Brief Information of the Compound and Protein
Compound Name
2-[(4-oxo-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]-N-[6-(trifluoromethyl)-1,3-benzothiazol-2-yl]acetamide
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PubChem ID
CID: 71716255
Canonical SMILES
FC(F)(F)c1ccc2nc(NC(=O)CSc3nc4CCSc4c(=O)n3-c3ccccc3)sc2c1
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Compound Formula C22H15F3N4O2S3
Compound Structure
Protein Name
Protein-serine O-palmitoleoyltransferase porcupine
Protein Classification
Enzyme
>
Transferase
Uniprot ID
Q9JJJ7
Gene Name
PORCN
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000309 NCTC clone 929 Mus musculus (Mouse)  1
1
EC50 = 40 nM
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