| Compound ID |
Compound Name |
Compound Formula |
|
CP0222270
|
(2S)-N-(tert-Butyl)-2-{[4-({[5-(phenylsulfonyl)-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]carbonyl}pyrrolidine-1-carboxamide
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|
C28H35F3N4O6S2
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0198695
|
(S)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluoromethyl)phenylsulfonamido)piperidine-1-carbonyl)pyrrolidine-1-carboxylate
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|
C28H34F3N3O7S2
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0198692
|
tert-butyl (2S)-2-[4-[[5-(benzenesulfonyl)-2-(trifluoromethyl)phenyl]sulfonylamino]piperidine-1-carbonyl]-5-oxopyrrolidine-1-carboxylate
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|
C28H32F3N3O8S2
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0264359
|
(2S)-N-Ethyl-2-{[4-({[5-(phenylsulfonyl)-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]carbonyl}pyrrolidine-1-carboxamide
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|
C26H31F3N4O6S2
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0289969
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-(2-methylpropanoyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C27H32F3N3O6S2
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0198696
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-(3,3-dimethylbutanoyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C29H36F3N3O6S2
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0264360
|
(2S)-N,N-Dimethyl-2-{[4-({[5-(phenylsulfonyl)-2-(trifluoromethyl)phenyl]sulfonyl}amino)piperidin-1-yl]carbonyl}pyrrolidine-1-carboxamide
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|
C26H31F3N4O6S2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0310846
|
5-(benzenesulfonyl)-N-[1-(2-morpholin-4-ylacetyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C24H28F3N3O6S2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0333299
|
5-(Phenylsulfonyl)-N-[1-(pyrrolidin-1-ylacetyl)piperidin-4-yl]-2-(trifluoro-methyl)benzenesulfonamide
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|
C24H28F3N3O5S2
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0212060
|
(R)-tert-butyl 2-(4-(5-(phenylsulfonyl)-2-(trifluoromethyl)phenylsulfonamido)piperidine-1-carbonyl)pyrrolidine-1-carboxylate
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|
C28H34F3N3O7S2
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0222295
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-methylpyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C24H28F3N3O5S2
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0345060
|
5-(benzenesulfonyl)-N-[1-(2-imidazol-1-ylacetyl)piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C23H23F3N4O5S2
|
1
|
| 1 |
EC50 = 230 nM
|
|
|
|
CP0310847
|
5-(benzenesulfonyl)-N-[1-[(2S)-5-oxopyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C23H24F3N3O6S2
|
1
|
| 1 |
EC50 = 240 nM
|
|
|
|
CP0222293
|
5-(Phenylsulfonyl)-N-[1-(piperazin-1-ylacetyl)piperidin-4-yl]-2-(trifluoro-methyl)benzenesulfonamide
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|
C24H29F3N4O5S2
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0310849
|
N-[1-[(2S)-1-acetylpyrrolidine-2-carbonyl]piperidin-4-yl]-5-(benzenesulfonyl)-2-(trifluoromethyl)benzenesulfonamide
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|
C25H28F3N3O6S2
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0333308
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-(2,2-dimethylpropanoyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C28H34F3N3O6S2
|
1
|
| 1 |
EC50 = 270 nM
|
|
|
|
CP0322892
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-(morpholine-4-carbonyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C28H33F3N4O7S2
|
1
|
| 1 |
EC50 = 280 nM
|
|
|
|
CP0345059
|
5-(benzenesulfonyl)-N-[1-[2-(dimethylamino)acetyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C22H26F3N3O5S2
|
1
|
| 1 |
EC50 = 280 nM
|
|
|
|
CP0269762
|
(2S)-N-Phenyl-2-{[4-({[5-(phenylsulfonyl)-2-(trifluoromethyl)-phenyl]sulfonyl}amino)piperidin-1-yl]carbonyl}pyrrolidine-1-carboxamide
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|
C30H31F3N4O6S2
|
1
|
| 1 |
EC50 = 310 nM
|
|
|
|
CP0289971
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-[2-(dimethylamino)acetyl]pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C27H33F3N4O6S2
|
1
|
| 1 |
EC50 = 310 nM
|
|
|
|
CP0198693
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-(cyclohexylmethyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C30H38F3N3O5S2
|
1
|
| 1 |
EC50 = 320 nM
|
|
|
|
CP0265627
|
(S)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbonyl)piperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C23H26F3N3O5S2
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0289973
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-(pyridine-4-carbonyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C29H29F3N4O6S2
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0222294
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-benzoylpyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
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|
C30H30F3N3O6S2
|
1
|
| 1 |
EC50 = 380 nM
|
|
|
|
CP0068037
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-(3,3-dimethylbutyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C29H38F3N3O5S2
|
1
|
| 1 |
EC50 = 450 nM
|
|
|
|
CP0333309
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-(cyclohexanecarbonyl)pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C30H36F3N3O6S2
|
1
|
| 1 |
EC50 = 460 nM
|
|
|
|
CP0264358
|
5-(benzenesulfonyl)-N-[1-[2-(methylamino)acetyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C21H24F3N3O5S2
|
1
|
| 1 |
EC50 = 620 nM
|
|
|
|
CP0204968
|
5-(Phenylsulfonyl)-N-piperidin-4-yl-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C18H19F3N2O4S2
|
1
|
| 1 |
EC50 = 650 nM
|
|
|
|
CP0192160
|
(R)-5-(phenylsulfonyl)-N-(1-(pyrrolidine-2-carbonyl)piperidin-4-yl)-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C23H26F3N3O5S2
|
1
|
| 1 |
EC50 = 710 nM
|
|
|
|
CP0198694
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-benzylpyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C30H32F3N3O5S2
|
1
|
| 1 |
EC50 = 720 nM
|
|
|
|
CP0347767
|
5-(benzenesulfonyl)-N-[1-[(2S)-1-[4-(dimethylamino)benzoyl]pyrrolidine-2-carbonyl]piperidin-4-yl]-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C32H35F3N4O6S2
|
1
|
| 1 |
EC50 = 830 nM
|
|
|
