| Compound ID |
Compound Name |
Compound Formula |
|
CP0545538
|
[(1R)-2-(1-benzofuran-3-yl)-1-[[(1S,2R,4R)-7-oxabicyclo[2.2.1]heptane-2-carbonyl]amino]ethyl]boronic acid
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|
C17H20BNO5
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0550598
|
US10294246, Compound No. 92
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|
C19H20BNO5
|
1
|
| 1 |
IC50 = 8.9 nM
|
|
|
|
CP0564533
|
[(1R)-2-(1-benzofuran-3-yl)-1-(3-methoxypropanoylamino)ethyl]boronic acid
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|
C14H18BNO5
|
1
|
| 1 |
IC50 = 10.6 nM
|
|
|
|
CP0547336
|
[(1R)-2-(1-benzofuran-3-yl)-1-[[(3R)-oxolane-3-carbonyl]amino]ethyl]boronic acid
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|
C15H18BNO5
|
1
|
| 1 |
IC50 = 13.7 nM
|
|
|
|
CP0545536
|
US10294246, Compound No. 6
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|
C18H18BNO4
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0570106
|
US10294246, Compound No. 20
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|
C16H16BN3O4
|
1
|
| 1 |
IC50 = 15.5 nM
|
|
|
|
CP0571391
|
US10294246, Compound No. 18
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|
C16H16BN3O4
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0575636
|
[(1R)-2-(1-benzofuran-3-yl)-1-[[(1R,2S,4S)-7-oxabicyclo[2.2.1]heptane-2-carbonyl]amino]ethyl]boronic acid
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|
C17H20BNO5
|
1
|
| 1 |
IC50 = 19.6 nM
|
|
|
|
CP0564531
|
US10294246, Compound No. 105
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|
C19H19BN2O4
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0547335
|
US10294246, Compound No. 125
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|
C18H17BFNO4
|
1
|
| 1 |
IC50 = 22.8 nM
|
|
|
|
CP0575635
|
US10294246, Compound No. 8
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|
C17H17BN2O4
|
1
|
| 1 |
IC50 = 24.7 nM
|
|
|
|
CP0571153
|
US10294246, Compound No. 132
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|
C18H19BClNO4
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0550601
|
[(1R)-2-(1-benzofuran-3-yl)-1-[(2-methoxyacetyl)amino]ethyl]boronic acid
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|
C13H16BNO5
|
1
|
| 1 |
IC50 = 26.7 nM
|
|
|
|
CP0564532
|
[(1R)-1-acetamido-2-(1-benzofuran-3-yl)ethyl]boronic acid
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|
C12H14BNO4
|
1
|
| 1 |
IC50 = 27.1 nM
|
|
|
|
CP0575641
|
US10294246, Compound No. 75
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|
C19H20BNO4
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0576763
|
[(1R)-2-(1-benzofuran-3-yl)-1-[(2-pyrazol-1-ylacetyl)amino]ethyl]boronic acid
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|
C15H16BN3O4
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0564529
|
[(1R)-2-(1-benzofuran-3-yl)-1-[[(2R)-oxolane-2-carbonyl]amino]ethyl]boronic acid
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|
C15H18BNO5
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0569314
|
US10294246, Compound No. 85
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|
C18H17BClNO4
|
1
|
| 1 |
IC50 = 41.5 nM
|
|
|
|
CP0575644
|
US10294246, Compound No. 90
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|
C19H17BN2O4
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0550599
|
US10294246, Compound No. 134
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|
C19H18BClN2O4
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0571390
|
US10294246, Compound No. 124
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|
C19H22BNO4
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0545537
|
[(1R)-2-(1-benzofuran-3-yl)-1-[[(3S)-oxolane-3-carbonyl]amino]ethyl]boronic acid
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|
C15H18BNO5
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0572729
|
US10294246, Compound No. 130
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|
C20H21BN2O4
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0570105
|
US10294246, Compound No. 19
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|
C17H17BN2O4
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0572728
|
US10294246, Compound No. 126
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|
C19H19BClNO4
|
1
|
| 1 |
IC50 = 164 nM
|
|
|
|
CP0564534
|
[(1R)-2-(1-benzofuran-3-yl)-1-[[(2S)-oxolane-2-carbonyl]amino]ethyl]boronic acid
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|
C15H18BNO5
|
1
|
| 1 |
IC50 = 400 nM
|
|
|
|
CP0572727
|
[(1R)-2-(3,4-dimethylphenyl)-1-[(2-phenylacetyl)amino]ethyl]boronic acid
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|
C18H22BNO3
|
1
|
| 1 |
IC50 = 434 nM
|
|
|
|
CP0575637
|
US10294246, Compound No. 14
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|
C17H20BNO3
|
1
|
| 1 |
IC50 = 438 nM
|
|
|
|
CP0577158
|
[(1R)-2-phenyl-1-[(2-phenylacetyl)amino]ethyl]boronic acid
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|
C16H18BNO3
|
1
|
| 1 |
IC50 = 643 nM
|
|
|
|
CP0575639
|
US10294246, Compound No. 73
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|
C18H17BClNO4
|
1
|
| 1 |
IC50 = 824 nM
|
|
|
|
CP0579795
|
US10294246, Compound No. 110
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|
C18H18BNO4
|
1
|
| 1 |
IC50 = 824 nM
|
|
|
|
CP0573716
|
US10294246, Compound No. 29
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|
C18H22BNO3
|
1
|
| 1 |
IC50 = 896 nM
|
|
|
|
CP0571152
|
[(1R)-2-(4-chlorophenyl)-1-[(2-phenylacetyl)amino]ethyl]boronic acid
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|
C16H17BClNO3
|
1
|
| 1 |
IC50 = 983 nM
|
|
|
|
CP0571392
|
[(1S)-2-(3,4-dimethylphenyl)-1-[(2-phenylacetyl)amino]ethyl]boronic acid
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|
C18H22BNO3
|
1
|
| 1 |
IC50 = 1407 nM
|
|
|
|
CP0550600
|
[(1R)-3-methyl-1-[(2-phenylacetyl)amino]butyl]boronic acid
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|
C13H20BNO3
|
1
|
| 1 |
IC50 = 3300 nM
|
|
|
|
CP0564530
|
US10294246, Compound No. 133
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|
C18H19BClNO4
|
1
|
| 1 |
IC50 = 9670 nM
|
|
|
