| Compound ID |
Compound Name |
Compound Formula |
|
CP0669565
|
(S)-2-(1-(6-chloro-7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)ethylamino)-4-methoxypyrimidine-5-carbonitrile
Show/Hide
|
C18H16ClN5O3
|
5
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 3 nM
|
|
|
| 3 |
IC50 = 4 nM
|
|
|
| 4 |
IC50 = 5 nM
|
|
|
| 5 |
IC50 = 129 nM
|
|
|
|
CP0117201
|
Ft-2102
Show/Hide
|
C18H15ClN4O2
|
4
|
| 1 |
IC50 = 6 nM
|
|
|
| 2 |
IC50 = 9 nM
|
|
|
| 3 |
IC50 = 39 nM
|
|
|
| 4 |
IC50 = 42 nM
|
|
|
|
CP0714073
|
(S)-2-((1-(6-Chloro-2-oxo-1,2-dihydroquinolin-3-yl)ethyl)amino)-4-methoxypyrimidine-5-carbonitrile
Show/Hide
|
C17H14ClN5O2
|
5
|
| 1 |
IC50 = 18 nM
|
|
|
| 2 |
IC50 = 60 nM
|
|
|
| 3 |
IC50 = 120 nM
|
|
|
| 4 |
IC50 = 130 nM
|
|
|
| 5 |
IC50 = 1490 nM
|
|
|
|
CP0096015
|
(2S)-2-(2-chlorophenyl)-2-[[2-[(2S)-1-(4-cyanopyridin-2-yl)-5-oxopyrrolidin-2-yl]acetyl]-(5-fluoropyridin-3-yl)amino]-N-(3,3-difluorocyclobutyl)acetamide
Show/Hide
|
C29H24ClF3N6O3
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0069129
|
US10028961, Compound 121
Show/Hide
|
C17H22F3N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0076794
|
US10028961, Compound 101
Show/Hide
|
C14H13ClF6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0179549
|
US10028961, Compound 128
Show/Hide
|
C15H13F7N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0179571
|
US10028961, Compound 105
Show/Hide
|
C20H22F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0233887
|
US10028961, Compound 160
Show/Hide
|
C20H22F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387374
|
US10028961, Compound 141
Show/Hide
|
C13H12F9N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387375
|
US10028961, Compound 178
Show/Hide
|
C20H15F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387376
|
US10028961, Compound 183
Show/Hide
|
C19H21F7N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387380
|
US10028961, Compound 404
Show/Hide
|
C13H11F9N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387381
|
US10028961, Compound 120
Show/Hide
|
C17H12ClF4N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387382
|
US10028961, Compound 129
Show/Hide
|
C17H18ClF4N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387383
|
US10028961, Compound 186
Show/Hide
|
C20H23F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387384
|
US10028961, Compound 216
Show/Hide
|
C19H19F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387385
|
US10028961, Compound 217
Show/Hide
|
C23H17F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387386
|
US10028961, Compound 109
Show/Hide
|
C18H14ClF4N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387387
|
US10028961, Compound 110
Show/Hide
|
C20H27ClN6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387390
|
US10028961, Compound 407
Show/Hide
|
C17H14F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387391
|
US10028961, Compound 158
Show/Hide
|
C20H15F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387392
|
US10028961, Compound 199
Show/Hide
|
C24H22F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387393
|
US10946023, Compound 201
Show/Hide
|
C19H15F6N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387394
|
US10028961, Compound 230
Show/Hide
|
C24H22F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387396
|
US10028961, Compound 372
Show/Hide
|
C23H20F4N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387397
|
US10028961, Compound 378
Show/Hide
|
C22H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387398
|
US10028961, Compound 386
Show/Hide
|
C14H12F9N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387399
|
US10028961, Compound 245
Show/Hide
|
C19H16F4N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387400
|
US10028961, Compound 298
Show/Hide
|
C18H17F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387401
|
US10028961, Compound 104
Show/Hide
|
C16H17ClF6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387405
|
US10028961, Compound 211
Show/Hide
|
C25H24F4N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387408
|
US10946023, Compound 342
Show/Hide
|
C22H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387411
|
US10028961, Compound 413
Show/Hide
|
C17H11F7N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387412
|
US10028961, Compound 102
Show/Hide
|
C19H19F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387413
|
US10028961, Compound 115
Show/Hide
|
C19H15ClF5N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387414
|
US10028961, Compound 116
Show/Hide
|
C19H14F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387415
|
US10028961, Compound 155
Show/Hide
|
C18H20F6N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387416
|
US10028961, Compound 156
Show/Hide
|
C13H12ClF6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387418
|
US10028961, Compound 184
Show/Hide
|
C25H25F5N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387438
|
US10028961, Compound 113
Show/Hide
|
C18H19ClF4N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387439
|
US10028961, Compound 119
Show/Hide
|
C17H11F7N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0387440
|
US10028961, Compound 123
Show/Hide
|
C20H15F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393388
|
US10028961, Compound 136
Show/Hide
|
C14H13ClF6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393543
|
US10028961, Compound 125
Show/Hide
|
C21H17F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393561
|
US10028961, Compound 138
Show/Hide
|
C18H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393562
|
US10028961, Compound 147
Show/Hide
|
C19H22ClF4N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393564
|
US10946023, Compound 151
Show/Hide
|
C23H19F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393566
|
US10028961, Compound 159
Show/Hide
|
C18H13F7N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393567
|
US10028961, Compound 163
Show/Hide
|
C21H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393568
|
US10028961, Compound 164
Show/Hide
|
C22H17F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393570
|
US10946023, Compound 168
Show/Hide
|
C22H17F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393572
|
US10946023, Compound 175
Show/Hide
|
C20H15F4N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393573
|
US10028961, Compound 193
Show/Hide
|
C21H25F3N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393574
|
US10028961, Compound 214
Show/Hide
|
C18H20F3N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0393575
|
US10028961, Compound 221
Show/Hide
|
C20H15F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0394779
|
US10946023, Compound 392
Show/Hide
|
C19H15F6N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0394780
|
US10028961, Compound 402
Show/Hide
|
C17H18F6N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0394782
|
US10028961, Compound 410
Show/Hide
|
C18H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401742
|
US10028961, Compound 103
Show/Hide
|
C16H17ClF6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401743
|
US10028961, Compound 130
Show/Hide
|
C14H13ClF6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401744
|
US10028961, Compound 133
Show/Hide
|
C23H19F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401745
|
US10028961, Compound 139
Show/Hide
|
C19H14F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401746
|
US10028961, Compound 140
Show/Hide
|
C18H12F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401747
|
US10028961, Compound 146
Show/Hide
|
C17H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401748
|
US10028961, Compound 148
Show/Hide
|
C17H17F7N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401749
|
US10028961, Compound 152
Show/Hide
|
C23H21F5N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401751
|
US10028961, Compound 157
Show/Hide
|
C18H19ClF4N6
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0401753
|
US10946023, Compound 169
Show/Hide
|
C20H16F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401754
|
US10028961, Compound 170
Show/Hide
|
C15H13F7N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401755
|
US10028961, Compound 171
Show/Hide
|
C18H12F9N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401756
|
US10946023, Compound 174
Show/Hide
|
C21H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401758
|
US10028961, Compound 179
Show/Hide
|
C18H14F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401759
|
US10946023, Compound 189
Show/Hide
|
C24H21F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401760
|
US10028961, Compound 192
Show/Hide
|
C21H17F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401761
|
US10028961, Compound 203
Show/Hide
|
C17H18F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401763
|
US10028961, Compound 209
Show/Hide
|
C16H16F6N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401764
|
US10028961, Compound 218
Show/Hide
|
C22H26F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401765
|
US10028961, Compound 223
Show/Hide
|
C19H21F7N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401766
|
US10028961, Compound 232
Show/Hide
|
C17H10F9N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401768
|
US10028961, Compound 252
Show/Hide
|
C19H19F7N6O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401769
|
US10028961, Compound 259
Show/Hide
|
C22H21F3N8O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401771
|
US10028961, Compound 293
Show/Hide
|
C20H22F7N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0401783
|
US10028961, Compound 167
Show/Hide
|
C22H21ClN8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401784
|
US10028961, Compound 182
Show/Hide
|
C23H20ClF5N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401785
|
US10028961, Compound 224
Show/Hide
|
C21H24F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401786
|
US10028961, Compound 253
Show/Hide
|
C19H15F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401787
|
US10028961, Compound 260
Show/Hide
|
C20H16F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401850
|
US10028961, Compound 261
Show/Hide
|
C22H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401852
|
US10028961, Compound 289
Show/Hide
|
C19H19F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401864
|
US10028961, Compound 344
Show/Hide
|
C14H12F9N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0401865
|
US10028961, Compound 355
Show/Hide
|
C21H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401867
|
US10028961, Compound 375
Show/Hide
|
C22H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401868
|
US10028961, Compound 108
Show/Hide
|
C18H14F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401869
|
US10028961, Compound 124
Show/Hide
|
C21H15F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401870
|
US10028961, Compound 144
Show/Hide
|
C15H14ClF4N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0401871
|
US10028961, Compound 162
Show/Hide
|
C19H17F3N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405654
|
US10028961, Compound 153
Show/Hide
|
C19H16F5N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405662
|
US10028961, Compound 370
Show/Hide
|
C19H21F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405663
|
US10028961, Compound 380
Show/Hide
|
C21H16F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405664
|
US10028961, Compound 409
Show/Hide
|
C16H15F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405665
|
US10028961, Compound 411
Show/Hide
|
C16H15F6N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0405666
|
US10028961, Compound 127
Show/Hide
|
C22H19ClF2N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405667
|
US10028961, Compound 197
Show/Hide
|
C17H12F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405668
|
US10028961, Compound 200
Show/Hide
|
C18H15ClF3N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405670
|
US10028961, Compound 349
Show/Hide
|
C19H15F6N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405671
|
US10946023, Compound 382
Show/Hide
|
C22H20F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405696
|
US10028961, Compound 390
Show/Hide
|
C18H12F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0405697
|
US10946023, Compound 394
Show/Hide
|
C23H20F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412011
|
US10028961, Compound 389
Show/Hide
|
C20H16F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412014
|
US10028961, Compound 161
Show/Hide
|
C16H14F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412018
|
US10028961, Compound 210
Show/Hide
|
C17H12F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412019
|
US10028961, Compound 213
Show/Hide
|
C19H13F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412020
|
US10946023, Compound 226
Show/Hide
|
C20H14F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412023
|
US10028961, Compound 400
Show/Hide
|
C16H11F9N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412024
|
US10028961, Compound 401
Show/Hide
|
C21H16F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412025
|
US10028961, Compound 137
Show/Hide
|
C23H19F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412686
|
US10028961, Compound 360
Show/Hide
|
C21H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412689
|
US10028961, Compound 190
Show/Hide
|
C19H13F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0412692
|
US10946023, Compound 215
Show/Hide
|
C19H14ClF3N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0420686
|
US10028961, Compound 142
Show/Hide
|
C14H13ClF6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0424115
|
US10028961, Compound 2
Show/Hide
|
C19H23F3N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0427569
|
US10028961, Compound 1
Show/Hide
|
C17H19F3N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0429242
|
US10028961, Compound 393
Show/Hide
|
C18H14F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0429244
|
US10028961, Compound 195
Show/Hide
|
C18H12F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0429882
|
US10028961, Compound 145
Show/Hide
|
C17H16F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0429883
|
US10028961, Compound 154
Show/Hide
|
C20H13F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0429886
|
US10028961, Compound 391
Show/Hide
|
C19H14F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0445766
|
US10028961, Compound 207
Show/Hide
|
C16H11F6N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446178
|
US10028961, Compound 114
Show/Hide
|
C13H11F9N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446195
|
US10028961, Compound 185
Show/Hide
|
C21H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446197
|
US10028961, Compound 231
Show/Hide
|
C21H19F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446200
|
US10028961, Compound 126
Show/Hide
|
C15H14F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446203
|
US10028961, Compound 228
Show/Hide
|
C22H23F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446204
|
US10028961, Compound 257
Show/Hide
|
C22H17F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446209
|
US10946023, Compound 341
Show/Hide
|
C22H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446210
|
US10028961, Compound 356
Show/Hide
|
C16H11F9N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446211
|
US10028961, Compound 376
Show/Hide
|
C22H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446212
|
US10028961, Compound 387
Show/Hide
|
C18H14F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446214
|
US10028961, Compound 176
Show/Hide
|
C19H22F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446215
|
US10028961, Compound 181
Show/Hide
|
C20H15F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446216
|
US10028961, Compound 198
Show/Hide
|
C19H24F2N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446217
|
US10946023, Compound 229
Show/Hide
|
C25H21F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446218
|
US10028961, Compound 237
Show/Hide
|
C18H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446219
|
US10028961, Compound 248
Show/Hide
|
C19H18ClF3N6O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446221
|
US10028961, Compound 354
Show/Hide
|
C17H15F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446222
|
US10028961, Compound 357
Show/Hide
|
C20H24F6N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446223
|
US10028961, Compound 381
Show/Hide
|
C18H14F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446224
|
US10028961, Compound 384
Show/Hide
|
C24H22F4N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446225
|
US10028961, Compound 398
Show/Hide
|
C21H20F3N7O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0446228
|
US10028961, Compound 267
Show/Hide
|
C21H19F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450646
|
US10028961, Compound 352
Show/Hide
|
C21H16F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450647
|
US10028961, Compound 365
Show/Hide
|
C19H13F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450650
|
US10028961, Compound 403
Show/Hide
|
C15H14F6N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450651
|
US10028961, Compound 118
Show/Hide
|
C19H19F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450653
|
US10028961, Compound 122
Show/Hide
|
C18H11F6N7S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450659
|
US10028961, Compound 106
Show/Hide
|
C17H12F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450660
|
US10028961, Compound 350
Show/Hide
|
C21H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450673
|
US10028961, Compound 172
Show/Hide
|
C20H15F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450674
|
US10028961, Compound 205
Show/Hide
|
C19H22F6N6S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450675
|
US10028961, Compound 256
Show/Hide
|
C16H14F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450679
|
US10028961, Compound 246
Show/Hide
|
C22H23F3N6O
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0450709
|
US10028961, Compound 191
Show/Hide
|
C21H21F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450958
|
US10028961, Compound 194
Show/Hide
|
C18H18F7N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0450962
|
US10028961, Compound 377
Show/Hide
|
C20H15F6N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450963
|
US10028961, Compound 75
Show/Hide
|
C18H23F3N6O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0450965
|
US10028961, Compound 177
Show/Hide
|
C16H11F9N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0457656
|
US10028961, Compound 72
Show/Hide
|
C18H19ClN6O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0457657
|
US10028961, Compound 74
Show/Hide
|
C16H25N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0457658
|
US10028961, Compound 111
Show/Hide
|
C19H19F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0457659
|
US10028961, Compound 117
Show/Hide
|
C20H18F3N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0457660
|
US10028961, Compound 150
Show/Hide
|
C23H20F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0457661
|
US10028961, Compound 187
Show/Hide
|
C18H18F6N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0457662
|
US10028961, Compound 268
Show/Hide
|
C18H22F3N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0457665
|
US10028961, Compound 363
Show/Hide
|
C15H16F9N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0457666
|
US10028961, Compound 405
Show/Hide
|
C20H15F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0458083
|
US10028961, Compound 143
Show/Hide
|
C19H19F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0458085
|
US10028961, Compound 258
Show/Hide
|
C21H24F4N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0466620
|
US10028961, Compound 351
Show/Hide
|
C21H16F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0466622
|
US10028961, Compound 366
Show/Hide
|
C17H17F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0466623
|
US10028961, Compound 374
Show/Hide
|
C21H25F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0466681
|
US10028961, Compound 368
Show/Hide
|
C19H14F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0471768
|
US10028961, Compound 361
Show/Hide
|
C22H20F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0471769
|
US10028961, Compound 369
Show/Hide
|
C19H14F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0471770
|
US10946023, Compound 373
Show/Hide
|
C22H18F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473719
|
US10028961, Compound 202
Show/Hide
|
C25H20F5N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473720
|
US10028961, Compound 399
Show/Hide
|
C18H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473721
|
US10028961, Compound 408
Show/Hide
|
C18H19F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473722
|
US10028961, Compound 73
Show/Hide
|
C18H29N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0473723
|
US10028961, Compound 343
Show/Hide
|
C19H14F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473724
|
US10028961, Compound 358
Show/Hide
|
C20H16F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473725
|
US10028961, Compound 359
Show/Hide
|
C23H17F6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473726
|
US10028961, Compound 367
Show/Hide
|
C20H16F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473727
|
US10946023, Compound 132
Show/Hide
|
C19H13F6N7S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473728
|
US10028961, Compound 165
Show/Hide
|
C20H18F5N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473729
|
US10028961, Compound 204
Show/Hide
|
C21H17F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0473730
|
US10028961, Compound 220
Show/Hide
|
C26H22F5N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0473733
|
US10028961, Compound 395
Show/Hide
|
C20H21F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0476930
|
US10028961, Compound 149
Show/Hide
|
C17H15F7N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477101
|
US10028961, Compound 340
Show/Hide
|
C19H14F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477102
|
US10028961, Compound 347
Show/Hide
|
C22H19F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477103
|
US10028961, Compound 348
Show/Hide
|
C22H19F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477105
|
US10028961, Compound 364
Show/Hide
|
C23H16ClF6N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477106
|
US10028961, Compound 379
Show/Hide
|
C17H13F6N7S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477107
|
US10946023, Compound 383
Show/Hide
|
C24H16F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477111
|
US10028961, Compound 212
Show/Hide
|
C20H23ClF4N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477112
|
US10028961, Compound 250
Show/Hide
|
C20H17F5N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477113
|
US10028961, Compound 277
Show/Hide
|
C17H15F7N6O
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0477122
|
US10028961, Compound 353
Show/Hide
|
C18H13F8N7S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477123
|
US10028961, Compound 388
Show/Hide
|
C17H11F8N7S
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0477124
|
US10028961, Compound 406
Show/Hide
|
C18H18F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0479003
|
US10028961, Compound 112
Show/Hide
|
C19H14F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0479004
|
US10028961, Compound 131
Show/Hide
|
C22H27ClN6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0484674
|
US10028961, Compound 346
Show/Hide
|
C17H17F9N6
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0484687
|
US10028961, Compound 385
Show/Hide
|
C24H20F5N9
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0494043
|
US10028961, Compound 420
Show/Hide
|
C20H24F3N5
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0494046
|
US10028961, Compound 107
Show/Hide
|
C16H11F8N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0513506
|
US10028961, Compound 339
Show/Hide
|
C16H16F9N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0517883
|
US10028961, Compound 173
Show/Hide
|
C18H14F8N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0517893
|
US10028961, Compound 244
Show/Hide
|
C20H17F4N7O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0517901
|
US10028961, Compound 412
Show/Hide
|
C18H19F6N7
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0534801
|
US10028961, Compound 397
Show/Hide
|
C21H20F6N6O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0539506
|
US10028961, Compound 325
Show/Hide
|
C18H16F5N7O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0539510
|
US10028961, Compound 371
Show/Hide
|
C23H16F7N7
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0851745
|
2-(4-(3,5-difluorophenylamino)-6-(3-(trifluoromethyl)-1H-pyrazol-1-yl)-1,3,5-triazin-2-ylamino)-1,1-difluoroethanol
Show/Hide
|
C15H10F7N7O
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0859550
|
2-methyl-2-(4-(6-(trifluoromethyl)pyridin-2-yl)-6-(2-(trifluoromethyl)pyridin-4-ylamino)-1,3,5-triazin-2-ylamino)propanenitrile
Show/Hide
|
C19H14F6N8
|
1
|
| 1 |
IC50 < 50 nM
|
|
|
|
CP0860895
|
N2,N4-di(3-oxabicyclo[3.1.0]hexan-6-yl)-6-phenyl-1,3,5-triazine-2,4-diamine
Show/Hide
|
C19H21N5O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0865294
|
1-(4-(4-(6-(trifluoromethyl)pyridin-2-yl)-6-(1,1,1-trifluoropropan-2-ylamino)-1,3,5-triazin-2-ylamino)pyridin-2-yl)cyclopropanecarbonitrile
Show/Hide
|
C21H16F6N8
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1
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| 1 |
IC50 < 50 nM
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CP0887458
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2-(4-(3-chloro-5-fluorophenylamino)-6-(3-(1,1-difluoroethyl)-1H-pyrazol-1-yl)-1,3,5-triazin-2-ylamino)-1,1-difluoroethanol
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C16H13ClF5N7O
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1
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| 1 |
IC50 < 50 nM
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CP0928973
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N2,N4-di(but-3-enyl)-6-phenyl-1,3,5-triazine-2,4-diamine
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C17H21N5
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1
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| 1 |
IC50 = 50 nM
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CP0057375
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N-cyclohexyl-2-(3-fluoro-N-[2-(2-methylimidazol-1-yl)acetyl]anilino)-2-(2-methylphenyl)acetamide
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C27H31FN4O2
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1
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| 1 |
IC50 = 70 nM
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CP0387388
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US10028961, Compound 308
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C20H23F6N7
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1
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| 1 |
IC50 = 100 nM
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CP0387395
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US10028961, Compound 272
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C29H25F5N6
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1
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| 1 |
IC50 = 100 nM
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CP0387417
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US10028961, Compound 180
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C16H17ClF6N6
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1
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| 1 |
IC50 = 100 nM
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CP0387420
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US10028961, Compound 227
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C22H22F5N9
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1
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| 1 |
IC50 = 100 nM
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CP0394783
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US10028961, Compound 222
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C23H23F5N8
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1
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| 1 |
IC50 = 100 nM
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CP0401767
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US10028961, Compound 249
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C20H24F5N7
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1
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| 1 |
IC50 = 100 nM
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CP0401770
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US10028961, Compound 270
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C20H22F7N7
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1
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| 1 |
IC50 = 100 nM
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CP0405669
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US10028961, Compound 279
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C16H22IN7
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1
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| 1 |
IC50 = 100 nM
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CP0446196
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US10028961, Compound 196
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C16H17ClF6N6
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1
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| 1 |
IC50 = 100 nM
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CP0446199
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US10028961, Compound 251
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C16H14F7N7
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1
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| 1 |
IC50 = 100 nM
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CP0446206
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US10028961, Compound 283
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C20H24F6N6S
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1
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| 1 |
IC50 = 100 nM
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CP0446207
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US10028961, Compound 288
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C19H17F3N8O
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1
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| 1 |
IC50 = 100 nM
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CP0450636
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US10028961, Compound 419
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C18H20F3N5
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1
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| 1 |
IC50 = 100 nM
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CP0457663
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US10028961, Compound 302
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C18H22ClF4N7
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1
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| 1 |
IC50 = 100 nM
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CP0466682
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US10028961, Compound 287
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C19H23F5N6O
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1
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| 1 |
IC50 = 100 nM
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CP0477121
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US10028961, Compound 345
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C16H16F9N7
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1
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| 1 |
IC50 = 100 nM
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CP0928972
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N2-isopropyl-6-phenyl-N4-(tetrahydro-2H-pyran-3-yl)-1,3,5-triazine-2,4-diamine
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C17H23N5O
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1
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| 1 |
IC50 = 100 nM
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CP0070790
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N-cyclohexyl-2-(3-fluoro-N-(2-thiophen-2-ylacetyl)anilino)-2-(2-methylphenyl)acetamide
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C27H29FN2O2S
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1
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| 1 |
IC50 = 190 nM
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CP0286878
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N-cyclohexyl-2-(3-fluoro-N-(2-pyridin-4-ylacetyl)anilino)-2-(2-methylphenyl)acetamide
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C28H30FN3O2
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1
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| 1 |
IC50 = 210 nM
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CP0057374
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N-cyclohexyl-2-(3-fluoro-N-[2-(2-methylbenzimidazol-1-yl)acetyl]anilino)-2-(2-methylphenyl)acetamide
Show/Hide
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C31H33FN4O2
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1
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| 1 |
IC50 = 240 nM
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CP0165474
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6-{[(6-chloro-2-oxo-1,2-
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C17H13ClN4O
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2
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| 1 |
IC50 = 258 nM
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| 2 |
IC50 = 274 nM
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CP0283017
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N-cyclohexyl-2-(3-fluoro-N-[2-(1,3-thiazol-4-yl)acetyl]anilino)-2-(2-methylphenyl)acetamide
Show/Hide
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C26H28FN3O2S
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1
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| 1 |
IC50 = 290 nM
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CP0225556
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4-{[(6-chloro-2-oxo-1,2-
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C18H14ClN3O2
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2
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| 1 |
IC50 = 316 nM
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| 2 |
IC50 = 1250 nM
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CP0070645
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N-cyclohexyl-2-(3-fluoro-N-[2-(1H-indol-3-yl)acetyl]anilino)-2-(2-methylphenyl)acetamide
Show/Hide
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C31H32FN3O2
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1
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| 1 |
IC50 = 360 nM
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CP0176272
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N-cyclohexyl-2-(3-fluoro-N-(2-indol-1-ylacetyl)anilino)-2-(2-methylphenyl)acetamide
Show/Hide
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C31H32FN3O2
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1
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| 1 |
IC50 = 370 nM
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CP0070647
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N-cyclopentyl-2-(3-fluoro-N-(2-thiophen-2-ylacetyl)anilino)-2-(2-methylphenyl)acetamide
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C26H27FN2O2S
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1
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| 1 |
IC50 = 580 nM
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CP0446220
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US10028961, Compound 285
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C18H25N7
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1
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| 1 |
IC50 >= 1000 nM
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CP0477100
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US10028961, Compound 278
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C18H23ClN6
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1
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| 1 |
IC50 >= 1000 nM
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CP0494045
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US10028961, Compound 326
Show/Hide
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C19H22F5N7
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1
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| 1 |
IC50 >= 1000 nM
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