Brief Information of the Cell Line and Protein
Cell Line ID: CL000041 , LTK-
 Cell Line Info 
Category Transformed cell line
Organism
Mus musculus (Mouse)
Cellosaurus ID
CVCL_3392
Protein ID: PT02075 , Alpha-1D adrenergic receptor
 Protein Info 
Gene Name ADRA1D
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P23944
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000041
 Cell Line Info 
 Protein ID: PT02075
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0035002
 Compound Info 
(R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-2-methoxybenzenesulfonamide
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C20H28N2O5S
  1
1
Ki = 0.07 nM
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CP0300622
 Compound Info 
7-Methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C24H27N3O4
  1
1
Ki = 0.21 nM
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CP0277233
 Compound Info 
6-Methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione
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C22H25N3O4S
  1
1
Ki = 0.24 nM
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CP0150194
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-benzo[4,5]thieno[3,2-d]pyrimidine-7-carboxylic acid amide
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C26H26N4O4S
  1
1
Ki = 0.27 nM
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CP0285996
 Compound Info 
2-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4H-9-thia-2,4,6-triaza-fluorene-1,3-dione
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C24H24N4O3S
  1
1
Ki = 0.28 nM
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CP0257880
 Compound Info 
8-Chloro-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C25H24ClN3O3S
  1
1
Ki = 0.31 nM
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CP0215556
 Compound Info 
5-[2-[(3aR,9bR)-6-methoxy-1,3,3a,4,5,9b-hexahydrobenzo[e]isoindol-2-yl]ethyl]-8-thia-3,5,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),10,12-tetraene-4,6-dione
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C24H24N4O3S
  1
1
Ki = 0.37 nM
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CP0107697
 Compound Info 
N-[3-[2-[(3aR,9bR)-6-methoxy-1,3,3a,4,5,9b-hexahydrobenzo[e]isoindol-2-yl]ethyl]-2,4-dioxo-1H-quinazolin-7-yl]acetamide
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C25H28N4O4
  1
1
Ki = 0.41 nM
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CP0087515
 Compound Info 
2-[2-((3aR,9bR)-6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4H-9-thia-2,4,5-triaza-fluorene-1,3-dione
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C24H24N4O3S
  1
1
Ki = 0.51 nM
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CP0306128
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-benzo[4,5]thieno[3,2-d]pyrimidine-8-carboxylic acid amide
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C26H26N4O4S
  1
1
Ki = 0.51 nM
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CP0111306
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-thieno[3,4-d]pyrimidine-2,4-dione
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C21H23N3O3S
  1
1
Ki = 0.52 nM
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CP0117377
 Compound Info 
7-Chloro-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C23H24ClN3O3
  1
1
Ki = 0.58 nM
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CP0306296
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-benzo[4,5]thieno[3,2-d]pyrimidine-8-carbonitrile
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C26H24N4O3S
  1
1
Ki = 0.59 nM
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CP0272523
 Compound Info 
6-Chloro-2-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4H-9-thia-2,4,5-triaza-fluorene-1,3-dione
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C24H23ClN4O3S
  1
1
Ki = 0.61 nM
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CP0111505
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C23H25N3O3
  1
1
Ki = 0.62 nM
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CP0181767
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-benzo[4,5]thieno[3,2-d]pyrimidine-8-carboxylic acid dimethylamide
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C28H30N4O4S
  1
1
Ki = 0.63 nM
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CP0105963
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-7-phenyl-1H-thieno[3,2-d]pyrimidine-2,4-dione
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C27H27N3O3S
  1
1
Ki = 0.66 nM
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CP0306109
 Compound Info 
(Cis)3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-benzo[4,5]furo[3,2-d]pyrimidine-2,4-dione
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C25H25N3O4
  1
1
Ki = 0.68 nM
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CP0303772
 Compound Info 
7,8-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C25H29N3O5
  1
1
Ki = 0.68 nM
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CP0278691
 Compound Info 
7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-5H-9-thia-1,5,7-triaza-fluorene-6,8-dione
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C24H24N4O3S
  1
1
Ki = 0.69 nM
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CP0366100
 Compound Info 
5-Chloro-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C23H24ClN3O3
  1
1
Ki = 0.69 nM
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CP0339131
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-7-methyl-1H-thieno[3,2-d]pyrimidine-2,4-dione
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C22H25N3O3S
  1
1
Ki = 0.71 nM
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CP0272442
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-6,7-dimethyl-1H-quinazoline-2,4-dione
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C25H29N3O3
  1
1
Ki = 0.73 nM
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CP0111500
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-benzo[4,5]thieno[3,2-d]pyrimidine-7-carbonitrile
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C26H24N4O3S
  1
1
Ki = 0.74 nM
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CP0172953
 Compound Info 
(Cis)2-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4,9-dihydro-2,4,9-triaza-fluorene-1,3-dione
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C25H26N4O3
  1
1
Ki = 0.74 nM
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CP0311747
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-quinazoline-7-carbonitrile
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C24H24N4O3
  1
1
Ki = 0.77 nM
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CP0339119
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-quinazoline-7-carboxylic acid methyl ester
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C25H27N3O5
  1
1
Ki = 0.77 nM
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CP0172104
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-9-methyl-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C26H27N3O3S
  1
1
Ki = 0.88 nM
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CP0334603
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-7,8-dimethyl-1H-quinazoline-2,4-dione
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C25H29N3O3
  1
1
Ki = 0.89 nM
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CP0277241
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione
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C21H23N3O3S
  1
1
Ki = 0.92 nM
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CP0816886
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione
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C21H23N3O3S
  1
1
Ki = 0.92 nM
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CP0049024
 Compound Info 
1-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-4-((tetrahydro-2-furanyl)carbonyl)piperazine
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C19H25N5O4
  1
1
Ki = 1.01 nM
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CP0339125
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-thieno[2,3-d]pyrimidine-2,4-dione
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C21H23N3O3S
  1
1
Ki = 1.01 nM
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CP0208716
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-8-methyl-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C26H27N3O3S
  1
1
Ki = 1.04 nM
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CP0215114
 Compound Info 
9-Methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C26H27N3O4S
  1
1
Ki = 1.07 nM
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CP0200691
 Compound Info 
3-Methoxy-7-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-5H-9-thia-1,4,5,7-tetraaza-fluorene-6,8-dione
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C24H25N5O4S
  1
1
Ki = 1.1 nM
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CP0290436
 Compound Info 
6-Methoxy-2-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4H-9-thia-2,4,5-triaza-fluorene-1,3-dione
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C25H26N4O4S
  1
1
Ki = 1.1 nM
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CP0104354
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-5-methyl-1H-quinazoline-2,4-dione
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C24H27N3O3
  1
1
Ki = 1.13 nM
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CP0281096
 Compound Info 
6-Methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C24H27N3O4
  1
1
Ki = 1.13 nM
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CP0318718
 Compound Info 
8-Methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C24H27N3O4
  1
1
Ki = 1.15 nM
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CP0308881
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-7-nitro-1H-quinazoline-2,4-dione
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C23H24N4O5
  1
1
Ki = 1.2 nM
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CP0107696
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-8-nitro-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C25H24N4O5S
  1
1
Ki = 1.31 nM
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CP0200627
 Compound Info 
9-Chloro-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C25H24ClN3O3S
  1
1
Ki = 1.32 nM
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CP0306131
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-thieno[3,2-d]pyrimidine-6-carboxylic acid methyl ester
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C23H25N3O5S
  1
1
Ki = 1.38 nM
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CP0146707
 Compound Info 
6,7-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C25H29N3O5
  1
1
Ki = 1.4 nM
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CP0244629
 Compound Info 
8-Methoxy-2-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4H-9-thia-2,4,5-triaza-fluorene-1,3-dione
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C25H26N4O4S
  1
1
Ki = 1.41 nM
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CP0339071
 Compound Info 
6-Methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-7-methyl-1H-thieno[3,2-d]pyrimidine-2,4-dione
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C23H27N3O4S
  1
1
Ki = 1.45 nM
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CP0293490
 Compound Info 
7-Isopropyl-6-methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-thieno[3,2-d]pyrimidine-2,4-dione
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C25H31N3O4S
  1
1
Ki = 1.5 nM
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CP0316626
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1,7-dihydro-pyrrolo[2,3-d]pyrimidine-2,4-dione
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C21H24N4O3
  1
1
Ki = 1.67 nM
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CP0334602
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-pyrido[3,4-d]pyrimidine-2,4-dione
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C22H24N4O3
  1
1
Ki = 1.78 nM
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CP0251350
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-pyrido[2,3-d]pyrimidine-2,4-dione
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C22H24N4O3
  1
1
Ki = 1.99 nM
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CP0193838
 Compound Info 
7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-5H-9-thia-1,4,5,7-tetraaza-fluorene-6,8-dione
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C23H23N5O3S
  1
1
Ki = 2.06 nM
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CP0334912
 Compound Info 
7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-5H-9-thia-1,3,5,7-tetraaza-fluorene-6,8-dione
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C23H23N5O3S
  1
1
Ki = 2.08 nM
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CP0363623
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-benzo[4,5]thieno[3,2-d]pyrimidine-6-carbonitrile
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C26H24N4O3S
  1
1
Ki = 2.08 nM
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CP0251349
 Compound Info 
7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2-methyl-5H-9-thia-1,4,5,7-tetraaza-fluorene-6,8-dione
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C24H25N5O3S
  1
1
Ki = 2.31 nM
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CP0220027
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-pyrido[3,2-d]pyrimidine-2,4-dione
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C22H24N4O3
  1
1
Ki = 2.5 nM
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CP0300093
 Compound Info 
6-Chloro-7-methoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-quinazoline-2,4-dione
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C24H26ClN3O4
  1
1
Ki = 2.71 nM
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CP0101288
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-benzo[4,5]thieno[3,2-d]pyrimidine-8-carboxylic acid methyl ester
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C27H27N3O5S
  1
1
Ki = 2.84 nM
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CP0099011
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-6,8-dimethyl-1H-quinazoline-2,4-dione
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C25H29N3O3
  1
1
Ki = 2.86 nM
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CP0281405
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-pyrido[4,3-d]pyrimidine-2,4-dione
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C22H24N4O3
  1
1
Ki = 2.87 nM
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CP0278639
 Compound Info 
7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,3-dimethyl-5H-9-thia-1,4,5,7-tetraaza-fluorene-6,8-dione
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C25H27N5O3S
  1
1
Ki = 3.28 nM
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CP0094875
 Compound Info 
6,7-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1-methyl-1H-quinazoline-2,4-dione
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C26H31N3O5
  1
1
Ki = 3.71 nM
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CP0507035
 Compound Info 
2-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4H-9-thia-2,4,5,7-tetraaza-fluorene-1,3-dione
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C23H23N5O3S
  1
1
Ki = 3.74 nM
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CP0200084
 Compound Info 
3-Chloro-7-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-5H-9-thia-1,4,5,7-tetraaza-fluorene-6,8-dione
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C23H22ClN5O3S
  1
1
Ki = 3.83 nM
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CP0405674
 Compound Info 
8-Chloro-2-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-4H-9-thia-2,4,5-triaza-fluorene-1,3-dione
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C24H23ClN4O3S
  1
1
Ki = 4.16 nM
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CP0193331
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-6-phenyl-1H-thieno[3,2-d]pyrimidine-2,4-dione
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C27H27N3O3S
  1
1
Ki = 4.4 nM
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CP0117265
 Compound Info 
(Cis)3-[4-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-butyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C27H29N3O3S
  1
1
Ki = 4.77 nM
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CP0278803
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-pteridine-2,4-dione
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C21H23N5O3
  1
1
Ki = 5.49 nM
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CP0296008
 Compound Info 
(Cis)3-[2-(8-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C25H25N3O3S
  1
1
Ki = 5.76 nM
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CP0081691
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,4-dioxo-1,2,3,4-tetrahydro-benzo[4,5]thieno[3,2-d]pyrimidine-9-carbonitrile
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C26H24N4O3S
  1
1
Ki = 6.6 nM
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CP0352054
 Compound Info 
3-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-7-trifluoromethyl-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C26H24F3N3O3S
  1
1
Ki = 6.84 nM
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CP0257865
 Compound Info 
(Cis)3-[3-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-propyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C26H27N3O3S
  1
1
Ki = 7.7 nM
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CP0272620
 Compound Info 
6,7-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-3H-quinazolin-4-one
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C25H29N3O4
  1
1
Ki = 7.79 nM
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CP0331914
 Compound Info 
(Cis)3-[2-(9-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C25H25N3O3S
  1
1
Ki = 8.67 nM
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CP0299620
 Compound Info 
7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-3-phenyl-5H-9-thia-1,4,5,7-tetraaza-fluorene-6,8-dione
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C29H27N5O3S
  1
1
Ki = 19.8 nM
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CP0214818
 Compound Info 
6-Chloro-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C25H24ClN3O3S
  1
1
Ki = 25 nM
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CP0104415
 Compound Info 
2-Amino-4,5-dimethoxy-N-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-benzamide
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C24H31N3O4
  1
1
Ki = 32.65 nM
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CP0300109
 Compound Info 
(Cis)3-[2-(7-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-1H-benzo[4,5]thieno[3,2-d]pyrimidine-2,4-dione
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C25H25N3O3S
  1
1
Ki = 47 nM
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CP0339046
 Compound Info 
6,7-Dimethoxy-2-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-3,4-dihydro-2H-isoquinolin-1-one
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C26H32N2O4
  1
1
Ki = 58.4 nM
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CP0350146
 Compound Info 
6,7-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2,3-dihydro-1H-quinazolin-4-one
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C25H31N3O4
  1
1
Ki = 71.97 nM
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CP0311748
 Compound Info 
2-[2-(6,7-Dimethoxy-3,4-dihydro-1H-isoquinolin-2-yl)-ethyl]-6-methoxy-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]isoindole
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C26H34N2O3
  1
1
Ki = 83.4 nM
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CP0307684
 Compound Info 
7-[2-(6-Methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-2-phenyl-5H-9-thia-1,4,5,7-tetraaza-fluorene-6,8-dione
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C29H27N5O3S
  1
1
Ki = 160 nM
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CP0103803
 Compound Info 
6,7-Dimethoxy-3-[2-(6-methoxy-1,3,3a,4,5,9b-hexahydro-benzo[e]isoindol-2-yl)-ethyl]-3,4-dihydro-1H-quinazolin-2-one
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C25H31N3O4
  1
1
Ki = 168.2 nM
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CP0280474
 Compound Info 
2-[2-(6,7-Dimethoxy-1,4-dihydro-2H-quinazolin-3-yl)-ethyl]-6-methoxy-2,3,3a,4,5,9b-hexahydro-1H-benzo[e]isoindole
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C25H33N3O3
  1
1
Ki = 189 nM
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