| Compound ID |
Compound Name |
Compound Formula |
|
CP0440127
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(5-thiophen-2-ylpyridin-2-yl)acetamide
Show/Hide
|
C23H18N4O2S3
|
1
|
| 1 |
EC50 = 0.3 nM
|
|
|
|
CP0517856
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(6-phenylpyridin-3-yl)acetamide
Show/Hide
|
C25H20N4O2S2
|
1
|
| 1 |
EC50 = 0.3 nM
|
|
|
|
CP0440130
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(4-pyridin-3-ylphenyl)acetamide
Show/Hide
|
C25H20N4O2S2
|
1
|
| 1 |
EC50 = 0.45 nM
|
|
|
|
CP0142329
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(5-phenylpyridin-2-yl)acetamide
Show/Hide
|
C25H20N4O2S2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0515505
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(4-phenylphenyl)acetamide
Show/Hide
|
C26H21N3O2S2
|
1
|
| 1 |
EC50 = 0.75 nM
|
|
|
|
CP0440129
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(5-pyridin-3-ylpyridin-2-yl)acetamide
Show/Hide
|
C24H19N5O2S2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0515502
|
N-[5-(furan-3-yl)pyridin-2-yl]-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C23H18N4O3S2
|
1
|
| 1 |
EC50 = 1.5 nM
|
|
|
|
CP0521828
|
N-[5-(furan-3-yl)pyrimidin-2-yl]-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C22H17N5O3S2
|
1
|
| 1 |
EC50 = 1.5 nM
|
|
|
|
CP0515500
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(5-thiophen-3-ylpyridin-2-yl)acetamide
Show/Hide
|
C23H18N4O2S3
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0418001
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(4-pyridin-4-ylphenyl)acetamide
Show/Hide
|
C25H20N4O2S2
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0440128
|
N-[5-(furan-2-yl)pyridin-2-yl]-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C23H18N4O3S2
|
1
|
| 1 |
EC50 = 3.5 nM
|
|
|
|
CP0481455
|
N-[5-(furan-2-yl)pyrimidin-2-yl]-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C22H17N5O3S2
|
1
|
| 1 |
EC50 = 3.5 nM
|
|
|
|
CP0418002
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(4-pyridin-2-ylphenyl)acetamide
Show/Hide
|
C25H20N4O2S2
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0515503
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(5-pyrimidin-5-ylpyridin-2-yl)acetamide
Show/Hide
|
C23H18N6O2S2
|
1
|
| 1 |
EC50 = 5.5 nM
|
|
|
|
CP0515509
|
2-[(3,6-dimethyl-4-oxidanylidene-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(6-methyl-1,3-benzothiazol-2-yl)ethanamide
Show/Hide
|
C18H18N4O2S3
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0521829
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(5-phenylpyrimidin-2-yl)acetamide
Show/Hide
|
C24H19N5O2S2
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0528628
|
N-[2-[(6-chloro-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-3-(4-methoxyphenyl)-4-oxophthalazine-1-carboxamide
Show/Hide
|
C25H18ClN5O4S
|
1
|
| 1 |
EC50 = 15 nM
|
|
|
|
CP0145450
|
2-[[3-(2-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]-N-(6-methyl-1,3-benzothiazol-2-yl)acetamide
Show/Hide
|
C23H20N4O3S3
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0515495
|
N-[2-[(6-chloro-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-3-(4-fluorophenyl)-4-oxophthalazine-1-carboxamide
Show/Hide
|
C24H15ClFN5O3S
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0528629
|
3-(4-methoxyphenyl)-N-[2-[(6-methyl-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-4-oxophthalazine-1-carboxamide
Show/Hide
|
C26H21N5O4S
|
1
|
| 1 |
EC50 = 25 nM
|
|
|
|
CP0076082
|
N-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C22H18N4O2S3
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0428120
|
2-[[3-(2-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]-N-[6-(trifluoromethyl)-1,3-benzothiazol-2-yl]acetamide
Show/Hide
|
C23H17F3N4O3S3
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0481456
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(4-piperidin-1-ylphenyl)acetamide
Show/Hide
|
C25H26N4O2S2
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0515496
|
N-[2-[(6-chloro-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-4-oxo-3-phenylphthalazine-1-carboxamide
Show/Hide
|
C24H16ClN5O3S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0522902
|
N-(6-chloro-1,3-benzothiazol-2-yl)-2-[[3-(4-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]acetamide
Show/Hide
|
C22H17ClN4O3S3
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0528630
|
N-[2-[(6-methyl-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-4-oxo-3-phenylphthalazine-1-carboxamide
Show/Hide
|
C25H19N5O3S
|
1
|
| 1 |
EC50 = 35 nM
|
|
|
|
CP0145449
|
2-[[3-(4-fluorophenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]-N-(6-methyl-1,3-benzothiazol-2-yl)acetamide
Show/Hide
|
C22H17FN4O2S3
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0145451
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-[6-(trifluoromethyl)-1,3-benzothiazol-2-yl]acetamide
Show/Hide
|
C22H15F3N4O2S3
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0482408
|
N-(6-chloro-1,3-benzothiazol-2-yl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C21H15ClN4O2S3
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0528631
|
N-(6-methoxy-1,3-benzothiazol-2-yl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C22H18N4O3S3
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0515499
|
N-(6-methoxy-1,3-benzothiazol-2-yl)-2-[[3-(2-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]acetamide
Show/Hide
|
C23H20N4O4S3
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0522879
|
N-(6-chloro-1,3-benzothiazol-2-yl)-2-[[3-(2-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]acetamide
Show/Hide
|
C22H17ClN4O3S3
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0426152
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(5-phenyl-1,3-thiazol-2-yl)acetamide
Show/Hide
|
C23H18N4O2S3
|
1
|
| 1 |
EC50 = 55 nM
|
|
|
|
CP0440132
|
N-[2-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-3-(4-methoxyphenyl)-4-oxophthalazine-1-carboxamide
Show/Hide
|
C26H21N5O5S
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0481454
|
3-(4-fluorophenyl)-N-[2-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-4-oxophthalazine-1-carboxamide
Show/Hide
|
C25H18FN5O4S
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0511560
|
3-(4-fluorophenyl)-4-oxo-N-[2-oxo-2-[[6-(trifluoromethyl)-1,3-benzothiazol-2-yl]amino]ethyl]phthalazine-1-carboxamide
Show/Hide
|
C25H15F4N5O3S
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0528632
|
N-[2-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-3-(2-methoxyphenyl)-4-oxophthalazine-1-carboxamide
Show/Hide
|
C26H21N5O5S
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0428119
|
2-[[3-(4-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]-N-[6-(trifluoromethyl)-1,3-benzothiazol-2-yl]acetamide
Show/Hide
|
C23H17F3N4O3S3
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0433805
|
2-[[3-(4-fluorophenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]-N-[6-(trifluoromethyl)-1,3-benzothiazol-2-yl]acetamide
Show/Hide
|
C22H14F4N4O2S3
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0438728
|
3-(4-fluorophenyl)-N-[2-[(6-methyl-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-4-oxophthalazine-1-carboxamide
Show/Hide
|
C25H18FN5O3S
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0489917
|
4-oxo-N-[2-oxo-2-[[6-(trifluoromethyl)-1,3-benzothiazol-2-yl]amino]ethyl]-3-phenylphthalazine-1-carboxamide
Show/Hide
|
C25H16F3N5O3S
|
1
|
| 1 |
EC50 = 110 nM
|
|
|
|
CP0543986
|
N-(6-methoxy-1,3-benzothiazol-2-yl)-2-[[3-(4-methoxyphenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]acetamide
Show/Hide
|
C23H20N4O4S3
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0511561
|
N-(6-chloro-1,3-benzothiazol-2-yl)-2-[[3-(4-fluorophenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]acetamide
Show/Hide
|
C21H14ClFN4O2S3
|
1
|
| 1 |
EC50 = 175 nM
|
|
|
|
CP0426147
|
N-[2-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-4-oxo-3-phenylphthalazine-1-carboxamide
Show/Hide
|
C25H19N5O4S
|
1
|
| 1 |
EC50 = 210 nM
|
|
|
|
CP0489916
|
N-[2-[(6-nitro-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-4-oxo-3-phenylphthalazine-1-carboxamide
Show/Hide
|
C24H16N6O5S
|
1
|
| 1 |
EC50 = 240 nM
|
|
|
|
CP0438729
|
2-[[3-(4-fluorophenyl)-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl]sulfanyl]-N-(6-methoxy-1,3-benzothiazol-2-yl)acetamide
Show/Hide
|
C22H17FN4O3S3
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0481458
|
ethyl 4-[[2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetyl]amino]benzoate
Show/Hide
|
C23H21N3O4S2
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0440131
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(4-phenyl-1,3-thiazol-2-yl)acetamide
Show/Hide
|
C23H18N4O2S3
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0515497
|
N-[2-[(6-fluoro-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-4-oxo-3-phenylphthalazine-1-carboxamide
Show/Hide
|
C24H16FN5O3S
|
1
|
| 1 |
EC50 = 470 nM
|
|
|
|
CP0515507
|
N-(6-methoxyquinolin-2-yl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C24H20N4O3S2
|
1
|
| 1 |
EC50 = 580 nM
|
|
|
|
CP0426151
|
N-(4-ethoxyphenyl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C22H21N3O3S2
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0440126
|
N-[2-(1,3-benzothiazol-2-ylamino)-2-oxoethyl]-4-oxo-3-phenylphthalazine-1-carboxamide
Show/Hide
|
C24H17N5O3S
|
1
|
| 1 |
EC50 = 2600 nM
|
|
|
|
CP0478008
|
N-(1,3-benzothiazol-2-yl)-2-[(3-ethyl-6-methyl-4-oxo-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C18H18N4O2S3
|
1
|
| 1 |
EC50 = 4000 nM
|
|
|
|
CP0481453
|
N-[2-(1,3-benzothiazol-2-ylamino)-2-oxoethyl]-3-(2-methoxyphenyl)-4-oxophthalazine-1-carboxamide
Show/Hide
|
C25H19N5O4S
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0428118
|
ethyl 2-[[2-[(4-oxo-3-phenylphthalazine-1-carbonyl)amino]acetyl]amino]-1,3-benzothiazole-6-carboxylate
Show/Hide
|
C27H21N5O5S
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0449279
|
N-[2-(1,3-benzothiazol-2-ylamino)-2-oxoethyl]-3-(4-fluorophenyl)-4-oxophthalazine-1-carboxamide
Show/Hide
|
C24H16FN5O3S
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0449281
|
4-oxo-N-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-3-phenylphthalazine-1-carboxamide
Show/Hide
|
C20H15N5O3S
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0481452
|
N-[2-(1,3-benzothiazol-2-ylamino)-2-oxoethyl]-3-(4-methoxyphenyl)-4-oxophthalazine-1-carboxamide
Show/Hide
|
C25H19N5O4S
|
1
|
| 1 |
EC50 = 25000 nM
|
|
|
|
CP0515508
|
N-[2-[(6-methoxy-1,3-benzothiazol-2-yl)amino]-2-oxoethyl]-6-oxo-1-phenylpyridine-3-carboxamide
Show/Hide
|
C22H18N4O4S
|
1
|
| 1 |
EC50 > 25000 nM
|
|
|
|
CP0449280
|
N-[4-(dimethylamino)phenyl]-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C22H22N4O2S2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0481457
|
N-(4-acetylphenyl)-2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]acetamide
Show/Hide
|
C22H19N3O3S2
|
1
|
| 1 |
EC50 > 1000 nM
|
|
|
|
CP0387025
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(3-phenylphenyl)acetamide
Show/Hide
|
C26H21N3O2S2
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
|
CP0528633
|
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-(2-phenylphenyl)acetamide
Show/Hide
|
C26H21N3O2S2
|
1
|
| 1 |
EC50 > 5000 nM
|
|
|
