| Compound ID |
Compound Name |
Compound Formula |
|
CP0253979
|
US10435369, Example 137
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|
C26H25F8NO4S
|
1
|
| 1 |
EC50 = 2.7 nM
|
|
|
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CP0129837
|
(1R,3S,4R)-4-[[(3aR,9bR)-9b-(4-fluorophenyl)sulfonyl-7-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)-2,3a,4,5-tetrahydro-1H-benzo[e]indol-3-yl]amino]-3-methylcyclohexane-1-carboxylic acid
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|
C29H30F8N2O4S
|
1
|
| 1 |
EC50 = 11 nM
|
|
|
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CP0558225
|
N-[3,5-dichloro-4-(6-methoxy-5-propan-2-ylpyridin-3-yl)oxyphenyl]-2-(1-methylsulfonylpiperidin-4-yl)acetamide
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|
C23H29Cl2N3O5S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
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CP0553176
|
N-[3,5-dichloro-4-(4-methoxy-3-propan-2-ylphenoxy)phenyl]-2-(4-methylsulfonylpiperazin-1-yl)acetamide
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|
C23H29Cl2N3O5S
|
1
|
| 1 |
EC50 = 34 nM
|
|
|
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CP0556947
|
N-[3,5-dichloro-4-(4-methoxy-3-propan-2-ylphenoxy)phenyl]-2-pyridin-4-ylacetamide
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|
C23H22Cl2N2O3
|
1
|
| 1 |
EC50 = 81 nM
|
|
|
|
CP0334320
|
N-[1-[2-(2,4-dichlorophenyl)ethyl]indol-5-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C26H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0493777
|
2-(4-ethylsulfonylphenyl)-N-[1-[2-[4-(trifluoromethyl)phenyl]ethyl]indol-5-yl]acetamide
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|
C27H25F3N2O3S
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0493776
|
N-[1-[2-(3,4-dichlorophenyl)ethyl]indol-5-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C26H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0486773
|
2-(4-ethylsulfonylphenyl)-N-[1-[2-(4-propan-2-yloxyphenyl)ethyl]indol-5-yl]acetamide
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|
C29H32N2O4S
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0066901
|
N-[5-[4-chloro-2-(trifluoromethyl)phenoxy]-4-(3-cyanophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C27H19ClF3N3O4S2
|
1
|
| 1 |
IC50 = 158.49 nM
|
|
|
|
CP0538990
|
N-[1-[2-(4-chlorophenyl)ethyl]indol-5-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C26H25ClN2O3S
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0059071
|
N-[4-(3-cyanophenyl)-5-[2-(trifluoromethyl)phenoxy]-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C27H20F3N3O4S2
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0066706
|
2-(4-ethylsulfonylphenyl)-N-[5-(2-methoxyphenoxy)-4-phenyl-1,3-thiazol-2-yl]acetamide
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|
C26H24N2O5S2
|
1
|
| 1 |
IC50 = 251.19 nM
|
|
|
|
CP0519322
|
2-(4-ethylsulfonylphenyl)-N-[4-[[propyl-[[4-(trifluoromethyl)phenyl]methyl]amino]methyl]phenyl]acetamide
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|
C28H31F3N2O3S
|
1
|
| 1 |
IC50 = 320 nM
|
|
|
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CP0059072
|
N-[5-[2-chloro-4-(trifluoromethyl)phenoxy]-4-(3-cyanophenyl)-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C27H19ClF3N3O4S2
|
1
|
| 1 |
IC50 = 398.11 nM
|
|
|
|
CP0519321
|
N-[1-[2-(4-cyanophenyl)ethyl]indol-5-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C27H25N3O3S
|
1
|
| 1 |
IC50 = 457 nM
|
|
|
|
CP0175161
|
2-(4-ethylsulfonylphenyl)-N-[4-phenyl-5-[4-(trifluoromethyl)phenoxy]-1,3-thiazol-2-yl]acetamide
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|
C26H21F3N2O4S2
|
1
|
| 1 |
IC50 = 630.96 nM
|
|
|
|
CP0486774
|
2-(4-ethylsulfonylphenyl)-N-[4-[propyl-[2-[4-(trifluoromethyl)phenyl]ethyl]amino]phenyl]acetamide
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|
C28H31F3N2O3S
|
1
|
| 1 |
IC50 = 733 nM
|
|
|
|
CP0247829
|
2-(4-ethylsulfonylphenyl)-N-[4-phenyl-5-[2-(trifluoromethyl)phenoxy]-1,3-thiazol-2-yl]acetamide
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|
C26H21F3N2O4S2
|
1
|
| 1 |
IC50 = 1000 nM
|
|
|
|
CP0420736
|
N-[3-chloro-4-[2-[4-(trifluoromethyl)phenyl]ethylamino]phenyl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C25H24ClF3N2O3S
|
1
|
| 1 |
IC50 = 1023 nM
|
|
|
|
CP0059070
|
N-[4-(3-chlorophenyl)-5-phenoxy-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C25H21ClN2O4S2
|
1
|
| 1 |
IC50 = 1584.89 nM
|
|
|
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CP0066703
|
N-[5-(4-chlorophenoxy)-4-phenyl-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C25H21ClN2O4S2
|
1
|
| 1 |
IC50 = 1584.89 nM
|
|
|
|
CP0067836
|
N-[5-(2-chlorophenoxy)-4-phenyl-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C25H21ClN2O4S2
|
1
|
| 1 |
IC50 = 1584.89 nM
|
|
|
|
CP0101927
|
N-[4-(3-chlorophenyl)-5-[2-(trifluoromethyl)phenoxy]-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C26H20ClF3N2O4S2
|
1
|
| 1 |
IC50 = 1995.26 nM
|
|
|
|
CP0071666
|
N-[4-(4-chlorophenyl)-5-phenoxy-1,3-thiazol-2-yl]-2-(4-ethylsulfonylphenyl)acetamide
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|
C25H21ClN2O4S2
|
1
|
| 1 |
IC50 = 3981.07 nM
|
|
|
|
CP0514635
|
2-(4-ethylsulfonylphenyl)-N-[4-[[[4-(trifluoromethyl)phenyl]methylamino]methyl]phenyl]acetamide
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|
C25H25F3N2O3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0066702
|
2-(4-ethylsulfonylphenyl)-N-[5-(4-methoxyphenoxy)-4-phenyl-1,3-thiazol-2-yl]acetamide
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|
C26H24N2O5S2
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
