-D-ribofuranosyl(1H)pyrimidine-2,4-dione 5'-triphosphate
   Show/Hide
C12H21N2O15P3
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0408415
6-methyl-3-beta-D-ribofuranosyl(1H)pyrimidine-2,4-dione 5'-diphosphate
   Show/Hide
C10H16N2O12P2
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0433478
3-phenacyl-1-beta-D-ribofuranosylpyrimidine-2,4-dione 2'-Monophosphate-5'-triphosphate
   Show/Hide
C17H22N2O19P4
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0453590
3-METHYLURIDINE-5'-MONOPHOSHATE
   Show/Hide
C10H15N2O9P
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0453591
6-propyl-3-beta-D-ribofuranosyl(1H)pyrimidine-2,4-dione 2',3'-(cyclic phosphate) 5'-triphosphate
   Show/Hide
C12H20N2O17P4
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0464525
6-methyl-3-beta-D-ribofuranosyl(1H)pyrimidine-2,4-dione 5'-monophosphate
   Show/Hide
C10H15N2O9P
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0499963
3-phenacyl-1-beta-D-ribofuranosylpyrimidine-2,4-dione 5'-monophosphate
   Show/Hide
C17H19N2O10P
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0425864
2-Propylthio-1-beta-D-ribofuranosylpyrimidine-4-one-5'-monophosphate
   Show/Hide
C12H19N2O8PS
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0425865
2-Phenylethylthio-1-beta-D-ribofuranosylpyrimidine-4-one-5'-monophosphate
   Show/Hide
C17H21N2O8PS
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0438971
2-Methoxy-1-beta-D-ribofuranosylpyrimidine-4-one-5'-monophosphate
   Show/Hide
C10H15N2O9P
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0438972
((2R,3S,4R,5R)-3,4-dihydroxy-5-(2-(methylamino)-4-oxopyrimidin-1(4H)-yl)tetrahydrofuran-2-yl)methyl dihydrogen phosphate
   Show/Hide
C10H16N3O8P
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0438974
5-Bromo-1-beta-D-ribofuranosyl(3H)pyrimidine-2,4-dione 5'-(gamma-phenylamino)triphosphate
   Show/Hide
C15H19BrN3O14P3
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0466203
2-Benzylthio-1-beta-D-ribofuranosylpyrimidine-4-one-5'-monophosphate
   Show/Hide
C16H19N2O8PS
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0466204
[dichloro-[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-hydroxyphosphoryl]methyl]phosphonic acid
   Show/Hide
C10H15Cl2N2O14P3
 1
1
EC50 >= 100000 nM
   TI
   LI
   LO
   TS
CP0478598
2-Methylamino-1-beta-D-ribofuranosylpyrimidine-4-one-5'-diphosphate
   Show/Hide
C10H17N3O11P2
 1
1
EC50 >= 100000 nM
   TI
   LI
   LO
   TS
CP0478599
(((((2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl)methoxy)(hydroxy)phosphoryloxy)(hydroxy)phosphoryl)difluoromethylphosphonic acid
   Show/Hide
C10H15F2N2O14P3
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0478646
2-phenylethylthio-1-beta-D-ribofuranosylpyrimidine-4-one-5'-diphosphate
   Show/Hide
C17H22N2O11P2S
 1
1
EC50 >= 100000 nM
   TI
   LI
   LO
   TS
CP0503314
2-Methylthio-1-beta-D-ribofuranosylpyrimidine-4-one-5'-monophosphate
   Show/Hide
C10H15N2O8PS
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0503382
2-amino-1-beta-D-ribofuranosylpyrimidine-4-one-5'-diphosphate
   Show/Hide
C9H15N3O11P2
 1
1
EC50 >= 100000 nM
   TI
   LI
   LO
   TS
CP0504974
((2R,3S,4R,5R)-3,4-dihydroxy-5-(2-oxo-4-thioxo-3,4-dihydropyrimidin-1(2H)-yl)tetrahydrofuran-2-yl)methyl dihydrogen phosphate
   Show/Hide
C9H13N2O8PS
 1
1
EC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0376580
(2R,3R,4S,5R)-1-(3,4-dihydroxy-5-(diphosphoryloxymethyl)-tetrahydrofuran-2-yl)-2-thioxo-2,3-dihydropyrimidin-4(1H)-one ammonium salt
   Show/Hide
C9H14N2O11P2S
 1
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0394412
3-phenacyl-1-beta-D-ribofuranosylpyrimidine-2,4-dione 5'-triphosphate
   Show/Hide
C17H21N2O16P3
 1
1
EC50 > 1000 nM
   TI
   LI
   LO
   TS
CP0894768
Sodium 1-Amino-4-[4-(2,4-dimethylphenylthio)phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C28H21N2NaO5S2
 1
1
IC50 = 233 nM
   TI
   LI
   LO
   TS
CP0885815
Sodium 1-Amino-4-[4-(4-chlorophenoxy)phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C26H16ClN2NaO6S
 1
1
IC50 = 373 nM
   TI
   LI
   LO
   TS
CP0854864
Sodium 1-Amino-4-[4-(2,5-dimethylphenylthio)phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C28H21N2NaO5S2
 1
1
IC50 = 395 nM
   TI
   LI
   LO
   TS
CP0893862
Sodium 1-Amino-4-[4-(3-pyridin-3-ylmethylthio)phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C26H18N3NaO5S2
 1
1
IC50 = 409 nM
   TI
   LI
   LO
   TS
CP0885816
Sodium 1-Amino-4-[4-(3,4-dimethylphenylthio)phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C28H21N2NaO5S2
 1
1
IC50 = 482 nM
   TI
   LI
   LO
   TS
CP0713911
SID50106952
   Show/Hide
C29H17ClN7Na3O11S3
 1
1
IC50 = 625 nM
   TI
   LI
   LO
   TS
CP0893864
Sodium 1-Amino-4-(4-hydroxy-3-methylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H15N2NaO6S
 1
1
IC50 = 746 nM
   TI
   LI
   LO
   TS
CP0652101
Reactive Blue-2
   Show/Hide
C29H17ClN7Na3O11S3
 2
1
IC50 = 1140 nM
   TI
   LI
   LO
   TS
2
IC50 = 9790 nM
   TI
   LI
   LO
   TS
CP0946904
sodium 1-amino-9,10-dioxo-4-(4-(phenylthio)phenylamino)-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C26H17N2NaO5S2
 1
1
IC50 = 1180 nM
   TI
   LI
   LO
   TS
CP0893860
Sodium 1-amino-4-(3-fluorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C20H12FN2NaO5S
 1
1
IC50 = 1390 nM
   TI
   LI
   LO
   TS
CP0849079
sodium 1-amino-4-(3-carboxy-5-(4,6-dichloro-1,3,5-triazin-2-ylamino)phenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C24H13Cl2N6NaO7S
 1
1
IC50 = 1450 nM
   TI
   LI
   LO
   TS
CP0968181
Sodium 1-amino-4-(3-ethylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO5S
 1
1
IC50 = 1510 nM
   TI
   LI
   LO
   TS
CP0893861
Sodium 1-Amino-4-(4-fluoro-3-methoxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H14FN2NaO6S
 1
1
IC50 = 1540 nM
   TI
   LI
   LO
   TS
CP0958824
Sodium 1-Amino-4-(4-chloro-3-methylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H14ClN2NaO5S
 1
1
IC50 = 1650 nM
   TI
   LI
   LO
   TS
CP0921084
Sodium 1-Amino-4-[4-(4-fluorophenoxy)phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C26H16FN2NaO6S
 1
1
IC50 = 1690 nM
   TI
   LI
   LO
   TS
CP0918930
sodium 1-amino-4-(3-methoxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H15N2NaO6S
 2
1
IC50 = 1700 nM
   TI
   LI
   LO
   TS
2
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0963902
Sodium 1-Amino-4-[4-(4-bromophenoxy)phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C26H16BrN2NaO6S
 1
1
IC50 = 1760 nM
   TI
   LI
   LO
   TS
CP0874902
sodium 1-amino-9,10-dioxo-4-(4-(phenylamino)phenylamino)-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C26H18N3NaO5S
 1
1
IC50 = 1910 nM
   TI
   LI
   LO
   TS
CP0868055
sodium 1-amino-9,10-dioxo-4-(4-phenoxyphenylamino)-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C26H17N2NaO6S
 1
1
IC50 = 1940 nM
   TI
   LI
   LO
   TS
CP0652102
sodium 1-amino-9,10-dioxo-4-(phenylamino)-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C20H13N2NaO5S
 2
1
IC50 = 1970 nM
   TI
   LI
   LO
   TS
2
IC50 = 25800 nM
   TI
   LI
   LO
   TS
CP0963224
Sodium 1-Amino-4-(4-chloro-2-methylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H14ClN2NaO5S
 1
1
IC50 = 2200 nM
   TI
   LI
   LO
   TS
CP0652104
sodium 1-amino-4-(4-hydroxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C20H13N2NaO6S
 2
1
IC50 = 2220 nM
   TI
   LI
   LO
   TS
2
IC50 = 3160 nM
   TI
   LI
   LO
   TS
CP0849078
sodium 1-amino-9,10-dioxo-4-(m-tolylamino)-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H15N2NaO5S
 2
1
IC50 = 2220 nM
   TI
   LI
   LO
   TS
2
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0929924
sodium 1-amino-4-(3-chlorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C20H12ClN2NaO5S
 2
1
IC50 = 2340 nM
   TI
   LI
   LO
   TS
2
IC50 = 21800 nM
   TI
   LI
   LO
   TS
CP0785160
sodium 1-amino-4-(4-methoxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H15N2NaO6S
 1
1
IC50 = 2590 nM
   TI
   LI
   LO
   TS
CP0878492
sodium 1-amino-4-(2,3-dimethylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO5S
 1
1
IC50 = 2630 nM
   TI
   LI
   LO
   TS
CP0846170
sodium 1-amino-4-(2-carboxy-5-chlorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H12ClN2NaO7S
 1
1
IC50 = 2760 nM
   TI
   LI
   LO
   TS
CP0874900
sodium 1-amino-9,10-dioxo-4-(p-tolylamino)-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H15N2NaO5S
 1
1
IC50 = 2820 nM
   TI
   LI
   LO
   TS
CP0963379
Sodium 1-Amino-4-(3-propylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C23H19N2NaO5S
 1
1
IC50 = 2990 nM
   TI
   LI
   LO
   TS
CP0791547
SID50112916
   Show/Hide
C20H12ClN2NaO5S
 1
1
IC50 = 3030 nM
   TI
   LI
   LO
   TS
CP0875994
Sodium 1-Amino-4-(4-ethylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO5S
 1
1
IC50 = 3210 nM
   TI
   LI
   LO
   TS
CP0868045
sodium 1-amino-4-(4-bromophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C20H12BrN2NaO5S
 1
1
IC50 = 3300 nM
   TI
   LI
   LO
   TS
CP0960958
Sodium 1-Amino-4-(4-chloro-3-methoxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H14ClN2NaO6S
 1
1
IC50 = 3370 nM
   TI
   LI
   LO
   TS
CP0885813
sodium 1-amino-4-(4-benzylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C27H19N2NaO5S
 1
1
IC50 = 3450 nM
   TI
   LI
   LO
   TS
CP0878493
sodium 1-amino-9,10-dioxo-4-(o-tolylamino)-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H15N2NaO5S
 1
1
IC50 = 3490 nM
   TI
   LI
   LO
   TS
CP0854449
sodium 1-amino-4-(2-ethylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO5S
 1
1
IC50 = 3530 nM
   TI
   LI
   LO
   TS
CP0854848
sodium 1-amino-4-(2,4-dimethylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO5S
 1
1
IC50 = 3580 nM
   TI
   LI
   LO
   TS
CP0655729
sodium 1-amino-4-(2-methoxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H15N2NaO6S
 1
1
IC50 = 3980 nM
   TI
   LI
   LO
   TS
CP0887290
sodium 1-amino-4-(4-fluorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C20H12FN2NaO5S
 1
1
IC50 = 4040 nM
   TI
   LI
   LO
   TS
CP0854849
Sodium 1-Amino-4-(3-methoxy-4-methylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO6S
 1
1
IC50 = 4130 nM
   TI
   LI
   LO
   TS
CP0903424
Sodium 1-Amino-4-(3,4-dimethoxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO7S
 1
1
IC50 = 4980 nM
   TI
   LI
   LO
   TS
CP0848945
sodium 1-amino-4-(2-carboxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H13N2NaO7S
 1
1
IC50 = 6100 nM
   TI
   LI
   LO
   TS
CP0944606
sodium 1-amino-4-(3,5-dimethylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO5S
 1
1
IC50 = 6450 nM
   TI
   LI
   LO
   TS
CP0963223
sodium 1-amino-4-(3-bromophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C20H12BrN2NaO5S
 1
1
IC50 = 6960 nM
   TI
   LI
   LO
   TS
CP0921115
sodium 1-amino-9,10-dioxo-4-(phenethylamino)-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C22H17N2NaO5S
 1
1
IC50 = 7180 nM
   TI
   LI
   LO
   TS
CP0661524
SID50112917
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C24H15N2NaO5S
 1
1
IC50 = 7420 nM
   TI
   LI
   LO
   TS
CP0963901
Sodium 1-amino-4-(3,5-dimethoxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C22H17N2NaO7S
 1
1
IC50 = 9250 nM
   TI
   LI
   LO
   TS
CP0903423
Sodium 1-Amino-4-(2-chlorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C20H12ClN2NaO5S
 1
1
IC50 = 9340 nM
   TI
   LI
   LO
   TS
CP0849076
Disodium 1-Amino-4-[3-(4,6-dichloro[1,3,5]triazine-2-ylamino)-4-sulfophenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C23H12Cl2N6Na2O8S2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0849080
Sodium1-Amino-4-(3-benzylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C27H19N2NaO5S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0878441
Sodium 1-Amino-4-[3-(4,6-dichloro[1,3,5]triazine-2-ylamino)-phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C23H13Cl2N6NaO5S
 1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0903821
Sodium 1-Amino-4-[4-(4,6-dihydroxy[1,3,5]triazine-2-ylamino)-phenylamino]-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C23H15N6NaO7S
 1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0911840
sodium 1-amino-4-(4-(4,6-dichloro-1,3,5-triazin-2-ylamino)phenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C23H13Cl2N6NaO5S
 1
1
IC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0917863
sodium 1-amino-4-(4-(4,6-dihydroxy-1,3,5-triazin-2-ylamino)phenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C24H15ClN6Na2O9S2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0448653
1-amino-4-(3-methoxyanilino)-9,10-dioxoanthracene-2-sulfonic acid
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C21H16N2O6S
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0032210
4-(4-piperidin-4-ylphenyl)-7-[4-(trifluoromethyl)phenyl]naphthalene-2-carboxylic acid
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C29H24F3NO2
 1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0846903
Sodium 1-Amino-4-(2,5-dimethylphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C22H17N2NaO5S
 1
1
IC50 = 11200 nM
   TI
   LI
   LO
   TS
CP0946902
Sodium 1-amino-4-(3,5-difluorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C20H11F2N2NaO5S
 1
1
IC50 = 12500 nM
   TI
   LI
   LO
   TS
CP0846904
sodium 1-amino-4-(benzylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C21H15N2NaO5S
 1
1
IC50 = 14400 nM
   TI
   LI
   LO
   TS
CP0968373
Sodium 1-Amino-4-(2-carboxy-4-hydroxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C21H13N2NaO8S
 1
1
IC50 = 21100 nM
   TI
   LI
   LO
   TS
CP0895171
sodium 1-amino-4-(3-carboxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C21H13N2NaO7S
 1
1
IC50 = 23400 nM
   TI
   LI
   LO
   TS
CP0458434
1-amino-4-(3-methoxyanilino)-2-methylanthracene-9,10-dione
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C22H18N2O3
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0458435
1-amino-4-(3-fluoroanilino)-2-methylanthracene-9,10-dione
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C21H15FN2O2
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0460436
1-amino-4-(3-fluoroanilino)-9,10-dioxoanthracene-2-sulfonic acid
   Show/Hide
C20H13FN2O5S
 1
1
IC50 = 30000 nM
   TI
   LI
   LO
   TS
CP0874901
sodium 1-amino-4-(4-carboxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H13N2NaO7S
 1
1
IC50 = 30000 nM
   TI
   LI
   LO
   TS
CP0946903
Sodium 1-Amino-4-(2-carboxy-4-nitrophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H12N3NaO9S
 1
1
IC50 > 30000 nM
   TI
   LI
   LO
   TS
CP0448652
2-[(4-amino-3-methyl-9,10-dioxoanthracen-1-yl)amino]-5-fluorobenzoic acid
   Show/Hide
C22H15FN2O4
 1
1
IC50 = 100000 nM
   TI
   LI
   LO
   TS
CP0448654
2-[(4-amino-9,10-dioxo-3-sulfoanthracen-1-yl)amino]-5-fluorobenzoic acid
   Show/Hide
C21H13FN2O7S
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0658680
sodium 1-amino-4-(2-carboxy-4-fluorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C21H12FN2NaO7S
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0846902
sodium 1-amino-4-(4-bromo-2-carboxyphenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
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C21H12BrN2NaO7S
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0852887
sodium 1-amino-4-(2-carboxy-5-fluorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H12FN2NaO7S
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0873841
sodium 1-amino-4-(2-carboxy-4-chlorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H12ClN2NaO7S
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0893863
Sodium 1-Amino-4 (2-carboxy-3-fluorophenylamino)-9,10-dioxo-9,10-dihydroanthracene-2-sulfonate
   Show/Hide
C21H12FN2NaO7S
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
Clinical Information about the Protein
Target 1 ( P2Y purinoceptor 4 (P2RY4) )
Target Type Discontinued Target
Disease 1 Target-related Disease  1
1 Lung cancer [ICD-11: 2C25.0]
Discontinued Drug(s) 1 Discontinued Drug  1
1 INS 316 Discontinued in Phase 3
Lung cancer