| Compound ID |
Compound Name |
Compound Formula |
|
CP0885654
|
(S)-N-((S)-3-(biphenyl-4-yl)-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-(4-methoxyphenyl)-2-((R)-2-(2-morpholinoacetamido)propanamido)propanamide
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|
C37H44N4O7
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
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CP0945818
|
N-((S)-1-((S)-1-((S)-3-(biphenyl-4-yl)-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-ylamino)-3-(4-methoxyphenyl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
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|
C42H43N3O6
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
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CP0907723
|
(S)-N-((S)-3-(biphenyl-4-yl)-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-(4-methoxyphenyl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
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|
C37H44N4O7
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0945819
|
(S)-N-((S)-3-(biphenyl-4-yl)-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-(1H-indol-3-yl)-2-((R)-2-(2-morpholinoacetamido)propanamido)propanamide
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|
C38H43N5O6
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0847941
|
N-((R)-1-((S)-3-(1H-indol-3-yl)-1-((S)-1-((R)-2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
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|
C37H38N4O5
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0400353
|
N-[(2S)-1-[[(2S)-1-[[(2S)-3-cyclohexyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-3-(4-methoxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-3-methyl-1H-indene-2-carboxamide
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|
C36H45N3O6
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0859992
|
N-((R)-1-((S)-3-(4-methoxyphenyl)-1-((S)-1-((R)-2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
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|
C36H39N3O6
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0949827
|
(S)-3-(4-methoxyphenyl)-N-((S)-1-((R)-2-methyloxiran-2-yl)-3-(naphthalen-2-yl)-1-oxopropan-2-yl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
Show/Hide
|
C35H42N4O7
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0945962
|
N-((R)-1-((S)-1-((S)-3-(biphenyl-4-yl)-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-ylamino)-3-(4-methoxyphenyl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
Show/Hide
|
C42H43N3O6
|
1
|
| 1 |
IC50 = 3.3 nM
|
|
|
|
CP0448435
|
N-[(2S)-1-[[(2S)-3-(4-methoxyphenyl)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-3-methyl-1H-indene-2-carboxamide
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|
C36H39N3O6
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0958709
|
N-((R)-1-((S)-1-((S)-3-(biphenyl-4-yl)-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
Show/Hide
|
C43H42N4O5
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0062987
|
(2S)-3-(4-methoxyphenyl)-N-[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxo-3-phenylpropan-2-yl]-2-[[(2S)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide
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|
C31H40N4O7
|
1
|
| 1 |
IC50 = 5.7 nM
|
|
|
|
CP0885679
|
(S)-N-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-(4-methoxyphenyl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
Show/Hide
|
C31H46N4O7
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
|
CP0868641
|
N-((R)-1-((S)-1-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
Show/Hide
|
C37H44N4O5
|
1
|
| 1 |
IC50 = 8.3 nM
|
|
|
|
CP0411613
|
N-[(2R)-1-[[(2S)-1-[[(2S)-3-cyclohexyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-3-(4-methoxyphenyl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]-3-methyl-1H-indene-2-carboxamide
Show/Hide
|
C36H45N3O6
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0864817
|
(S)-3-(1H-indol-3-yl)-N-((S)-1-((R)-2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-yl)-2-((R)-2-(2-morpholinoacetamido)propanamido)propanamide
Show/Hide
|
C32H39N5O6
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0907724
|
(S)-3-(4-methoxyphenyl)-N-((S)-1-((R)-2-methyloxiran-2-yl)-1-oxo-3-phenylpropan-2-yl)-2-((R)-2-(2-morpholinoacetamido)propanamido)propanamide
Show/Hide
|
C31H40N4O7
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0864816
|
(S)-N-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-yl)-3-(1H-indol-3-yl)-2-((R)-2-(2-morpholinoacetamido)propanamido)propanamide
Show/Hide
|
C32H45N5O6
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0386861
|
(2S)-N-[(2S)-3-cyclohexyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]-3-(4-methoxyphenyl)-2-[[(2R)-2-[(2-morpholin-4-ylacetyl)amino]propanoyl]amino]propanamide
Show/Hide
|
C31H46N4O7
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0850423
|
N-((R)-1-((S)-3-(1H-indol-3-yl)-1-((S)-4-(methylsulfonyl)-1-phenylbut-3-en-2-ylamino)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
Show/Hide
|
C36H38N4O5S
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0955124
|
(S)-3-(4-methoxyphenyl)-N-((S)-1-((R)-2-methyloxiran-2-yl)-3-(naphthalen-1-yl)-1-oxopropan-2-yl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
Show/Hide
|
C35H42N4O7
|
1
|
| 1 |
IC50 = 244 nM
|
|
|
|
CP0966265
|
(S)-3-(4-methoxyphenyl)-N-((S)-4-(methylsulfonyl)-1-phenylbut-3-en-2-yl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
Show/Hide
|
C30H40N4O7S
|
1
|
| 1 |
IC50 = 392 nM
|
|
|
|
CP0955125
|
N-((R)-1-((S)-1-((S)-1-cyclohexyl-4-(methylsulfonyl)but-3-en-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
Show/Hide
|
C36H44N4O5S
|
1
|
| 1 |
IC50 = 632 nM
|
|
|
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CP0907725
|
(S)-N-((S)-1-cyclohexyl-4-(methylsulfonyl)but-3-en-2-yl)-3-(4-methoxyphenyl)-2-((S)-2-(2-morpholinoacetamido)propanamido)propanamide
Show/Hide
|
C30H46N4O7S
|
1
|
| 1 |
IC50 = 5700 nM
|
|
|
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CP0859169
|
(S)-N-[(S)-1-Adamantan-1-ylmethyl-2-((R)-2-methyl-oxiranyl)-2-oxo-ethyl]-3-(4-methoxy-phenyl)-2-[(S)-2-(2-morpholin-4-yl-acetylamino)-propionylamino]-propionamide
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|
C35H50N4O7
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
